Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
05/2002
05/15/2002EP1204657A1 Piperidine and pyrrolidine derivatives displaying neuronal activity
05/15/2002EP1204652A1 Novel succinate derivative compounds useful as cysteine protease inhibitors
05/15/2002EP1204645A2 Melanocortin-4 receptor binding compounds and methods of use thereof
05/15/2002EP1204639A1 Synthesis of a novel paramagnetic amino acid derivative (epm-5) for labelling chemical and biological macromolecules
05/15/2002EP1049694B1 Derivatives of benzoxadiazoles, benzothiadiazoles, benzotriazoles and quinoxalines
05/15/2002CN1349535A Bicyclic heteroaromatic compounds useful as LH agonists
05/15/2002CN1349498A Alkenyl-and alkynyl-containing metalloprotease inhibitors
05/15/2002CN1349485A 糖皮质激素受体调制剂 Glucocorticoid receptor modulators
05/15/2002CN1348954A Prepn of N-bromosuccinimide
05/15/2002CN1084744C N-substituted azaheterocyclic compounds
05/15/2002CN1084734C Anhydrous crystals
05/14/2002US6388123 Substituted phenyl keto enols as pesticides and herbicides
05/14/2002US6388122 Tryptase inhibitor and novel guanidino derivatives
05/14/2002US6387949 Substituted urea compounds useful in pain management
05/14/2002US6387941 Antiserotonine agents
05/14/2002US6387937 Indole derivatives
05/10/2002WO2002036641A2 Improved productivity catalysts and microstructure control
05/10/2002WO2002036585A2 Process for the preparation of ligands for olefin polymerization catalysts
05/10/2002WO2002036561A1 Bis-heterocyclic compounds with antitumour and chemosensitising activity
05/10/2002WO2002036560A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
05/10/2002WO2002036555A1 Sulfamides as gamma-secretase inhibitors
05/10/2002WO2002036554A2 Amidino-urea serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their snythesis
05/10/2002WO2002036544A1 Method of resolving optical isomers of amino acid derivative
05/10/2002CA2427565A1 Bis-heterocyclic compounds with antitumour and chemosensitising activity
05/10/2002CA2425286A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
05/10/2002CA2425285A1 Amidino-urea serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their snythesis
05/09/2002US20020055631 N-acylsulfonamide apoptosis promoters
05/09/2002US20020055616 Peptide-containing alpha-ketoamide cysteine and serine protease inhibitors
05/09/2002US20020055543 Inhibit phosphodiesterase type IV or inhibit the production of tumor necrosis factor; useful in treating diseases including asthma, arthritis, and sepsis.
05/09/2002US20020055534 Method for treating neurodegeneration
05/09/2002US20020055469 Anticoagulants
05/08/2002EP1203767A1 Heterocyclic-substituted alkylamide acat inhibitors
05/08/2002EP1203766A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors
05/08/2002EP1203585A1 Anti-ischemic agent
05/08/2002EP1203047A1 Electrically conductive polymers capable of being covalently grafted on by light, method for obtaining same and uses as supports in probes for specific identification in electronic biosensors
05/08/2002EP1202990A2 Neurotrophic pyrrolidines and piperidines, and related compositions containing them
05/08/2002EP1202968A2 Antibacterial agents
05/08/2002EP1202962A1 Pyrrolidine compounds and their use for treating hyperproliferative diseases and tumor diseases
05/08/2002EP1202961A1 Arylsulfonamido-substituted hydroxamic acid derivatives
05/08/2002EP1202956A1 Therapeutically and/or nutritionally enhanced derivatives of active ingredients and orally administrable compositions containing same
05/08/2002EP1202718A2 Substituted guanidines for the treatment of cancer and pain
05/08/2002EP1202626A1 Alpha-hydroxy-gamma-[[(carbocyclic-or heterocyclic-substituted)amino]carbonyl]alkanamide derivatives and uses thereof
05/08/2002DE10053796A1 Aminonaphthalene N-phenylsulfonamide derivatives, useful for treating central nervous system disorders, e.g. Alzheimer's disease, dementia, Parkinson's disease, are 5-HT6 receptor antagonists
05/08/2002CN1347693A Noval compound, its synthetizing process and therapeutic use
05/07/2002US6384236 N-(aroyl)glycine hydroxamic acid derivatives and related compounds
05/07/2002US6384080 Anthranilic acid derivatives as inhibitors of the cGMP-phosphodiesterase
05/07/2002US6384075 Treating diseases in which mast cell dysfunction is involved
05/07/2002US6384069 Brain disorders chronic pain, hypoglycemia, hypoxia, trauma, alzheimer's disease, aids-associated dementia, amyotrophic lateral sclerosis, parkinson's disease, and chronic alcoholism, comprising administering to a patient in need a
05/07/2002US6384063 Compound having effect of promoting neuron differentiation
05/07/2002US6384056 Cognition activators and nerve and vision disorders
05/02/2002WO2002042244A2 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds
05/02/2002WO2002034711A1 Biaryl compounds as serine protease inhibitors
05/02/2002WO2002034698A2 Phosgene-free process for preparing carbamates
05/02/2002WO2002004416A3 Lactam metalloprotease inhibitors
05/02/2002WO2001085675A3 Fluorous tagging compounds and their use
05/02/2002WO2001052829A3 Statin-type bone growth stimulators
05/02/2002US20020052514 1-(phenylmethyl)sulfonyl-2-hydroxymethyl pyrrolidine for example; use treating neurological disorders including physically damaged nerves and neurodegenerative diseases; treating alopecia and promoting hair growth
05/02/2002US20020052512 Diaminopropionic acid derivatives
05/02/2002US20020052510 N-linked sulfonamides of n-heterocyclic carboxylic acids or carboxylic acid isosteres
05/02/2002US20020052502 Cis-substituted aminocyclopropane derivative
05/02/2002US20020052410 Administering to the animal suffering from neurological disorders an amide compound having an affinity for FKBP-type immunophilins
05/02/2002US20020052399 In particular as inhibitors of HIV protease.
05/02/2002US20020052398 Pharmaceutical composition of 6-amino EM-12
05/02/2002US20020052378 Novel compounds and compositions as protease inhibitors
05/02/2002US20020052370 Including the treatment of female sexual dysfunction especially female sexual arousal disorder
05/02/2002US20020052349 p-(sulfonyl) aryl and heteroarylamines as anti-inflammatory agents
05/02/2002US20020052003 Composition for use in the adhesion of particle to surfaces
05/02/2002EP1201650A2 Ionic malonitril derivatives and their uses
05/02/2002EP1201649A1 Glucocorticoid receptor modulators
05/02/2002EP1201239A1 Cyclic amine ccr3 antagonists
05/02/2002EP1200457A2 Cysteine protease inhibitors
05/02/2002EP1200406A1 Cyclic amides and imides having selective antagonist activity at alpha-1d adrenergic receptor
05/02/2002EP1200402A1 Substituted 1,5-dihydropyrrol-2-on derivatives as nmda receptor antagonists for the treatment of pain
05/02/2002EP1200401A1 Method for producing protected acyl guanidines by way of mukaiyama reaction
05/02/2002EP1200400A1 Substituted pyrrolidin-2,3,4-trion-3-oxime derivatives useful as nmda-receptor antagonists
05/02/2002EP1200395A1 Urea derivatives as inhibitors of ccr-3 receptor
05/02/2002EP1200083A1 Antibiotic compound
05/02/2002CA2427473A1 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds
05/02/2002CA2426466A1 Phosgene-free process for preparing carbamates
05/02/2002CA2426430A1 Biaryl compounds as serine protease inhibitors
05/01/2002CN1347423A Catalyst contg. N-pyrrolyl substd. nitrogen donors
04/2002
04/30/2002US6380398 Compounds such as (s,s)1-(2-amino-3,3-dimethyl-butyryl)-2,5-dihydro-1h-pyrrole-2 -carbonitrile administered as antidiabetic agents; dipeptidyl peptidase-iv (dpp-iv)
04/30/2002US6380258 Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
04/30/2002US6380246 For combating pests and weeds
04/30/2002US6380243 Including human cytomegalovirus, herpes simplex viruses, epstein-barr virus, varicella-zoster virus, human herpesviruses- 6 and -7, and kaposi herpesvirus.
04/30/2002US6380241 For therapy of coronary angina, cerebral vasospasm, acute and chronic renal failure, gastric ulceration, cyclosporin-induced nephrotoxicity, endotoxin-induced toxicity, asthma, lpl-related lipoprotein disorders, proliferative diseases
04/30/2002US6380223 For therapy of diseases, such as obesity, diabetes, inflammation
04/30/2002US6380181 Synthetic catechol derivatives, method for production and use thereof
04/30/2002US6380149 Using mono-, di-, or trialkoxy-substituted perfluoroalkane, perfluorocycloalkane, and perfluorocycloalkyl(ene)-containing perfluoroalkane, optionally with catenary heteroatoms, and a cosolvent; good solvency, ozone depletion potential of zero
04/30/2002US6379655 For protection of human skin and/or hair against the damaging effects of ultraviolet irradiation
04/30/2002US6379588 Stabilized monomer composition
04/27/2002CA2539147A1 Process for the preparation of non-steroidal glucocorticoid receptor modulators
04/25/2002WO2002033026A1 Blends of quinone alkide and nitroxyl compounds as polymerization inhibitors
04/25/2002WO2002032874A2 Substituted heterocyclic compounds for treating multidrug resistance
04/25/2002WO2002032872A1 Nitrogenous aromatic ring compounds
04/25/2002WO2002032871A2 Compounds and methods for treating multidrug resistance
04/25/2002WO2002032869A2 Substituted heterocyclic compounds for treating multidrug resistance
04/25/2002WO2002032868A2 2-substituted heterocyclic compounds and their use in treating multidrug resistance
04/25/2002WO2002032864A1 Pharmaceutically active sulfanilide derivatives
04/25/2002WO2002032376A2 Bile-acid conjugates for providing sustained systemic concentrations of drugs