Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
04/2004
04/01/2004US20040062927 Fluorinated dendrons and self-organizing ultrahigh density nanocylinder compositions
04/01/2004US20040062713 Dye; photosensitive stimulant; using eye
04/01/2004CA2498946A1 2,4-substituted indoles and their use as 5-ht6 modulators
04/01/2004CA2498781A1 Indolinones substituted by heterocycles, their preparation thereof and their use as medicaments
04/01/2004CA2496765A1 2,7-substituted indoles and their use as 5-ht6 modulators
03/2004
03/31/2004EP1403303A1 Methods for the preparation of poly(etherimide)s
03/31/2004EP1403277A1 Method for synthesis of (2S,3aS,7aS)-1-((S)-alanyl)-octahydro-1H-indole-2-carboxylic acid derivatives and use in the synthesis of perindopril
03/31/2004EP1403275A1 Process for the synthesis of perindopril and its pharmaceutically acceptable salts
03/31/2004EP1403267A1 Process for preparing glycidylphthalimide
03/31/2004EP1402890A1 Sulfonamide derivatives
03/31/2004EP1401813A1 New indole derivatives with 5-ht6 receptor affinity
03/31/2004EP1401812A1 4-piperazinylindole derivatives with 5-ht6 receptor affinity
03/31/2004EP1401801A1 Selective androgen receptor modulators and methods of use thereof
03/31/2004EP1401575A1 Hydroxylation of beta-dicarbonyls with zirconium catalysts
03/31/2004EP1401434A1 Modulators of peroxisome proliferator activated receptors (ppar)
03/31/2004EP1299401B1 Chiral ligands for asymmetric catalysis
03/31/2004EP1242327B1 Pigmented vitreous material its precursor glass items coated therewith and method of its preparation
03/31/2004EP1232144B1 Novel il-8 receptor antagonists
03/31/2004EP1177186B1 Ureas and their use as cell adhesion modulators
03/31/2004EP1051398B1 Thermodynamically stable form of (r)-3- (4-fluorophenyl) sulphonyl]amino] -1,2,3,4- tetrahydro -9h-carbazole -9-propanoic acid (ramatroban)
03/31/2004EP1037865A4 Synthesis of cc-1065/duocarmycin analogs
03/31/2004EP0901470B1 Indole derivatives useful as endothelin receptor antagonists
03/31/2004EP0871439B1 Substituted (aryl, heteroaryl, arylmethyl or heteroarylmethyl) hydroxamic acid compounds
03/31/2004CN1486300A 1,4-disubstituted piperazine derivatives useful as uro-selective dollar g(a)1-adrenoceptor blockers
03/31/2004CN1486299A Substituted bis-indole derivatives useful as contrast agents, pharmaceutical compositions containing them and intermediates for producing them
03/31/2004CN1143854C Novel 2-(iminomethyl) amino-phenyl derivatives,the preparation thereof, application as medicines and pharmaceutical compositions containing same
03/31/2004CN1143847C Thio-oxindole derivatives
03/30/2004US6713645 Substituted tricyclics
03/30/2004US6713473 6-carbamate-1,2,3,4-tetrahydrocarbazole derivatives; affinity for neuropeptide y receptors
03/30/2004CA2091058C Methylen-oxindole derivatives and process for their preparation
03/25/2004WO2004024896A2 Phenyl-indole compounds
03/25/2004WO2004024702A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
03/25/2004WO2004024688A1 Substituted spirocyclic ketoenols
03/25/2004WO2004024687A1 Benzoyl compounds having imino group and herbicides
03/25/2004WO2004024681A2 Novel compounds comprising a thiocarbonyl-sulfanyl group, which can be used for the radical synthesis of alpha-perfluoroalkylamines
03/25/2004WO2004024676A1 Compounds for modulating the glycolosis enzyme complex and/or transaminase complex
03/25/2004WO2004024139A1 Melanin extinguisher
03/25/2004WO2003087050A3 Novel perindopril salt and pharmaceutical compositions containing same
03/25/2004WO2003086318A3 Improved prodrugs of cc-1065 analogs
03/25/2004WO2003082271A3 Indole derivatives having anti-angiogenetic activity
03/25/2004WO2003072528A3 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
03/25/2004WO2003069350A3 Small molecule modulators of apoptosis
03/25/2004WO2003048106A3 1,3-diarylprop-2-en-1-ones, compositions containing same and use thereof
03/25/2004US20040059132 Reacting an indolin-2-one derivative with substituted benzyl halide to form substituted N-benzyl indolin-2-one derivatives have an affinity for oxytocin receptors
03/25/2004US20040059131 Methylation and benzylation of the indole nitrogen in nearly quantitative yields using 1,4-diazabicyclo(2.2.2)octane as a base in catalytic amount under microwave irradiation
03/25/2004US20040059130 Benz(f)indole compounds useful for Inflammatory Diseases
03/25/2004US20040058979 Indoline derivative and process for producing the same
03/25/2004US20040058978 Novel substituted indolines with an inhibitory effect on various kinases and complexes of CDKs
03/25/2004US20040058977 Cyclooxygenase inhibitors; antiinflamamtory agents
03/25/2004US20040058971 Substituted dipeptides as growth hormone secretagogues
03/25/2004US20040058936 Dietetics, sexual disorders, antidiabetic agents
03/25/2004US20040058933 Aryl carbamate derivatives, preperation and use thereof
03/25/2004US20040058913 Cyclic diamine compound with condensed-ring groups
03/25/2004US20040058901 Crystalline ethanolate solvate form of zafirluskast process for manufacture and pharmaceutical compositions thereof
03/25/2004US20040058877 Somatostatin antagonists and agonists that act at the sst subtype 2 receptor
03/25/2004US20040058820 Central nervous system disorders; psychological disorders; antiinflammatory agents; multiple sclerosis
03/25/2004CA2498493A1 Phenyl-indole compounds
03/25/2004CA2498045A1 Compounds for modulating the glycolosis enzyme complex and/or transaminase complex
03/25/2004CA2496563A1 New carboxamide compounds having mch-antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture
03/24/2004EP1400510A1 Cyclic diamine compounds having fused-ring groups
03/24/2004EP1400241A1 Fused cyclic compounds and medicinal use thereof
03/24/2004EP1399445A2 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists
03/24/2004EP1399411A1 Aloe-emodin derivatives and their use in the treatment of neoplastic pathologies
03/24/2004EP1399155A2 Small molecules useful in the treatment of inflammatory disease
03/24/2004EP1399146A1 Novel compounds and compositions as cathepsin inhibitors
03/24/2004EP1280796B1 Pyrimidinyl methyl indole derivatives with antibacterial activity
03/24/2004EP1117641B1 Indolin derivatives as sun protection agents
03/24/2004EP0904079B1 Antidiabetic agents
03/24/2004CN1484638A I-aryl-or-I-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-b ligands
03/24/2004CN1142911C Compounds with growth hormone releasing properties
03/24/2004CN1142909C Indole derivatives with antiviral activity
03/24/2004CN1142904C One-step process synthetizing 2-oxazolidone derivative interediate and preparation process thereof
03/23/2004US6710185 Process for the preparation of cell proliferation inhibitors
03/23/2004US6710184 Crystalline solids of carvedilol and processes for their preparation
03/23/2004US6710089 Substituted N-fused-phenyl-N-benzyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
03/23/2004US6710080 Substituted 2-dialkylaminoalkylbiphenyl derivatives
03/23/2004US6710069 1-aryl- or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
03/23/2004US6710068 Phenylsulfonylinodles useful for the treatment of hiv in humans and other host animals
03/23/2004US6710055 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbo quinoline-8-sulfonylamino)-indole
03/20/2004CA2406504A1 Method of treating resistant tumors
03/18/2004WO2004022712A2 INDOLE-TYPE DERIVATIVES AS INHIBITORS OF p38 KINASE
03/18/2004WO2004022541A1 1,4-substituted cyclohexane derivatives
03/18/2004WO2004022538A1 Crystal for oral solid drug and oral solid drug for dysuria treatment containing the same
03/18/2004WO2004022529A2 Diarylurea derivatives and their use as chloride channel blockers
03/18/2004WO2004022526A1 Cathepsin cysteine protease inhibitors
03/18/2004WO2004022525A1 Amide derivatives and their use as chloride channel blockers
03/18/2004WO2004022524A2 N-vinylformamide derivatives, polymers formed therefrom and synthesis thereof
03/18/2004WO2004022523A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
03/18/2004WO2004022061A1 Use of indolyl derivatives for the manufacture of a medicament for the treatment allergic rhinitis
03/18/2004WO2004006355A3 Charge transport compositions which are quinazoline derivatives and electronic devices made with such compositions
03/18/2004WO2003018535A3 Novel aminobenzoephenones
03/18/2004WO2002060867A3 Carbazole derivatives and their uses as heparanase inhibitors
03/18/2004US20040054168 Anticancer agents
03/18/2004US20040053987 Bis-heterocyclic compounds with antitumour and chemosensitising activity
03/18/2004US20040053983 1, 2, 4-tribsubstituted benzenes as inhibitors of 15-lipoxygenase
03/18/2004US20040053931 Kinase inhibitors; angiogenesis inhibitors, anticancer agents, antiinflammatory agents and chronic obstructive pulmonary disease inhibitors
03/18/2004US20040053920 Administering to a patient suffering from caspase mediated diseses, an effective amount of a mono,bi or tri-heterocyclic ring containing nitrogen atom attached to ester or thioester to form carbamate group, as caspase inhibitor
03/18/2004US20040053911 Reacting a substituted bis- indole compound with a chelating agent
03/18/2004US20040053907 Cell adhesion inhibitors
03/18/2004US20040053382 Oxidizing an alpha-amino-carboxylic acid, hydrate, or salt thereof using a L-amino acid deaminase or oxidase and subsequently reducing the product thereof using a dehydrogenase