Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
10/2003
10/23/2003US20030199566 Phenolic acid derivatives and composition for preventing or treating blood lipid level-related diseases comprising the same
10/23/2003US20030199552 Amide derivatives as NMDA receptor antagonists
10/23/2003US20030199540 Fluoroalkyoxybenzylamino derivatives of nitrogen containing heterocycles
10/23/2003US20030199531 Biodegradation-resistant mimics of pentapeptide tyrosine-isoleucine-glycine-serine-arginine (YIGSR) binding site for laminin binding protein
10/23/2003US20030199520 Sulfonamide hydroxamates
10/23/2003US20030199519 Prodrugs of CC-1065 analogs
10/23/2003US20030199510 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
10/23/2003US20030199499 Novel guanidinobenzamides
10/23/2003US20030199497 Novel calcium receptor active molecules and method for preparing same
10/23/2003US20030199482 Anticholesterol agents; a drug mixture for treating hypercholesterolemia comprising an apical sodium co-dependent bile acid transport inhibitor, enzyme inhibitors of a cyclooxygenase-2
10/23/2003US20030199478 For modulating tyrosine kinase signal transduction in order to regulate, modulate and/or inhibit abnormal cell proliferation
10/23/2003CA2481313A1 Bicyclic amides
10/23/2003CA2480856A1 Substituted aryl amides
10/23/2003CA2480832A1 Nitric oxide donors, compositions and methods of use
10/23/2003CA2480759A1 Improved prodrugs of cc-1065 analogs
10/22/2003EP1354887A1 Ligands for metals and improved metal-catalyzed processes based thereon
10/22/2003EP1354876A1 Method for synthesis of (2S,3aS,7aS)-perhydroindole-2-carboxylic acid and esters thereof; and use in the synthesis of perindopril
10/22/2003EP1354875A1 Method for synthesis of (2S,3aS,7aS)-perhydroindole-2-carboxylic acid and esters thereof; and use in the synthesis of perindopril
10/22/2003EP1354874A1 Method for synthesis of (2S,3aS,7aS)-perhydroindole-2-carboxylic acid and esters thereof; and use in the synthesis of perindopril
10/22/2003EP1354873A1 Salt of perindopril and pharmaceutical compositions containing it
10/22/2003EP1354865A1 Process for the preparation of aromatic aldehydes via ozonolysis of aromatic alkenes
10/22/2003EP1353906A1 Process for the preparation of (3-cyano-1h-indol-7-yl)(4-(4-fluorophenethyl)piperazin-1-yl)-methanone and salts thereof
10/22/2003EP1353904A1 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
10/22/2003EP1353898A2 Compounds to treat alzheimer's disease
10/22/2003EP1353890A1 Obtaining anthracene and carbazole by melt-crystallization
10/22/2003EP1353673A1 Camptothecin derivatives
10/22/2003EP1353662A2 Methods for the treatment of diseases using malonyl-coa decarbox ylase inhibitors
10/22/2003EP1097136B1 Process for the preparation of an indole derivative
10/22/2003CN1451014A Peptidomimetic protease inhibitors
10/22/2003CN1450991A Hydroxamate derives useful as deacetylase inhibitors
10/22/2003CN1450896A Use of indole derivatives for intracular pressure for reducing
10/22/2003CN1450893A Method for treatment of sepsis
10/22/2003CN1450049A N-arylating method using amino-acid as additives
10/22/2003CN1125071C Phthalocyanine and use of phthalocyanine as marking agent
10/22/2003CN1125047C Thermodynamically stable modification of 1-(4-carbazolyloxy)-3-[2-(2-methoxyphenoxy) ethylamino]-2-propanole process for its preparation and pharmaceutical use
10/22/2003CN1125040C Therapeutic compound-fatty acid conjugates
10/21/2003US6635771 N-benzhydryl indole compounds
10/21/2003US6635673 1-Aminomethyl-3,4-dimethyl-cyclopentyl acetic acid; epilepsy; neurodegenerative, neuropathological and gastrointestinal disorders; depression, anxiety, panic, pain
10/21/2003US6635670 Such as N-(2-((3-(Aminooxoacetyl)-2-ethyl-1-(phenylmethyl)-1H-indol-4 -yl)oxy)acetyl)glycine; inflammatory diseases
10/21/2003US6635669 Kinase inhibitor; benign prostatic hyperplasia
10/21/2003US6635668 Imidazoline receptor binding compounds
10/21/2003US6635655 Agonists or antagonists of peroxisome proliferator-activated receptors
10/21/2003US6635650 Such as N-(2-(7-(2-((8-(2-(acetyl-amino)ethyl)-2-naphthyl) oxy)ethoxy)-1-napthyl)ethyl)acetamide for treating or preventing melatoninergic disorders
10/21/2003US6635642 Poly(ADP-ribose) polymerase inhibitors; tissue damage treatment
10/21/2003US6635639 Use of N-alkylamino-heterocylic compounds for the treatment of migraine
10/21/2003CA2240136C Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
10/21/2003CA2153979C Compounds having both potent calcium antagonist and antioxidant activity and use thereof as cytoprotective agents
10/21/2003CA2037100C 6-substituted-hexahydrobenz ¢cd! indoles
10/16/2003WO2003084956A1 Novel 1,2,3-substituted indolizine derivatives, inhibitors of fgfs, method for making same and pharmaceutical compositions containing same
10/16/2003WO2003084943A2 Terphenyl derivatives, preparation thereof, compositions containing same
10/16/2003WO2003084928A1 Alpha, omega-dicarboximide derivatives as useful uro-selective α1α adrenoceptor blockers
10/16/2003WO2003084927A1 Haloalkenes, process for production thereof, and pest controllers containing the same
10/16/2003WO2003084916A2 Compounds that modulate ppar activity and methods for their preparation
10/16/2003WO2003084915A1 Novel thyroid receptor ligands
10/16/2003WO2003053922A3 Heteroaryl substituted imidazole modulators of metabotropic glutamate receptor-5
10/16/2003WO2003027314A3 Protected linker compounds
10/16/2003US20030195365 CC-1065 analog synthesis
10/16/2003US20030195361 Bicyclic pyrrolyl amides as glycogen phosphorylase inhibitors
10/16/2003US20030195360 For therapy of oncoses
10/16/2003US20030195355 Indole-type derivatives as inhibitors of p38 kinase
10/16/2003US20030195258 Taxol enhancer compounds
10/16/2003US20030195244 Nitrogen compounds such as (6-Methoxy-1H-indol-3-yl)-(3,4,5-trimethoxy-phenyl)-methanone, administered for prophylaxis of cancer; angiogenesis inhibitors
10/16/2003US20030195238 Enzyme inhibitors
10/16/2003US20030195234 Substituted oxindole derivatives as tyrosine kinase inhibitors
10/16/2003US20030195226 Nitrogen compounds such as pyridine-3-carbaldehyde, O-(((4-undecyloxy-phenyl)amino)carbonyl)oxime, used for prophylaxis of vision, eating or cardiovascular disorders, and as anxiolytic and antiemetic agents
10/16/2003US20030195223 Antithrombotic agents
10/16/2003US20030195212 An amide derivatives for treating obesity, anorexia, inflammation, mental diseases associated with the melanocyte stimulating hormones
10/16/2003US20030195208 Phthalimido derivatives and a process for their preparation
10/16/2003US20030195201 Vanilloid receptor ligands and their use in treatments
10/16/2003US20030195187 For therapy of obesity or type II diabetes
10/16/2003US20030195159 HIV protease inhibitors based on amino acid derivatives
10/16/2003US20030194740 System and method for nucleic acid sequencing by polymerase synthesis
10/16/2003CA2481976A1 Novel thyroid receptor ligands
10/16/2003CA2481888A1 Alpha, omega-dicarboximide derivatives as useful uro-selective a1a adrenoceptor blockers
10/16/2003CA2481392A1 Terphenyl derivatives, preparation thereof, compositions containing same
10/15/2003EP1352650A1 Inhibitors against the production and release of inflammatory cytokines
10/15/2003EP1351946A2 Materials and methods to potentiate cancer treatment
10/15/2003EP1351934A1 Naphthalene derivatives which bind to the ep4 receptor
10/15/2003EP1351924A2 Diamines as modulators of chemokine receptor activity
10/15/2003EP1228041B1 Indole derivatives and their use as 5ht2a ligands
10/15/2003EP1051374B1 The use of compressed carbon dioxide in chemical reactions
10/15/2003EP0950047B1 Indolin-2-one derivatives, method for preparing them and pharmaceutical compositions containing them
10/15/2003EP0861246B1 Prolyl endopeptidase inhibitors, their preparation and their pharmaceutical use
10/15/2003CN1449385A Aza-bridged-bicyclic amino acid derivatives as alpha4 integrin antagonists
10/15/2003CN1449287A Fused pyrrolocarbazoles against inflammation
10/15/2003CN1449286A Carvedilol
10/15/2003CN1124265C Method for producing aromatic bisimides
10/15/2003CN1124262C Indole derivatives useful as endothelin receptor antagonists
10/14/2003US6632962 Caspase inhibitors and uses thereof
10/14/2003US6632836 To treat autoimmune disorders, cardiac arrhythmias and the like
10/14/2003US6632834 Compositions and methods for treating conditions responsive to estrogen
10/14/2003US6632830 ACE-2 inhibiting compounds and methods of use thereof
10/14/2003US6632825 Picornaviral 3C protease enzyme inhibitors; amide ester or amide acid derivatives
10/14/2003US6632810 Cyclic diamine compound with condensed-ring groups
10/09/2003WO2003083063A2 Common ligand mimics: naphtoates
10/09/2003WO2003082928A1 Control agents for living-type free radical polymerization and methods of polymerizing
10/09/2003WO2003082874A2 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino[4,5-b]indole-1-acetamide derivatives, preparation and use thereof in medicaments
10/09/2003WO2003082860A1 Processes for producing indole compound
10/09/2003WO2003082853A1 New compounds
10/09/2003WO2003082835A1 Process for the preparation of morpholine derivatives and intermediates therefore