Patents
Patents for C07D 239 - Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings (42,619)
08/2009
08/12/2009EP2086947A1 Pyrimidines and their use as cxcr2 receptor antagonists
08/12/2009EP2086946A2 Rosuvastatin dehydroabietylamine salt
08/12/2009EP2086945A2 Novel process for the preparation of statins and their pharmaceutically acceptable salts thereof
08/12/2009EP2086329A2 Aquaporin modulators and methods of using them for the treatment of edema and fluid imbalance
08/12/2009CN101506177A 2, 4 -di (arylaminio) -pyrimidine-5-carboxamide compounds as JAK kinases inhibitors
08/12/2009CN101506176A 2-anilino-4-aminoalkyleneaminopyrimidines
08/12/2009CN101506175A 2-anilino-4-(heterocyclic)amino-pyrimidines as inhibitors of protein kinase C-alpha
08/12/2009CN101506168A Positively charged water-soluble prodrugs of n-arylanthranilic acids with very fast skin penetration rate
08/12/2009CN101503402A 2-aniline pyrimidine derivative, as well as preparation and uses thereof
08/12/2009CN100526982C Positive-working photoimageable bottom antireflective coating
08/12/2009CN100526308C Arylvinylazacycloalkane compounds and methods of preparation and use thereof
08/12/2009CN100526298C Amide derivative and medicine
08/12/2009CN100525768C Novel compounds
08/11/2009US7572911 Azotization of 5-amino-3-t-butyl-4-cyanopyrazole, then reacting with couplers and alkylation or arylation, to form azo dyes, used as inks having colorfastness; liquid crystal displays and plasma display panels; excellent color reproducibility
08/11/2009US7572817 Carboxypeptidase U inhibitors; thrombosis, atherosclerosis, adhesions, dermal scarring, cancer, fibrotic conditions, inflammatory diseases; e.g. 2-[(6-Aminopyridin-3-yl)methyl]-3-mercapto-5-[3-(pyrrolidin-1-ylcarbonyl)phenyl]pentanoic acid
08/11/2009US7572816 Therapeutic agents for the treatment of cancer, metabolic diseases and skin disorders
08/11/2009US7572802 For central nervous system diseases, in particular Parkinson's disease, Extra Pyramidal Syndrome, restless legs syndrome and attention deficit hyperactivity disorder
08/11/2009US7572798 Combi-molecules having signal transduction inhibitory properties and DNA damaging properties
08/11/2009US7572793 Tau protein kinase 1 inhibitors; treatment for neurodegenerative disorders; Alzheimer's Disease, Parkinson's disease, Pick's Disease, vision defects; antiischemic, antidiabetic, anticarcinogenic, antitumor agents, antidepressants
08/11/2009CA2368688C Novel inhibitors of formation of advanced glycation endproducts (age's)
08/06/2009WO2009097578A1 Oxim derivatives as hsp90 inhibitors
08/06/2009WO2009096667A2 Novel quinazoline-2,4-dione derivative, and medical compositions for the prophylaxis and treatment of cranial nerve disease containing the same
08/06/2009WO2009096526A1 Carboxylic acid compound or salt thereof
08/06/2009WO2009096198A1 Novel biaryl derivative
08/06/2009WO2009095773A2 Novel heterocycles
08/06/2009WO2009094867A1 Nitrogenous heterocyclic compound with insecticidal activity and its preparation and use
08/06/2009WO2009094831A1 Heteroaromatic compounds, the preparation method and the use thereof
08/06/2009WO2009024323A3 Process for preparing pyrimidine derivatives
08/06/2009WO2008103354A3 Modulators of acetyl-coenzyme a carboxylase and methods of use thereof
08/06/2009US20090197902 Use of Pyrimidine Compounds in the Preparation of Parasiticides
08/06/2009US20090197901 Variolin derivatives and their use as antitumor agents
08/06/2009CA2715069A1 Novel heterocycles
08/06/2009CA2713658A1 Oxim derivatives as hsp90 inhibitors
08/06/2009CA2712819A1 Novel quinazoline-2,4-dione derivative, and medical compositions for the prophylaxis and treatment of cranial nerve disease containing the same
08/05/2009EP1631292B1 4-anilino-quinazoline derivatives as antiproliferative agents
08/05/2009EP1473289B1 Preventives or remedies for alzheimer's disease or amyloid protein fibrosis inhibitors containing nitrogen-containing heteroaryl compounds
08/05/2009EP1383731B1 Biaryl compounds as serine protease inhibitors
08/05/2009EP1249233B9 Npyy5 antagonists
08/05/2009CN101501007A Quinazoline derivative
08/05/2009CN100522952C Insecticidal phthalamide derivatives
08/05/2009CN100522172C Non-sedating barbiturate compounds as neuroprotective agents
08/05/2009CN100522171C 1-benzoyl-piperazine derivatives as glycine uptake inhibitors for the treatment of psychoses
08/04/2009US7569678 Protease inhibitor conjugates and antibodies useful in immunoassay
08/04/2009US7569601 Such as (2E)-3-{4-[1-ethyl-2,2-bis(4-hydroxyphenyl)ethenyl]phenyl}-2-propenoic acid; for selective estrogen receptor modulation; menopausal or postmenopausal disorders, vasomotor symptoms, urogenital or vulvar vaginal atrophy, atrophic vaginitis, female sexual dysfunction, breast cancer, osteoporosis
08/04/2009US7569578 Heterocyclic anti-migraine agents
08/04/2009US7569577 (2S)-1-[4-({4-[3-chloro-2-fluoroanilino]-6-methoxyquinazolin-7-yl}oxy)piperidin-1-yl]-1-oxopropan-2-ol; antiproliferative agents; for treatment of cancers mediated by erbB receptor EGFR tyrosine kinases; psoriasis
08/04/2009US7569575 Synthesis of locked nucleic acid derivatives
08/04/2009CA2425984C 2-pyrimidinyloxy-n-aryl-benzylamine derivatives, their preparation processes and uses
08/04/2009CA2356212C Crystalline bis[(e)-7- [ 4-(4- fluorophenyl)- 6-isopropyl-2- [methyl (methylsulfonyl) amino] pyrimidin -5-yl] (3r,5s)-3, 5-dihydroxyhept -6-enoic acid]calcium salt
07/2009
07/30/2009WO2009094528A1 TRICYCLIC COMPOUNDS AS MODULATORS OF TNF-α SYNTHESIS AND AS PDE4 INHIBITORS
07/30/2009WO2009094442A2 5-fluoro pyrimidine derivatives as fungicides
07/30/2009WO2009092702A2 ((2s,4r)-4,6-dihydroxytetrahydro-2h-pyran-2-yl)methyl carboxylate and process for the production employing a 2-deoxyribose-5-phosphate aldolase
07/30/2009WO2009067600A3 Biaryl pde4 inhibitors for treating inflammation
07/30/2009US20090192122 Inflammatory cytokine release inhibitor
07/30/2009US20090188305 Reference standard for characterization of rosuvastatin
07/30/2009CA2713009A1 ((2s,4r)-4,6-dihydroxytetrahydro-2h-pyran-2-yl)methyl carboxylate and process for the production thereof
07/30/2009CA2712777A1 5-fluoro pyrimidine derivatives as fungicides
07/29/2009EP2081914A2 Crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2h)-pyrimidinyl]-4-fluoro-n-[[methyl-(1-methyl-ethyl)amino]sulphonyl]benzamide
07/29/2009EP1701944B1 2-(amino-substituted)-4-aryl pyramidines and related compounds useful for treating inflammatory diseases
07/29/2009EP1686119B1 Pyrimidine-5-one derivatives as LDL-PLA2 inhibitors
07/29/2009EP1678166B1 Protein kinase inhibitors
07/29/2009EP1268443B1 2-hydroxy-mutilin carbamate derivatives for antibacterial use
07/29/2009CN101495462A Pyrimidine derivatives and their use as pesticides
07/29/2009CN101495461A Novel HIV reverse transcriptase inhibitors
07/29/2009CN101495460A HSP90 inhibitor
07/29/2009CN101492425A Compounds of PARP restrainer
07/29/2009CN101492416A Compounds effecting glucokinase
07/29/2009CN100519540C S-DABO compound, synthesizing method and usage
07/29/2009CN100519527C Inhibitors of histone deacetylase
07/28/2009US7566782 Process for the preparation of rosuvastatin
07/28/2009US7566730 Substituted aminoethers for the treatment of Alzheimer's disease
07/28/2009US7566724 Glycine derivative and use thereof
07/28/2009US7566723 1-phenyl1-3,4-dihydropyrimidin-2(1H)-one derivatives and their use
07/28/2009US7566453 Methods for treating melanomas
07/28/2009CA2472008C Combined therapy against tumors comprising substituted acryloyl distamycin derivatives and protein kinase (serine/threonine kinase) inhibitors
07/23/2009WO2009091962A1 A novel intermediate for the preparation of paliperidone
07/23/2009WO2009091732A1 Compounds for the treatment of metabolic disorders
07/23/2009WO2009090661A1 6.7-dialkoxy ouinazoline derivatives useful for treatment of cancer related disorders
07/23/2009WO2009089851A1 Sulphoximine-substituted quinazoline derivatives as immunomodulators, their preparation and use as medicaments
07/23/2009WO2009013348A3 Pyrimidine derivatives useful for the treatment of inflammatory or allergic conditions
07/23/2009WO2009002808A3 Quinazolinone compounds and methods of use thereof
07/23/2009WO2008103351A3 Heterocyclic aspartyl protease inhibitors
07/23/2009US20090186913 Tetrahalogenated compounds useful as inhibitors of angiogenesis
07/23/2009US20090186912 Anti-infective agents and uses thereof
07/23/2009US20090186911 (RS)-S-[3-({[6-Bromo-4-(isopropylamino)quinazolin-7-yl]oxy}methyl)phenyl] N-(ethoxycarbonyl)-S-ethylsulphoximide, used for the treatment of chronic inflammatory diseases, such as rheumatoid arthritis, Crohn's disease, asthma and multiple sclerosis
07/23/2009US20090186890 Pharmaceutical Formulation of Iressa Comprising a Water-Soluble Cellulose Derivative
07/23/2009US20090186881 1(R)-1-(4-methyl-2-oxo-2,3-dihydro-benzoxazol-6-ylmethyl)-2-oxo-2-[4-(tetrahydropyran-4-yl)-piperazin-1-yl]-ethyl 4-(2-oxo-1,2,4,5-tetrahydro-1,3-benzodiazepin-3-yl); calcitonin gene related peptide antagonist; analgesic, antidiabetic agent; migraine or cluster headaches, non-insulin-dependent diabetes
07/23/2009CA2712367A1 Sulphoximine-substituted quinazoline derivatives as immunomodulators, their preparation and use as medicaments
07/23/2009CA2711737A1 6,7-dialkoxy quinazoline derivatives useful for treatment of cancer related disorders
07/22/2009EP2080744A1 Reaction reagent for trifluoromethylation
07/22/2009EP2079714A1 Hydrates of 2-chloro-5-ý3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoro-methyl)-1-(2h)-pyrimidinyl¨-4-fluoro-n-ýýmethyl-(1-methylethyl)-amino¨sulphonyl¨benzamide
07/22/2009EP2079713A1 Process for synthesis of phenoxy diaminopyrimidine derivatives
07/22/2009EP2079712A2 An improved process for preparing rosuvastatin calcium
07/22/2009EP2079711A2 2-phenyl-6-aminocarbonyl-pyrimidine derivatives and their use as p2y12 receptor antagonists
07/22/2009EP1644337B1 Melanocortin-4 receptor binding compounds and methods of use thereof
07/22/2009EP1477481B1 Process for producing quinazolin-4-one derivative
07/22/2009EP1169293B1 Liquid crystal compounds
07/22/2009CN101490016A 2,4-substituted quinazolines as lipid kinase inhibitors
07/22/2009CN101490015A 瑞舒伐他汀锌盐 Rosuvastatin zinc salt
07/22/2009CN101486685A Microwave extracting process for 4(3H) quinazolone in dyers woad leaf