Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
08/2002
08/28/2002EP0846110B1 Thf-containing sulfonamide inhibitors of aspartyl protease
08/28/2002CN1366518A Biphenyl butyric acid derivative as matrix metalloproteinase inhibitor
08/28/2002CN1365970A Process for separating and purifying N-ethyl carbazole
08/28/2002CN1089755C Distamycin derivatives, processe for preparing them, and their use as antitumor and antiviral agents
08/28/2002CN1089754C Derivatives from itaconic acid as component of polymer
08/27/2002US6441194 Two step, one pot alkylation in presence of bronstead acid catalyst; reacting pyrrole-2-carbaldehyde with vilsmeir reagent, such as oxalyl chloride and dimethylforamide, then alkylating agent, such as tertbutyl choride
08/27/2002US6441177 (4-bromo-phenyl)-(4-(6-(cyclopropyl-methyl-amino)-hexyloxy)-2-fluoro -phenyl)-methanone; antimycotic and cholesterol lowering activity
08/27/2002US6441023 For therapy of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone disease, diabetes (insulin resistance) and hiv infection
08/27/2002US6441001 2-substituted-4-nitrogen heterocycles as modulators of chemokine receptor activity
08/27/2002US6440937 Competitive inhibitors of trypsin-like serin proteases, especially thrombin and kininogenases such as kallikrein; thrombin inhibitors, anticoagulants, and antiinflammatory agents
08/22/2002WO2002064644A1 Complexed compounds and use thereof for the polymerisation of olefins
08/22/2002WO2002064563A1 Novel benzoylguanidine salt
08/22/2002WO2002064562A1 Pyrrolecarboxamides for the use as fungicides
08/22/2002WO2002064561A1 $g(d)1-pyrrolines used in pest control
08/22/2002WO2002064550A1 Glucocorticoid receptor modulators
08/22/2002WO2002064546A2 Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
08/22/2002WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals
08/22/2002WO2002032869A3 Substituted heterocyclic compounds for treating multidrug resistance
08/22/2002US20020115863 Hydroxamate derivatives that inhibit peptidyl deformylase (PDF), antimicrobials and antibiotics
08/22/2002US20020115806 Olefin polymerization catalyst system is a reaction product of a metallocenes and a cocatalyst containing fluoroaryl substituted secondary amine or phsophine compound and an anion containing group 13 element which is noncoordinatig
08/22/2002US20020115709 Atorvastatin hemi-calcium form VII
08/22/2002US20020115653 Retinoic acid mimetic anilides
08/22/2002US20020115576 Condensates of hydroxy aromatic compounds, an aldehyde and an amine
08/22/2002DE10114425C1 Diaminobenzol-Derivate und diese Verbindungen enthaltende Haarfärbemittel Diaminobenzene derivatives and compositions containing these compounds hair dye
08/22/2002CA2436271A1 Pyrrolecarboxamides for the use as fungicides
08/21/2002EP1233013A1 Novel phenylalanine derivatives
08/21/2002EP1232150A1 Urea derivatives as anti-inflammatory agents
08/21/2002EP1231939A2 Oncolytic combinations for the treatment of cancer
08/21/2002EP0829472B1 Improved process for producing 4-hydroxy-2-pyrrolidone
08/21/2002EP0675715B1 Cell differentiation induction with mevalonate and mevalonolactone derivatives
08/21/2002CN1365347A Anthracene derivatives and organic electroleuminescents device made by using the same
08/21/2002CN1089437C Neutral molecular detection method and device including using new compound and painting materials
08/20/2002US6437175 Process for racemization of n-acylamino acids by means of transition metal catalysts
08/20/2002US6437137 Naphthyl compounds, intermediates, processes, compositions, and methods
08/20/2002US6437009 Low foam n-alkyltartarimide and n-alkylmalimide wetting agents
08/20/2002US6436999 Diacyl-substituted guanidines, a process for their preparation, their use as medicine or diagnostic aid, and medicine containing them
08/20/2002US6436967 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
08/20/2002US6436957 Indole derivatives as 5-HT1 agonists
08/20/2002US6436921 Have low minimum inhibitory concentrations for grampositive and gramnegative strains, are stable against degradation by renal dehydropeptidase-i and have excellent bioavailability
08/20/2002US6436904 Treatment of inflammatory diseases in mammals
08/20/2002US6436243 Continuous distillation at controlled temperature; separation from n-(2-hydroxyethyl)-2-pyrrolidone starting material, water and by-products; inhibiting thermal polymerization or decomposition
08/20/2002US6436235 N-substituted perfluoroalkylated pyrrolidines and process for making them
08/20/2002US6436152 Substituted 2-aminoalky-1,4-diaminobenzene compounds and oxidation dye precursor compositions containing same
08/20/2002CA2150372C Stable oral ci-981 formulation and process of preparing same
08/20/2002CA2088367C Tri- and tetra-valent monospecific antigen-binding proteins
08/20/2002CA2071273C Tetrahydropyrrolo[1,2-a]pyrazine-4-spiro-3'-pyrrolidine derivatives, processes for the preparation thereof and pharmaceutical compositions containing the same
08/20/2002CA2043294C Preparation of n-substituted pyrrolidones
08/15/2002WO2002062778A2 Anti-thrombotic compounds, production and use thereof as medicaments
08/15/2002WO2002062777A2 Amino ceramide-like compounds and therapeutic methods of use
08/15/2002WO2002062757A1 Norbornene-based heterobifunctional monomers and uses therefor
08/15/2002WO2002062756A1 Aromatic sulfonyl alpha-cycloamino hydroxamates and their use as mmp inhibitors
08/15/2002WO2002062755A2 Polyamide analogs as dna minor groove binders
08/15/2002WO2002062748A1 Carboxylic amides, the production and use thereof as medicaments
08/15/2002WO2002044175A3 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit
08/15/2002WO2002042244A3 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds
08/15/2002WO2001072685B1 Polyamine analogues as cytotoxic agents
08/15/2002US20020111347 Nervous system disorders
08/15/2002US20020111340 Antiallergens
08/15/2002US20020111338 Bile-acid conjugates for providing sustained systemic concentrations of drugs
08/15/2002US20020111265 Group-15 cationic compounds for olefin polymerization catalysts
08/15/2002CA2436837A1 Carboxylic acid amides, the preparation thereof and their use as pharmaceutical compositions
08/15/2002CA2435492A1 Antithrombotic compounds, the preparation thereof and their use as pharmaceutical compositions
08/14/2002EP1230215A1 Pyrrole derivatives as phosphodiesterase vii inhibitors
08/14/2002EP1230210A1 Aminoalcohol derivatives useful for the treatment of gastrointestinal disorders
08/14/2002EP0790974B1 Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors
08/14/2002EP0722439B1 Hiv protease inhibitors
08/14/2002DE10107045A1 Verfahren zur Polymerisation von Olefinen A process for the polymerization of olefins
08/14/2002DE10106455A1 DELTA·1·-Pyrroline DELTA · 1 · -Pyrrolines
08/14/2002CN1364158A Mutilin derivatives and their use as antibacterials
08/14/2002CN1364155A N-Cyanomethyl amides as protease inhibitors
08/14/2002CN1363555A Percutaneous absorption promoter and its synthesizing process and application
08/13/2002US6433213 Process for the synthesis of 1,3-diols
08/13/2002US6433162 Method for synthesizing porphyrin compounds
08/13/2002US6433002 Pesticidal 1-polyarylpyrroles
08/13/2002US6432969 Non-insulin dependent diabetes, obesity, arthritis, and osteoporosis treatment
08/13/2002US6432933 Malaria therapy; alzheimer's disorders
08/13/2002US6432921 Oligopeptides
08/08/2002WO2002060858A1 Novel compound having maillard reaction inhibitory activity
08/08/2002WO2002060383A2 Cancer therapy
08/08/2002WO2002038541A9 Cyanopyrrolidine derivatives
08/08/2002WO2002006189A3 Aniline derivatives
08/08/2002WO2001098268A3 Piperidine amides as modulators of chemokine receptor activity
08/08/2002US20020107406 Calcium receptor-active compounds
08/08/2002US20020107345 Complex of a selected transition metal with a monoanionic ligand that has at least three atoms that may coordinate to the transition metal, one of which is an oxygen at and one of which is a nitrogen in an imine radical
08/08/2002US20020107290 Inhibiting activated blood-coagulation factor X
08/08/2002US20020107255 Potent and selective inhibitors of chemokine binding to its receptor CCR1 found on inflammatory and immunomodulatory cells (preferably leukocytes and lymphocytes).
08/08/2002US20020107241 N-heterocyclic derivatives useful for treating or preventing neuronal damage associated with neurological disease
08/08/2002US20020107239 Cyclized amide derivatives
08/08/2002US20020107235 Carbamate and hydroxy groups containing phenanthrene derivatives; useful to treat obesity, diabetes and inflammation
08/08/2002US20020106341 Primary intermediates for oxidative coloration of hair
08/08/2002DE10104598A1 Carbonsäureamide, deren Herstellung und deren Verwendung als Arzneimittel Carboxamides, their preparation and their use as medicaments
08/08/2002CA2436245A1 Medicament for protection in radiotherapy
08/07/2002EP1228067A1 5-membered n-heterocyclic compounds with hypogylcemic and hypolipidemic activity
08/07/2002EP1228061A1 Dipeptidyl peptidase iv inhibitors and methods of making and using dipeptidyl peptidase iv inhibitors
08/07/2002EP1228053A1 Substituted piperazine derivatives, the production and use thereof as inhibitors of the microsomal triglyceride transfer protein (mtp)
08/07/2002EP1227805A2 Mediators of hedgehog signaling pathways, compositions and uses related thereto
08/07/2002EP1087660B1 Composition for keeping away vermin
08/07/2002CN1362954A Sulfamato hydroxamic acid metalloprotease inhibitor
08/07/2002CN1362947A N-cyanomethylamides as protease inhibitors
08/07/2002CN1362877A Method for treating neurodegeneration