Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
01/2001
01/17/2001EP1068185A1 Compounds with activity on muscarinic receptors
01/17/2001EP0983258A4 N-hydroxy 4-sulfonyl butanamide compounds
01/17/2001CN1280572A Inhibiting platelet derivative growth factor and/or quinoline and quinowoline compounds of P56lek tyrosinkinase
01/17/2001CN1280569A 1,2-dihydro-2-oxoquinoline derivatives
01/16/2001US6175011 Preparing aryloxy arylamides of pyridine-, pyrimidine-, pyrazine- and 1,3,5-triazine-carboxylic acids by reacting the heteroaromatic dihalide with an aromatic hydroxy then with carbon monoxide and an arylamine using diphosphine catalyst
01/16/2001US6174905 As carcinostatic agent to a hematologic malignancy and a solid carcinoma
01/16/2001US6174887 Amide compounds and use of the same
01/11/2001WO2001002381A1 Piperazine derivatives as modulators of chemokine receptor activity
01/11/2001WO2001002372A1 Cyclized amino acid derivatives
01/11/2001WO2001002371A1 Optically active piperazine compounds, intermediates for the preparation of the same and processes for the preparation of both
01/11/2001WO2001002354A1 Phthalamide derivatives, intermediates in the production thereof, and agricultural/horticultural insecticides and method of using the same
01/11/2001WO2001002349A1 Phenyl sulfamate derivatives
01/11/2001WO2001002345A2 Mono and multifunctional alkoxyamines for the preparation of functionalized macromers
01/11/2001CA2375806A1 Mono and multifunctional alkoxyamines for the preparation of functionalized macromers
01/10/2001EP1066290A1 PYRROLO[1,2-a]PYRAZINE sPLA 2 INHIBITOR
01/10/2001EP1066247A1 Inhibitors of serine proteases, particularly hepatitis c virus ns3 protease
01/10/2001EP1066246A1 Novel cationic couplers and their use for oxidation dyeing
01/10/2001EP1066245A1 Novel local anesthetic compounds and uses
01/10/2001EP1066022A1 Compositions for oxidation dyeing keratin fibres comprising a cationic coupler, novel cationic couplers, their use for oxidation dyeing and dyeing methods
01/10/2001CN1279682A bicyclic kinase inhibitors
01/09/2001US6172229 1-phenyl-4-benzylpiperazines; dopamine receptor subtype specific ligands
01/09/2001US6172065 Central nervous system disorders
01/09/2001US6172058 Nervous system disorders; psychological disorders
01/09/2001US6171522 Heterocyclic aromatic anion salts, and their uses as ionic conducting materials
01/04/2001WO2001000654A2 Purification and stabilization of peptide and proteins in pharmaceutical agents
01/04/2001WO2001000578A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
01/04/2001WO2001000575A1 Heterocyclic dicarboxylic acid diamide derivatives, agricultural/horticultural insecticides and method of using the same
01/04/2001WO2001000214A1 Src kinase inhibitor compounds
01/04/2001CA2377204A1 Purification and stabilization of peptide and protein pharmaceutical agents
01/04/2001CA2376951A1 Src kinase inhibitor compounds
01/04/2001CA2370500A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
01/03/2001EP1065203A2 Heterocyclic compounds as retinoic acid receptor antagonists
01/03/2001EP1064274A1 Benzenesulfonamide derivatives and their use as medicaments
01/03/2001CN1278807A Herbicidal N-alkenyl Heteroaryloxyacetamides
01/03/2001CN1278721A IL-8 receptor antagonists
01/03/2001CN1060172C Substituted biphenyl sulfonamide endothelin antagonists
01/03/2001CN1060161C N-substituted phenylcarbamic acid derivatives, process for production thereof, agricultural and horticultural fungicides, intermediats of derlvatives and process for production thereof
01/02/2001US6169095 For prevention and/or treatment of bradykinin or its analogues mediated diseases in the eye, such as allergy, inflammation and pain of the eye
01/02/2001CA2068064C Fibrinogen receptor antagonists
01/02/2001CA1341163C Oxime ether derivatives, their preparation and fungicides containing these derivatives
01/02/2001CA1341159C Pure enantiomers of 4,5-disubstituted .alpha.-butyrolactams, process for their preparation, and their use
12/2000
12/28/2000WO2000078746A1 Antiviral agents
12/28/2000WO2000078319A1 Dihydropyrazine derivatives as npy antagonists
12/28/2000CA2377698A1 Dihydropyrazine derivatives as npy antagonists
12/28/2000CA2375211A1 Antiviral agents
12/27/2000EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
12/27/2000EP1062199A1 Modulators of protein tyrosine phosphatases (ptpases)
12/27/2000EP0821671B1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors
12/27/2000CN1278244A Dipeptide nitriles
12/27/2000CN1278242A Iron alkali salt of S, S-ethylenediamine-n,n'-disuccinic acid, and process for producing same
12/26/2000US6166053 Antiproliferative agent for treating cancer
12/26/2000US6166008 Treatment of schizophrenia with ampakines and neuroleptics
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors
12/26/2000US6166004 Treatment of aids
12/21/2000WO2000077519A1 Solid phase synthesis of n,n-disubstituted diazacycloalkylcarboxy derivatives
12/21/2000WO2000077027A2 Serine protease inhibitors
12/21/2000WO2000076984A2 Novel compounds, their use and preparation
12/21/2000WO2000076980A1 Novel nitrogen-contaiing heterocyclic derivatives or salts thereof
12/21/2000WO2000076976A1 Process for the production of 2-pyridylpyridine derivatives
12/21/2000WO2000076974A2 Oligomers and polymers of cyclic imino carboxylic acids
12/21/2000WO2000076971A2 Serine protease inhibitors
12/21/2000WO2000076970A2 Serine protease inhibitors
12/21/2000WO2000076957A1 N-alkoxyalkyl-n,n-dialkylamine derivatives or salts thereof, and remedies for nerve degeneration diseases containing the same
12/21/2000WO2000044709A3 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
12/21/2000CA2383008A1 Compounds
12/21/2000CA2375920A1 Compounds
12/20/2000EP1060175A2 Tryptase inhibitors
12/20/2000EP1060171A2 Tryptase inhibitors
12/14/2000WO2000075121A2 Process for preparing 10,11-methanobenzosuberane derivatives
12/14/2000WO2000075113A1 Novel heterocyclic carboxamide derivatives
12/14/2000CA2378735A1 Process for preparing 10,11-methanobenzosuberane derivatives
12/13/2000EP1058698A1 Preparation for prevention and healing of inflammation affections
12/12/2000US6160126 Useful in preparing guanidine derivatives useful as insecticides and miticides
12/12/2000US6160118 Process for the synthesis of substituted piperazinones via Mitsunobu reaction
12/12/2000US6159995 Substituted diaminocarboxylic acids
12/12/2000US6159980 Anxiolytic agents, antidepressants; psychological and eating disorders
12/12/2000US6159978 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
12/07/2000WO2000073283A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
12/07/2000WO2000073260A1 Squaric acid derivatives as cell adhesion molecules
12/07/2000WO2000072801A2 Alpha v integrin receptor antagonists
12/07/2000CA2376024A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
12/07/2000CA2375218A1 Squaric acid derivatives as cell adhesion molecules
12/07/2000CA2373937A1 Alpha v integrin receptor antagonists
12/06/2000EP1057816A1 Method for producing heteroaromatic aldehydes
12/06/2000EP1056728A1 Dihydro-benzo(1,4)oxazines and tetrahydroquinoxalines
12/06/2000EP1056727A1 Solid support synthesis of 2-oxopiperazines
12/06/2000CN1275981A Novel pharmaceutically active compounds, their preparation and use as ECE-inhibitors
12/05/2000US6156895 Using chiral hydrogenation, intermediate for an hiv protease inhibitor.
12/05/2000US6156761 Substituted tetralone derivatives for enhancing cognition
11/2000
11/30/2000WO2000071572A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
11/30/2000WO2000071518A2 Heterocyclic analgesic compounds and their use
11/30/2000WO2000071516A2 INHIBITORS OF FACTOR Xa
11/30/2000WO2000071515A2 INHIBITORS OF FACTOR Xa
11/30/2000WO2000071506A2 Naphthalene ureas as glucose uptake enhancers
11/30/2000WO2000032583A9 Antitumor dibenzofluorene derivatives
11/30/2000CA2374788A1 Inhibitors of factor xa
11/30/2000CA2374225A1 Naphthalene ureas as glucose uptake enhancers
11/30/2000CA2372887A1 Heterocyclic analgesic compounds and their use
11/30/2000CA2371904A1 Inhibitors of factor xa
11/29/2000EP1054858A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted-alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors