Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
03/2001
03/15/2001CA2383086A1 Non-peptidic cyclophilin binding compounds and their use
03/14/2001EP1082362A1 Supported group 8-10 transition metal olefin polymerization catalysts
03/14/2001EP1082289A1 Methods for identifying novel multimeric agents that modulate receptors
03/14/2001EP1082121A1 Hiv integrase inhibitors
03/14/2001EP1082110A1 Use of compounds for the elevation of pyruvate dehydrogenase activity
03/13/2001US6200972 Heterocyclic esters and amides
03/13/2001US6200925 As polymerization catalyst
03/08/2001WO2001016121A1 Heterocyclic compounds and methods of use thereof
03/08/2001WO1999063930A8 Novel angiotensin receptor modulators and their uses
03/07/2001EP1081137A1 Selective inhibitors of aggrecanase in osteoarthritis treatment
03/07/2001EP1080080A1 Novel therapeutic agents that modulate neurokinin receptors
03/07/2001EP1080068A1 Modulators of protein tyrosine phosphatases
03/07/2001EP1079835A1 Pyrazinone thrombin inhibitors
03/07/2001EP0641325B1 Retroviral protease inhibitors
03/07/2001CN1286684A Carboxamide derivs. of pyrrolidine, piperidine and hexahydroazepine for treatment of thrombosis disorders
03/07/2001CN1286254A Aromatic amino ether as analgesics
03/07/2001CN1062865C Process for production of amidinobenzofuran and amidinobenzothiophen derivs. and salt thereof
03/06/2001US6197773 N-acyl and N-aroyl aralkyl amides as serotonergic agents
03/01/2001WO2001014371A1 N-heterocyclic derivatives as nos inhibitors
03/01/2001WO2001014355A1 Substituted piperazine derivatives, the production thereof and their utilization as medicaments
03/01/2001WO2001014339A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
03/01/2001WO2000071516B1 INHIBITORS OF FACTOR Xa
03/01/2001CA2382311A1 Substituted piperazine derivatives, the preparation thereof and their use as medicaments
03/01/2001CA2376275A1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
02/2001
02/28/2001EP1077978A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors
02/28/2001CN1285820A Metabotropic glutamate receptor antagonists for treating central nervous system disease
02/27/2001US6194574 Selectively bind to corticotropin-releasing factor (crf1) receptors; for treating stress related disorders such as post traumatic stress disorder (ptsd) as well as depression, headache and anxiety
02/27/2001US6194416 Central nervous system disorders; alzheimer's disease
02/27/2001US6194412 Mixtures derived from grains of Eugenia Jambolana Lamarck preparation and use of said mixtures and some of their constituents as medicaments
02/27/2001CA2101316C Gnrh analogs
02/22/2001WO2001012614A1 N-oxyl radicals
02/22/2001WO2001012600A1 INHIBITORS OF FACTOR Xa
02/22/2001WO2001012591A1 Novel naphthylsulfonic acids and related compounds as glucose uptake agonists
02/22/2001WO2001012233A2 Sustained release formulation of a peptide
02/22/2001WO1999063996A8 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
02/22/2001DE19939745A1 New 1-carboxyalkyl-4-(hetero)aryl-piperazine derivatives as microsomal triglyceride transfer protein inhibitors, useful for reducing plasma atherogenic lipoprotein levels, e.g. in treatment of hyperlipidemia
02/22/2001DE19939516A1 New 1-carboxyalkyl-4-(hetero)aryl-piperazine derivatives, as microsomal triglyceride transfer protein inhibitors useful for reducing plasma atherogenic lipoprotein levels, e.g. in treatment of hyperlipidemia
02/22/2001DE19939031A1 N-Oxyl-Radikale N-oxyl radicals
02/21/2001CN1284953A Method of preparing enantiomerically-enriched tetrahydrobenzothiepine oxides
02/20/2001US6191182 Subjecting p-halophenyl alkyl ketone to aminolysis with cyclic secondary amine to form cyclic amine-substituted phenyl alkyl ketone; halogination and reacting with amine compound; stevens rearrangement under basic condition
02/20/2001US6191134 Stroke therapy, antiischemic agents, brain disorders
02/20/2001US6191132 Use of quisqualate receptor antagonists
02/20/2001US6190852 Coupler provides a desirably narrow spectrographic absorption curve.
02/15/2001WO2001010842A2 Melanocortin-4 receptor binding compounds and methods of use thereof
02/15/2001WO2001010834A2 Antibacterial agents
02/15/2001WO2001010799A1 Methods for preparing n-[(aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
02/15/2001CA2381008A1 Melanocortin-4 receptor binding compounds and methods of use thereof
02/14/2001EP1075469A1 Piperazine derivatives and process for the preparation thereof
02/14/2001EP1075468A1 Method for producing high melting point crystals of phenoxypropionic acid derivative
02/13/2001US6187944 A phenyl acrylonitrile compounds useful as active ingredients of an insecticide, a miticide, a nematicide, a soil pesticide, a fungicide and a marine antifouling agent
02/13/2001US6187943 Catalyzing the reaction in the presence of a metal oxide catalyst containing vanadium and/or molybdenum in a fluidized bed
02/13/2001US6187812 For controlling animal pests or harmful fungi; (e,e,e)-2-methoxyimino-2-(2'-(1?-methyl, 1?-(1?'-ethoxyiminoethyl))iminooxymethyl)phenylacetic acid monomethylamide, for example
02/13/2001US6187776 Heterocyclic compounds and their use
02/08/2001WO2000076984A3 Novel compounds, their use and preparation
02/07/2001EP1073644A1 Solid supported synthesis of sulfonated 2-oxopiperazines
02/07/2001EP1073638A1 Heterocyclically substituted amides, their production and their use
02/07/2001EP1073626A1 Azine used as fungicides
02/07/2001EP0538422B1 New use of diphenylbutylpiperazinecarboxamides in the treatment of substance disorders
02/07/2001CN1283195A 1-(2-naphthyl) and 1(2-azanaphthyl)-4-(1-phenylmethyl)piperazines being dopamine D4 receptor subtype ligands
02/07/2001CN1283180A Inhibition of raf kinase using symmerical and unsymmerical substituted diphenyl ureas
02/06/2001US6184224 Drug resistance and side effect reduction
02/06/2001CA2027349C Light polarizing materials and suspensions thereof
02/01/2001WO2001007436A2 Substituted oxoazaheterocyclyl compounds
02/01/2001WO2001007419A1 Novel thiazine or pyrazine derivatives
02/01/2001WO2001007411A1 Biarylurea derivatives
02/01/2001CA2382755A1 Substituted oxoazaheterocyclyl compounds
02/01/2001CA2380389A1 Biarylurea derivatives
02/01/2001CA2380218A1 Novel thiazine or pyrazine derivatives
01/2001
01/31/2001EP1071669A1 Bicyclic compounds having an anti-thrombitic effect
01/31/2001EP1071666A1 Azacycloalkane derivatives, preparation and therapeutic application
01/31/2001CN1061350C 2.7-substituted octahydro-pyrrolo (1.2-A) pyrazine derivatives
01/30/2001US6180646 Retroviral protease inhibitors
01/30/2001US6180632 Use of these compounds for treating disorders/conditions involving cellular differentiation, proliferation, extracellular matrix production or mediator release and/or t cell activation and proliferation
01/30/2001US6180623 Used as analgesics and anti-pruritic agents
01/30/2001US6180619 Prenyl transferase inhibitors
01/25/2001WO2001005773A1 Conjugates of sodium channel blockers and methods of using the same
01/25/2001WO2001005772A1 Pyrazinones, compositions containing such compounds
01/25/2001WO2001005769A2 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/25/2001WO2001005748A1 Oligomeric amino acid derivatives useful as nitric oxide synthase inhibitors
01/25/2001WO2001005398A1 Phosphate transport inhibitors
01/25/2001WO2001005390A2 Method for treating chronic pain using mek inhibitors
01/25/2001WO2001005354A2 Improved process for the preparation of benzenesulfonylureas as oral hypoglycemic agents of the second generation
01/25/2001WO2000071515A3 INHIBITORS OF FACTOR Xa
01/25/2001WO2000058293A3 Glucokinase activators
01/25/2001CA2379657A1 Phosphate transport inhibitors
01/25/2001CA2378181A1 Conjugates of sodium channel blockers and methods of using the same
01/25/2001CA2377092A1 Method for treating chronic pain using mek inhibitors
01/24/2001EP1070084A1 PIPERAZINES AS INHIBITORS OF FRUCTOSE-1,6-BISPHOSPHATASE (FBPase)
01/24/2001EP1070065A1 Azabicyclic 5ht1 receptor ligands
01/24/2001EP1070054A1 Amine compounds, their production and their use as somatostatin receptor antagonists or agonists
01/24/2001CN1281449A Crystalline antifungal polymorph
01/24/2001CN1281436A N-Benzyl-3-indenylacetamides derivatives for treating neoplasia
01/24/2001CN1281335A Treatment of schizophrenia with ampakines and neuroleptics
01/23/2001US6177429 Dihydropyrazine derivatives as NPY antagonists
01/23/2001US6177401 Use of organic compounds for the inhibition of Flk-1 mediated vasculogenesis and angiogenesis
01/23/2001CA2128202C Alkyl derivatives of trazodone with cns activity
01/18/2001WO2001004097A2 Cyclic delocalized cations connected by spacer groups
01/18/2001WO2000071516A3 INHIBITORS OF FACTOR Xa
01/17/2001EP1068200A1 2,4,4-trisubstituted-1,3-dioxolane antifungals
01/17/2001EP1068190A1 Quinoxalinones as serine protease inhibitors such as factor xa and thrombin