Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619) |
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10/06/2009 | US7598383 mitogen activated protein kinase inhibitors; 4-(2-fluoro-4-methylphenylamino)-1,3-dimethyl-6,7-dihydro-1H-pyrrolo[3,4-b]pyridine-2,5-dione; used in the treatment of hyperproliferative diseases, such as cancer and inflammation in mammals |
10/06/2009 | US7598379 Methods for the synthesis of unsymmetrical cycloalkyl substituted xanthines |
10/06/2009 | US7598260 CDK-inhibitory pyrimidines, their production and use as pharmaceutical agents |
10/06/2009 | US7598259 mGluR1 antagonists as therapeutic agents |
10/06/2009 | US7598255 Pyrimidine compounds as serotonin receptor modulators |
10/06/2009 | US7598236 Diazabicyclic central nervous system active agents |
10/06/2009 | CA2402431C 1,2,3,4-tetrahydroisoquinoline derivatives |
10/06/2009 | CA2301377C N-aroylphenylalanine derivatives |
10/01/2009 | WO2009121042A1 Quinazoline derivatives and methods of treatment |
10/01/2009 | WO2009118598A1 Process for the manufacture of rosuvastatin calcium with high purity |
10/01/2009 | WO2009118384A1 Quinazolinone derivatives as tubulin polymerization inhibitors |
10/01/2009 | WO2009117985A1 Pirinixic acid derivatives as prostglandin e2 synthesis inhibitors for treating inflammatory diseases |
10/01/2009 | WO2009117899A1 The polymorphs of 4-anilinoquinazoline derivatives, the preparation methods and uses thereof |
10/01/2009 | WO2009080638A3 Sulfamides as zap-70 inhibitors |
10/01/2009 | WO2009060835A8 Novel ubiquilin-binding small molecule |
10/01/2009 | US20090247555 5,7-Disubstituted[1,3]Thiazolo[4,5-D]Pyrimidin-2(3H)-One Derivatives 258 |
10/01/2009 | US20090247553 Highly Pure Paliperidone or a Pharmaceutically Acceptable Salt Thereof Substantially Free of Keto Impurity |
10/01/2009 | US20090247534 New compounds |
10/01/2009 | US20090247524 HSP90 Inhibitor |
10/01/2009 | US20090247519 Amino-ethyl-amino-aryl (aeaa) compounds and their use |
10/01/2009 | US20090247509 for treating central nervous system disorders such as psychological disorders, drug dependence and abuse, dyskinesia, dementia, anxiety disorders, sleep disorders and mood disorders |
10/01/2009 | US20090247506 Antibacterial agents |
10/01/2009 | CA2716088A1 Quinazolinone derivatives as tubulin polymerization inhibitors |
09/30/2009 | EP2105435A1 Hydrazone derivative |
09/30/2009 | CN101547910A Crystalline erlotinib |
09/30/2009 | CN101544609A Crystallization form of 4-anilinoquinazoline derivatives |
09/29/2009 | US7595501 Electroluminescent iridium compounds with fluorinated phenylpryidines, phenylpyrimidines, and phenylquinolines and devices made with such compounds |
09/29/2009 | US7595400 Synthesis of antitumor agents including camptothecin derivative 9-ethyl-9-hydroxy-1-pentyl-1H,12H-pyrano[3'',4'':6',7']-indolizino[1',2':6,5]pyrido[4,3,2-de]quinazoline-10,13(9H,15H)-dione |
09/29/2009 | US7595343 Inhibitors of histone deacetylase |
09/29/2009 | US7595332 Such as N-(4-tert-butylphenyl)-4-(2-pyridinyl)benzamide for treatment of urinary incontinence, pain, inflammatory thermal hyperalgesia, and/or bladder overactivity |
09/29/2009 | US7595326 1-[4-(5-Bromopyrimidin-2-ylsulfanyl)phenyl]-3-(2-nitrobenzoyl)-urea; antiproliferative, water soluble compound with high bioavailability |
09/29/2009 | US7595323 N-phenyl-2-pyrimidine-amine derivatives and process for the preparation thereof |
09/29/2009 | US7595317 Antiarthritic agents; rheumatoid and osteoarthritis; corneal, epidermal, or gastric ulceration; tumor metastasis or invasion; periodontal disease; and bone disease; 4-[(2-methyl-4-quinolinyl)methoxy]-N-(1,3,5-trioxo-2,4-diazaspiro[5.5]undec-7-yl)benzamide trifluoroacetate, for example |
09/29/2009 | US7595316 2-(1-Cyclopentylpiperidin-4-yloxy)-5-(4-cyanophenyl)pyrimidine, for example; exhibits histamine receptor H3 antagonist or inverse agonist activity and is useful for the treatment and/or prevention of obesity, diabetes, hormonal secretion abnormality, sleep disorders |
09/29/2009 | US7595309 For therapy of bacterial infections and neoplasms, |
09/29/2009 | CA2550372C Alpha-hydroxy amides as bradykinin antagonists or inverse agonists |
09/29/2009 | CA2375670C 5-phenyl-pyrimidine derivatives |
09/29/2009 | CA2349330C Nitrogen containing heterobicycles as factor xa inhibitors |
09/29/2009 | CA2334923C Aryl substituted olefinic amines and their use as cholinergic receptors agonists |
09/29/2009 | CA2328280C Thienopyrimidines |
09/29/2009 | CA2311922C Thienopyrimidines |
09/24/2009 | WO2009117080A1 Quinazoline derivatives as raf kinase modulators and methods of use thereof |
09/24/2009 | WO2009115587A1 Regioselective preparation of substituted pyrimidines |
09/24/2009 | WO2009115583A1 Regioselective preparation of substituted pyrimidines |
09/24/2009 | WO2009083608A9 Quinazolines and related heterocyclic compounds, and their therapeutic use |
09/24/2009 | WO2009057139A3 Novel 4-(tetrazol-5-yl)-quinazoline derivatives as anti cancer agents |
09/24/2009 | WO2009032668A3 2 -biphenylamino-4 -aminopyrimidine derivatives as kinase inhibitors |
09/24/2009 | WO2009005674A3 Novel hiv reverse transcriptase inhibitors |
09/24/2009 | US20090240054 Rosuvastatin calcium with a low salt content |
09/24/2009 | US20090240053 2-(4-(1-methyl-4-piperidinoxy)benzylamino)-2-methyl-propanamide; nervous system disorders; analgesics; anticonvulsants; sodium channel moderators; antidepressants, antiarrhythmics and for the treatment or prevention of diabetic neuropathy |
09/24/2009 | US20090240027 Intermediates for macrocyclic compounds |
09/24/2009 | US20090239841 Diaryl Ureas as CB1 Antagonists |
09/24/2009 | US20090239829 Thioaryl substituted inhibitors of zinc proteases and their use |
09/24/2009 | US20090239811 Polycationic compounds and uses thereof |
09/24/2009 | CA2755235A1 Nucleotide analogues with quaternary carbon stereogenic centers and methods of use |
09/24/2009 | CA2718892A1 Selective preparation of substituted pyrimidines |
09/24/2009 | CA2718858A1 Selective synthesis of substituted pyrimidines |
09/24/2009 | CA2718123A1 Quinazoline derivatives as raf kinase modulators and methods of use thereof |
09/23/2009 | EP2103601A1 Process for production of phenylalanine derivatives having quinazolinedione skeletons and intermediates for the production |
09/23/2009 | EP2102199A1 Antibacterial polycyclic urea compounds |
09/23/2009 | EP2102174A1 Process for the preparation of substituted cynophenoxy-pyrimidinyloxy-phenyl acrylate derivatives |
09/23/2009 | EP2102173A1 Pyrimidyl derivatives as protein kinase inhibitors |
09/23/2009 | EP2102172A1 Synthesis of 4-amino-pyrimidines |
09/23/2009 | EP2101986A1 Dithiolene metal complex colorless ir absorbers |
09/23/2009 | EP2101777A1 Composition for treating a pulmonary hypertension |
09/23/2009 | CN101541767A Pyrimidines and their use as CXCR2 receptor antagonists |
09/23/2009 | CN101541766A Pyrimidyl derivatives as protein kinase inhibitors |
09/23/2009 | CN101541765A 3-piperidin-4-yl-indole ORL-1 receptor modulators |
09/23/2009 | CN101541764A Pyrimidylmethyl-sulfonamide compounds useful as fungicides and against arthropods |
09/23/2009 | CN101538254A Derivatives of 1-piperazine- and 1-homopiperazine-carboxylates, preparation method thereof and use of same as inhibitors of the faah enzyme |
09/23/2009 | CN101538247A Alkaloid compound and preparation method thereof |
09/23/2009 | CN101538246A Pyrimidine amide compounds as pgds inhibitors |
09/23/2009 | CN101538230A Beta-amino ketones compound with anti-diabetic activity |
09/22/2009 | US7592452 Reacting an aryl or heteroaryl halide with a cyanide donor,potassium hexacyanoferrate(II) or (III), in the presence of a copper compound and a 1-alkyl imidazole as a catalyst stabilizer); nontoxic; industrial scale; cost efficiency; chemical intermediates for agrochemicals and pharmaceuticals |
09/22/2009 | US7592450 used to inhibit proliferative conditions, such as cancer and psoriasis, with improved bioavailability and stability |
09/22/2009 | US7592446 Synthesis of selenium-derivatized nucleosides, nucleotides, phosphoramidites, triphosphates and nucleic acids |
09/22/2009 | US7592349 Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors |
09/22/2009 | US7592348 Heterocyclic aspartyl protease inhibitors |
09/22/2009 | US7592337 Di-aryl substituted tetrazole modulators of metabotropic glutamate receptor-5 |
09/22/2009 | US7592177 Compositions and methods for inducing cell dedifferentiation |
09/22/2009 | CA2398274C Adenosine receptor modulators |
09/17/2009 | WO2009114575A1 Tricyclic spiro pyrimidine derivatives as histamine h4 ligand |
09/17/2009 | WO2009113320A1 Mmp inhibitor |
09/17/2009 | WO2009112691A2 Derivatives of tetrahydroquinoxaline urea, preparation thereof and therapeutic application thereof |
09/17/2009 | WO2009112490A1 Sulfonamides as zap-70 inhibitors |
09/17/2009 | WO2009112461A1 Novel triaryl derivatives useful as modulators of nicotinic acetylcholine receptors |
09/17/2009 | WO2009111943A1 The compounds as the estrogen related receptors modulators and the uses thereof |
09/17/2009 | WO2009111893A1 Substituted pyrimidine compounds and their use as ifnar mediators |
09/17/2009 | US20090234119 Pyrimidinium cation and fluoroalkylsulfonate or fluoroalkylsulfonimide anions; solvents and catalysts |
09/17/2009 | US20090233949 Isoserine derivatives for use as coagulation factor ixa inhibitors |
09/17/2009 | US20090233924 Quinazoline derivatives |
09/17/2009 | US20090233904 Macrocyclic Spiro Pyrimidine Derivatives |
09/17/2009 | CA2750859A1 The compounds as the estrogen related receptors modulators and the uses thereof |
09/17/2009 | CA2718241A1 Novel triaryl derivatives useful as modulators of nicotinic acetylcholine receptors |
09/17/2009 | CA2717529A1 Sulfonamides as zap-70 inhibitors |
09/17/2009 | CA2713367A1 Derivatives of tetrahydroquinoxaline urea, preparation thereof and therapeutic application thereof |
09/16/2009 | EP2100881A1 Pyrimidyl- or pyridinylaminobenzoic acid derivatives |
09/16/2009 | EP2100507A1 Substance capable of inhibiting cytokinin signaling |
09/16/2009 | EP2099772A2 Hydrates of erlotinib hydrochloride |
09/16/2009 | EP2099771A1 Pyrimidine kinase inhibitors |