| Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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| 03/18/2004 | DE10242350A1 New 3-aminomethylene-indoline-2-(thi)one derivatives, are kinase inhibitors useful for treating proliferative diseases e.g. tumors, rheumatoid arthritis, neovascular glaucoma and arteriosclerosis |
| 03/18/2004 | CA2497979A1 1, 3-diamino-2-hydroxypropane prodrug derivatives |
| 03/18/2004 | CA2497829A1 Method to treat allergic rhinitis |
| 03/18/2004 | CA2497408A1 Indole-type derivatives as inhibitors of p38 kinase |
| 03/18/2004 | CA2495939A1 Cathepsin cysteine protease inhibitors |
| 03/18/2004 | CA2495284A1 Diarylurea derivatives and their use as chloride channel blockers |
| 03/17/2004 | EP1398027A1 Use of matrix metalloproteinase inhibitors for treating or preventing glomerulopathy |
| 03/17/2004 | EP1397360A1 Azaindoles |
| 03/17/2004 | EP1397356A1 Substituted naphthyl indole derivatives as inhibitors of plasminogen activator inhibitor type-1 (pai-1) |
| 03/17/2004 | EP1397348A2 Factor xa inhibitor |
| 03/17/2004 | EP1397341A1 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (pai-1) |
| 03/17/2004 | EP1397136A1 Heterocyclic beta-aminoacids and their use as anti-epileptogenic agents |
| 03/17/2004 | EP1397130A1 Substituted indole acid derivatives as inhibitors of plasminogen activator inhibitor-1 (pai-1) |
| 03/17/2004 | EP1397129A1 Heteroaryloxy 3-substituted propanamines s serotonin and norepinephrine reuptake inhibitors |
| 03/17/2004 | EP1305318B1 Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b] [1,3]benzothiazepines |
| 03/17/2004 | EP1246816B1 Substituted phenyl-piperazine derivatives, their preparation and use |
| 03/17/2004 | EP1246815B1 Phenylpiperazinyl derivatives |
| 03/17/2004 | EP1144496B1 Polymeric stabilizers having low polydispersity |
| 03/17/2004 | EP1140936B1 Tricyclic inhibitors of poly(adp-ribose) polymerases |
| 03/17/2004 | EP1140802B1 Substituted aryl and heteroaryl derivatives, their production and their use as medicines |
| 03/17/2004 | EP1137739B1 Catalytic cracking process using an mcm-68 catalyst |
| 03/17/2004 | EP1100792B1 Tricyclic sulfonamides and their derivatives as inhibitors of matrix metalloproteinases |
| 03/17/2004 | CN1483024A Vla-4 inhibitors |
| 03/17/2004 | CN1483023A 3-arylindole derivatives and their use as cb2 receptor agonists |
| 03/17/2004 | CN1482118A Novel 5-hydroxy-3-carboxylate indoles derivant and method for preparing the same |
| 03/17/2004 | CN1142140C Acylation method |
| 03/16/2004 | US6706929 Reacting phenol with dimethyl carbonate in presence of 1,4-diazabicyclo(2.2.2)octane catalyst |
| 03/16/2004 | US6706890 Reduction of 3-oxa-indolin-2-one with hydrazine hydrate in tertiary amine catalyst presence |
| 03/16/2004 | US6706853 Compound for use as a mineral fibre binder and process for providing such |
| 03/16/2004 | US6706765 Aminoguanidines and alkoxyguanidines as protease inhibitors |
| 03/16/2004 | US6706753 Integrin receptor inhibitors |
| 03/16/2004 | US6706752 Human non-pancreatic secretory phospholipase a2 inhibitors for inhibiting spla2 mediated release of fatty acids for treatment of inflammatory diseases such as septic shock |
| 03/16/2004 | US6706751 Dihydroindole and tetrahydroquinoline derivatives |
| 03/16/2004 | US6706750 Useful in treating obesity and other disorders |
| 03/16/2004 | US6706744 Hypoglycemic agents; antidiabetic agents |
| 03/16/2004 | US6706712 Cyclic derivatives as modulators of chemokine receptor activity |
| 03/16/2004 | US6706709 Treating, for example, proliferative disorders including cancer |
| 03/16/2004 | US6706707 Phenylethynyl and styryl derivatives of imidazole and fused ring heterocycles |
| 03/16/2004 | US6706254 Cyanine dye bioconjugates useful for diagnostic imaging and therapy |
| 03/11/2004 | WO2004020422A1 1, 4- substituted piperidine derivatives and use thereof as base-inhibitors in treatment of alzheimer's disease |
| 03/11/2004 | WO2004020409A1 Indoles having anti-diabetic activity |
| 03/11/2004 | WO2004020408A1 Indoles having anti-diabetic activity |
| 03/11/2004 | WO2004020373A1 Spiro compound and organic luminescence device using the same |
| 03/11/2004 | WO2004019935A1 -3 (sulfonamidoethyl) -indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases |
| 03/11/2004 | WO2004019869A2 Indoles having anti-diabetic activity |
| 03/11/2004 | WO2004005279A3 Substituted anthranilic amide derivatives and methods of use |
| 03/11/2004 | WO2003091396A3 Polypeptides and biosynthetic pathways |
| 03/11/2004 | WO2003074091A3 Near infrared fluorescent contrast agent and method for fluorescence imaging |
| 03/11/2004 | WO2003065789A3 N-biphenylmethyl aminocycloalkanecarboxamide derivatives |
| 03/11/2004 | WO2003053945A3 Urea derivatives and their use as vanilloid receptor antagonists |
| 03/11/2004 | US20040049065 Substituted 3-phenoxy-1-phenyl acetylene derivatives), herbicides |
| 03/11/2004 | US20040049054 Process for preparation of fused pyrroles |
| 03/11/2004 | US20040049030 Such as naphthalenes, anthracenes, phenanthrenes, tetracenes, perylenes, terrylenes, quaterrylenes, pentarylenes, hexarylenes, anthraquinones, indanthrones, and N-substituted naphthalene-1,8-dicarboxylic monoimides |
| 03/11/2004 | US20040048916 3-(Guanidinylcarbonylmethyl)-substituted; inhibit the cellular sodium-proton antiporter, in particular NHE1; antiarrhythmic agents;cardioprotective for infarction prophylaxis and treatment; preventing ischemia-induced damage |
| 03/11/2004 | US20040048858 Chalcone derivatives and their use to treat diseases |
| 03/11/2004 | US20040048797 Regulation of TNF-alpha |
| 03/11/2004 | US20040048346 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds |
| 03/11/2004 | DE10238865A1 New carboxamides are melanin-concentrating hormone receptor antagonists, useful for treating e.g. metabolic diseases, diabetes, eating disorders, cardiovascular disease, emotional disorders, reproductive and memory disorders |
| 03/11/2004 | CA2496580A1 3-(sulfonamidoethyl)-indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases |
| 03/11/2004 | CA2495915A1 Indoles having anti-diabetic activity |
| 03/10/2004 | EP1396490A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives |
| 03/10/2004 | EP1395615A1 Oxime ester photoinitiators having a combined structure |
| 03/10/2004 | EP1395578A1 Carbazole derivatives and their use for the preparation of pharmaceutical compositions for the treatment of npy related diseases |
| 03/10/2004 | EP1395554A1 Substituted carbazoles as inhibitors of spla2 |
| 03/10/2004 | EP1395551A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases |
| 03/10/2004 | EP1395548A1 Derivatives of diphenylurea, diphenyloxalic acid diamide and diphenylsulfuric acid diamide and their use as medicaments |
| 03/10/2004 | EP1395258A1 Oral controlled release pharmaceutical composition for one-a-day therapy for the treatment and prophylaxis of cardiac and circulatory diseases |
| 03/10/2004 | EP1395242A1 Liquid pharmaceutical composition |
| 03/10/2004 | EP1081132B1 Hydroxamic acid derivatives and medicinal utilization thereof |
| 03/10/2004 | CN1481382A Isoindolin-1-one glucokinase activators |
| 03/10/2004 | CN1481366A Dihydroindole and tetrahydroquinoline derivatives |
| 03/10/2004 | CN1481358A Carboxylic acid amide derivatives and their use in treatment of thromboembolic diseases and tumours |
| 03/10/2004 | CN1141295C Indoline derivatives as progesterohe antagonists |
| 03/09/2004 | US6703410 Crystal forms of 3-(2,4-dichlorobenzyl)-2-methyl-n-(pentylsulfonyl)-3h-benzimidazole-5-carboxamide |
| 03/09/2004 | US6703397 Pyrimidinyl methyl indole derivatives with antibacterial activity |
| 03/09/2004 | US6703379 Benzene derivatives and pharmaceutical use thereof |
| 03/09/2004 | US6703338 Heterocyclic compound combined with alumoxane or alkylaluminum |
| 03/09/2004 | US6703042 Salts of L-carnitine and lower alkanoyl L-carnitine |
| 03/09/2004 | CA2272463C Treating or preventing the early stages of degeneration of articular cartilage or subchondral bone in mammals using carprofen and derivatives |
| 03/04/2004 | WO2004018475A2 Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventive agents |
| 03/04/2004 | WO2004018461A2 Antibacterial benzoic acid derivatives |
| 03/04/2004 | WO2004018436A2 Compounds derived from aryl carbamates, preparation thereof and uses of same |
| 03/04/2004 | WO2004018428A1 Antibacterial benzoic acid derivatives |
| 03/04/2004 | WO2004018422A1 Fluoro and sulphonylamino containing 3,6-disubstituted azabicyclo (3.1.0) hexane derivatives as muscarinic receptor antagonists |
| 03/04/2004 | WO2004018421A1 Idol derivatives as new thyroid receptor agonist ligands and methods |
| 03/04/2004 | WO2004018420A1 Indolylalkylamino-methylidenecarbamate derivatives useful as gnrh antagonists |
| 03/04/2004 | WO2004018414A2 Antibacterial agents |
| 03/04/2004 | WO2003088917A3 Regulation of tnf-alpha |
| 03/04/2004 | WO2003075907A3 Small molecule entry inhibitors |
| 03/04/2004 | WO2003068157A3 Kinase inhibitors and methods of use thereof |
| 03/04/2004 | WO2002096867A3 Inhibitors of protein kinase for the treatment of disease |
| 03/04/2004 | US20040044258 Substituted phenylalkanoic acid derivatives and use thereof |
| 03/04/2004 | US20040044250 Transition-metal-catalyzed carbon-nitrogen bond-forming methods using carbene ligands |
| 03/04/2004 | US20040044222 New substituted indolinones, preparation thereof and their use as pharmaceutical compositions |
| 03/04/2004 | US20040044075 Alpha acyloxyacetamides for kallikrein and urokinase inhibition |
| 03/04/2004 | US20040044066 Active ingredient combinations comprising insecticidal and acaricidal properties |
| 03/04/2004 | US20040044053 Antitumor agents; kinase inhibitor |
| 03/04/2004 | US20040044051 Cannabinoid receptor agonists |
| 03/04/2004 | US20040044047 Alpha and beta-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors |
| 03/04/2004 | US20040044037 Sleep disorders; antidepressants; analgesics; central nervous system disorders |