Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
10/2004
10/13/2004EP1465854A2 Chalcone derivatives and their use to treat diseases
10/13/2004EP1465629A1 5-ht3 receptor antagonists and methods of use
10/13/2004EP1465623A1 Urea derivatives
10/13/2004EP1280771B1 Novel prodrugs von 6-hydroxy-2,3-dihydro-1h-indoles, 5-hydroxy-1,2-dihydro-3h-pyrrolo 3,2-e]indoles and 5-hydroxy-1,2-dihydro-3h-benzo(e)indoles as well as of 6-hydroxy-1,2,3,4-tetrahydro-benzo f]quinoline derivatives for use in selective cancer therapy
10/13/2004EP1202965B1 Indole derivatives, processes for their preparation, pharmaceutical compositions containing them and their medicinal application
10/13/2004EP1150954B1 Anti-imflammatory indole derivatives
10/13/2004EP1086086B1 Imidazolyl derivatives and their use as somatostatin receptor ligands
10/13/2004EP0736036B1 Kininogen inhibitors
10/13/2004CN1537100A Substituted 2-pyrrole cyclohexan-1,4-diamine derivatives
10/13/2004CN1537099A Process for preparation of 3-spiro'cyclohexam-1, 3'-'3H indolin-2'-one derivatives
10/13/2004CN1537094A Retinoid derivatives with antiangiogenic, antitumoral and proapoptotic activities
10/13/2004CN1536999A Crystalline forms
10/13/2004CN1536992A Carbamates of 2-heterocyclic-1, 2-ethanediols
10/13/2004CN1535965A cyanine compound, filter and optical recording material
10/13/2004CN1535956A Substituted phenyl keto-enol pesticide and weedicide
10/13/2004CN1170813C N2 phenylamidine derivatives and fungicidal composition and use
10/13/2004CN1170536C Use of preparing medicine for preventing vomit using tetrahydrobenzo [cd] indole-6-formylamine compound
10/12/2004USRE38624 Hydroxyindoles, their use as inhibitors of phosphodiesterase 4 and process for their preparation
10/12/2004US6803362 Heterocyclic compounds
10/07/2004WO2004085539A2 Cyanine dye labelling reagents with meso-substitution
10/07/2004WO2004085396A1 Preventive or therapeutic agent for ischemia/reperfusion injury, organ preservative, and screening method
10/07/2004WO2004085395A1 Melatonin derivatives and their use for treating neurological dysfunctions
10/07/2004WO2004085394A1 7-nitroindoline derivatives and their uses
10/07/2004WO2004085393A1 Novel crystalline forms of tegaserod maleate
10/07/2004WO2004085392A1 Melatonin derivatives and their use for treating neurological dysfunctions
10/07/2004WO2004085385A2 Cannabinoid receptor ligands
10/07/2004WO2004085382A1 Compound inhibiting in vivo phosphorus transport and medicine containing the same
10/07/2004WO2004085361A1 Bioreductively activated stilbene prodrugs
10/07/2004WO2004026829A3 Heterocyclically substituted indolinones and their use as receptor tyrosine kinase inhibitors
10/07/2004US20040198982 such as (4S)-1-(3-bromophenyl)-N-cyanomethyl)-4-methyl-prolinamide; for treatment of osteoporosis
10/07/2004US20040198812 Pseudopolymorphic forms of carvedilol
10/07/2004US20040198802 Antiproliferative agents
10/07/2004US20040198801 Antiinflammatory agents; sepsis
10/07/2004US20040198793 Chemical process and new intermediates
10/07/2004US20040198734 2-(4-Aryl or heteroaryl-piperazin-1-ylmethyl)-1H-indole derivatives interacting with the dopamine
10/07/2004US20040198733 Obesity; antidiabetic agents; cardiovascular disorders; antilipemic agentsl circadian rhythm disorders; hypotensive agents; antidepressants; anxiolytic agents
10/07/2004US20040198732 Aminoalkyl-substituted aromatic bicyclic compounds, methods for their preparation and their use as pharmaceuticals
10/07/2004US20040198731 Antidiabetic agents; cardiovascular disorders; anticholesterol agents; antidepressants; schizophrenia; antilipemic agents; circidian rhythm disorders
10/07/2004US20040198720 3-(Arylamino)methylene-1, 3-dihydro-2H-indol-2-ones as kinase inhibitors
10/07/2004US20040197705 Cyanide compound, optical filter, and optical recording material
10/07/2004US20040197400 Immediate release medicinal compositions for oral use
10/07/2004CA2519401A1 Cannabinoid receptor ligands
10/06/2004EP1464678A1 Cyanine compound, optical filter, and optical recording material
10/06/2004EP1464641A1 4-Phenyl-piperazinyl, -piperidinyl and tetrahydropyridyl derivatives as dopamine D4 antagonists
10/06/2004EP1464638A1 Process for producing erythro-3-amino-2-hydroxybutyric acid derivatives
10/06/2004EP1463719A2 Eponemycin and epoxomicin analogs and uses thereof
10/06/2004EP1463715A1 Novel glucagon antagonists
10/06/2004EP1463714A2 Vanilloid receptor ligands and their use in treatments
10/06/2004EP1165516B1 Heterocyclic urea and related compounds useful as anti-inflammatory agents
10/06/2004EP1098864B1 Method for hydrogenating unsaturated heterocyclic compounds
10/06/2004EP1032424B9 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
10/06/2004EP1018878B1 Novel indolecarboxamides, pharmaceutical compositions and methodsof inhibiting calpain
10/06/2004EP0821551B1 Screening assay for the identification of inhibitors of macrophage migration inhibitory factor
10/06/2004CN1535146A 5-halo-tryptamine derivatives used as ligands of 5-HT 6 and/or 5-HT7 serotonin receptors
10/06/2004CN1534076A Red light emitted compound used for organic electroluminous device and orgainic electroluminous device using same
10/06/2004CN1169805C Esters and amides of non-steroidal anti-inflammatory carboxylic acids which may be used as anti-oxidants, 5-lipoxygenase inhibitors and non-steroidal anti-inflammatory products
10/06/2004CN1169789C Aminoalkoxy carbazoles for treatment of CNS diseases
10/06/2004CN1169759C Process for producing substituted aromatic compound
10/05/2004US6800762 Indolin derivaties as sun protection agents
10/05/2004US6800660 Bis(thio-hydrazide amide) compounds; anticancer agents
10/05/2004US6800658 A potent and safe inhibitors of mammalian cell proliferation for treating or preventing cancer, blood vessel proliferative disorders, fibrotic disorders and arteriosclerotic conditions
10/05/2004US6800656 Tricyclic compounds and method of treating herpes virus
10/05/2004US6800655 Analogs of indole-3-carbinol metabolites as chemotherapeutic and chemopreventive agents
10/05/2004US6800654 Substituted naphthyl indole derivatives as inhibitors of plasminogen activator inhibitor type-1 (PAI-1)
10/05/2004US6800645 Substituted azabicyclic compounds
10/05/2004CA2282834C Novel hexanoic acid derivatives
10/05/2004CA2103836C 7-(substituted)-9-[(substituted glycyl)-amido]-6-demethyl-6-deoxytetracyclines
09/2004
09/30/2004WO2004083238A1 Novel method for the synthesis of perindopril and the pharmaceutically-acceptable salts thereof
09/30/2004WO2004083237A1 Novel method for the synthesis of (2s, 3as, 7as)-perhydroindole-2-carboxylic acid and the esters thereof and application to the synthesis of perindopril
09/30/2004WO2004083194A1 Blue light-emitting compound, method for producing same and light-emitting device utilizing same
09/30/2004WO2004083174A2 Sulfonyl-amidino containing and tetrahydropyrimidino containing compounds as factor xa inhibitors
09/30/2004WO2004082565A2 Asymmetric cyclization in the presence of substituted pseudophedrines
09/30/2004WO2004082357A2 Novel method for the synthesis of derivatives of (2s, 3as, 7as)-1-[(s)-alanyl]-octahydro-1h-indole-2-carboxylic acid and application thereof to the synthesis of perindopril
09/30/2004WO2004050084A3 Ace-inhibitors having antioxidant and nitricoxid-donor activity
09/30/2004WO2004050014A3 Seterocyclic quinones as pharmaceutical agents
09/30/2004WO2003072535A8 Substituted hydroxyethylamines
09/30/2004US20040192911 Reacting 3-chloro-3-carboxylate indole compound with 3-chloropropanol in presence of acid catalyst
09/30/2004US20040192779 2-amino-2-alkyl-4 hexenoic and hexynoic acid derivatives useful as nitric oxide synthase inhibitors
09/30/2004US20040192755 Immediate release medicinal compositions for oral use
09/30/2004US20040192749 1-Aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
09/30/2004US20040192745 Method of treating amytrophic lateral sclerosis using melatonin
09/30/2004US20040192744 Inhibition of Histone Deacetylase; antiproliferative; antitumor: cell differentiation; 3,5-Dimethyl-isoxazole-4-carboxylic acid (2-amino-4,5-dichloro-phenyl)-amide
09/30/2004US20040192702 Heteroaryl alkyl piperazine derivatives
09/30/2004US20040192693 Antidiabetic agents; arteriosclerosis; cardiovascular disorders; anticholesterol agents; antidepressants; schizophrenia; antilipemic agents
09/30/2004US20040192681 N-acylsulfonamide apoptosis promoters
09/30/2004US20040192623 Aloe-emodin derivatives and their use in the treatment of neoplasias
09/30/2004US20040191210 Compounds
09/29/2004EP1462103A1 NO donors, combination products and uses as modulators of neurotransmitter release
09/29/2004EP1461311A2 Urea derivatives as vr1-antagonists
09/29/2004EP1461038A1 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders
09/29/2004EP0713702B1 Anxiolytic agent
09/29/2004CN1533374A Substitutled cyclohexane-1,4-diamine derivatives
09/29/2004CN1168716C Optical active tetrahydrobenzindole derivatives
09/29/2004CN1168715C Novel benzene amine compound, its prepn. process and medicinal compsns. contg. them
09/28/2004US6797848 Anthracene derivative and organic electroluminescence device using the derivative
09/28/2004US6797825 Protein kinase inhibitors
09/28/2004US6797731 Resorcinol derivatives
09/28/2004US6797708 Enzyme inhibitors such as 4-(2-(1-benzhydryl-2-(2-((benzyl-sulfonyl)amino)ethyl)-5-chloro-1h-indol-3 -yl)ethoxy) benzoic acid, used as analgesics or antiinflammatory agents
09/28/2004US6797699 Exemplified by n'-l-arginylspermidine
09/28/2004US6797449 For planographic printing plate precursors, color proofs, photoresists and color filters; high infrared radiation absorption; semiconductor lasers