Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
07/2009
07/01/2009CN100506803C Polymorph of {6,7-bis(2-methoxy-ethoxy)-quinazolin-4-yl}-(3e)
07/01/2009CN100506802C Formyl peptide-like acceptor-1 regulator and its Preparation and use
07/01/2009CN100506801C Inhibitors of glycogen synthase kinase 3
07/01/2009CN100506800C Tetrahydropyrimidine-2-one derivatives and their uses
06/2009
06/30/2009US7553976 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
06/30/2009US7553971 Aryl aniline β2 adrenergic receptor agonists
06/30/2009US7553966 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/30/2009US7553876 angiogenesis inhibitors; a salicylamides; amphiphilic compounds; used with various antiinflammatory and cytotoxic agents as well as with radio-therapeutic agents to treat tumor growth and metastasis
06/30/2009US7553872 Compounds and compositions for delivering active agents
06/30/2009US7553852 Caspase inhibitors and uses thereof
06/30/2009US7553840 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use
06/30/2009US7553826 Cytarabine monophosphate prodrugs
06/30/2009CA2406088C Novel phenyl-propargylether derivatives
06/30/2009CA2330447C N-(3-ethynylphenyl-6,7-bis(2-methoxyethoxy)-4-quinazolinamine mesylate anhydrate and monohydrate
06/30/2009CA2254693C Process for the preparation of aminoalcohol derivatives and their further conversion to (1r,4s)-4-((2-amino-6-chloro-5-formamido-4-pyrimidinyl)amino)-2-cyclopentenyl-1-methanol
06/25/2009WO2009079597A1 Piperazinyl derivatives useful as modulators of the neuropeptide y2 receptor
06/25/2009WO2009079490A1 Process and intermediates for the synthesis of heterocyclic substituted piperazines with cxcr3 antagonist activity
06/25/2009WO2009076747A1 Viral polymerase inhibitors
06/25/2009WO2009076743A1 Preparations containing amino acids and orotic acid
06/25/2009US20090163712 Processes for preparing hiv reverse transcriptase inhibitors
06/25/2009US20090163525 Substituted quinazolines with anti-cancer activity
06/25/2009US20090163516 Carboxamides for controlling undesired micro-organisms in plant protection
06/25/2009US20090163515 Compounds Which Bind to the Active Site of Protein Kinase Enzymes
06/25/2009US20090163496 Antibacterial agents
06/25/2009US20090163485 Heteroaryl derivatives as orexin receptor antagonists
06/25/2009US20090163463 Organic Compounds
06/25/2009US20090163457 Compositions and methods for delivering a biologically active agent
06/25/2009US20090160326 Organic electroluminescence material and element using the same
06/25/2009DE102007061766A1 New 4-(4-cyano-2-thioaryl)-dihydro-pyrimidinone compounds are human neutrophil elastase inhibitor, useful for the treatment or prevention of e.g. pulmonary arterial hypertonia, acute lung injury and diseases of the cardiovascular system
06/25/2009DE102007061757A1 Substituierte 2-Phenylpyrimidin-5-carbonsäuren und ihre Verwendung Substituted 2-phenyl-pyrimidine-5-carboxylic acids and their use
06/25/2009DE102007061756A1 Substituierte 4-Aminopyrimidin-5-carbonsäuren und ihre Verwendung Substituted 4-aminopyrimidine-5-carboxylic acids and their use
06/25/2009CA2708324A1 Viral polymerase inhibitors
06/24/2009EP2072503A2 Process for the preparation of bosentan
06/24/2009EP2072502A1 Sulfoximide substituted chinolin and chinazolin derivatives as kinase inhibitors
06/24/2009EP1844004B1 Quinazoline derivates as antiviral agents
06/24/2009EP1781614B1 Compounds which potentiate glutamate receptor and uses thereof in medicine
06/24/2009EP1611109A4 Novel quinazoline derivatives and methods of treatment related to the use thereof
06/24/2009EP1483247B1 Aryl substituted pyrimidines and the use thereof
06/24/2009CN101463015A Preparation of 5,6,7-trialkoxy-N-aryl substituted-4-amino quinazoline derivative and compound synthesized thereby
06/24/2009CN101463014A Diaryl benzo pyridine derivative, and preparation and use thereof
06/24/2009CN101463013A Preparation of erlotinid hydrochloride
06/24/2009CN101463012A Preparation of gefitinib
06/24/2009CN101463011A Process for synthesizing 3,4-dihydropyrimidine-2-keto
06/24/2009CN100503600C Pesticidal heterocycles
06/24/2009CN100503599C Carbonylamino-derivatives as novel inhibitors of histone deacetylase
06/24/2009CN100503580C Irreversible inhibitor of tyrosine kinase
06/24/2009CN100503579C Process for producing substituted aniline compound
06/24/2009CN100503578C N-2-pyrimidinyl oxy-benzyl substituted cyclic amine compound, its preparation process and uses
06/24/2009CN100503572C Caspase inhibitors and uses thereof
06/24/2009CN100503560C Substituted cyclohexane derivatives
06/23/2009US7550590 Such as 2-[2-(3-Amino-piperidin-1-yl)4-oxo-4H-quinazolin-3-ylmethyl]-benzonitrile; type 2 diabetes mellitus, diabetic dislipidemia, impaired glucose tolerance
06/23/2009US7550489 N-[3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide and phentermine, metformin, or bupropion; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists
06/23/2009US7550473 Pyrimidine derivatives useful as inhibitors of PKC-theta
06/23/2009US7550461 Benzofuran and benzothiophene compounds useful in treating cytokine mediated diseases
06/23/2009US7550460 2,4-pyrimidinediamine compounds and their uses
06/23/2009CA2402991C Drugs for the diagnosis of tissue-reproductive activity or the treatment of proliferative diseases
06/23/2009CA2384354C Pyrimidine derivatives and herbicides containing them
06/23/2009CA2214131C Trisubstituted phenyl derivatives
06/18/2009WO2009075835A1 CYCLIC UREA INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE 1
06/18/2009WO2009075277A1 4-aminopyrimidine derivative and medicinal composition containing the compound
06/18/2009WO2009075080A1 Fluoroalkylsulfide derivative and pest control agent
06/18/2009WO2009074749A2 Nicotinamide derivatives, preparation thereof and therapeutic use thereof
06/18/2009WO2009074487A1 Inhibitors of stearoyl-coa desaturase
06/18/2009WO2009074333A1 Synthesis of paliperidone
06/18/2009WO2009053748A3 Novel crystalline forms
06/18/2009WO2009044018A3 Derivatives of 1-oxo-1,2-dihydroisoquinoline-5-carboxamides and of 4-oxo-3,4-dihydroquinazoline-8-carboxamides, preparation thereof and application thereof in therapeutics
06/18/2009WO2009036996A3 Small molecule bradykinin b1 receptor antagonists
06/18/2009WO2009025919A3 5-propargyl-pyrimidine derivatives as inhibitors of dihydrofolate reductase with antibacterial antiprotozoal, antifungal and anticancer properties
06/18/2009WO2007027532A3 Niacin receptor agonists, compositions containing such compounds and methods of treatment
06/18/2009US20090156812 Preparations containing amino acids and orotic acid
06/18/2009US20090156804 Intermediate compound for synthesizing pharmaceutical agent and production method thereof
06/18/2009US20090156622 2,4-pyrimidinediamine compounds and their uses
06/18/2009US20090156616 Therapeutic agents
06/18/2009US20090156601 kinase inhibitor; immunotherapy; viricides; function or behavior associated with PI3 kinase such as cancer, immune, cardiovascular, nervous system, metabolism/endocrine and neurological diseases, viral infection, inflammation; 2-(3-hydroxyphenyl)-4-(morpholin-4-yl)-6-(pyridin-3-ylmethylamino) pyrimidine
06/18/2009US20090155917 Method for analyzing nucleobases on a single molecular basis
06/18/2009US20090155787 Mutations in the BCR-ABL tyrosine kinase associated with resistance to STI-571
06/18/2009CA2708303A1 Cyclic urea inhibitors of 11.beta.-hydroxysteroid dehydrogenase 1
06/18/2009CA2707105A1 Inhibitors of stearoyl-coa desaturase
06/18/2009CA2700559A1 Nicotinamide derivatives, preparation thereof and therapeutic use thereof
06/18/2009CA2646795A1 Process for the preparation of bosentan
06/17/2009EP2070914A1 New antagonist derivatives of the vitronectin receiver, method for preparing same, application of same as medicine and pharmaceutical compositions containing them
06/17/2009EP2069316A1 2,4-diaminoquinazolines for spinal muscular atrophy
06/17/2009EP2069315A2 Quinazolinone and isoquinolinone acetamide derivatives
06/17/2009EP2069314A1 Pyrimidines derivatives and their use as kinase inhibitors
06/17/2009EP2069313A2 Metalloprotease inhibitors
06/17/2009EP2069305A2 Nicotinic acid derivatives as modulators of metabotropic glutamate receptors
06/17/2009EP2069289A1 ISOSERINE DERIVATIVES FOR USE AS COAGULATION FACTOR IXa INHIBITORS
06/17/2009EP2069022A2 Agent for dyeing fibers comprising keratin
06/17/2009CN101456845A 4,5-diaryl-2-sulfhydryl miazines compounds and synthetic method thereof and pharmaceutical use
06/16/2009US7547782 Met kinase inhibitors
06/16/2009US7547781 inhibitors of epidermal growth factor receptor tyrosine kinase and histone deacetylase; 2-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquinazolin-6-yloxy)-N-hydroxyacetamide; anticarcinogenic agent
06/16/2009US7547780 Dihydropteridione intermediate compounds
06/16/2009US7547709 Prevent free radical cellular damage; oxidation resistant additive for fuels, lubricants, rubbers, polymers, solvents, chemical and foodstuff; lipid and water soluble vitamin c, vitamin e
06/16/2009US7547706 1H-pyrimido[4,5-b]indole derivatives, their preparation and therapeutic use
06/16/2009US7547705 Ethyl-1'-[(2S)-2-hydroxy-2-phenylethyl]-6'-oxo-8'-(pyridin-4-yl)-1',3',4',6'-tetrahydro-1H-spiro[piperidine-4,2'-pyrimido[1,2-a]pyrimidine]-1-carbox; glycogen synthase kinase-3 beta, amyloid precursor protein, tau protein hyperphosphorylation inhibitor; neurodegenerative disease, type II diabetes
06/16/2009US7547704 Hepatitis C; antivirals; cytosine, uracil or thymine bases on a cyclopentane ring with optional amino acid ester to form hydroxy or phosphate in vivo
06/16/2009US7547702 Glycoprotein antagonist; anticholesterol agents; cardiovascular disorders; strokes; antiischemic agents
06/16/2009US7547274 Radioactive member and method of making
06/16/2009CA2574904C Antiretroviral enantiomeric nucleotide analogs
06/16/2009CA2452217C Hiv inhibiting pyrimidines derivatives