Patents
Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550)
02/2005
02/03/2005US20050026875 Treating bacterial, viral, or fungal infections, cancer, a lung injury, an eye disorder, neurological disorder or stroke
02/03/2005DE10330358A1 New arylalkanol derivatives used for treating e.g. respiratory diseases, joint diseases, vascular inflammations, skin disorders, kidney and liver diseases and neurological diseases
02/03/2005DE10130504B4 Xanthin- und Phenazon-Acesulfam-H-Komplexe mit verbessertem Geschmack, Verfahren zu ihrer Herstellung und ihre Verwendung Xanthine-phenazone and acesulfame-H-complexes with improved taste, process for their preparation and their use
02/03/2005CA2744317A1 Substituted tetracycline compounds
02/03/2005CA2533494A1 Aryl heteroaromatic products, compositions comprising the same and use thereof
02/03/2005CA2533392A1 Diphenyl substituted cycloalkanes, compositions containing such compounds and methods of use
02/03/2005CA2532403A1 Ppar active compounds
02/03/2005CA2532231A1 Aminopyrazole compounds and use as chk1 inhibitors
02/03/2005CA2529036A1 Indane derivates as muscarinic receptor agonists
02/02/2005EP1501841A2 Non nucleoside reverse transcriptase inhibitors
02/02/2005EP1501810A1 Ionic liquids
02/02/2005EP1501805A1 Substituted pyrazolyl compounds for the treatment of inflammation
02/02/2005EP1299389A4 A process for preparing pyrazolopyrimidinone derivatives for the treatment of impotence
02/02/2005CN1575279A Substituted thioacetamides
02/02/2005CN1575273A 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor antagonists
02/02/2005CN1572792A Pyrazolo [4, 3-d] pyrimidine derivatives
02/02/2005CN1187335C Benzoylpyrazols and their use as herbicides
02/01/2005US6849745 Fluorescent dye for use in the detection of preferential compounds
02/01/2005US6849653 Substituted pyrazolyl benzenesulfamide compounds for the treatment of inflammation
02/01/2005US6849649 N-phenpropylcyclopentyl-substituted glutaramide derivatives as inhibitors of neutral endopeptidase
02/01/2005US6849631 Semicarbazides and their uses
02/01/2005US6849623 For use as human and veterinary medicine
02/01/2005US6849618 Herbicidal compositions for the desiccation/ defoliation of plants
02/01/2005US6849617 Administering Tissue factor pathway inhibitors for prophylaxis of thrombosis and cardiovascular disorders; anticoagulants
01/2005
01/27/2005WO2005007635A2 Combretastatin derivatives with cytotoxic action
01/27/2005WO2005007621A2 Ubiquitin ligase inhibitors
01/27/2005WO2005007620A2 New n-hydroxy-4-(3-phenyl-5-methyl-isoxazole-4-yl)-benzenesulfonamide solvates
01/27/2005WO2004098518A3 Pyrazole-amide compounds useful as kinase inhibitors
01/27/2005WO2004096757A8 Aminopropanol derivatives as sphingosine-1-phosphate receptor modulators
01/27/2005US20050020659 Substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists
01/27/2005US20050020602 Bone disorders; reduction concentration of parathyroid hormone in blood
01/27/2005US20050020593 Anticancer agents
01/27/2005US20050020584 Benzamide derivatives as antagonists of orexin receptors
01/27/2005US20050020564 Pyrazole-amides and sulfonamides as sodium channel modulators
01/27/2005US20050015893 Hair dyes, oxidation color dyes for human hair
01/27/2005DE10331496A1 Verfahren zum Herstellen von Difluoracetessigsäurealkylestern A process for producing Difluoracetessigsäurealkylestern
01/27/2005CA2531389A1 Combretastatin derivatives with cytotoxic action
01/27/2005CA2530175A1 New n-hydroxy-4-(3-phenyl-5-methyl-isoxazole-4-yl)-benzenesulfonamide solvates
01/26/2005EP1499600A1 Heteroaryl substituted biphenyl derivatives as p38 kinase inhibitors
01/26/2005EP1499597A2 Compounds and methods for inducing apoptosis in proliferating cells
01/26/2005CN1186342C Substituted (4-bromopyrazole-3-yl) indole
01/26/2005CN1186332C New thryoid receptor ligands and process II
01/25/2005US6846935 Reacting 1,1,1-trifluoro-4-(2,4-difluorophenyl)-3-buten-2-one with phenylhydrazine chlorhydrate, to form 1-phenyl-5-(2,4-difluorophenyl)-4,5-dihydro-3-trifluoromethyl-1H-pyrazole, then resolving into stereoisomers; enzyme inhibitors
01/25/2005US6846919 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof
01/25/2005US6846825 Antibacterial agents
01/25/2005CA2191647C Process improvement in the synthesis of n-[3-(3-cyanopyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-n-ethylacetamide
01/25/2005CA2068224C Novel potent inducers of terminal differentiation and method of use thereof
01/20/2005WO2005005393A2 Cck-1 receptor modulators
01/20/2005WO2005004810A2 Arylsulfonamide derivatives
01/20/2005WO2004069158A3 Substituted pyrazoles, compositions containing such compounds and methods of use
01/20/2005US20050014813 High yield; synthetic pharmaceutical intermediate; diabetes, insulin sensitizers
01/20/2005US20050014805 Hypotensive agents; antidiabetic agents; cardiovascular disorders; anticholesterol agents; anticancer agents
01/20/2005US20050014787 5-amidino-2-hydroxybenzenesulfonamide derivatives medicinal compoistions containing the same medicinal use thereof and intermediates in the production thereof
01/20/2005US20050014649 Herbicides; and synthesis thereof
01/20/2005CA2530737A1 Cck-1 receptor modulators
01/19/2005EP1496900A2 New pharmaceutical compositions based on anticholinergics and p38 kinase inhibitors
01/19/2005EP1496892A2 1h-benzo(f)indazol-5-yl derivatives as selective glucocorticoid receptor modulators
01/19/2005EP1496838A2 Substituted amides
01/19/2005EP1230244B1 Pyrazolecarboxylic acid tricyclic derivatives, preparation and pharmaceutical compositions containing same
01/19/2005CN1568185A Compounds effecting glucokinase
01/19/2005CN1566096A Prostaglandin agonists and their use to treat bonedisorders
01/19/2005CN1185234C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives
01/18/2005US6844436 Chlorosulfonation, cyclization, salt formation'; impotency; cardiovascular disorders; antidiabetic agents; central nervous system disorders
01/18/2005US6844407 Nitrogen-nitrogen bond covalently bonded to a thiocarbonyl moiety
01/16/2005WO2005000281A2 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
01/16/2005CA2529436A1 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
01/13/2005WO2005003098A1 Heterocyclically substituted pentanol derivatives, method for the production thereof, and use thereof as anti-inflammatory agents
01/13/2005WO2005003077A1 Method for producing difluoro-acetyl-acetic acid alkylesters
01/13/2005WO2005002574A1 Pyrazolidinedione derivatives and their use as platelet aggregation inhibitors
01/13/2005WO2004099134A3 Glutaminyl based dp iv-inhibitors
01/13/2005US20050009900 3-Substituted with a heterocyclic group, e.g., 2-Chloro-5-[1-(2,3-dihydroxy-propyl)-5-methyl-1H-pyrazol-3-yl]-N-(1-hydroxy-cycloheptylmethyl)-benzamide; treatment of IL-1 mediated disorders, including osteo- and rheumatoid arthritis, allergies, asthma, COPD, cancer, and reperfusion or ischemia in stroke
01/13/2005US20050009896 Drugs comprising combination of antithrombotic agent with pyrazolone derivative
01/13/2005US20050009876 Indazole compounds, compositions thereof and methods of treatment therewith
01/13/2005US20050009871 Ubiquitin ligase inhibitors
01/13/2005US20050009834 E.g., 3-(2-chloro-6-fluorophenyl)-1-[4-(3,5-dichloropyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole and 3-(3-chloropyridin-2-yl)-1-[4-(3-chloro-5-trifluoromethylpyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole; for use as pesticides, especially insecticides and acaricides
01/13/2005US20050009819 1-Aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
01/13/2005CA2531060A1 Heterocyclically-substitued pentanol derivatives, process for their production and their use as anti-inflammatory agents
01/12/2005EP1495035A1 Method for the production of bis(perfluoroalkyl)phosphinic acids and the salts thereof
01/12/2005EP1495015A1 3-aminophenol derivatives and dyes that contain these compounds while serving to dye keratin fibers
01/12/2005EP1495005A1 Pyrazole compounds as anti-inflammatory and analgesic agents
01/12/2005EP1494997A1 Substituted aryl amides
01/12/2005EP1494993A2 Novel curcumin analogues and uses thereof
01/12/2005EP1494989A2 Compounds that modulate ppar activity and methods for their preparation
01/12/2005EP1494673A1 Compounds having unique cb1 receptor binding selectivity and methods for their production and use
01/12/2005EP1494666A1 Orally deliverable pharmaceutical composition comprising an active compound having an aminosulfonyl group (cox-2 inhibitor), a polyethylene glycol and a free-radical scavenging antioxidant
01/12/2005EP1494645A2 Method of treating mucus hypersecretion
01/12/2005EP0944604B1 Guanidinyl heterocycle compounds useful as alpha-2 adrenoceptor agonists
01/12/2005CN1562976A Method for synthesizing 1-methyl-benzdiazole-3-formic acid
01/12/2005CN1184207C Process for producing insecticide intermediate
01/12/2005CN1184206C Prepn process of pyrazole derivative
01/11/2005US6841624 Subjecting mixture of one or more monomers, at least one free radical source and a control agent to polymerization condition, wherein control agent contains at least one N-N bond covalently bonded to a thiocarbonyl group
01/11/2005CA2284051C Pharmaceutical composition for oral administration of a n-piperidino-3-pyrazolecarboxamide derivative, its salts and their solvates
01/06/2005WO2005002293A2 Cox-2-targeted imaging agents
01/06/2005WO2005000820A2 4-cyanopyrazole-3-carboxamide derivatives preparation and application thereof as cb1 cannabinoid antagonists
01/06/2005WO2005000813A1 Heteroarylamino-phenylketone derivatives and their use as kinase inhibitors
01/06/2005WO2005000800A1 Cathepsin cysteine protease inhibitors
01/06/2005WO2005000309A2 Chemical compounds
01/06/2005US20050004176 Pyrazole-amide compounds useful as kinase inhibitors
01/06/2005US20050004135 Pyrazole ether derivatives as anti-inflammatory/analgesic agents
01/06/2005US20050004133 Inhibiting ligand gated ion channel vanilloid receptor (VR1); pain relievers; such as 6-(3,4-dichloro-phenyl)-N-(2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-nicotinamide