Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
02/2004
02/19/2004US20040034088 For treating microbial/fungal infections
02/19/2004US20040034055 For treating central nervous system disorders, immunomodulatory disorders, antimalaria, viral disease of Borna virus, Hepatitis; a 6-azatricyclo(6.3.1.01,6)dodecane derivatives
02/19/2004US20040034052 Antitumor agents
02/19/2004US20040034019 Piperazine and piperidine derivatives
02/19/2004US20040033995 Nitrogen compounds, stereoisomers and/or racemic mixtures used as enzyme inhibitors for prophylaxis of inflammatory diseases
02/19/2004US20040033962 Antibody directed enzyme prodrug therapy
02/19/2004US20040033910 Bicyclic thioamides as additives for lubricating oils
02/19/2004DE10235945A1 New 4-(3-substituted benzoyl)-pyrazol-5-one derivatives, useful as broad-spectrum, pre- and post-emergence herbicides especially for selective weed control in crops e.g. wheat, maize and rice
02/19/2004DE10233500A1 3-Z-[1-(4-(N-((4-Methyl-piperazin-1-yl)-methylcarbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylen]-6-methoxycarbonyl-2-indolinon-Monoethansulfonat und dessen Verwendung als Arzneimittel and its use as a medicament
02/19/2004CA2495108A1 Therapeutic use of aryl amino acid derivatives
02/19/2004CA2494086A1 Metallic complexes covalently bound to conjugated polymers and electronic devices containing such compositions
02/19/2004CA2493575A1 Tyrosine kinase inhibitors
02/19/2004CA2493143A1 2,3-dihydro-isoindol-1-ones with mao-b inhibiting activity
02/18/2004EP1389203A2 Analogs of thalidomide as potential angiogenesis inhibitors
02/18/2004EP1389189A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
02/18/2004EP1389185A2 Aminoalcohol derivatives
02/18/2004EP1389104A2 3-aminoalkyl-2-aryl-indole derivatives and their use as gnrh antagonists
02/18/2004EP1389103A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
02/18/2004EP1178958B1 N-cyanomethyl amides as protease inhibitors
02/18/2004EP1171416B1 3-bicycloaryl-2-aminomethyl bicycloalkanes as serotonine reuptake inhibitors
02/18/2004EP0946166B1 Use of matrix metalloproteinase inhibitors for promoting wound healing
02/18/2004EP0918781B1 Asymmetric synthesis catalyzed by transition metal complexes with cyclic chiral phosphine ligands
02/18/2004EP0851857B1 Inhibitors of tumor necrosis factor alpha
02/18/2004CN1476432A Indole and dihydroindole derivatives
02/18/2004CN1138789C Method of producing network structure of polymer
02/18/2004CN1138755C Cyclic amino acids and derivs thereof useful as pharmaceutical agents
02/17/2004US6693199 Deprotecting carbamate group and amidating in presence of such as hydroxybenzotriazole hydrate promoter
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/17/2004US6693111 Indole-2,3-dione-3-oxime derivatives
02/17/2004US6693105 Using xanthinyl derivatives to reduce treatment induced toxicity; inhibiting cellular signaling through second messenger pathway; reducing cellular level of nonarachi-donate phosphatidic acid and diacylglycerol
02/17/2004US6693098 Carboxylic acid or tetrazole derivatives containing carbamate groups are useful for treating the conditions associated with the urinary tract, pain, inflammation, respiratory states, edema formation of hypotensive vascular diseases
02/17/2004US6693092 Herbicides; pesticides
02/12/2004WO2004013282A2 Bis (amino acid) molecular scaffolds
02/12/2004WO2004013127A1 Method for producing highly pure hydroxy indolyl glyoxylic acid amides
02/12/2004WO2004013117A1 Bicyclic cylopentanone and cyclopentenone derivatives as potent activators of hsf
02/12/2004WO2004013099A1 3-z-[1-(4-(n-((4-methyl-piperazin-1-yl)-methylcarbonyl)-n-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone-monoethanesulphonate and the use thereof as a pharmaceutical composition
02/12/2004WO2004013094A2 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/12/2004WO2004013087A1 Anthranyl derivatives having an anticholecystokinin activity (anti-cck-1), a process for their preparation, and pharmaceutical use thereof
02/12/2004WO2004013085A1 3-amino-2-hrydroxyalkanoic acids and their prodrugs
02/12/2004WO2004013072A2 Copper catalyzed arylation
02/12/2004WO2004012722A2 Bicifadine formulation
02/12/2004WO2004012648A2 Substituted diaryl heterocycles, method for the production and use thereof as medicaments
02/12/2004WO2003049702A3 Vanilloid receptor ligands and their use in treatments
02/12/2004WO2002030406A3 Use of antagonists or partial agonists of 5ht1a receptors for the preparation of a medicament for treatment and prevention of gastrointestinal diseases
02/12/2004US20040030154 Isolation of tryptophan; controlling nervous system response; contactor with porous carriers; agitation aqueous solution
02/12/2004US20040030072 Using coordination catalyst
02/12/2004US20040029950 Nervous system and psychological disorders
02/12/2004US20040029948 Antiinflammatory agents; sepsis shock; rheumatic disorders
02/12/2004US20040029913 Halogenated selective androgen receptor modulators and methods of use thereof
02/12/2004US20040029889 Bone disorders; antiarrhythmia agents; cardiovascular disorders
02/12/2004US20040029871 Pharmaceutical compounds for treating copd
02/12/2004US20040029814 Cathepins inhibitor; antiinflammatory agents; antiarthritic agents
02/12/2004US20040029813 Cardiovascular disorders; hypotensive agents; angiotensin converting enzyme inhibitor
02/12/2004DE10233817A1 Substituierte Diarylheterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Substituted Diarylheterocyclen, processes for their preparation and their use as medicaments
02/12/2004DE10233366A1 In 6-Stellung substituierte Indolinonderivate, ihre Herstellung und ihre Verwendung als Arzneimittel In the 6-position substituted indolinone derivatives, their preparation and their use as medicaments
02/12/2004CA2494632A1 3-amino-2-hrydroxyalkanoic acids and their prodrugs
02/12/2004CA2494404A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/12/2004CA2494142A1 Copper catalyzed arylation
02/12/2004CA2493982A1 Method for producing highly pure hydroxy indolyl glyoxylic acid amides
02/12/2004CA2493593A1 Bicifadine formulation
02/11/2004EP1388535A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
02/11/2004EP1387827A2 Synthesis of cyclopentadiene derivatives
02/11/2004EP1387826A1 Novel 5-phenyl-1h-indole derivatives as antagonists of interleukine-8 receptors
02/11/2004EP1240157B1 Substituted n-benzyl-indol-3-yl glyoxylic acid derivatives having an anti-tumoral effect
02/11/2004EP1216239B1 Piperazine derivatives as 5-ht1b antagonists
02/11/2004EP1176987B1 Short-chain peptide dye conjugates used as contrast agents for optical diagnostics
02/11/2004EP1047411B1 Substituted diphenyl indanone, indane and indole compounds and analogues thereof useful for the treatment or prevention of diseases characterized by abnormal cell proliferation
02/11/2004EP1028725B1 Use of vasopressin antagonists for treating disturbances or illnesses of the inner ear
02/11/2004EP0812825B1 Propenone derivatives
02/11/2004CN1474804A 2-amino-2-alkyl-4-hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
02/11/2004CN1474691A Novel uses of combined 5-HT 1A agonists and serotonin reuptake inhibitor
02/11/2004CN1473814A Intemediate for preparing alkyl-dihalogeno phenyl substituted keto-enol
02/11/2004CN1137894C Pyridopyranoazepine derivatives, preparation and therapeutic use
02/11/2004CN1137884C Indazole compounds and pharmaceutical compositions for inhibiting protein kinases and methods for their use
02/10/2004US6689881 Method for preparing substituted [1,4]diazepino[6,7,1-hi]indol-4-ones
02/10/2004US6689806 Indolinone compounds as kinase inhibitors
02/10/2004US6689792 Useful for the treatment of schizophrenia and related psychotic disorders such as parkinson's disease and alzheimer's disease
02/10/2004US6689784 Controlling cell apoptosis
02/10/2004US6689523 Charge transport compound containing bis(3-formylcarbazolyl)-1,1'-(sulfonyldi-4, 1-phenylene)bis-hydrazones
02/05/2004WO2004011556A1 Site-specific labelling of proteins using cyanine dye reporters
02/05/2004WO2004011438A1 Diaryl-substituted cyclic urea derivatives having an mch-modulatory effect
02/05/2004WO2004011425A2 Indole, azaindole and related heterocyclic ureido and thioureido piperazine derivatives
02/05/2004WO2004011410A1 Chemical compounds
02/05/2004WO2004010761A2 Pesticidal cyanine dye derivatives
02/05/2004WO2003075857A3 Amino-methyl substituted tetracycline compounds
02/05/2004WO2003070703A3 Hydroxylated indirubin derivatives
02/05/2004WO2003064388A3 Process for the preparation of high purity perindopril and intermediates useful in the synthesis
02/05/2004US20040024211 Such as (3S)-N-(2-(2-(2,4-dichlorophenyl)ethyl)-1-oxo-2,3-dihydro-1H-isoindol-5-yl) -3-methyl-N'-((1S,2S,3S,5R)-2,6,6-trimethylbicyclo(3.1.1)hept-3 -yl)piperazine-1-carboximidamide for treatment of obesity or type II diabetes
02/05/2004US20040024190 Viral polymerase inhibitors
02/05/2004US20040024132 A free radical polymerization in presence of a sulfur based chain transfer agents, controlling during the synthesis of polystyrene, polymethyl acrylate, polymethyl methacrylate
02/05/2004US20040024067 Deacetylase inhibitors
02/05/2004US20040024057 Nitrosated nonsteroidal antiinflammatory compounds, compositions and methods of use related applications
02/05/2004US20040024045 Glucagon antagonists/inverse agonists
02/05/2004US20040024023 1-Heterocyclylalkyl-3-sulfonyl-indole or -indazole derivatives as 5-hydroxytryptamine-6 ligands
02/05/2004US20040024010 3-methylidenyl-2-indolinone modulators of protein kinase
02/05/2004US20040023999 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
02/05/2004US20040023890 Drugs for diabetes
02/05/2004US20040023060 Structure including at least three planar moieties, which are linearly configured such that one planar moiety is located between two neighboring planar moieties and shares an atom with each of the moieties
02/05/2004US20040022856 Carriers for drug delivery
02/05/2004US20040020791 Electrochemical assays