Patents
Patents for C07D 223 - Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom (8,732)
09/2006
09/06/2006CN1827601A Crystalline form gamma-d of the chlorohydrate of ivabradine, process for its preparation and pharmaceutical compositions containing it
09/06/2006CN1827600A Crystalline form beta of the chlorhydrate of ivabradine, process for its preparation and pharamcetuical composition containing it
09/06/2006CN1827599A Crystalline form beta-d of the chlorohydrate of ivabradine, process for its preparation and pharmaceutical compositions containing it
09/05/2006US7101870 2R,3S) N1-[6,7-dihydro-5-(3-phenoxybenzyl)-6-oxo-5H-dibenz[b,d]azepin-7-yl]-2-(2-methylpropyl)-3-(propyl)-butanediamide; treating Alzheimer's disease and Down's Syndrome by inhibiting production of A beta -peptide
08/2006
08/31/2006WO2006091301A2 Passcodes
08/31/2006WO2006090044A1 Lactam production method
08/31/2006WO2006056696A3 2-alcoxy-3,4,5-trihydroxy-alkylamides, preparation thereof, compositions containing them and use thereof
08/31/2006WO2006023187A3 Cycloalkylamine derivatives as nk-1 /ssri antagonists
08/31/2006US20060194967 Process for the preparation of Fenoldopam Mesylate
08/31/2006US20060194964 Gamma d-Crystalline form of ivabradine hydrochloride, a process for its preparation and pharmaceutical compositions containing it
08/31/2006US20060194963 Procoralan; brandycardial agent: angina pectoris, myocardial infarct, heart failure, myocardial ischaemia, supraventricular rhythm disturbances; stability and processability
08/31/2006US20060194962 Beta-crystalline form of ivabradine hydrochloride, a process for its preparation and pharmaceutical compositions containing it
08/31/2006US20060194790 Bridged bicyclic amine derivatives useful as CCR-3 receptor antagonists
08/31/2006US20060194787 substituted 1,1,4-1l6-trioxo[1,2]thiazepan-4-ylamide-derived protease inhibitors which inhibit the likes of cathepsin K; treating osteoporosis, osteo- and rheumatoid arthritis and periodontal disease; inhibiting excessive cartilage or matrix degradation
08/31/2006US20060194786 Process and intermediates for preparing benzazepines
08/30/2006EP1695965A1 Crystalline form beta of the chlorhydrate of ivabradine, process for its preparation and pharamcetuical composition containing it
08/30/2006EP1694334A1 Tetrahydrobenzazepines and their use in the modulation of the dopamine d3 receptor
08/29/2006US7098203 and selective serotonin reuptake inhibitors; 4-benzyloxymethyl-4-phenylazepanes; antidepressants; anxiety
08/29/2006CA2112779C Arylsulfonamido-substituted hydroxamic acids
08/24/2006WO2006075925A3 Method for preparation of 10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide
08/23/2006EP1692129A1 Keto lactam compounds and use thereof
08/23/2006EP1691814A2 Anti-inflammatory agents
08/23/2006CN1823059A Selective D1/dD receptor antagonists for the treatment of obesity and CNS disorders
08/23/2006CN1823047A Method for racemisation of (S)-(+)- and (R)-(-)-10,11-dihydro-10-hydroxy-5h-dibenz[b,f]azepine-5-carboxamide and optically enriched mixtures thereof
08/23/2006CN1271167C Organic electroluminescent element
08/23/2006CN1271057C Method for preparing 1-methyl-3-ethyl-3-(3-hydroxy phenyl)-hexa hydrogen-1 H azepin hydrochloride
08/22/2006US7094896 Diaminothiazoles having antiproliferative activity
08/22/2006US7094778 Nervous system disorders; muscular disorders; urogenital disorders; gastrointestinal disorders; repiratory system disorders; antiallergens; side effect reduction
08/17/2006WO2006085688A1 Psychogenic pain therapeutic agent
08/17/2006WO2006021213A3 Vasopressin v1a antagonists
08/17/2006US20060183896 Optically active quaternary ammonium salt, process for producing the same, and process for producing optically active alpha-amino acid derivative with the same
08/17/2006US20060183732 Novel lactams and uses thereof
08/16/2006EP1019075B9 Beta 2-adrenergic receptor agonists
08/16/2006CN1820000A A method for the preparation of enantiomerically pure mirtazapine
08/16/2006CN1817865A Preparation of sinomontanine and its hydrobromide
08/16/2006CN1269807C Aryl substituted piperazine for curing benign prostatauxe
08/16/2006CN1269804C Metalloproteinase inhibitors
08/16/2006CN1269803C Process for preparing epsilon-caprolactam
08/15/2006US7091339 Reacting the dibenz(b,f)azepaine with Group 1a, Group 2a cyanide
08/10/2006US20060178362 Substituted heterocyle fused gamma-carbolines
08/09/2006EP1688418A2 Chemokine receptor antagonists and methods of use thereof
08/09/2006EP1688393A1 High silica cds-1 zeolite
08/09/2006EP1687279A1 7- [4-(4-chlorobenzyloxy) benzenesulfonyl]-8-methoxy-3-methyl-2,3,4,5-tetrahydro-1h-3-benzazepinium maleate or tosylate as antipsychotics
08/09/2006EP1687005A1 7-phenylsulfonyl-tetrahydro-3-benzazepine derivatives as antipsychotic agents
08/09/2006EP1453832B1 Ring fused pyrazole derivatives
08/09/2006CN1268627C Process for preparing 1.8-diazadicyclo [5,4,0] -7 undecene
08/08/2006US7087596 2-oxo-piperidinyl- and 2-oxo-azepanyl alkanoic acid derivatives for the treatment of epilepsy and other neurological disorders
08/02/2006EP1685103A1 3-aminopyrrolidone derivatives
08/02/2006EP1014966B1 Pharmaceutical for treatment of neurological and neuropsychiatric disorders
08/02/2006CN1810786A Synthesis of caprolactam and its oligomer
08/02/2006CN1267099C Medicament with protective effect against oxidative-toxic substances, particularly against cardiotoxin substances
08/01/2006US7084154 Reducing pain
07/2006
07/27/2006WO2006078753A1 N-substituted heterocyclic sulfonamides
07/27/2006US20060166968 Crystalline form of oxcarbazepine
07/27/2006US20060166966 4-amino-azepan-3-one compounds as cathepsin k inhibitors useful in the treatment of osteoporosis
07/27/2006US20060165648 Compounds, compositions, and methods for controlling biofilms
07/27/2006CA2595173A1 N-substituted heterocyclic sulfonamides
07/27/2006CA2593667A1 Process for the preparation of fenoldopam mesylate
07/26/2006CN1809532A Method for making caprolactam
07/26/2006CN1807429A Use of fern in extracting harringtonine or homoharringtonine
07/26/2006CN1266136C Kinetic resolution of intermediate for preparing benazepril and its analogues
07/25/2006US7081458 Small molecule, non-peptide antagonists; antidiabetic agents; obesity; {5-[1-4-Methoxy-2,3-dimethyl-phenyl)-ethyl]-(1S,4S)-2,5-diaza-bicyclo[2.2.1]hept-2-yl}-(4-trifluoromethyl-phenyl)-methanone
07/25/2006US7081455 sleep disorders associated with 5-HT2A serotonin receptor modulation; antagonists or agonists
07/20/2006WO2006075925A2 Method for preparation of 10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide
07/20/2006US20060160894 Benzamides as ppar modulators
07/20/2006CA2594869A1 Method for preparation of 10,11-dihydro-10-hydroxy-5h-dibenz/b,f/azepine-5-carboxamide
07/19/2006EP1681291A1 Process for the preparation of norgalanthamine, its isomers, salts and hydrates
07/19/2006EP1680406A1 N-substituted benzene sulfonamides
07/19/2006EP1680405A1 Bengamide derivatives, method for the production thereof and use thereof for the treatment of cancer
07/19/2006EP1680400A2 Derivatives of n-[ phenyl(pyrrolidine-2-yl)methyl]benzamide and n-[ (azepan-2-yl)phenylmethyl]benzamide, preparation method thereof and application of same in therapeutics
07/19/2006EP1680127A1 Benzazepine derivatives as mao-b inhibitors
07/19/2006EP1370556B1 Metalloproteinase inhibitors
07/19/2006EP1325054B1 Twisted polymers, uses thereof and processes for the preparation of statistical copolymers
07/19/2006CN1805939A Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases
07/19/2006CN1805938A Benzazepine derivatives useful for the treatment of 5HT2C receptor associated diseases
07/19/2006CN1803760A N-arylation process with hydrazone as ligand in aqueous phase system
07/19/2006CN1264808C Production of alkyl 6-aminocaproate
07/18/2006US7078424 Central nervous system disorders; alopecia
07/13/2006WO2006073967A1 Piperidine derivatives as prodrugs of potassium channel inhibitors
07/13/2006US20060154872 chemical intermediate for Hemiasterlin, first isolated from the sponge Hemiasterella; anticarcinogenic agent for treatment of colon cancer, tumor; prevention of restenosis of blood vessels subject to traumas such as angioplasty and stenting
07/12/2006EP1679303A1 Process for preparing 1-alkoxycarbonyl-3-phenylpropyl derivative
07/12/2006EP1679069A1 Novel piperidine derivative
07/12/2006EP1678140A2 Novel process for preparation of 10-oxo-10, 11-dihydro-5h-dibenz [b,f]azepine-5-carboxamide (oxcarbazepine) via intermediate, 10-methoxy-5h-dibenz [b,f] azepine-5-carbonylchloride
07/12/2006EP1441718B1 Use of carbinols for the treatment of neuropathic dysfunction
07/12/2006CN1802356A Alkylated iminodibenzyls as antioxidants
07/12/2006CN1802159A 2-phenoxy- and 2-phenylsulfomamide derivatives with CCR3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders
07/11/2006US7074920 Process for the synthesis of 1,3-dihydro-2H-3-benzazepin-2-one compounds, and to the application thereof in the synthesis of ivabradine and addition salts thereof with a pharmaceutically acceptable acid
07/11/2006US7074782 Administering to a patient suffering from caspase mediated diseses, an effective amount of a mono,bi or tri-heterocyclic ring containing nitrogen atom attached to ester or thioester to form carbamate group, as caspase inhibitor
07/06/2006WO2006046039A3 Tetracyclic indole derivatives as antiviral agents
07/06/2006US20060148808 N'-methyl-2-[(p-fluorophenyl)-4-oxo-butyl]piperazino[1,2-fg]gamma-carboline; N'-methyl-2-[p-fluorophenoxypropyl]piperazino[1,2-fg]gamma-carboline; serotonin modulators; sleep disorders; central nervous system disorders
07/05/2006EP1676846A2 Hydantoin derivatives as MMP inhibitors
07/04/2006US7071211 Vision disorders; adjustment activation of gelatinase
07/04/2006US7071186 Drug abuse; antiserotonine agents; central nervous system disorders; sleep disorders
07/04/2006US7071184 Protease inhibitors
07/04/2006CA2130797C 2,3,4,5-tetrahydro-1h-3-benzazepines having anti-psychotic activity, and synthesis of .alpha.-substituted-arylacetamides
06/2006
06/29/2006US20060142566 Enantioselective process for the preparation of both enantiomers of 10,11-dihydro-10-hydroxy-5h-dibenz[b,f]azepine-5-carboxamide and new crystal forms thereof
06/29/2006US20060142264 Novel amide derivatives
06/29/2006CA2589988A1 Crystalline forms of (r)-8-chloro-1-methyl- 2,3,4,5-tetrahydro-1h-3-benzazepine hydrochloride
06/28/2006EP1674099A1 Therapeutic combination of amlodipine and benazepril / benazeprilat
06/28/2006EP1673347A1 Substituted dibenzo-azepine and benzo-diazepine derivatives useful as gamma-secretase inhibitors
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