Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273) |
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12/12/2002 | US20020188122 Such as pyridine-4-carboxaldehyde-(4-Morpholinylprop-3-yl) imine for use in therapy as cytokine inhibitors |
12/12/2002 | US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV |
12/12/2002 | US20020188015 Method and composition for rejuvinating cells, tissues organs, hair and nails |
12/12/2002 | CA2449942A1 Characterising polypeptides |
12/12/2002 | CA2449813A1 Process for preparing chiral diol sulfones and dihydroxy acid hmg coa reductase inhibitors |
12/12/2002 | CA2449021A1 Novel compounds and compositions as cathepsin inhibitors |
12/12/2002 | CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases |
12/12/2002 | CA2446719A1 Benzoylsulfonamides and sulfonylbenzamidines for use as antitumour agents |
12/11/2002 | EP1264827A1 Process for the preparation of Tosylbenzylformamides |
12/11/2002 | EP1264825A1 Beta-Hydroxyalkylpicoliniumsalts |
12/11/2002 | EP1264820A1 Novel amide compounds |
12/11/2002 | EP1263755A2 Cyclic beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha |
12/11/2002 | EP1263732A1 Corticotropin releasing factor antagonists |
12/11/2002 | EP1263731A1 Method for producing 5-aryl nicotinaldehydes |
12/11/2002 | EP1263714A1 Novel phenylheteroalkylamine derivatives |
12/11/2002 | EP1263712A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds |
12/11/2002 | EP1263711A1 Novel use of phenylheteroalkylamine derivatives |
12/11/2002 | EP1100805B1 Medicine nitrate salts |
12/11/2002 | EP1058678B1 Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes |
12/11/2002 | EP0966441B1 Process for preparing 2-hydroxy-6-trifluoromethylpyridine |
12/11/2002 | EP0966436B1 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases |
12/11/2002 | EP0920456B1 Phosgenated oxime resins and their preparation |
12/11/2002 | EP0863891B1 (methylsulfonyl)phenyl-2-(5h)-furanones as cox-2 inhibitors |
12/11/2002 | EP0805796B1 Cell adhesion inhibitors |
12/11/2002 | EP0628030B1 2,3,4,5-TETRAHYDRO-1H --3-BENZAZEPINES HAVING ANTI-PSYCHOTIC ACTIVITY, AND SYNTHESIS OF $g(a)-SUBSTITUTED-ARYLACETAMIDES |
12/11/2002 | EP0624155B2 Carbamates and plant-protecting agents containing them |
12/11/2002 | CN1384870A Method of bleaching stained fabrics |
12/11/2002 | CN1384869A Method of pretreating and bleaching stained fabrics |
12/11/2002 | CN1384837A Ligand and complex for catalytically bleaching substrate |
12/11/2002 | CN1384742A Use of bis-sulfonamides for producing medicaments used for preventing or treating hyperlipidaemia |
12/11/2002 | CN1095692C Halogenation catalyst |
12/10/2002 | US6492562 Invention also relates to novel intermediates and the resulting modified polyketides and antibiotics. |
12/10/2002 | US6492539 Preparation of preparing substituted indanones |
12/10/2002 | US6492524 Process for the synthesis of an aryl pyridine base using a zeolite catalyst |
12/10/2002 | US6492519 Chemical intermediate for antihistamine |
12/10/2002 | US6492502 Reduction of a quaternary ammonium containing nitro compound, to form an intermediate, oxidizing to give azo compound; useful for dyeing hair |
12/10/2002 | US6492423 Hepatitis c and b viricides |
12/10/2002 | US6492412 Prevention of loss and restoration of bone mass by certain prostaglandin agonists |
12/10/2002 | US6492405 Compounds containing sulfhydryl, disulfide, or group(s) capable of being converted in-vivo to a sulfhydryl group, and at least one nitrate group; use as substitutes for existing tolerance-inducing nitric oxide donors |
12/10/2002 | US6492399 Pharmaceutical compositions and methods for use |
12/10/2002 | US6492396 Substituted thioacetamides |
12/10/2002 | US6492393 Compounds useful as anti-inflammatory agents |
12/10/2002 | US6492372 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 |
12/10/2002 | US6492368 Benzamidine derivatives as factor XA inhibitors |
12/10/2002 | US6492363 2-(4-bromo or 4-iodo phenylamino) benzoic acid derivatives |
12/10/2002 | US6492362 Compounds and compositions as cathepsin S inhibitors |
12/10/2002 | US6492351 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
12/10/2002 | US6492293 Polymerisation catalyst |
12/10/2002 | US6491989 Fluorinated naphthalene derivatives and their use in liquid crystal mixtures |
12/10/2002 | CA2109934C Substituted indoles as anti-aids pharmaceuticals |
12/09/2002 | WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments |
12/09/2002 | CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments |
12/05/2002 | WO2002097393A2 Cleavable surfactants and methods of use thereof |
12/05/2002 | WO2002096901A2 1,3-dihydroxybenzene derivatives and colorants containing said compounds |
12/05/2002 | WO2002096882A1 Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage |
12/05/2002 | WO2002096879A1 Aminoquinoline and aminopyridine derivatives and their use as adenosine a3 ligands |
12/05/2002 | WO2002096878A1 A short synthesis of pyridine-based pharmaceutical intermediates with sulfur-containing groups at the 2- and 3-positions |
12/05/2002 | WO2002096877A1 5-chloro-3-(4-methanesulfonylphenyl)-6'-methyl-[2,3']bipyridinyl in pure crystalline form and process for synthesis |
12/05/2002 | WO2002096876A1 Carbamate and oxamide compounds as inhibitors of cytokine production |
12/05/2002 | WO2002096867A2 Inhibitors of protein kinase for the treatment of disease |
12/05/2002 | WO2002096864A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments |
12/05/2002 | WO2002096858A1 Cinnamide derivatives as kcnq potassium channel modulators |
12/05/2002 | WO2002096516A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease |
12/05/2002 | WO2002096421A1 5-substituted-2-arylpyridines as crf1 modulators |
12/05/2002 | WO2002078693A3 N-(2-arylethyl)benzylamines as antagonists of the 5-ht6 receptor |
12/05/2002 | WO2002064547A3 Isophthalic acid derivatives as matrix metalloproteinase inhibitors |
12/05/2002 | WO2002011707A3 Drugs for incontinence |
12/05/2002 | US20020183517 Reacting dihydric alcohol characterized by four to six carbons, preferably 1,5-pentanediol, with excess ammonia in presence of ZSM-5 catalyst modified with nickel, copper or cobalt |
12/05/2002 | US20020183397 Substituted n-phenyl-n-fused-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity |
12/05/2002 | US20020183365 Therapy or ameliorating an indication of the invention in an animal, including a human, comprising administering heteroaryl compond |
12/05/2002 | US20020183362 2-Fluorobenzenesulfonyl compounds for the treatment of inflammation |
12/05/2002 | US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm |
12/05/2002 | US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder |
12/05/2002 | US20020183324 Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors |
12/05/2002 | US20020183323 For therpay of inflammatory bowel disease, cerebral ischemia and arthritis, adult respiratory distress syndrome (ARDS) and myocarditis, as adjuvants to short term immunosuppression in transplant therapy |
12/05/2002 | US20020183321 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof |
12/05/2002 | US20020183316 Amidoalkyl-piperidine and amidoalkyl-piperazine derivatives useful for the treatment of nervous system disorders |
12/05/2002 | DE10127041A1 New glycine N-(1-biphenyl-4-yl-2-substituted-ethyl)-amides, are integrin receptor inhibitors useful for treating e.g. angiogenic, cardiovascular, inflammatory and osteolytic or tumor diseases |
12/05/2002 | DE10125567A1 New N-aroyl-N'-(carbamoyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibiting hypoglycemic agents, especially useful for treating type II diabetes |
12/05/2002 | CA2448899A1 A short synthesis of pyridine-based pharmaceutical intermediates with sulfur-containing groups at the 2- and 3-positions |
12/05/2002 | CA2448894A1 Cinnamide derivatives as kcnq potassium channel modulators |
12/05/2002 | CA2448626A1 Carbamate and oxamide compounds as inhibitors of cytokine production |
12/05/2002 | CA2448198A1 5-substituted-2-arylpyridines as crf1 modulators |
12/05/2002 | CA2448023A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments |
12/05/2002 | CA2447657A1 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease |
12/05/2002 | CA2445647A1 1,3-dihydroxybenzene derivatives and colorants containing said compounds |
12/04/2002 | EP1261595A1 Arylpiperazines and arylpiperidines and their use as metalloproteinase inhibiting agents |
12/04/2002 | EP1261590A1 Piperidine- and piperazine substituted n-hydroxyformamides as inhibitors of metalloproteinases |
12/04/2002 | EP1261579A1 Dehydroamino acids |
12/04/2002 | EP1261338A1 Compositions and methods for treatment of epilepsy |
12/04/2002 | EP1261336A2 Il-8 receptor antagonists |
12/04/2002 | EP1261327A2 Adenosine receptor modulators |
12/04/2002 | EP1261321A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof |
12/04/2002 | EP1001930B1 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases |
12/04/2002 | CN1383425A Uracil substituted phenyl sulfamoyl carboxamides |
12/04/2002 | CN1383424A Aryl and heteroacrylcyclopropyl oxime ethers and their use as fungicides |
12/03/2002 | US6489497 Manufacture of α-olefins |
12/03/2002 | US6489485 Para-amine substituted phenylamide glucokinase activators |
12/03/2002 | US6489483 Reacting acetyl-substituted pyridine derivative with 3-aminoacrolein, reacting reaction product with ammonia or ammonium salt |
12/03/2002 | US6489481 Compounds used for treatment and/or prevention of neuronal apoptosis and/or excitotoxicity related neurological disorders |