Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
01/2009
01/14/2009EP2013173A2 Pyridine-, isoxazole, thiophenecarboxamide compounds having activity at the glycine transporter glyt1 and uses thereof
01/14/2009EP1258484B1 Novel isoxazole and thiazole compounds and use thereof as drugs
01/14/2009CN101346358A Estrogen modulators
01/13/2009US7476744 Polymorphic crystalline forms of celecoxib
01/13/2009US7476688 Cyclic amidine derivatives
01/13/2009US7476686 e.g. 1-(Benzofuran-2-carbonyl-3-(3-phenoxy-phenyl)-thiourea; viricides; Hepatitis C infection
01/08/2009WO2009005015A1 Substituted isoxazoline or enone oxime compound, and pest control agent
01/08/2009WO2009003719A2 Indane-amine derivatives, their preparation and use as medicaments
01/08/2009CA2692513A1 Indane-amine derivatives, their preparation and use as medicaments
01/07/2009EP2011786A1 Indane-amine derivatives, their preparation and use as medicaments
01/07/2009EP2010507A2 Novel isooxazole derivatives and their uses
01/07/2009EP1569916B1 Substituted aralkyl derivatives
01/06/2009CA2120319C Pharmaceutical for the treatment of skin disorders
01/01/2009US20090005594 Z=reacting Z-C(O) CH2 C(O)-Z ( Z= Cl)or HO C(O) CH2 (CO) OH and a carboxylic acid activating agent e.g. dicyclohexyl carbodiimide with a thiohydrazide compound ; enhances the desirable tumor attacking properties of anticancer agents without further increasing undesirable side-effects
01/01/2009US20090005418 such as 2-benzyl-5-(2,5-difluorophenyl)-3-phenyl-2,3-dihydroisoxazole, useful for treating cellular proliferative diseases such as cancer, hyperplasias, restenosis, cardiac hypertrophy, immune disorders and inflammation in mammals
01/01/2009US20090005370 Isoxazole-imidazole derivatives
01/01/2009US20090005350 Cyclooxygenase-2 selective inhibitors, compositions and methods of use
12/2008
12/31/2008WO2009001942A1 Method for production of 3-hydroxypropan-1-one compound, method for production of 2-propen-1-one compound, and method for production of isoxazoline compound
12/31/2008WO2008115149A8 N-HETEROCYCLIC CARBENE CATALYZED SYNTHESIS OF N-PHENYLISOXAZOLIDIN-5-ONE DERIVATIVE AND SYNTHESIS OF β -AMINO ACID ESTER DERIVATIVE
12/31/2008EP2007759A1 Isoxazole derivatives as calcium channel blockers
12/31/2008EP2007717A1 Novel sulfonamide compounds
12/31/2008CN100446767C Use of GAL3 receptor antagonists for treatment of. depression and/or anxiety and compounds useful in such methods
12/31/2008CA2684632A1 Naphthalene isoxazoline invertebrate pest control agents
12/30/2008US7470807 Suppress production of both prostaglandins and leukotrienes and have reduced side effects; treatment of various inflammatory diseases, autoimmune diseases, allergic diseases, pain and fibrosis; for example, methyl 3-[3-acetylamino-4-cyclopentyloxy-5-(naphthalen-2-yl)phenyl]propionate
12/30/2008US7470715 (+-)-4-{5-[1-(1-Hydroxy-ethyl)-cyclopropyl]-4-phenyl-isoxazol-3-yl}-phenol;new class of isoxazole derivative; breast cancer, migraine, incontinence, vaginal atrophy, bladder infection, senile gynecomastia, diabetes, hypoglycemia, melanoma, impotence, inflammatory bowel disease, CNS and GI disorders
12/24/2008WO2008156601A1 Tricyclic inhibitors of hydroxysteroid dehydrogenases
12/24/2008WO2008156142A1 Novel malonic acid sulfonamide derivative and pharmaceutical use thereof
12/24/2008WO2008126665A3 Isoxazoline compounds and their use in pest control
12/24/2008EP2006286A2 Isoxazole derivative and isothiazole derivative having inhibitory activity on 11 beta -hydroxysteroid dehydrogenase type i
12/24/2008EP2004619A1 1-phenylsulfonyl-diaza heterocyclic amide compounds and their uses as modulators of hydroxsteroid dehydrogenases
12/24/2008EP2004192A2 Modified macrophage migration inhibitory factor inhibitors
12/24/2008EP1687314B1 PREPARATION OF 1-AZA-2-OXA-DIBENZO [e,h] AZULENES AND THEIR USE FOR THE MANUFACTURE OF PHARMACEUTICAL FORMULATIONS FOR THE TREATMENT AND PREVENTION OF CENTRAL NERVOUS SYSTEM DISEASES AND DISORDERS
12/24/2008CN101331114A 2-adamantylurea derivatives as selective 11beta-HSD1 inhibitors
12/24/2008CN100445276C Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
12/24/2008CA2691309A1 Tricyclic inhibitors of hydroxysteroid dehydrogenases
12/23/2008US7468393 Diarylsulfones as 5-HT2A antagonists
12/23/2008CA2331685C Use of compounds for the elevation of pyruvate dehydrogenase activity
12/23/2008CA2245267C Crystal form of n-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamide
12/18/2008WO2008152081A2 Anthelmintic benzo[d]isoxazolyl benzamide derivatives
12/18/2008WO2008130320A3 Novel n- (8-heteroaryltetrahydronaphtalene-2yl) or n- (5- heteroarylchromane-3-yl) carboxamide derivatives for the treatment of pain
12/18/2008WO2008079339A3 Tetracycline derivatives for the treatment of bacterial, viral and parasitic infections
12/18/2008US20080312301 Substituted N-Benzo[D]Isoxazol-3-Yl-Amine Compounds as Inhibitors of Mglur5, Serotonin (5-Ht) and Noradrenaline Receptors, and Uses Thereof
12/18/2008US20080311212 Crystalline isoxazole derivative and pharmaceutical preparation thereof
12/18/2008US20080311113 Method for treating adamts-5-associated disease
12/18/2008CA2691987A1 Antibacterial agents
12/18/2008CA2684671A1 Isoxazoline insecticides
12/17/2008EP2002837A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
12/17/2008EP2001851A2 Amide derivatives and their application for the treament of g protein related diseases
12/17/2008CN100443467C Substituted aromatic amide derivative intemediate thereof, agrohorticultral insecticide containing thereof and method for use thereof
12/16/2008US7465806 N-(1-alkyl-4-piperidinyl)-2-pyrrolecarboxamides, e.g., 1-[5-(5-Chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-1H-pyrrole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide; treating vascular restenosis following angioplasty
12/16/2008US7465805 Isoxazoline derivatives and their use as herbicides
12/11/2008WO2008150231A1 New heterocyclic compounds for treatment of respiratory, airway or inflammatory disorders
12/11/2008US20080306258 Cyclopropane compounds and pharmaceutical use thereof
12/11/2008US20080306127 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners
12/11/2008US20080306125 nuclear receptor modulators such as 6-{4-[3-(2,6-Dichloro-phenyl)-5-isopropyl-isoxazol-4-ylmethoxy]-phenyl}-1-isopropyl-1H-indole-3-carboxylic acid, used for treating dyslipidemia, atherosclerosis, diabetes, raising plasma high density lipoproteins, lowering low density lipoproteins and triglycerides
12/11/2008US20080306124 Polycyclic Oxadiazoles or I Soxazoles and Their Use as Sip Receptor Ligands
12/11/2008US20080306117 Ep4 receptor antagonists
12/11/2008US20080306066 Non-imidazole heterocyclic compounds
12/10/2008EP1999119A2 Novel acetyl-coa carboxylase (acc) inhibitors and their use in diabetes, obesity and metabolic syndrome
12/10/2008EP1756052B1 Improved method for preparing 3-hydroxy-4-hydroxymethyl-pyrrolidine compounds
12/10/2008EP1094816B1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
12/09/2008US7462636 Broadspectrum substituted benzisoxazole sulfonamide HIV protease inhibitors
12/09/2008CA2379061C Antibacterial agents
12/04/2008WO2008035315A3 Inhibitors of phosphodiesterase type-iv
12/04/2008US20080300288 Alkenyldiarylmethanes, Fused Analogs And Syntheses Thereof
12/03/2008EP1997813A1 Substituted isoxazoline compound and pest control agent
12/03/2008EP1997811A2 Indazole, benzoxazole and pyrazolopyridine derivatives as P38 kinase inhibitors
12/03/2008EP1997810A2 Indazole, benzoxazole and pyrazolopyridine derivatives for medical use
12/03/2008EP1997809A2 Indazole, benzoxazole and pyrazolopyridine derivatives for medical use
12/03/2008EP1997807A1 Heterocyclyl-substituted-ethylamino-phenyl derivatives, their preparation and use as medicaments
12/03/2008EP1761262B1 Marine compounds with calcium channel blocking properties for the treatment of cognitive or neurodegenerative diseases
12/02/2008US7459564 thromboembolic and/or inflammatory disorders; 4-Aminomethyl-cyclohexanecarboxylic acid (1-biphenyl-3-yl-2-phenyl-ethyl)-amide; selective inhibitors of serine protease enzymes of the coagulation cascade and/or contact activation system; improved pharmacological properties, plasma kallikrein activity
12/02/2008US7459477 Chemical intermediate for agriculture, horticulture compounds; insecticide, fungicides, miticides
12/02/2008CA2305548C Prostaglandin agonists and their use to treat bone disorders
11/2008
11/27/2008WO2008142134A1 Benzisoxazole derivatives as potassium channel modulators for the treatment of e.g. respiratory diseases, epilepsy and convulsions
11/27/2008WO2008046072A3 Chemical inducers of neurogenesis
11/27/2008US20080293915 Nanoscale Neuromodulating Platform For Retina Neuron Activation Apparatus and Method
11/27/2008US20080293741 Tricyclo Substituted Amides as Glucokinase Modulators
11/27/2008US20080293730 Tricyclo Substituted Amides
11/26/2008EP1995241A1 Inhibitors of ion channels
11/26/2008EP1802566B1 Hexafluoroisopropanol substituted ether derivatives
11/25/2008US7456133 Substituted arylketones
11/20/2008WO2007129019A8 Sulfonamide compounds useful as edg receptor modulators
11/19/2008EP1991542A1 Herbicidal isoxazoline compounds
11/19/2008CN101309909A 2-phenylethylamino derivatives as calcium and/or sodium channel modulators
11/19/2008CN101307017A Amino-methyl substituted tetracycline compounds
11/18/2008US7453001 Such as, ethyl 3-(2-hydroxyphenyl)-6-methyl4-oxo4,5,6,7-tetrahydrobenzo[d]isoxazole-5-carboxylate; intermediates
11/18/2008US7452878 Biaromatic compounds which activate PPARγ type receptors and cosmetic/pharmaceutical compositions comprised thereof
11/18/2008CA2278331C 3-heterocyclyl-substituted benzoyl derivatives
11/13/2008US20080280875 Fused phenyl amido heterocyclic compounds
11/13/2008US20080280334 Method for Preparing 3-Hydroxy-4-Hydroxymethyl-Pyrrolidine Compounds
11/11/2008US7449481 Thio-substituted biaryl-methanesulfinyl derivatives
11/06/2008WO2008116663A3 Heterocyclyl-substituted-tetrahydro-naphthalen-amine derivatives, their preparation and use as medicaments
11/06/2008WO2007110068A3 Novel isooxazole derivatives and their uses
11/06/2008US20080275249 Process for Production of (4,5-Dihydroisoxazol-3-Yl) Thio-Carboxamidine Salts
11/06/2008US20080275070 Aryl Ether Compounds and Their Preparation and Use Thereof
11/05/2008EP1988085A1 Process for production of 3-[5-[4-(cyclopentyloxy)-2-hydroxybenzoyl]-2-[(3-hydroxy-1,2-bezisoxazol-6-yl)methoxy]phenyl]propionate ester and intermediate for the process
11/05/2008EP1987831A1 Compounds effecting glucokinase
11/05/2008CN100430052C Cathepsin cysteine protease inhibitors
11/04/2008US7446222 2-benzyloxy-5-chloro-[1,1';2',1'']terphenyl-3''-carboxylic acid; neuropathic pain; chronic articular pain (e.g. rheumatoid arthritis, osteoarthritis, rheumatoid spondylitis, gouty arthritis and juvenile arthritis) including the property of disease modification and joint structure preservation
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