Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
02/2003
02/06/2003US20030026521 Optical interleaver
02/06/2003CA2454903A1 Substituted piperazines as modulators of the melanocortin receptor
02/06/2003CA2452159A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods
02/05/2003EP1281703A1 Process for the preparation of 5-alkoxy-oxazoles as well as of pyridoxines
02/05/2003EP1281702A2 Calcium receptor active molecules
02/05/2003EP1280799A1 Ortho-substituted anthranilic acid amides and their use as medicaments
02/05/2003EP1280797A1 Inhibitors of dipeptidyl peptidase iv
02/05/2003EP1280776A1 Substituted benzoic acid amides and use thereof for the inhibition of angiogenesis
02/05/2003EP1280765A2 Fluorous tagging compounds and their use
02/05/2003EP1280764A2 Inhibitors of histone deacetylase
02/05/2003EP1280757A2 New gamma selective retinoids
02/05/2003EP1086078B1 Neuropeptide y5 receptor antagonists
02/05/2003EP1082121A4 Hiv integrase inhibitors
02/05/2003EP1037868B1 $g(a)-HYDROXY, -AMINO, AND HALO DERIVATIVES OF $g(b)-SULFONYL HYDROXAMIC ACIDS AS MATRIX METALLOPROTEINASES INHIBITORS
02/05/2003EP0742201B1 Process for producing aromatic or heteroaromatic sulfur compounds
02/05/2003CN1395566A Corticotropin releasing factor antagonists
02/05/2003CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
02/05/2003CN1394859A Intermediate for preparing cyclopentane formamide compound and its preparation method
02/05/2003CN1394855A Substituted heterocyclic compound
02/05/2003CN1394854A Polysubstituted pyridine salt compound and its preparation method
02/05/2003CN1100777C N-heterocyclic derivatives as NOS inhibitor
02/05/2003CN1100760C Process for preparation of arylamides of heteroarometic carboxylic acids
02/05/2003CN1100758C Process for preparing [(5,6-dicarboxy 3-pyridyl) methyl] ammonium halides
02/05/2003CN1100540C Protein tyrosine kinase aryl and heteroaryl quinazoline compounds having selective inhibition of HER-2 autophosphorylation properties
02/04/2003US6515134 Substituted acetylpridine derivatives and process for the preparation of intermediates for optically active beta-3 agonist by the use of the same
02/04/2003US6515130 The invention relates to a process of preparing (S-(R*,S*))-beta -(((1-(1-oxo-3-(4-piperidinyl)propyl)-3-piperidinyl) carbonyl)amino)-3-pyridinepropanoic acid derivatives represented by the antagonists of the platelet fibrinogen
02/04/2003US6515128 Dissolving 6-hydroxy-3,4-dihydroquinolinone and a base in water; dissolving a 1-cyclohexyl-5- (4-halobutyl)-tetrazole in water-immiscible solvent, mixing aqueous phase and organic phase in presence of phase transfer catalyst; recovering
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6515028 Glucamine compounds for treating hepatitis virus infections
02/04/2003US6515026 Potentiators of glutamate receptor function
02/04/2003US6515024 Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
02/04/2003US6515023 Thrombin receptor antagonists
02/04/2003US6515021 The compounds according to the invention have pronounced activity in the fields of cell differentiation and cell proliferation
02/04/2003US6514997 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
02/04/2003US6514995 Metal complex is capable of forming a benzenoid diradical under physiological conditions and/or under photothermal conditions
02/04/2003US6514985 Induce the biosynthesis of cytokines such as interferon and tumor necrosis factor; exhibit antiviral and antitumor properties
02/04/2003US6514976 Arylpiperazines having activity at the serotonin 1A receptor
02/04/2003US6514964 Treating diseases, conditions or disorders mediated by integrin receptors, such as vitronectin and fibronectin receptors
02/03/2003WO2002016312A2 Novel compounds inhibiting factor xa activity
02/03/2003CA2418283A1 Novel compounds inhibiting factor xa activity
01/2003
01/31/2003WO2002012169A1 Amino diphenyl ethers and amido diphenyl ethers
01/31/2003CA2417880A1 Amino diphenyl ethers and amido diphenyl ethers
01/30/2003WO2003008559A2 Novel analogs of choline for neuroprotection and cognitive enhancement in neurodegenerative disorders
01/30/2003WO2003008384A1 Substituted 2-thio-3, 5-dicyano-4-phenyl-6-aminopyridines and their use as adenosine receptor-selective ligands
01/30/2003WO2003008383A1 Production of enantiomer pure 3r, 5s- (+) natrium erythro- (e) 7-'4-(4-fluorophenyl)-2, 6-diisopropyl-5-methoxymethyl-pyrid-3-yl!-3, 5-dihydroxy-hept-6-e-noate
01/30/2003WO2003008372A1 Diamine derivative, process for producing the same, and bactericide containing the same as active ingredient
01/30/2003WO2003007954A2 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
01/30/2003WO2003007951A1 A synergistic pharmaceutical combination for the prevention or treatment of diabetes
01/30/2003WO2003007950A1 (pyridinyl and pyrimidyl) trienoic acid derivatives as retinoid x receptor modulators
01/30/2003WO2003007942A1 Substituted isoindoles and the use thereof
01/30/2003WO2003007931A1 Sulfonamide derivatives
01/30/2003WO2003002522A8 Peptide deformylase inhibitors
01/30/2003WO2002070510A3 Amino dicarboxylic acid derivatives with pharmaceutical properties
01/30/2003US20030023088 To produce medicament for therapy and prophylaxis of cancer
01/30/2003US20030023087 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
01/30/2003US20030023084 For use in the oral hygiene
01/30/2003US20030022944 Self-emulsifying formulations of cholesteryl ester transfer protein inhibitors
01/30/2003US20030022935 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical agents
01/30/2003US20030022921 Stable pharmaceutical formulation comprising torsemide modification II
01/30/2003US20030022903 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
01/30/2003US20030022902 Based upon 2-(N-(7-benzyl-9-methyl-1,5-dioxonan-2,6-dione-3-yl)amido)-3-hydroxy-4 -methoxypyridine; use as agricultural fungicide
01/30/2003US20030022893 Hydroxamic and carboxylic acid derivatives
01/30/2003US20030022891 Melanin-concentrating hormone (MCH); treating metabolic and eating disorders, such as hyperphagia, and diabetes; urea, thiourea and cyano-guanidine compounds of given formula
01/30/2003US20030022887 Unsymmetrical cyclic diamine compound
01/30/2003US20030022886 Bis (2-aryl-5-pyridyl) derivatives
01/30/2003US20030022884 Heterocycle derivatives and drugs
01/30/2003US20030022266 Novel agents for replacement of NAD+/NADH system in enzymatic reactions
01/30/2003CA2682251A1 A synergistic pharmaceutical combination for the prevention or treatment of diabetes
01/30/2003CA2453650A1 Substituted isoindoles and the use thereof
01/30/2003CA2453613A1 Sulfonyl aryl hydroxamates and their use as matrix metalloprotease inhibitors
01/30/2003CA2452541A1 (pyridinyl and pyrimidyl) trienoic acid derivatives as retinoid x receptor modulators
01/29/2003EP1279656A2 Process for preparing unsymmetrical biaryls and alkylated aromatic compounds from arylnitriles
01/29/2003EP1278758A1 Combretastatin a-1 phosphate and combretastatin b-1 phosphate prodrugs
01/29/2003EP1278734A2 Method of treatment using phenyl and biaryl derivatives as prostaglandin e inhibitors and compounds useful therefore
01/29/2003EP1278723A2 P-(sulfonyl)-aryl and -heteroaryl amines
01/29/2003EP1278722A1 Aryl and heteroaryl sulfonates
01/29/2003EP1278716A1 Cyclohexylamine derivative as subtype selective nmda receptor antagonists
01/29/2003EP1278526A2 Treatment of cerebrovascular disease
01/29/2003EP1192145A4 Process for preparing chiral cyclopropane carboxylic acids and acyl guanidines
01/29/2003EP0994831B1 Manufacture of alpha-olefins
01/29/2003EP0973735B1 Polyaromatic antiviral compositions
01/29/2003EP0832081B1 Bicyclic-aromatic compounds
01/29/2003EP0817772B1 Pyrrolidinyl hydroxamic acid compounds and their production process
01/29/2003EP0708769B1 Substituted 2-fused phenylpyridines with herbicidal activity
01/29/2003CN1394241A Selective electrochemical reduction of halogenated 4-aminopicolinic acids
01/29/2003CN1394203A Piperidine and piperazine derivatives which function as 5-HT2A receptor antagonists
01/29/2003CN1394202A Picolinic acid derivatives and their use as fungicides
01/29/2003CN1100058C Novel intermediates and process for manufacture of camptothecin derivatives (CPT-11) and related compounds
01/28/2003US6512002 Methods of treatment for premature ejaculation in a male
01/28/2003US6511995 Inhibits collagen synthesis, which is useful for prophylaxis or treatment of fibrosis
01/28/2003US6511992 For treating pain or memory deficiencies related to Alzheimer's disease and other neurodegenerative disorders associated with aging
01/28/2003US6511990 Class of cytodifferentiating agents and histone deacetylase inhibitors, and methods of use thereof
01/28/2003US6511988 Prevention binding of transcription factor tozinc finger binding compounds
01/28/2003US6511980 For therapy of gastrointestinal reflux disorders, eating disorders leading to obesity and irritable bowel disorder
01/27/2003WO2002010127A1 Acetamide derivatives and the use thereof as inhibitors of coagulation factors xa and viia
01/27/2003CA2417427A1 Acetamide derivatives and the use thereof as inhibitors of coagulation factors xa and viia
01/23/2003WO2003006462A1 Processes for the manufacture of thrombin inhibitors and n-pyridin-4-yl-oxazolidin-2-ones as intermediate therefor
01/23/2003WO2003006457A1 Variolin derivatives and their use as antitumor agents
01/23/2003WO2003006456A1 4-substituted-picolinic acid amide derivates useful as fungicides
01/23/2003WO2003006454A2 Heterocyclic carboxamides and their use as fungicides