Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
06/2009
06/16/2009CA2447640C Substituted anilide derivative, intermediate thereof, agricultural and horticultural chemical and its usage
06/11/2009WO2009071726A1 Method for the preparation of capecitabine and intermediates used in said method
06/11/2009WO2009071535A1 Diaminopyridines for the treatment of diseases which are characterised by excessive or anomal cell proliferation
06/11/2009WO2009071449A1 Pyridylmethyl-sulfonamide compounds
06/11/2009WO2009071448A1 Pyridylmethyl-sulfonamide compounds
06/11/2009WO2008093325A3 Polymorphs of 3-(e)-2-{2-[6-(2-cyanophenoxy) pyrimidin-4-yloxy]phenyl}-3-methoxyacrylate
06/11/2009US20090149487 4,5-diphenyl-pyrimidinylamino substituted carboxylic acids, method for the production and use thereof as medicaments
06/11/2009US20090149486 4,5-diphenyl-pyrimidinyl-oxy or -mercapto substituted carboxylic acids, method for the production and use thereof as medicaments
06/11/2009US20090149485 Pyrimidinediones as tyrosine kinase inhibitors
06/11/2009US20090149484 Quinazolin-4-one derivatives, process for their preparation and pharmaceutical compositions containing them
06/11/2009US20090149477 use for lowering blood glucose, treating diabetes, or increasing insulin release; 7-(4,5-Diphenylpyrimidin-2-yl)-6-heptynoic Acid
06/11/2009US20090149476 3-[[6-[4-(1,2,3,4-tetrahydro-1,8-naphthyridin-7-yl)-1-piperidinyl]-2,5-dimethyl-4-pyrimidinyl]amino]-N-[(phenylmethoxy)carbonyl]alanine, used for the treatment of osteoporosis, restenosis, arteriosclerosis, nephropathy or retinopathy
06/11/2009US20090149469 Phenyl-[4-(3-phenyl-1h-pyrazol-4-yl)-pyrimidin-2-yl]-amine derivatives as igf-ir inhibitors
06/11/2009US20090149468 Substituted heterocyclic compounds and methods of use
06/11/2009US20090149456 2-Pyrimidinyl Pyrazolopyridine ErbB Kinase Inhibitors
06/11/2009US20090148531 Rate-controlled particles
06/11/2009CA2707653A1 Diaminopyridines for the treatment of diseases which are characterised by excessive or anomal cell proliferation
06/11/2009CA2705489A1 Pyridylmethyl-sulfonamide compounds
06/10/2009EP2066645A2 2 amino-pyrimidine derivatives as h4 receptor antagonists, processes for preparing them and their use in pharmaceutical compositions
06/10/2009EP2066644A2 Salts of rosuvastatin and processes for their preparation
06/10/2009EP2066632A1 Benzophenone derivatives useful for inhibiting formation of microtubule
06/10/2009EP1597251B1 Pyrimidine compounds
06/10/2009CN101454294A Quinazolines for pdk1 inhibition
06/10/2009CN101450934A Sulfonyl-derivatives as novel inhibitors of histone deacetylase
06/10/2009CN100497326C Derivatives of 1-piperazine- and 1-homopiperazine-carboxylates, preparation method thereof and use of same in therapeutics
06/10/2009CN100497318C Method for preparing 2,4,6-trichloro pyrimidine
06/09/2009US7544799 Crystal modification of a N-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
06/09/2009US7544691 Guanidine derivatives
06/09/2009US7544690 MCH receptor antagonists
06/09/2009US7544688 Hetereoaryl nitrile derivatives
06/09/2009US7544675 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
06/09/2009CA2583764C Thrombopoietin activity modulating compounds and methods
06/09/2009CA2403721C Combined treatment with keratinocyte growth factor and epidermal growth factor inhibitor
06/09/2009CA2162900C New peptide derivatives
06/04/2009WO2009069291A1 Prophylactic and/or therapeutic composition for disease caused by inhalation of tobacco smoke
06/04/2009WO2009068512A1 2 -amino-pyrimidine derivatives as histamine h4 antagonists
06/04/2009WO2009007300A3 Substituted amino-quinazolinones, medicaments comprising said compound, their use and their method of manufacture
06/04/2009WO2008155669A3 Arylamide pyrimidone derivatives for the treatment of neurodegenerative diseases
06/04/2009US20090143579 Heterocyclic Inhibitors of MEK and Methods of Use Thereof
06/04/2009US20090143414 Quinazoline Derivatives Having Tyrosine Kinase Inhibitory Activity
06/04/2009US20090143389 Heterocyclic inhibitors of mek and methods of use thereof
06/04/2009US20090143384 2,4,6-Trisubstituted Pyrimidines as Phosphotidylinositol (Pi) 3-Kinase Inhibitors and Their Use in the Treatment of Cancer
06/04/2009US20090143376 Fused Heterocyclic Compounds and Their Use as Sirtuin Modulators
06/04/2009US20090143365 Derivatives of alkylpiperazine- and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors
06/03/2009EP2064191A1 Aspartyl protease inhibitors
06/03/2009EP2064190A1 Pyrimidylmethyl-sulfonamide compounds useful as fungicides and against arthropods
06/03/2009EP2064177A2 Protease inhibitors
06/03/2009CN101448794A Pyrimidine derivatives for the treatment of amyloid-related diseases
06/03/2009CN101445487A Preparation method of 3H-quinazoline-4-ketones compounds
06/03/2009CN101445486A Derivatives of aryl-quinazoline/aryl-2-amino-phenyl methanone which promote the release of parathyroid hormone
06/03/2009CN101445485A Synthesis method of 4,6-dichloro-5-fluoropyrimidine compound
06/03/2009CN100494183C Preparation process of key intermediate 2-cyano pyrimidine of bosentan
06/03/2009CN100494177C Bi-amido heterocyclic derivative with antitumour activity and its preparation method and use
06/02/2009US7541465 Substituted 2-aminoacetamides and the use thereof
06/02/2009US7541369 Amino-derivatives as novel inhibitors of histone deacetylase
06/02/2009US7541361 N-[4,5-diphenylpyrimidin-2-yl)methyl]amine derivatives, the preparation thereof and their therapeutic use
06/02/2009US7541360 2-amino-4-N-cyclohexylmethylamino-6-(L-erythro-1,2-dihydroxypropyl)-7,8-dihydro-pteridine; treatment of pathological blood pressure decreases, such as occur in septic or hemorrhagic shock, in tumor or cancer therapy with cytokines, liver cirrhosis; ulcerative colitis; NO synthase inhibitor
06/02/2009CA2503900C Purine compounds and use thereof as cannabinoid receptor ligands
06/02/2009CA2452253C Novel crystal of arylethenesulfonamide derivative and preparation process thereof
06/02/2009CA2362594C Process for the production of tert-butyl (e)-(6-[2- [4-(4-fluorophenyl) -6-isopropyl-2-[ methyl (methylsulfonyl) amino] pyrimidin-5-yl] vinyl](4r, 6s)-2,2-dimethyl [1,3]dioxan-4-yl) acetate
06/02/2009CA2116421C Inhibitors of hydroxyphenylpyruvate dioxygenase and an assay for identification of inhibitors
05/2009
05/28/2009WO2009067621A1 Biaryl pde4 inhibitors for treating pulmonary and cardiovascular disorders
05/28/2009WO2009067600A2 Biaryl pde4 inhibitors for treating inflammation
05/28/2009WO2009067081A1 Pyrimidine derivatives for the treatment of asthma, copd, allergic rhinitis, allergic conjunctivitis, atopic dermatitis, cancer, hepatitis b, hepatitis c, hiv, hpv, bacterial infections and dermatosis
05/28/2009WO2009066084A1 2 -morpholinopyrimidines and their use as pi3 kinase inhibitors
05/28/2009WO2009048752A3 Insecticidal substituted azinyl derivatives
05/28/2009WO2009030467A3 Saturated and insaturated bi- or tricyclic aryloxyacetamide derivatives and their use as fungicides
05/28/2009WO2007050381A3 3-piperidin-4-yl-indole orl-1 receptor modulators
05/28/2009US20090137804 Compounds and Compositions as Protein Kinase Inhibitors
05/28/2009US20090137803 5-protected aminopyrimidine compound, production method thereof and intermediate therefor
05/28/2009US20090137802 A2b adenosine receptor antagonists
05/28/2009US20090137611 Fungicide N-Cyclopropyl-Sulfonylamide Derivatives
05/28/2009US20090137589 Stereoisomerically Enriched 3-Aminocarbonyl Bicycloheptene Pyrimidinediamine Compounds And Their Uses
05/28/2009US20090137588 Heteroaryl compounds and uses thereof
05/28/2009US20090137585 N-acylsulfonamide apoptosis promoters
05/28/2009US20090137583 2-aminoquinazoline derivatives
05/28/2009US20090137575 Fused Tetracyclic mGluR1 Antagonists as Therapeutic Agents
05/28/2009US20090137567 Methods for Treating Blood Disorders
05/28/2009US20090137557 Calcilytic Compounds
05/28/2009US20090137021 Anti-inflammatory medicaments
05/28/2009US20090136473 Biaryl pde4 inhibitors for treating pulmonary and cardiovascular disorders
05/28/2009US20090133318 Anthranilamide insecticides
05/28/2009CA2722611A1 Biaryl pde4 inhibitors for treating pulmonary and cardiovascular disorders
05/28/2009CA2722582A1 Biaryl pde4 inhibitors for treating inflammation
05/28/2009CA2704214A1 Pyrimidine derivatives for the treatment of asthma, copd, allergic rhinitis, allergic conjunctivitis, atopic dermatitis, cancer, hepatitis b, hepatitis c, hiv, hpv, bacterial infections and dermatosis
05/27/2009EP2061773A2 Quinazoline based egfr inhibitors containing a zinc binding moiety
05/27/2009EP2061771A1 Aspartyl protease inhibitors containing a tricyclic ring system
05/27/2009EP2061770A1 Piperazine compounds with herbicidal action
05/27/2009EP2061764A1 Heterocyclic derivatives binding to the peripheral-type benzodiazepine receptor (pbr)
05/27/2009EP2061760A1 Benzo-fused compounds for use in treating metabolic disorders
05/27/2009EP2061469A2 Quinazoline based egfr inhibitors containing a zinc binding moiety
05/27/2009EP1663241B1 5-arylpyrimidines as anticancer agents
05/27/2009EP0934287B1 Heterocyclic esters and amides
05/27/2009CN101443664A Mass tags for quantitative analyses
05/27/2009CN101443318A Heterobicyclic carboxamides as inhibitors for kinases
05/27/2009CN101440066A Benzodiazepinic amine nitrite compound, preparation and use thereof
05/27/2009CN100491371C Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (GSK3 inhibitors)
05/27/2009CN100491358C Pyrimidinone compounds, compositions and methods
05/27/2009CN100491356C Compounds exhibiting thrombopoietin receptor agaonism
05/27/2009CN100491353C Carboxylic acid derivative capable of inhibiting combination of integrin and its receptor