Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459) |
---|
11/05/2009 | US20090274632 Identification of human T2R receptors that respond to bitter compounds that elicit the bitter taste in compositions, and the use thereof in assays to identify compounds that inhibit (block) bitter taste in composition and use thereof |
11/05/2009 | CA2722733A1 Cyclopentylacrylamide derivative |
11/05/2009 | CA2722704A1 Cyclylamine derivatives as calcium channel blockers |
11/04/2009 | EP1784388B1 Biphenyloxyacetic acid derivatives for the treatment of respiratory disease |
11/03/2009 | US7612092 Nitrogen-containing aromatic derivatives |
11/03/2009 | CA2565660C Ortho substituted aryl or heteroaryl amide compounds |
11/03/2009 | CA2443724C Novel, arylsusfonamide compounds for the treatment of obesity, type ii diabetes and cns-disorders |
11/03/2009 | CA2383327C Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists |
10/29/2009 | WO2009131951A2 Compounds, compositions and methods comprising isoxazole derivatives |
10/29/2009 | WO2009130264A1 PROCESS FOR PREPARING A CRYSTALLINE FORM COMPOUND OF 3-BENZYL-2-METHYL-2,3,3a,4,5,6,7,7a-OCTAHYDROBENZO[d]ISOXAZOL-4-ONE |
10/29/2009 | WO2009130263A1 PROCESS FOR PREPARING A CRYSTALLINE FORM COMPOUND OF 3-BENZYL-2-METHYL-2,3,3a,4,5,6,7,7a-OCTAHYDROBENZO[d]ISOXAZOL-4-ONE |
10/29/2009 | CA2720818A1 Substituted phenoxybenzamides |
10/28/2009 | EP2112142A1 Process for preparing a crystalline form compound of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
10/27/2009 | US7608739 2,3-Dihydrooxadiazoles such as 3-acetyl-5-(2,5-difluorophenyl)-2-phenyl-2,3-dihydro-1,3,4-oxadiazole and 3-[3-acetyl-5-(2,5-difluorophenyl)-2-phenyl-2,3-dihydro-1,3,4-oxadiazol-2-yl]-N,N-dimethylpropan-1-amine that are useful for treating cancer |
10/27/2009 | US7608631 1-(4-{3-[2,6-Dichloro-4-(3,3-dichloro-allyloxy)-phenoxy]-propoxy}-phenyl)-1H-pyrrole, for example; protecting soybean plants against pests such as caterpillars |
10/27/2009 | US7608564 Herbicide; in crops such as wheat, rice, maize, soybeans and cotton they act against broad-leaved weeds and grass weeds without damaging the crop plants; compounds are based on 3-(5,5-disubstituted 2-isoxazolin-3-yl)benzoic acid, esters, thioesters and pyrazolyl ketones thereof |
10/22/2009 | WO2009127338A1 Oxo-heterocyclic substituted carboxylic acid derivates and the use thereof |
10/22/2009 | US20090264486 Compounds, Compositions and Methods Comprising Isoxazole Derivatives |
10/21/2009 | EP2109602A2 Tetracycline derivatives for the treatment of bacterial, viral and parasitic infections |
10/21/2009 | CN101559053A 5-membered heterocycle derivatives, production thereof and use thereof as medicaments |
10/20/2009 | US7605164 Compositions and methods for treating heart failure |
10/20/2009 | US7605150 Drug therapy for Celiac Sprue |
10/20/2009 | CA2585898C Use of (2s,3s,5s)-5-(n-(n-((n-methyl-n-((2-isopropyl-4-thaizolyl)methyl)amino)-carbonyl)valinyl)amino)-2-(n-((5-thiazolyl)methoxycarbonyl)amino)-1,6-diphenyl-3-hydroxyhexane in combination with another protease inhibitor for treating hiv infection |
10/20/2009 | CA2441798C Crystalline isoxazole derivative and medical preparation thereof |
10/15/2009 | WO2009126668A2 Method for preparing 3-trifluoromethyl chalcones |
10/15/2009 | WO2008145615A3 Aminoazoline and urea derivatives for combating animal pests |
10/15/2009 | WO2008115149A9 N-HETEROCYCLIC CARBENE CATALYZED SYNTHESIS OF N-PHENYLISOXAZOLIDIN-5-ONE DERIVATIVE AND SYNTHESIS OF β -AMINO ACID ESTER DERIVATIVE |
10/15/2009 | US20090258884 Substituted amides |
10/15/2009 | US20090258868 Heterocyclic aspartyl protease inhibitors |
10/15/2009 | CA2720530A1 Sulfonamides |
10/15/2009 | CA2718668A1 Method for preparing 3-trifluoromethyl chalcones |
10/14/2009 | EP1720829B1 Derivatives of heteroaryl-alkylcarbamates, preparation method thereof and use of same as faah enzyme inhibitors |
10/14/2009 | EP1658267B1 Inhibitors of cathepsin s |
10/14/2009 | CN100549003C 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers |
10/13/2009 | US7601674 α-oxygenated or α-thiolated carboxylic acid phenethylamide derivatives |
10/08/2009 | WO2009123241A1 Inhibitor of plasminogen activator inhibitor-1 |
10/08/2009 | WO2009122034A2 Novel hsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof |
10/08/2009 | US20090253659 Cycloalkylidene Compounds As Modulators of Estrogen Receptor |
10/08/2009 | US20090253656 Bcrp/abcg2 inhibitor |
10/08/2009 | CA2718488A1 Novel dhsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof |
10/07/2009 | EP2107052A1 Novel n-(2-aminophenyl)benzamide derivative having an urea structure |
10/06/2009 | US7598412 Cystic fibrosis transmembrane conductance regulator; ABC transporter mediated diseases like cystic fibrosis; 5-methoxy-N-((1-(3,4-dimethoxyphenyl)-cyclohexyl)methyl)benzofuran-2-carboxamide; or sulfonamide analogs; chloride or bicarbonate channel modulators |
10/06/2009 | US7598391 Heteroaryl-ureas and their use as glucokinase activators |
10/06/2009 | US7598389 Silylated carboxamides |
10/06/2009 | US7598283 Controlling cell proliferation, cell differentiation,autoimmune disease; N-[4-(3-amino-1,2-benzisoxazol-4-yl)phenyl]-N'-(3-methylphenyl)urea; 2-[4-(3-amino-1H-indazol-4-yl)phenyl]-N-(3-chlorophenyl)acetamide; N-[4-(3-amino-1,2-benzisothiazol-4-yl)phenyl]-N'-(3,5-dimethylphenyl)urea; anticarcinogenic |
10/06/2009 | US7598280 For the treatment, prevention and management of inflammatory and autoimmune diseases and disorders; for example, (1R,2S,3R)-1-(2-(5-methylisoxazol-3-yl)-1H-imidazol-5-yl)butane-1,2,3,4-tetraol |
10/06/2009 | US7598236 Diazabicyclic central nervous system active agents |
10/06/2009 | CA2301377C N-aroylphenylalanine derivatives |
10/01/2009 | WO2009119652A1 USE OF BENZOPHENONE DERIVATIVE OR SALT THEREOF AND TNF α INHIBITOR IN COMBINATION AND PHARMACEUTICAL COMPOSITION CONTAINING THE DERIVATIVE OR SALT THEREOF AND THE INHIBITOR |
10/01/2009 | WO2009118125A1 4-(3-aminobenzoyl)-5-cyclopropylisoxazoles effective as herbicides |
10/01/2009 | US20090247547 Hydroxamate-based inhibitors of deacetylases b |
10/01/2009 | US20090247509 for treating central nervous system disorders such as psychological disorders, drug dependence and abuse, dyskinesia, dementia, anxiety disorders, sleep disorders and mood disorders |
10/01/2009 | CA2719533A1 4-(3-aminobenzoyl)-5-cyclopropylisoxazoles effective as herbicides |
10/01/2009 | CA2719290A1 Use of benzophenone derivative or salt thereof and tnf.alpha. inhibitor in combination and pharmaceutical composition containing the derivative or salt thereof and the inhibitor |
09/30/2009 | EP2105437A1 4-(3-Aminobenzoyl)-5-cyclopropylisoxazols as herbicides |
09/30/2009 | EP2105435A1 Hydrazone derivative |
09/30/2009 | EP2104664A1 Tetrahydrobenzoisoxazole - and tetrahydroindazole derivatives as modulators of the mitotic motor protein |
09/30/2009 | EP1501361B1 3-heteroaryl substituted 5-methyloxymethyl isoxazolines used as herbicides |
09/29/2009 | US7595332 Such as N-(4-tert-butylphenyl)-4-(2-pyridinyl)benzamide for treatment of urinary incontinence, pain, inflammatory thermal hyperalgesia, and/or bladder overactivity |
09/29/2009 | US7595309 For therapy of bacterial infections and neoplasms, |
09/29/2009 | US7595162 Methods of labeling polynucleotides with energy transfer dyes |
09/24/2009 | WO2009076454A3 Compounds that modulate intracellular calcium |
09/24/2009 | WO2009035949A3 Soluble epoxide hydrolase inhibitors |
09/24/2009 | US20090239798 Compounds, Methods and Formulations for the Oral Delivery of a Glucagon-Like Peptide (Glp)-1 Compound or a Melanocortin-4 Receptor (Mc4) Agonist Peptide |
09/23/2009 | EP2102155A1 Aryl compounds as ppar ligands and their use |
09/23/2009 | EP1377288B1 2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase iv and use |
09/23/2009 | CN101538230A Beta-amino ketones compound with anti-diabetic activity |
09/23/2009 | CN100543017C Novel keto-oxadiazole derivatives as cathepsin inhibitors |
09/22/2009 | US7592456 Arylsulfonylnaphthalene derivatives as 5HT2A antagonists |
09/22/2009 | US7592354 Administering a stimulantfor the endogenous production/ release of somatotropins; 3-((1-(2-aminoprop-2-yl)carbonylamino-),2-(phenylmethoxymethyl-)ethyl-),5-(morpholino-carbonyloxymethyl-)-5,6,7,8-tetrahydro-1,2,4-triazolo(4,3-)pyridine; osteoporosis; obesity;improving bone densisty, muscle mass/strength |
09/17/2009 | WO2009112275A1 Pesticidal condensed - ring aryl compounds |
09/17/2009 | US20090233975 Hair resiliency/body improver and hair cosmetic |
09/17/2009 | US20090233915 mitogen-activated protein kinase inhibitors such as 3,4-difluoro-2-(2-fluoro-4-iodo-phenylamino)-N-(2-hydroxy-ethoxy)-5(2-hydroxy-ethoxymethyl)-benzamide, used to treat proliferative diseases, for example, cancers, psoriasis, restenosis, autoimmune diseases and atherosclerosis |
09/17/2009 | CA2718199A1 Pesticidal condensed-ring aryl compounds |
09/16/2009 | EP2100605A1 Bis(thio-hydrazide amide) compounds in combination with taxol for treating cancer |
09/16/2009 | EP1581488B1 Inhibitors of tace |
09/16/2009 | EP1478364B1 Selective antibacterial agents |
09/16/2009 | CN101535282A A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
09/16/2009 | CN101535281A A salt of 3-benzyl-2-methyl-2,3,3a,4,5,6,7,7a-octahydrobenzo[d]isoxazol-4-one |
09/16/2009 | CN100540534C N-alkynyl-2- (substituted aryloxy) alkylthioamide derivatives as fungicides |
09/15/2009 | US7589232 5-[(3-Cyclopentylpropanoyl)(4-dec-1-ynylbenzyl)amino]-2-hydroxybenzoic acid; inflammatory disorder, obesity and/or metabolic disorders mediated by insulin resistance or hyperglycemia, comprising diabetes, inadequate glucose tolerance, insulin resistance, hyperlipidemia, hypertriglycerimia |
09/15/2009 | US7589207 Chemokine receptors; inhibition of HIV replication; acquired immune deficiency syndrome (AIDS); cis N-(4-{2-[3-(2-methyl-1H-benzimidazol-1-yl)-8-azabicyclo[3.2.1]oct-8-yl]ethyl}-4-phenylcyclohexyl)-1H-pyrazole-4-carboxamide |
09/15/2009 | US7589102 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
09/15/2009 | US7589094 N- (3-amino-2-hydroxy-propyl) substituted alkylamide compounds |
09/15/2009 | US7589089 Inhibitors for GlyT-1 |
09/15/2009 | CA2429220C Gaba enhancers in the treatment of diseases relating to reduced neurosteroid activity |
09/11/2009 | WO2009111447A2 Isosorbide derivatives and their use as flavor modifiers, tastants, and taste enhancers |
09/11/2009 | CA2716741A1 Isosorbide derivatives and their use as flavor modifiers, tastants, and taste enhancers |
09/10/2009 | US20090227790 A kit for treating a disorder characterized by loss of dopaminergic and/or motoneurons, for treating Parkinson's disease, amyotrophic lateral sclerosis (ALS), or limiting damage to neuronal cells by Parkinsonian conditions |
09/10/2009 | US20090227645 Pharmaceutical compositions of valdecoxib |
09/10/2009 | US20090227604 Vitamin d receptor modulators |
09/10/2009 | US20090227592 Compounds effecting glucokinase |
09/09/2009 | EP2098517A1 Novel phenyl-isoxazol-3-ol derivative |
09/09/2009 | EP2097396A2 Process for the preparation of 5-hydroxyisoxazolidines, 5-isoxazolidinones, b-amino acids, b-amino aldehydes and derivatives thereof |
09/09/2009 | EP2097380A1 New haloalkylsulfone substituted compounds useful for treating obesity and diabetes |
09/09/2009 | CN101528716A Compounds and methods for inhibiting the interaction of BCL proteins with binding partners |
09/09/2009 | CN100537527C Aryl and biaryl compounds having MCH modulatory activity |
09/08/2009 | US7585859 PDE4B inhibitors and uses therefor |
09/03/2009 | WO2009105906A1 Flavor molecules |
09/03/2009 | WO2009068171A3 Chiral 3-(benzylsulfinyl)-5,5-dimethyl-4,5-dihydroisoxazole derivatives and 5,5-dimethyl-3-[(1h-pyrazol-4-ylmethyl)sulfinyl]-4,5-dihydroisoxazole derivatives, method for the production thereof, and use of same as herbicides and plant growth regulators |