Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
05/2001
05/10/2001CA2389773A1 Activators of soluble guanylate cyclase
05/09/2001EP1097970A2 Water-soluble monoazo compounds, process for their preparation and their use as dyestuffs
05/09/2001EP1097927A1 Cyanoiminoquinoxaline derivatives
05/09/2001EP1097145A1 Polyhydroalkylpyrazine derivatives and their preparation and medicines containing them
05/09/2001EP0745594B1 Process for producing 6-substituted 2(1h)-quinoxalinone
05/08/2001US6228942 Dehydration to esterify or amidate surface of oxidized or aminated carbon powder or fiber suspended in solution containing a monomer or polymer having amine, hydroxy, and/or viny ether groups
05/03/2001WO2001030749A1 Novel compounds
05/02/2001EP1095936A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
05/02/2001EP1095029A1 Piperazine derivatives inhibiting human immunodeficiency virus replication
05/02/2001EP1095015A2 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
05/02/2001EP1094826A1 Novel therapeutic agents that modulate alpha-1a adrenergic receptors
05/02/2001EP1094810A1 Use of prenyltransferase inhibitors for preparing a medicine for treating pathologies resulting from heterotrimeric g protein membrane fixation
05/02/2001EP0984959A4 Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds
05/02/2001EP0983257A4 Aromatic sulfonyl alpha-cycloamino hydroxamic acid compounds
05/02/2001EP0973392A4 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/02/2001CN1293666A Benzenesulfonamide-derivatives and their use as medicaments
05/01/2001US6225471 Preparing aqueous medium containing ammonium compound and acetoin compound; heating, refluxing and subliming simultaneously; cooling surface for collecting sublimation prodcut; collecting alkyl-pyrazine
05/01/2001US6225334 Glyoxylic acid derivatives
05/01/2001US6225329 Useful in the treatment of type i diabetes, type ii diabetes, impaired glucose tolerance, insulin autoimmunity diseases with dysfunctions of the coagulation system, allergic diseases
05/01/2001US6225074 Mixing test sample with reagent solution of chloramphenicol or derivative, an acyl coenzyme a compound, and a tetrazolium salt, then observing optical response; solution does not contain redox enzyme
04/2001
04/26/2001WO2000075121A3 Process for preparing 10,11-methanobenzosuberane derivatives
04/25/2001EP1093819A2 Compounds and compositions for delivering active agents
04/24/2001US6222062 Beta-ketoester compounds
04/24/2001US6221865 Inhibitors of protein farnesyltransferase and protein geranylgeranyltransferase.
04/22/2001WO2002102250A1 $g(in vivo) imaging
04/22/2001CA2422767A1 In vivo imaging
04/19/2001WO2001027096A1 Aminomethyl-(hetero)aryl derivatives and their use as tryptase inhibitors
04/19/2001US20010000344 N-(2-(R)-amino-3-mercaptopropyl)-L-penicillaminyl-1,2,3,4 -tetrahydro-3(S)-isoquinoline carbonyl methionine methylester cyclic disulfide, for example; administering as antitumor agent or to treat restenosis
04/18/2001EP1091943A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
04/18/2001EP1091737A2 Calcium channel blockers
04/18/2001EP0968250B1 Soluble chromophores having improved solubilising groups
04/18/2001EP0904265B1 Preparation of bis(fluoroalkylenesulfonyl)imides and (fluoroalkylsulfonyl) (fluorosulfonyl)imides
04/18/2001CN1291892A Substituted oxoazaheterocyclyl factor Xa inhibitors
04/17/2001US6218576 Process for producing a diarylamine
04/17/2001US6218551 N-(allyloxycarbonyl)proline derivatives
04/17/2001US6218544 Heterocyclic esters and amides
04/17/2001US6218393 Anthranilic acid derivatives as multi drug resistance modulators
04/17/2001US6218391 Triazinones and derivatives thereof
04/12/2001WO2001025244A1 Complexes of mid-transition metals and unsaturated nitrogenous ligands as single-site catalysts
04/12/2001WO2001025229A1 Amide compounds
04/12/2001WO2001025219A2 Piperazine compounds
04/12/2001WO2001025217A1 New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
04/12/2001WO2001025181A1 Carboxylic acid derivatives and drugs containing the same
04/12/2001CA2386157A1 Amide compounds
04/11/2001EP1090914A2 Processes and intermediates for manufacturing retroviral protease inhibiting compounds
04/11/2001EP1089979A1 Substituted quinoxalin-2(1h)-ones useful as hiv reverse transcriptase inhibitors
04/11/2001CN1291183A N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl-3-substituted-alkyl, aryl or heteroarylamides) as matrix metallo protein inhibitors
04/10/2001US6215030 Catalytic reduction of acids, esters and anhydrides to alcohols
04/10/2001US6214995 Synthetic polymer stabilized against thermal and photo deterioration with a 7,7,9,9-tetramethyl-1,3,8-triazaspiro(4,5)decan-2,4-dione derivative of given formula
04/10/2001US6214835 Dihalopropene compounds insecticides containing them as active ingredients, and intermediates for their production
04/04/2001EP1087981A2 Prenyl transferase inhibitors
04/04/2001EP1087953A1 Nitrate salts of antihypertensive medicines
04/04/2001EP1087941A2 Thiolesters and uses thereof
04/04/2001EP0824515B1 Substituted phenyl amidines, medicaments containing these compounds and process for producing them
04/04/2001CN1290255A Dihydroxyhexanoic acid derivatives
04/04/2001CN1290254A Sulfonamide derivatives process for producing the same and utilization thereof
04/04/2001CN1290252A Method for producing heteroaromatic aldehydes
04/03/2001US6211241 Aryl sulfonamides and sulfamide derivatives and uses thereof
04/03/2001US6211240 O-benzyl oxime ether derivatives and their use as pesticides
04/03/2001US6211196 Benzyloxy-substituted, fused N-heterocycles, processes for their preparation, and their use as bradykinin receptor antagonists
04/03/2001US6211183 Selective factor Xa inhibitors
03/2001
03/29/2001WO2001021584A1 Tyrosine derivatives
03/28/2001EP1086103A1 Pyrido 2,3-b]indolizine derivatives and aza analogues thereof; crf 1? specific ligands
03/28/2001EP1086076A1 Sulfonamide inhibitors of aspartyl protease
03/28/2001EP1085895A1 Bradykinin antagonists
03/28/2001EP1085894A1 Beta 3-adrenergic receptor agonists
03/28/2001EP1085889A2 Novel therapeutic agents that modulate endothelin receptors
03/28/2001EP1085887A2 Novel angiotensin receptor modulators and their uses
03/28/2001EP1085870A2 Multivalent agonists, partial agonists and antagonists of the gaba receptors
03/28/2001EP1085868A1 H1-histamine receptor antagonists
03/28/2001EP1085853A1 Heterocyclic ester and amide hair growth compositions and uses
03/28/2001EP1085847A2 Novel therapeutic agents that modulate estrogen receptors
03/28/2001EP0708762B1 Process for making hiv protease inhibitors
03/28/2001CN1289334A Benzothiadiazoles and derivatives
03/28/2001CN1289324A Method for preparing an N-[(aliphatic or aromatic) carbonyl]-2-aminoacetamide compound and a cyclyzed compound
03/27/2001US6207698 For therapy of osteoarthritis, rheumatoid arthritis, corneal ulceration, periodontitis, metastasis and invasion of tumor, and virus infection
03/27/2001US6207697 Amidinyl-substituted rings; anticoagulants; thromboembolic disorders; antiischemic and antiinflammatory agents; strokes; serine protease inhibitors
03/27/2001US6207693 Benzamide derivatives having a vasopressin antagonistic activity
03/27/2001US6207665 To treat inflammatory disorders in humans
03/22/2001WO2001019808A1 Chemical compounds and compositions and their use as cathepsin s inhibitors
03/22/2001WO2001019796A1 Compounds and pharmaceutical compositions as cathepsin s inhibitors
03/22/2001WO2000069862A3 Hemisynthetic method and intermediates thereof
03/22/2001WO2000001376A3 Pharmaceutical compositions and their uses for treatment of demyelinating disorders
03/22/2001WO1999063936A8 Novel therapeutic agents that modulate endothelin receptors
03/22/2001CA2384974A1 Compounds and pharmaceutical compositions as cathepsin s inhibitors
03/21/2001EP1083921A1 Novel leukotriene receptor antagonists and their uses
03/21/2001EP1083917A1 Novel analgesic agents
03/21/2001EP1083893A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the d 1? receptors
03/21/2001EP1083888A1 MULTIBINDING AGENTS THAT MODULATE PPARgamma AND RXR RECEPTORS
03/21/2001CN1288457A Inhibitors of & alpha; 4 mediated cell adhesion
03/21/2001CN1063444C Stable crystalline (65)-and (GR)-tetrahydrofolic acid
03/20/2001US6204293 Inhibitors of protein isoprenyl transferases
03/20/2001CA2213111C Substituted carboxanilide derivative and plant disease control agent comprising same as active ingredient
03/15/2001WO2001017982A1 Benzophenones as inhibitors of reverse transcriptase
03/15/2001WO2001017968A1 Integrase inhibitors containing aromatic heterocycle derivatives
03/15/2001WO2001017953A1 Non-peptidic cyclophilin binding compounds and their use
03/15/2001WO2001017942A1 Amides as inhibitors for pyruvate dehydrogenase
03/15/2001WO2000075113A8 Novel heterocyclic carboxamide derivatives
03/15/2001WO1999065870A3 Sulfonamide inhibitors of aspartyl protease
03/15/2001CA2383782A1 Compounds for the treatment of viral infections