Patents
Patents for C07D 213 - Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members (63,273)
09/2002
09/26/2002US20020137201 Detection of transmembrane potentials by optical methods
09/26/2002US20020134984 Transition metal complex and light-emitting device
09/26/2002DE10113976A1 Production of (hetero)aromatic nitriles, e.g. for pharmaceutical synthesis, involves reacting aryl halide with cyanide in presence of palladium compound, chelating di- or amino-phosphane ligand and chelating diamine
09/26/2002DE10113402A1 New N,N'-bis-(Aminocarbonyl)-hydrazine derivatives are Factor Xa and Factor VIIa inhibitors useful e.g. for treating thrombosis, myocardial infarction, inflammation, apoplexy, restenosis or tumors
09/26/2002DE10112771A1 New 3-acylamino-3-phenyl-propionic acid derivatives, are integrin inhibitors useful e.g. for treating thrombosis, cardiac infarction, angina pectoris, tumor diseases, inflammation, osteoporosis or infections
09/26/2002DE10112068A1 Use of sulfonylguanidine derivatives, mostly new compounds, for treating e.g. pain and neurodegeneration, have affinity for the gabapentin binding site
09/26/2002DE10100928A1 Kuppler/Entwickler- und Kuppler/Kuppler-Hybridfarbstoffe und -hybridfarbstoffvorprodukte Coupler / developer and coupler / coupler hybrid dyes and -hybridfarbstoffvorprodukte
09/26/2002CA2445754A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
09/26/2002CA2441427A1 Biurethane derivatives
09/26/2002CA2440482A1 Tryptase-inhibitors
09/26/2002CA2435847A1 Aniline derivatives useful as phosphodiesterase 4 inhibitors
09/26/2002CA2434030A1 Stabilized formulation of selective ligands of retinoic acid gamma-receptors
09/25/2002EP1243581A1 Pyridinium compounds useful for the treatment of AGE-related diseases
09/25/2002EP1243579A1 Process for the production of pyridine derivatives
09/25/2002EP1242399A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS
09/25/2002EP1242397A1 Trans olefinic glucokinase activators
09/25/2002EP1242390A1 Method for production of 1,3-disubstituted 2-nitroguanidines
09/25/2002EP1242380A1 Improved process for preparing carbamoyl pyridinium compounds
09/25/2002EP1242379A1 Curcumin analogues for treating cancer
09/25/2002EP1242366A1 Salicylamides as serine protease and factor xa inhibitors
09/25/2002EP1242352A2 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states
09/25/2002EP1242078A2 Use of flupirtine for alleviating pain caused by degenerative joint diseases in dogs and cats
09/25/2002EP0968179B1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
09/25/2002EP0835258B1 Novel camptothecin analogues, preparation methods therefor, use thereof as drugs, and pharmaceutical compositions containing said analogues
09/25/2002EP0835257B1 Intermediates and process for the manufacture of camptothecin derivatives (cpt-11) and related compounds
09/25/2002EP0746312B1 Guanylhydrazones for treating inflammatory conditions
09/25/2002CN1371367A Phenethyl-5-bromopyridyl thiourea (PBT) and dihydroalkoxybenzyloxopyrimidine (DABO) derivatives exhibiting spermicidal activity
09/25/2002CN1371366A Benzamide formulation with histone deacetylase inhibitor activity
09/25/2002CN1371364A Tetrahydropyridines as pesticides
09/25/2002CN1371357A Aminobenzoic acid derivatives
09/25/2002CN1371286A Use of cyclooxygenase-2 inhibitor matrix metallappoteinase inhibitor antineoplastic agent and optionally radiation as combination treatment of neoplasia
09/25/2002CN1370770A Pyridine recovering process
09/25/2002CN1091442C Method for preparing phenylpyridyl substituted urea
09/24/2002US6455701 Such as 4-((4'-tert-butyl-3'-(4?-trifluoromethyl)phenoxy) phenylethynyl)benzoic acid; side effect reduction
09/24/2002US6455660 Given annealed density, charpy impact, and dynamic storage modulus; made using a tridentate nitrogen-containing transition metal polymerization catalyst
09/24/2002US6455581 Inhibitors of hiv protease.
09/24/2002US6455554 Oxopyridinyl pharmaceutical compositions and methods for use
09/24/2002US6455551 Use of 1-hydroxy-2-pyridones for treating mucosa diseases which are difficult to treat
09/24/2002US6455550 N-alkanoylphenylalanine derivatives
09/24/2002US6455545 Gastrointestinal disorders
09/24/2002US6455528 Tumor necrosis factor antagonist and/or interleukin promoter; antiallergens, antiinflammatory agents; autoimmune disease treatment
09/24/2002US6455520 Benzamide derivatives and their use as cytokine inhibitors
09/24/2002US6455519 Use of substituted N, N-disubstituted fused-heterocyclo amino compounds for inhibiting cholesteryl ester transfer protein activity
09/24/2002US6455502 Compounds and compositions as protease inhibitors
09/20/2002WO2001070692A2 Heterocyclic acylsulfimides, a method for their production, agents containing the same and their use as pesticides
09/20/2002CA2403807A1 Heterocyclic acylsulfimides,processes for their preparation,compositionscomprising them and their use as pesticides
09/19/2002WO2002072869A2 Novel agents for replacement of nad+/nadh system in enzymatic ractions
09/19/2002WO2002072707A1 Pyridone dyes, a process for their preparation and their use in the production of coloured plastics or polymeric colour particles
09/19/2002WO2002072654A2 Polymers and oligomers, their synthesis, and electronic devices incorporating same
09/19/2002WO2002072564A1 N-phenylarylsulfonamide compound, drug containing the compound as active ingredient, intermediate for the compound, and processes for producing the same
09/19/2002WO2002072559A1 Process to intermediates for biologically active compounds
09/19/2002WO2002072553A1 Antiproliferative agents
09/19/2002WO2002072544A2 Multifluoro-substituted chalcones and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/19/2002WO2002072540A2 Improved methods of ortho alkylation
09/19/2002WO2002072532A1 7, 9-substituted tetracycline compounds
09/19/2002WO2002072518A2 Method for producing monocarbonyl compounds or biscarbonyl compounds or hydroxyl compounds
09/19/2002WO2002072511A1 'convenient and efficient suzuki-miyaura cross-coupling catalyzed by a palladium/diazabutadiene system'
09/19/2002WO2002072092A1 Method for increasing leptin levels using nicotinic acid compounds
09/19/2002WO2002072091A1 Anticancer drug-tolerance inhibitors
09/19/2002WO2002072084A2 Glycyrrhetinic acid derivatives, progesterone and progesterone derivatives and their use for the manufacture of a medicament to inhibit 11beta-hydroxysteroid dehydrogenase activity
09/19/2002WO2002029021A3 Biotechnological method for preparing carboxylic acids with a hydroxy-nitrogen heterocycle
09/19/2002WO2002024194A9 Use of statins (hmg-coa reductase inhibitors) for the preparation of medicament as a novel type of immunomodulator, immunosuppressor and anti-inflammatory agent
09/19/2002WO2002014311A3 Urea compounds and methods of uses
09/19/2002WO2001007020A3 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
09/19/2002US20020133023 Antitumor agents, osteoporosis
09/19/2002US20020133015 4-pyridinyl-N-acyl-L-phenylalanines
09/19/2002US20020133013 Reacting halobenzoic acid with 2,2,2-trifluoroethanol; thenhaloacetonitrile
09/19/2002US20020133005 Heterocyclic compounds and medical use thereof
09/19/2002US20020132888 Alkylthio-and aryl(heteroyl)thio-substituted p-phenylenediamines, their manufacture and their use in rubber
09/19/2002US20020132853 Diaryl piperazines and related compounds useful in the treatment of a chronic and acute pain conditions, itch and urinary incontinence.
09/19/2002US20020132852 Symmetrically disubstituted aromatic compounds and pharmaceutical compositions for inhibiting poly (ADP-ribose) glycohydrolase, and methods for their use
09/19/2002US20020132833 Caspase inhibitors and uses thereof
09/19/2002US20020132830 Use of beta 2 bronchodilator drugs
09/19/2002US20020132816 Estrogen agonists/antagonists for preventing breast cancer
09/19/2002US20020132807 Aryl phenylheterocyclyl sulfide derivatives and their use as cell adhesion-inhibiting anti-inflammatory and immune-suppressive agents
09/19/2002US20020132794 Compounds and methods for inhibition of HIV and related viruses
09/19/2002DE10113027A1 3-Diaminophenyl-acrylamide derivatives or their physiologically acceptable, water-soluble salts, used as developers in combination with couplers in oxidative dye formulations, especially for dyeing hair are new
09/19/2002DE10110754A1 Substituierte 2-Thio-3,5-dicyano-4-aryl-6-aminopyridine und ihre Verwendung Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and their use
09/19/2002DE10110438A1 Substituierte 2-Oxy-3,5-dicyano-4-aryl-6-aminopyridine und ihre Verwendung Substituted 2-oxy-3,5-dicyano-4-aryl-6-aminopyridines and their use
09/19/2002DE10109204A1 Use of new and known diphenylurea compounds for the preparation of a medicament for the inhibition of intracellular protein-degradation pathway
09/19/2002DE10058461A1 Substituierte Cyclohexanderivate und ihre Verwendung Substituted cyclohexane derivatives and their use
09/19/2002CA2441745A1 Polymers and oligomers, their synthesis, and electronic devices incorporating same
09/19/2002CA2437755A1 Improved methods of ortho alkylation
09/19/2002CA2434837A1 Pyridone dyes, a process for their preparation and their use in the production of coloured plastics or polymeric colour particles
09/18/2002EP1241170A2 Pyrazolopyrimidine derivatives
09/18/2002EP1240906A1 Preventives or remedies for arrhythmia
09/18/2002EP1240162A2 Novel derivatives of 3-imino-1,2-dithioles, method for producing them and pharmaceutical compositions containing the same
09/18/2002EP1240154A1 Serine protease inhibitors
09/18/2002EP1240147A1 Potassium channel inhibitors
09/18/2002EP1240145A2 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof
09/18/2002EP1240144A2 Compound having effect of promoting neuron differentiation
09/18/2002EP1240133A1 Methods of preparing substituted tetracyclines with transition metal-based chemistries
09/18/2002EP1036059B1 Adamantane derivatives
09/18/2002EP0950056B1 N-(pyridinylamino)isoindolines and related compounds
09/18/2002EP0888322B1 Electrophilic ketones for the treatment of herpesvirus infections
09/18/2002EP0865424B1 Pesticides
09/18/2002EP0823889B1 1,3-propane diol derivatives as bioactive compounds
09/18/2002EP0804427B1 Lta4 hydrolase inhibitors
09/18/2002EP0700388B1 Substituted beta-aryl and beta-heteroaryl-alpha-cyanoacrylamide derivatives as tyrosine kinase inhibitors
09/18/2002CN1370168A Novel spiro compounds