Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
11/1994
11/08/1994US5362912 Process for the preparation of a substituted diaminodiol
11/08/1994US5362902 Diuretics and treatment of cardiovascular disorders
11/02/1994EP0561863B1 Amidic derivatives of glutamic, aspartic and 2-amino adipic acids with antigastrin activity
11/01/1994US5360928 Synthesis and use of amino acid fluorides as peptide coupling reagents
11/01/1994US5360924 Process for preparing aromatic olefins
10/1994
10/30/1994CA2122227A1 Peptide analogs as irreversible interleukin-1.beta. protease inhibitors
10/27/1994WO1994023767A1 Oral drug delivery compositions and methods
10/26/1994CN1094057A Acetylglutaminylzinc and its preparation and usage
10/26/1994CN1094030A Diaminobenzoic acid derivatives
10/26/1994CN1094029A New acylamino acids
10/25/1994US5359120 Improvements relating to the production of prodrugs
10/25/1994US5359077 Process for preparation of 2-oxo-1 piperidinyl derivatives
10/19/1994EP0620210A1 Compounds with benzamidic structure active in gastro-intestinal pathologies
10/19/1994EP0619744A1 Nonionic x-ray contrast agents, compositions and methods
10/18/1994US5356613 X-ray contrast agents, compositions and methods
10/17/1994CA2120214A1 Compounds with benzamidic structure active in gastro-intestinal pathologies
10/13/1994WO1994022863A1 Second messenger cell signaling inhibitors
10/13/1994WO1994022811A1 New non ionic iodine-containing dimers useful as x-ray contrast agents, method for the preparation thereof, and galenical compositions containing them
10/13/1994WO1994022810A1 New non-ionic iodine-containing dimers useful as x-rays contrast agents, method for the preparation thereof, and galenical compositions containing them
10/13/1994WO1994022809A1 Substituted (arylalkylaminobenzyl)aminopropionamide derivatives, their preparation and use anti-epileptic, neuroprotective and antidepressant agents
10/13/1994WO1994022808A1 Substituted (arylalkoxybenzyl)aminopropanamide derivatives, their preparation and use as anti-epileptic, neuroprotective and antidepressant agents
10/13/1994WO1994022368A1 Perfluoro-1h-1h-neopentyl containing contrast agents and method to use same
10/13/1994WO1994019025A3 Contrast agents
10/13/1994CA2158279A1 Perfluoro-1h-1h-neopentyl containing contrast agents and method to use same
10/12/1994EP0619321A1 Very large scale immobilized peptide synthesis
10/12/1994EP0619297A1 Fungicides for the control of take-all desease of plants
10/12/1994EP0618926A1 New peptide derivatives
10/12/1994EP0618836A1 Purification of crude ioversol using reverse osmosis
10/11/1994US5354892 Biaryl substituted 4-amino-butyric acid amides
10/11/1994US5354884 Optically active N-α-fluoroacryloylamino acid derivatives for the resolution of racemates
10/11/1994US5354866 Treating HIV infections
10/11/1994CA1332422C Process for the preparation of bicyclic amino carboxylic acids, intermediates in this process, and their use
10/05/1994EP0618223A2 Peptides inhibiting interleukin 1-bêta release useful as antiinflammatory agents
10/05/1994EP0618190A1 9-[(Substituted glycyl)amido]-6-(substituted)-5-hydroxy-6-deoxytetracyclines
10/05/1994EP0618189A1 Iodinated aromatic propanedioates and their use as X-ray contrast agents
10/05/1994CN1093082A N,N-disubstituted arylcycloalkylamines, the salts thereof, pharmaceutical compositions containing these compounds...
09/1994
09/30/1994CA2119968A1 Iodinated aromatic propanedioates
09/29/1994WO1994021620A1 Amino-acid derivatives, their preparation and their use as renin inhibitors
09/29/1994WO1994021600A1 Novel polyiodinated compounds, preparation thereof and use thereof as radiological contrast agents
09/29/1994WO1994021599A1 Novel compound with platelet aggregation inhibitor activity
09/29/1994WO1994021595A1 Amine derivative and dermatologic preparation containing the same
09/29/1994CA2136243A1 New polyiodinated compounds, their preparation and their use as contrast media for radiology
09/28/1994EP0617009A1 Novel amino acid derivative
09/28/1994EP0616538A1 Novel macromolecular polyamine iodine-containing compound, process for its preparation and its use as a contrast agent
09/27/1994CA1332200C Non-linear optical active diols and polyurethanes prepared therefrom
09/21/1994EP0615969A1 2,4-Diamino-3-hydroxycarboxylic acid derivatives
09/21/1994EP0452377B1 Iodinated esters
09/21/1994CN1092410A Inhibitors of HIV protease useful for the treatment of aids
09/21/1994CN1092406A Compounds
09/15/1994WO1994020481A1 4-amino-2-(hetero)aryl-butanamides useful as 5-ht1a-antagonists
09/15/1994WO1994020463A1 Novel distamycin analogues
09/15/1994WO1994020455A1 Styryl derivatives, their preparation and use as pde-iv inhibitors
09/15/1994WO1994020454A1 New derivatives of glutamic and aspartic acids, a method of preparing them, and their use as drugs for enhancing memory and learning
09/15/1994WO1994020446A1 Trisubstituted phenyl derivatives as phosphodiesterase inhibitors and processes for their preparation
09/15/1994WO1994015598A3 Methods for the improvement of cognition with functional antagonists of the glycine nmda receptor complex
09/15/1994CA2157187A1 Novel distamycin analogues
09/14/1994EP0614661A2 Benzylidene- and cinnamylidine-malononitrile derivatives for the inhibition of proliferative processes in mammalian cells
09/14/1994EP0557345B1 1,3-bis- 3-(mono- or poly-hydroxy)acylamino-5-(mono- or poly-hydroxyalkyl)aminocarbonyl-2,4,6-triiodo-benzoyl-amino]-hydroxy- or hydroxyalkyl-propanes, their methods of preparation and x-ray contrast media containing them
09/14/1994EP0489032B1 Hydroxamic acid based collagenase inhibitors
09/13/1994US5347036 Substituted di-t-butylphenols
09/13/1994US5346907 Cholecystokinin antagonists used in treatment or prevention of disorders of gastrointestinal, central nervous, appetite regulating or pain regulating systems
09/13/1994CA2118876A1 2,4-diamino-3-hydroxycarboxylic acid derivatives
09/09/1994CA2117121A1 Peptides
09/07/1994EP0613883A1 Hydroxamic acid derivative
09/06/1994US5344845 Methyl 4(4-acetoxy-3-methoxycinnamanide and salts as an immunosuppressive drug for allergic reactions
09/06/1994US5344836 Fused benzeneoxyacetic acid derivatives
09/01/1994WO1994019344A1 Amide compounds with pharmacological activity
09/01/1994WO1994019314A1 Glycerol derivative, device and pharmaceutical composition
09/01/1994WO1994019025A2 Contrast agents
09/01/1994WO1994018987A1 Drug composition containing nucleic acid copolymer
09/01/1994WO1994018963A1 Method of reversing resistance of hiv-1 strains to zidovudine
09/01/1994CA2155829A1 Method of reversing resistance of hiv-1 strains to zidovudine
08/1994
08/31/1994EP0612751A2 Compounds for the preparation of cephem derivatives
08/31/1994EP0476014B1 Very large scale immobilized polymer synthesis
08/30/1994US5342835 Antifungal agents based on amides containing a phenyl group
08/24/1994EP0611756A2 Alcohol or aldehyde derivatives as cathepsin L inhibitor and bone resorption inhibitor
08/23/1994US5340807 Tricyclic compounds and intermediates thereof
08/23/1994CA1331626C Process for the preparation of 2,4,6-triiodo-5-amino-n-alkylisophthalamic acid
08/20/1994CA2115913A1 Alcohol or aldehyde derivatives and their use
08/18/1994WO1994018339A1 Compositions and methods for protein structural determinations
08/18/1994CA2129904A1 Compositions and methods for protein structural determinations
08/17/1994EP0610451A1 Ethynyl alanine amino diol compounds for treatment of hypertension
08/17/1994EP0610400A1 Hyperbranched aramids
08/16/1994US5338532 Starburst conjugates
08/16/1994US5338529 Chromatography detection, separation of fullerenes
08/16/1994CA1331450C Diethylenetriamine pentaacetic acid derivatives
08/10/1994EP0609625A1 Inhibitors of HIV protease useful for the treatment of AIDS
08/10/1994EP0575360B1 Process of concentration and purification of organic compounds
08/10/1994EP0564561A4 Peptides ketoamides, ketoacids, and ketoesters
08/10/1994CN1090572A New polyiodinated compounds, process of preparation, and contrast agent containing them.
08/09/1994CA1331419C Peptides with pharmaceutical activity
08/04/1994WO1994017125A1 Structured copolymers used as absorbents, gels and carriers of metal ions
08/04/1994WO1994017096A1 Peptides having anti-hiv activity
08/04/1994WO1994017035A1 Aminoacid derivates, medicaments containing these compounds and process for preparing the same
08/04/1994WO1994017034A1 Substituted amino compounds, their preparation and their use as inhibitors of thrombocyte aggregation
08/04/1994WO1993025583A3 Proteinoid carriers and methods for preparation and use thereof
08/04/1994CA2153582A1 Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
08/03/1994EP0608908A2 Dense star polymers and a process for producing dense star polymers
08/03/1994CN1090278A Renin Inhibiting N-(2-Amino-2-oxoethyl)-butanediamide derivatives
08/03/1994CN1090269A Fungicides