Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673) |
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10/19/1999 | US5968937 For treatment and/or prevention of hypertension, cardiac insufficiency, coronary vasospasm, cardiac ischemia, renal vasospasm, liver cirrhosis, congestive heart failure, nephrotic syndrome, brain edema, cerebral ischemia |
10/19/1999 | US5968930 Tricyclic diazepine vasopressin antagonists and oxytocin antagonists |
10/19/1999 | US5968929 Piperazino derivatives as neurokinin antagonists |
10/16/1999 | CA2269049A1 N-acyl and n-aroyl aralkyl amides |
10/14/1999 | WO1999051605A1 PYRROLO[1,2-a]PYRAZINE sPLA2 INHIBITOR |
10/14/1999 | WO1999051565A1 Novel local anesthetic compounds and uses |
10/14/1999 | CA2326522A1 Pyrrolo¬1,2-a|pyrazine spla2 inhibitor |
10/14/1999 | CA2315946A1 Novel local anesthetic compounds and uses |
10/13/1999 | EP0949242A1 Aromatic amine derivatives having nos inhibitory effect |
10/13/1999 | EP0948492A1 Process for the preparation of heteroaryl-phenylalanines |
10/13/1999 | EP0948489A1 Piperazine compounds as inhibitors of mmp or tnf |
10/13/1999 | CN1231661A Aralkyl and aralkylidene heterocyclic lactams and imides |
10/13/1999 | CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof |
10/13/1999 | CA2268621A1 2-pipirazinone-1-acetic acid derivative, production and use thereof |
10/12/1999 | US5965774 Substituted anilide derivative |
10/12/1999 | US5965558 2 or 2,3-di((2-carboxyethylenearyl)quinoxalines; purification of proteins and glycoproteins; units including protein tyrosine phosphatases and proteins with src-homology-2 domains; antidiabetics,-allergens,-coagulants |
10/12/1999 | US5965054 Comprising salts consisting of alkyl substituted, nitrogen-containing heterocyclic delocalized aromatic cations, and their perfluoro derivatives; high energy, high voltage |
10/07/1999 | WO1999050254A1 Quinoxalinones as serine protease inhibitors such as factor xa and thrombin |
10/07/1999 | WO1999050247A1 Compounds with activity on muscarinic receptors |
10/07/1999 | WO1999050230A1 Inhibitors of serine proteases, particularly hepatitis c virus ns3 protease |
10/06/1999 | EP0946524A1 Heterocyclic carboxylic acid derivatives, the production and use thereof as endothelin receptor antagonists |
10/06/1999 | EP0946519A1 Benzamide derivatives having a vasopressin antagonistic activity |
10/06/1999 | EP0946518A1 Modulators of proteins with phosphotyrosine recognition units |
10/06/1999 | EP0946501A1 Prevention of loss and restoration of bone mass by certain prostaglandin agonists |
10/06/1999 | CN1230540A Preparation of N-tert-butyl-2-piperazine carboxyl amides |
10/05/1999 | US5962695 Aromatic amidine derivatives and salts thereof |
10/05/1999 | US5962492 Antiasthma agents; antiinflammatory agents |
10/05/1999 | US5962489 Fungicides |
10/05/1999 | US5962483 Antiasthma agents; antiinflammatory agents |
10/05/1999 | CA2158824C N-substituted phenylcarbamic acid derivatives, a process for production thereof, agricultural and horticultural fungicides, intermediates of the derivatives and a process for production thereof |
09/29/1999 | EP0945444A1 Dihydrophenazinecarboxylic acid derivatives |
09/29/1999 | EP0945434A1 Process for producing halogenated heteroaryl compounds |
09/29/1999 | EP0945431A2 Process and intermediates for the preparation of phenylacetic derivatives |
09/29/1999 | EP0944582A1 Ketobenzamides as calpain inhibitors |
09/29/1999 | CN1230180A D4 receptor selectivity piperazine derivatives |
09/28/1999 | US5958959 Administering 5-methylisoxazole-4-carboxylic acid-(4-trifluoromethyl)anilide or 2-cyano-3-hydroxy-n-(4-(trifluoromethyl)phenyl)-2-butenamide |
09/28/1999 | US5958952 Substituted phenylamindines, medicaments containing these compounds and process for producing them |
09/28/1999 | US5958839 Herbicidal compounds |
09/23/1999 | WO1999047549A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase) |
09/23/1999 | WO1999047508A1 Benzenesulfonamide-derivatives and their use as medicaments |
09/23/1999 | CA2323783A1 Benzenesulfonamide-derivatives and their use as medicaments |
09/23/1999 | CA2289621A1 Piperazines as inhibitors of fructose-1,6-bisphosphatase (fbpase) |
09/22/1999 | EP0655063B1 Ethynyl alanine amino diol compounds having a piperazinyl-terminated group or a piperazinyl-alkylamino-terminated group for treatment of hypertension |
09/22/1999 | CN1229405A Novel acetamide derivatives and protease inhibitors |
09/21/1999 | US5955461 Quinoxalinedione derivatives, their production and use in pharmaceutical agents |
09/16/1999 | WO1999046268A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) |
09/16/1999 | WO1999046237A1 Modulators of protein tyrosine phosphatases |
09/16/1999 | WO1999046236A1 Modulators of protein tyrosine phosphatases (ptpases) |
09/16/1999 | WO1999028304A9 Pdgf receptor kinase inhibitory compounds, their preparation and compositions |
09/16/1999 | CA2323472A1 Modulators of protein tyrosine phosphatases |
09/15/1999 | EP0749421B1 Sulphonamide derivatives as aspartyl protease inhibitors |
09/15/1999 | EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors |
09/15/1999 | CN1228773A Heterocyclic metalloprotease inhibitors |
09/14/1999 | US5952503 Method for producing optically-active 2-piperazinecarboxylic acid derivatives |
09/14/1999 | US5952386 Excellent insecticidal activity for the control of noxious insects |
09/14/1999 | US5952359 Thiazoles and their agricultural compositions |
09/14/1999 | US5952316 2-amino-1,3-propanediol compound and immunosuppressant |
09/14/1999 | CA1340734C Substituted bridged-diazabicycloalkyl quinolone carboxylic acids |
09/08/1999 | EP0940139A2 Substituted guanidines and derivatives thereof as modulators of neurotransmitter release and novel methodology for identifying neurotransmitter release blockers |
09/08/1999 | CN1228090A Naphthyridines with affect IL-4 and G-CSF |
09/07/1999 | US5948790 Retroviral protease inhibitors |
09/07/1999 | US5948779 Substituted condensation products of n-benzyl-3-indenyl acetamides with heterocyclic aldehydes |
09/02/1999 | WO1999043662A1 Solid support synthesis of 2-oxopiperazines |
09/02/1999 | WO1999024460A3 Dipeptide nitriles |
09/02/1999 | WO1998034632A9 Compounds and compositions for delivering active agents |
09/02/1999 | CA2321302A1 Solid support synthesis of 2-oxopiperazines |
08/31/1999 | US5945534 Process for the preparation of optically active piperazine-2-carboxylic acid derivatives |
08/31/1999 | US5945443 Kappa agonist compounds and pharmaceutical formulations thereof |
08/31/1999 | US5945418 Administering to the mammal to inhibit a mammalian protein kinase p38 which causes cell proliferation, cell death and response to extracellular stimuli |
08/26/1999 | WO1999042463A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists |
08/26/1999 | WO1999042461A1 Substituted quinoxaline derivatives as interleukin-8 receptor antagonists |
08/26/1999 | WO1999042455A1 Antiviral agents |
08/26/1999 | WO1999042436A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors |
08/26/1999 | WO1999029700A3 Cyclohexadiene-derivatives as pesticides |
08/26/1999 | CA2320469A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors |
08/25/1999 | EP0937048A1 HETEROCYCLE DERIVATIVES WHICH INHIBIT FACTOR Xa |
08/25/1999 | CN1226594A Method for coal liquefaction |
08/24/1999 | US5942641 Fluorenone derivatives, process for preparing the same and central or peripheral nerve degeneration repair and protective agent |
08/19/1999 | WO1999041242A1 Di-substituted naphthyl derivatives, preparation thereof, pharmaceutical compositions containing them |
08/19/1999 | WO1999015894A3 Method of identification of leads or active compounds |
08/18/1999 | EP0936216A1 Novel acetamide derivatives and protease inhibitors |
08/18/1999 | EP0935599A1 2-methoxyphenylpiperazine derivatives |
08/18/1999 | EP0935597A2 Dihydropyrones with improved antiviral activity |
08/18/1999 | CN1226229A Glyoxalic acid derivative |
08/17/1999 | US5939563 Fungicides |
08/17/1999 | US5939549 From corresponding tetrahydropyrazine carboxylic acid nitriles and olefins |
08/17/1999 | US5939421 Treatment of immunoinflammatory and autoimmune diseases such as rheumatoid arthritis, transplant rejection; inhibit kinase(s) that regulate activation of transcription factors to prevent production of inflammatory proteins |
08/17/1999 | US5939381 4-(4-(phenoxyacetyl)aminophenyl)butyric acid as a carrier for drug delivery |
08/17/1999 | US5939359 Herbicidal pyrazine derivatives |
08/17/1999 | US5939268 Diels-alder reaction product of a diene and a dienophile; chemical intermediates for drugs, solid phase synthesis |
08/12/1999 | WO1999040089A1 Benzothiadiazoles and derivatives |
08/12/1999 | WO1999040083A2 Bifunctional tryptase inhibitors |
08/12/1999 | WO1999040075A1 Sulfonamide derivatives, process for producing the same and utilization thereof |
08/12/1999 | WO1999040073A2 Tryptase inhibitors |
08/12/1999 | WO1999040061A2 Novel dihydroxyhexanoic acid derivatives |
08/12/1999 | WO1999028304A3 Pdgf receptor kinase inhibitory compounds, their preparation and compositions |
08/12/1999 | CA2318977A1 Derivatives of benzoxadiazoles, benzothiadiazoles, benzotriazoles and quinoxalines |
08/12/1999 | CA2317017A1 Sulfonamide derivatives, their production and use |
08/11/1999 | EP0934992A1 Light-emitting material for organo-electroluminescence device and organic electroluminescence device |
08/11/1999 | EP0934920A2 Preparation of hydrogenated compounds using noble metal Raney catalysts |