Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
10/2002
10/08/2002USRE37873 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
10/08/2002US6462198 Used in the control or prevention of acute and/or chronic neurological disorders such as restricted brain function caused by bypass operations or transplants, poor blood supply to the brain, spinal cord injuries, head injuries, hypoxia,
10/08/2002US6462196 Preparation of a camptothecin derivative by intramolecular cyclization
10/08/2002US6462179 Conjugation to peptides, proteins, hormones, polysaccharides, nucleic acids, haptens, drugs, ligands, toxins, halophors, and other macromolecules
10/08/2002US6462092 Such as 3-((3-fluorophenyl)-((3-(trifluoromethyl)phenyl)-methyl)amino)-1,1,1 -trifluoro-2-propanol; cardiovascular disease, i.e. atherosclerosis and other coronary artery diseases
10/08/2002US6462086 Non-malignant disease treatment with Ras antagonists
10/08/2002US6462075 Chalcone and its analogs as agents for the inhibition of angiogensis and related disease states
10/08/2002US6462073 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
10/08/2002US6462059 Treatment of disorders associated with smooth muscle contraction; urinary incontinence, asthma, premature labor, irritable bowel syndrome, congestive heart failure, angina, and cerebral vascular disease
10/08/2002US6462057 Compounds for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
10/08/2002US6462053 Neuropeptide y receptor antagonists; cardiovascular and central nervous system disorders and metabolic diseases; hypertension, nephropathy, heart disease, vasospasm, arteriosclerosis
10/08/2002US6462044 Therapy for sexual disorders
10/08/2002US6462043 Method for producing substituted-2-nitroguanidine derivatives
10/08/2002US6462023 Cytostatic agents
10/08/2002US6461994 Transition metal complex compounds and polymerization catalysts based thereon, used in polymerization and copolymerization of olefins
10/08/2002US6461388 Diaminobenzene derivative compounds and dye compositions containing same
10/06/2002WO2003088897A2 Fab i inhibitors
10/06/2002CA2444597A1 Fab i inhibitors
10/03/2002WO2002077609A2 Identification of compounds for the treatment or prevention of proliferative diseases
10/03/2002WO2002076974A2 Process for the preparation of tetrasubstituted imidazole derivatives and novel crystalline structures thereof
10/03/2002WO2002076964A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
10/03/2002WO2002076939A2 Cysteine protease inhibitors
10/03/2002WO2002076929A1 Aryl and biaryl compounds having mch modulatory activity
10/03/2002WO2002076926A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists
10/03/2002WO2002076925A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002WO2002076447A1 Hallogenated aminobenzophenones and aminobenzoylpyridines as inhibitors of il-1 and tnf
10/03/2002WO2002076177A2 Design and synthesis of optimized ligands for ppar
10/03/2002WO2002058631A3 Primary intermediates for oxidative coloration of hair
10/03/2002WO2002030880A3 N-substituted amino acid derivatives (factor xa inhibitors)
10/03/2002WO2002026731A3 Quaternary amidino based inhibitors of factor xa
10/03/2002US20020143188 Nitrosated and nitrosylated potassium channel activators, compositions and methods of use
10/03/2002US20020143187 Nitric oxide donors and pharmaceutical compositions containing them
10/03/2002US20020143186 For prophylaxis and therapy of hyperglycemia, Type 1 diabetes, Type 2 diabetes, disorders of the lipid metabolism, such as dyslipidemia, and obesity
10/03/2002US20020143054 Cyclopentane(ENE)heptenoic or heptanoic acids and derivatives thereof useful as therapeutic agents
10/03/2002US20020143036 Pentafluorobenzenesulfonamides and analogs
10/03/2002US20020143034 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
10/03/2002US20020143025 For preventing free radical-mediated cellular damage or disruption; as oxidation inhibitors as additives to fuels, lubricants, rubber, polymers, chemicals, solvents and foodstuffs
10/03/2002US20020143020 Novel piperazine derivatives
10/03/2002US20020143011 Tri-substituted phenyl derivatives and processes for their preparation
10/03/2002US20020142969 Using didepsipeptide for the control of endoparasites in medicine and veterinary medicine
10/03/2002US20020142912 Substituted pyridyl amine complexes, and catalysts
10/03/2002US20020142045 Cyclooxygenase-2 inhibitor compositions having rapid onset of therapeutic effect
10/03/2002CA2442364A1 Process for the preparation of tetrasubstituted imidazole derivatives and novel crystalline structures thereof
10/03/2002CA2441080A1 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002CA2436351A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists
10/02/2002EP1245660A2 Liquid crystal compounds having bis(trifluoromethyl)phenyl rings, liquid crystal compositions and liquid crystal display devices
10/02/2002EP1244627A1 Picolinic acid derivatives and their use as fungicides
10/02/2002EP1244626A2 Caspase inhibitors and uses thereof
10/02/2002EP1244625A1 4-pyridinyl-n-acyl-l-phenylalanines
10/02/2002EP1086114B1 Morphine-6-glucuronide synthesis
10/02/2002EP0963484B1 Sizing of paper
10/02/2002EP0706521B1 Imides as tnf alpha inhibitors
10/02/2002EP0689534B1 Amide derivatives as 5-ht 1a? ligands
10/02/2002DE10115945A1 Substituierte 2-Carba-3,5-dicyano-4-aryl-6-aminopyridine und ihre Verwendung Substituted 2-carba-3,5-dicyano-4-aryl-6-aminopyridines and their use
10/02/2002DE10113587A1 Verfahren zur Herstellung von substituierten Pyrrolen A process for the preparation of substituted pyrroles
10/02/2002CN1372550A Process for the preparation of 2-cyanopyridines
10/02/2002CN1372549A Fungicidies
10/02/2002CN1372548A Heterocyclic compounds and medicinal use thereof
10/02/2002CN1372541A Sulfonyl carboxamide derivatives, method for their production and their use as medicaments
10/02/2002CN1091623C Crystallisation process
10/01/2002US6458998 Naphthaleneureas as antidiabetic agents
10/01/2002US6458982 Transition metal compound, catalyst, its production and its use for the polymerization of olefins
10/01/2002US6458957 α,α-dibromo-α-chloro-acetophenones as synthons
10/01/2002US6458951 For treatment of male erectile dysfunction, female sexual dysfunction
10/01/2002US6458852 Use of substituted N, N-bis-phenyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458849 Method of treating or preventing a ceip-mediated disorder in a subject by administering a therapeutically effective amount of a compound for strokes
10/01/2002US6458844 Antiinflammatory agents
10/01/2002US6458816 Anticancer agents
10/01/2002US6458815 Cardiovascular disorders, anticholesterol agent
10/01/2002US6458813 2-cyclohexyloxy-5-(2-chlorophenylcarbonylamino)pyridine, for example; treating inflammation, pain, diabetes, cancer
10/01/2002US6458806 Aryl alkenamides derivatives as MCP-1 antagonists
10/01/2002US6458803 Substituted N-phenyl-N-heteroaralkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
10/01/2002US6458794 Potassium channel inhibitors
10/01/2002US6458793 Heterocyclic derivatives which inhibit factor Xa
10/01/2002US6458789 2-aminopyridine derivatives and combinatorial libraries thereof
10/01/2002US6458775 NAALADase inhibitors useful as pharmaceutical compounds and compositions
10/01/2002US6458772 Prodrugs
10/01/2002US6458739 Polymerization catalysts
10/01/2002CA2209018C Sulfonamides and their use
10/01/2002CA2203850C Novel n-phenyl-n-phenyliminonethylbenzamidines and their analogues as muscarinic receptor agonists
09/2002
09/26/2002WO2002074757A1 Method for producing substituted pyrroles and furans
09/26/2002WO2002074735A2 Biurethane derivatives
09/26/2002WO2002074733A2 Tryptase-inhibitors
09/26/2002WO2002074731A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
09/26/2002WO2002074730A1 INHIBITORS OF INTEGRIN αvβ¿6?
09/26/2002WO2002074726A2 Aniline derivatives useful as phosphodiesterase 4 inhibitors
09/26/2002WO2002074310A2 Stabilized formulation of selective ligands of retinoic acid gamma-receptors
09/26/2002WO2002074296A1 Remedies for solid cancer containing hydroxamic acid derivatives as the active ingredient
09/26/2002WO2002036173A3 Simultaneous dual isotope imaging of cardiac perfusion and cardiac inflammation
09/26/2002WO2002032872A8 Nitrogenous aromatic ring compounds
09/26/2002WO2002024636A3 N-acylsulfonamide apoptosis promoters
09/26/2002WO2001087343A3 Combination therapy using cox-2 selective inhibitor and thromboxane inhibitor and compositions therefor
09/26/2002WO1997019953A8 New lh-rh antagonists with improved effectiveness
09/26/2002US20020137968 Treating with amides, ureas, amidines, carbamates, carboximidamides and other derivatives of given formula, e.g. (+)-N-((2,2-dimethylcyclopentyl)methyl)-4-hexyloxybenzamide
09/26/2002US20020137961 Use as skin lightening agents; 4-(1,4-Dioxaspiro(4.5)dec-8-yl)-1,3-benzenediol for example
09/26/2002US20020137939 Novel guanidinobenzamides
09/26/2002US20020137937 Process for preparing [S- (R*, S*) ] -beta- [ [ [1- [1-oxo-3- (4-piperidinyl) propyl] -3-piperidinyl] carbonyl]amino] -3-pyridinepropanoic acid and derivatives
09/26/2002US20020137845 Methods of copolymerizing ethylene and isobutylene and polymers made thereby
09/26/2002US20020137774 Carboxyaryl substituted diphenyl ureas as raf kinase inhibitors
09/26/2002US20020137687 Novel compounds that inhibit tryptase activity