Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
10/1999
10/19/1999US5968937 For treatment and/or prevention of hypertension, cardiac insufficiency, coronary vasospasm, cardiac ischemia, renal vasospasm, liver cirrhosis, congestive heart failure, nephrotic syndrome, brain edema, cerebral ischemia
10/19/1999US5968930 Tricyclic diazepine vasopressin antagonists and oxytocin antagonists
10/19/1999US5968929 Piperazino derivatives as neurokinin antagonists
10/16/1999CA2269049A1 N-acyl and n-aroyl aralkyl amides
10/14/1999WO1999051605A1 PYRROLO[1,2-a]PYRAZINE sPLA2 INHIBITOR
10/14/1999WO1999051565A1 Novel local anesthetic compounds and uses
10/14/1999CA2326522A1 Pyrrolo¬1,2-a|pyrazine spla2 inhibitor
10/14/1999CA2315946A1 Novel local anesthetic compounds and uses
10/13/1999EP0949242A1 Aromatic amine derivatives having nos inhibitory effect
10/13/1999EP0948492A1 Process for the preparation of heteroaryl-phenylalanines
10/13/1999EP0948489A1 Piperazine compounds as inhibitors of mmp or tnf
10/13/1999CN1231661A Aralkyl and aralkylidene heterocyclic lactams and imides
10/13/1999CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof
10/13/1999CA2268621A1 2-pipirazinone-1-acetic acid derivative, production and use thereof
10/12/1999US5965774 Substituted anilide derivative
10/12/1999US5965558 2 or 2,3-di((2-carboxyethylenearyl)quinoxalines; purification of proteins and glycoproteins; units including protein tyrosine phosphatases and proteins with src-homology-2 domains; antidiabetics,-allergens,-coagulants
10/12/1999US5965054 Comprising salts consisting of alkyl substituted, nitrogen-containing heterocyclic delocalized aromatic cations, and their perfluoro derivatives; high energy, high voltage
10/07/1999WO1999050254A1 Quinoxalinones as serine protease inhibitors such as factor xa and thrombin
10/07/1999WO1999050247A1 Compounds with activity on muscarinic receptors
10/07/1999WO1999050230A1 Inhibitors of serine proteases, particularly hepatitis c virus ns3 protease
10/06/1999EP0946524A1 Heterocyclic carboxylic acid derivatives, the production and use thereof as endothelin receptor antagonists
10/06/1999EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity
10/06/1999EP0946518A1 Modulators of proteins with phosphotyrosine recognition units
10/06/1999EP0946501A1 Prevention of loss and restoration of bone mass by certain prostaglandin agonists
10/06/1999CN1230540A Preparation of N-tert-butyl-2-piperazine carboxyl amides
10/05/1999US5962695 Aromatic amidine derivatives and salts thereof
10/05/1999US5962492 Antiasthma agents; antiinflammatory agents
10/05/1999US5962489 Fungicides
10/05/1999US5962483 Antiasthma agents; antiinflammatory agents
10/05/1999CA2158824C N-substituted phenylcarbamic acid derivatives, a process for production thereof, agricultural and horticultural fungicides, intermediates of the derivatives and a process for production thereof
09/1999
09/29/1999EP0945444A1 Dihydrophenazinecarboxylic acid derivatives
09/29/1999EP0945434A1 Process for producing halogenated heteroaryl compounds
09/29/1999EP0945431A2 Process and intermediates for the preparation of phenylacetic derivatives
09/29/1999EP0944582A1 Ketobenzamides as calpain inhibitors
09/29/1999CN1230180A D4 receptor selectivity piperazine derivatives
09/28/1999US5958959 Administering 5-methylisoxazole-4-carboxylic acid-(4-trifluoromethyl)anilide or 2-cyano-3-hydroxy-n-(4-(trifluoromethyl)phenyl)-2-butenamide
09/28/1999US5958952 Substituted phenylamindines, medicaments containing these compounds and process for producing them
09/28/1999US5958839 Herbicidal compounds
09/23/1999WO1999047549A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase)
09/23/1999WO1999047508A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999CA2323783A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999CA2289621A1 Piperazines as inhibitors of fructose-1,6-bisphosphatase (fbpase)
09/22/1999EP0655063B1 Ethynyl alanine amino diol compounds having a piperazinyl-terminated group or a piperazinyl-alkylamino-terminated group for treatment of hypertension
09/22/1999CN1229405A Novel acetamide derivatives and protease inhibitors
09/21/1999US5955461 Quinoxalinedione derivatives, their production and use in pharmaceutical agents
09/16/1999WO1999046268A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
09/16/1999WO1999046237A1 Modulators of protein tyrosine phosphatases
09/16/1999WO1999046236A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999028304A9 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
09/16/1999CA2323472A1 Modulators of protein tyrosine phosphatases
09/15/1999EP0749421B1 Sulphonamide derivatives as aspartyl protease inhibitors
09/15/1999EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors
09/15/1999CN1228773A Heterocyclic metalloprotease inhibitors
09/14/1999US5952503 Method for producing optically-active 2-piperazinecarboxylic acid derivatives
09/14/1999US5952386 Excellent insecticidal activity for the control of noxious insects
09/14/1999US5952359 Thiazoles and their agricultural compositions
09/14/1999US5952316 2-amino-1,3-propanediol compound and immunosuppressant
09/14/1999CA1340734C Substituted bridged-diazabicycloalkyl quinolone carboxylic acids
09/08/1999EP0940139A2 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers
09/08/1999CN1228090A Naphthyridines with affect IL-4 and G-CSF
09/07/1999US5948790 Retroviral protease inhibitors
09/07/1999US5948779 Substituted condensation products of n-benzyl-3-indenyl acetamides with heterocyclic aldehydes
09/02/1999WO1999043662A1 Solid support synthesis of 2-oxopiperazines
09/02/1999WO1999024460A3 Dipeptide nitriles
09/02/1999WO1998034632A9 Compounds and compositions for delivering active agents
09/02/1999CA2321302A1 Solid support synthesis of 2-oxopiperazines
08/1999
08/31/1999US5945534 Process for the preparation of optically active piperazine-2-carboxylic acid derivatives
08/31/1999US5945443 Kappa agonist compounds and pharmaceutical formulations thereof
08/31/1999US5945418 Administering to the mammal to inhibit a mammalian protein kinase p38 which causes cell proliferation, cell death and response to extracellular stimuli
08/26/1999WO1999042463A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042461A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists
08/26/1999WO1999042455A1 Antiviral agents
08/26/1999WO1999042436A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/26/1999WO1999029700A3 Cyclohexadiene-derivatives as pesticides
08/26/1999CA2320469A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
08/25/1999EP0937048A1 HETEROCYCLE DERIVATIVES WHICH INHIBIT FACTOR Xa
08/25/1999CN1226594A Method for coal liquefaction
08/24/1999US5942641 Fluorenone derivatives, process for preparing the same and central or peripheral nerve degeneration repair and protective agent
08/19/1999WO1999041242A1 Di-substituted naphthyl derivatives, preparation thereof, pharmaceutical compositions containing them
08/19/1999WO1999015894A3 Method of identification of leads or active compounds
08/18/1999EP0936216A1 Novel acetamide derivatives and protease inhibitors
08/18/1999EP0935599A1 2-methoxyphenylpiperazine derivatives
08/18/1999EP0935597A2 Dihydropyrones with improved antiviral activity
08/18/1999CN1226229A Glyoxalic acid derivative
08/17/1999US5939563 Fungicides
08/17/1999US5939549 From corresponding tetrahydropyrazine carboxylic acid nitriles and olefins
08/17/1999US5939421 Treatment of immunoinflammatory and autoimmune diseases such as rheumatoid arthritis, transplant rejection; inhibit kinase(s) that regulate activation of transcription factors to prevent production of inflammatory proteins
08/17/1999US5939381 4-(4-(phenoxyacetyl)aminophenyl)butyric acid as a carrier for drug delivery
08/17/1999US5939359 Herbicidal pyrazine derivatives
08/17/1999US5939268 Diels-alder reaction product of a diene and a dienophile; chemical intermediates for drugs, solid phase synthesis
08/12/1999WO1999040089A1 Benzothiadiazoles and derivatives
08/12/1999WO1999040083A2 Bifunctional tryptase inhibitors
08/12/1999WO1999040075A1 Sulfonamide derivatives, process for producing the same and utilization thereof
08/12/1999WO1999040073A2 Tryptase inhibitors
08/12/1999WO1999040061A2 Novel dihydroxyhexanoic acid derivatives
08/12/1999WO1999028304A3 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
08/12/1999CA2318977A1 Derivatives of benzoxadiazoles, benzothiadiazoles, benzotriazoles and quinoxalines
08/12/1999CA2317017A1 Sulfonamide derivatives, their production and use
08/11/1999EP0934992A1 Light-emitting material for organo-electroluminescence device and organic electroluminescence device
08/11/1999EP0934920A2 Preparation of hydrogenated compounds using noble metal Raney catalysts