Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
02/1995
02/02/1995WO1995003378A1 Reaction products of amino alkylene carboxylic acids and petroleum middle distillates containing them
02/02/1995WO1995003271A1 2-amino-4-phenyl-4-oxo-butyric acid derivatives with kynureninase and/or kynurenine-3-hydroxylase inhibiting activity
02/02/1995CA2144521A1 2-amino-4-phenyl-4-oxo-butyric acid derivatives with kynureninase and/or kynurenine-3-hydroxylase inhibiting activity
02/01/1995EP0636183A1 Compositions and methods for protein structural determinations
02/01/1995EP0636125A1 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists
02/01/1995EP0527983B1 Non-ionic surface active compounds
02/01/1995CN1098093A Arthropodicidal amides
02/01/1995CN1097949A L-aspartyl-d-alpha-aminoalkanoyl-(S)-N-alpha-alkylbenzyl amides useful as artificial sweeteners
01/1995
01/31/1995US5386041 Antibiotic
01/31/1995US5386040 Hydrolysis of an acetal resin; crosslinking agents
01/26/1995DE4324672A1 Compound with antibiotic activity, preparation process and composition containing the compound
01/25/1995EP0634995A1 Process and intermediate for the purification of oxytetracycline.
01/24/1995US5384331 Ketamine analogues for treatment of thrombocytopenia
01/24/1995US5384330 Pharmaceutically active 1,2,4-triamino-benzene derivatives, processes for their preparation and pharmaceutical compositions containing them
01/24/1995US5383942 Reaction of 4-alkyl-2-morpholinone and oxypolyalkylene amine to form amido alkanolamine as antideposit agents in fuel combustion
01/19/1995WO1995001966A1 Iodinated oligomeric compounds and diagnostic compositions containing the same
01/19/1995WO1995001956A1 Derivatives of valproic and 2-valproenoic acid amides and use as anticonvulsants
01/18/1995EP0634394A2 Organic fluorine compound
01/18/1995EP0633776A1 Compounds useful for treating allergic and inflammatory diseases
01/17/1995US5382683 Sedative, antiepileptic
01/17/1995US5382595 Antiischemic agents
01/12/1995WO1995001370A1 Higher order structure and binding of peptide nucleic acids
01/12/1995WO1995001369A1 Double-stranded peptide nucleic acids
01/12/1995WO1995001348A2 Imides as inhibitors of tnp alpha
01/12/1995WO1995001326A1 Anti-atherosclerotic diaryl compounds
01/12/1995WO1995001124A1 Functionalized tripodal ligands for imaging applications
01/12/1995DE4321897A1 Substituted amino acid derivatives, processes for their preparation, compositions comprising them, and their use
01/12/1995DE4321502A1 Alkynol-substituted peptides, processes for their preparation and their use as antiretroviral agents
01/12/1995CA2626178A1 Process for the preparation of thalidomide
01/12/1995CA2531868A1 Process for the preparation of thalidomide
01/12/1995CA2166462A1 Double-stranded peptide nucleic acids
01/12/1995CA2166461A1 Higher order structure and binding of peptide nucleic acids
01/12/1995CA2166413A1 Anti-atherosclerotic diaryl compounds
01/11/1995EP0633267A1 Process for the preparation of an alpha-amino acid amide for use in peptide synthesis
01/11/1995EP0633248A1 Butenoic acid derivatives
01/11/1995EP0632803A1 Arthropodicidal amides
01/10/1995US5380934 Process for producing alanylgutamine
01/10/1995US5380888 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
01/10/1995US5380818 High modulus aromatic polyamide film and production thereof
01/10/1995CA1333911C Dicarboxylic acid-bis(3,5-dicarbamoyl-2,4,6- triiodoanilides), process for their production as well as x-ray contrast media containing them
01/04/1995EP0632051A1 Anti-picornaviral agents
01/04/1995EP0632036A2 Amide and urea derivatives having anti-hypercholesteremic activity, their preparation and their therapeutic uses
01/04/1995EP0631570A1 Compounds
01/03/1995US5378729 Diamide derivatives
01/03/1995US5378728 Benzoic acid derivatives as antidiabetic agents
01/03/1995US5378712 Antithrombosis
01/02/1995CA2127187A1 Anti-picornaviral agents
12/1994
12/31/1994CA2126994A1 Amide and urea derivatives having anti-hypercholesteremic activity, their preparation and their therapeutic uses
12/28/1994EP0630959A1 Fuel composition
12/27/1994US5376155 Mineral oil middle distillate compositions
12/27/1994CA1333719C .alpha.-aminodicarboxylic acid derivatives, their preparation and their use
12/23/1994CA2123623A1 Fuel composition
12/22/1994WO1994029336A1 New peptide derivatives
12/22/1994WO1994029267A1 Arylacetamides, process for their preparation, compositions containing them and their use as fungicides
12/22/1994WO1994028878A1 Proteinoid carriers
12/22/1994WO1994025477A3 Novel peptide nucleic acids
12/22/1994CA2164957A1 Protenoid carriers and methods for preparation and use thereof
12/21/1994EP0629606A1 Amino acid derivative and anti-active-oxygen agent
12/21/1994EP0629196A1 Heterocyclic compounds, processes for their preparation and pharmaceutical compositions containing them
12/21/1994EP0586501B1 N-acyl derivatives of amino acid mixtures derived from cereal protein hydrolysates and applications thereof
12/20/1994US5374656 N-phenyl-n-alkoxycarbonylalkyl glycinamides, their preparation and the medicaments containing them
12/20/1994US5374623 Cysteine protease inhibitors effective for in vivo use
12/14/1994EP0628024A1 Synthesis of ioversol using a minimal excess of acetoxyacetylchloride
12/14/1994EP0498830B1 Glutamic and aspartic acid derivatives with antigastrin activity and a method for their preparation
12/13/1994US5373086 Inhibits precipitation of calcium carbonate and/or calcium phosphate and scale formation in cooling and boiler water treatment, reverse osmosis, flash evaporators, oil field recovery operation, plaque and tartar control and desalting
12/08/1994WO1994027954A1 Nitrobenzyl mustard quaternary salts and their use as hypoxia-selective cytotoxic agents
12/08/1994WO1994027644A1 Iodinated paramagnetic chelates, and their use as contrast agents
12/08/1994WO1994027584A2 Arylating medicaments
12/08/1994CA2163459A1 Arylating medicaments
12/07/1994EP0627410A1 N-acylglutamine derivative
12/07/1994EP0627406A1 2-amino-1,3-propanediol compound and immunosuppressant
12/06/1994US5371288 Branched alkyl-containing aminobenzamides as chain extenders in polyurethane-urea elastomers
12/06/1994US5371278 Increasing reaction solution concentration and temperature
12/06/1994US5371076 9-[(substituted glycyl)amido]-6-(substituted)-5-hydroxy-6-deoxytetracyclines
12/06/1994US5370877 Method for improving delivery and reducing toxicity of biologically active substances using novel α-amino dicarboxylic acid derivatives
12/06/1994US5370861 Intravascular administration; metabolizable to products which are soluble in body fluids
11/1994
11/30/1994CN1095725A N-acylaminoglutaricamide derivative
11/29/1994US5369123 Anticholesterol agents, treatment of atherosclerosis, antilipidemic agents and treatment of hyperlipoproteinaemia
11/29/1994US5369108 Potent inducers of terminal differentiation and methods of use thereof
11/24/1994WO1994026717A1 Hiv protease inhibitors useful for the treatment of aids
11/24/1994WO1994026695A1 Novel lupane derivatives, their preparation and pharmaceutical compositions containing same
11/24/1994WO1994026694A1 Method for the preparation of n-acylated aminoacids
11/24/1994CA2162702A1 Novel lupane derivatives, their preparation and pharmaceutical compositions containing same
11/24/1994CA2161334A1 Hiv protease inhibitors useful in the treatment of aids
11/22/1994US5366992 Benzoic acid substituted derivatives having cardiovascular activity
11/22/1994US5366982 Substituted bicyclic bis-aryl compounds exhibiting selective leukotriene B4 antagonist activity, their preparation and use in pharmaceutical compositions
11/15/1994US5364850 Substituted tyrosyl diamide compounds
11/13/1994CA2123261A1 Urethanes and ureas that induce cytokine production
11/10/1994WO1994025477A2 Novel peptide nucleic acids
11/10/1994WO1994025435A1 Peptidyl derivatives and their use as metalloproteinase inhibitors
11/10/1994WO1994025434A1 Peptidyl derivatives as metalloproteinase inhibitors
11/10/1994WO1994025429A1 4-amino-fluorobenzamides and their use as cytotoxic prodrugs
11/10/1994WO1994025051A1 Thrombin inhibitors
11/10/1994WO1994025015A1 Digestive symptom ameliorant
11/10/1994CA2161230A1 Novel peptide nucleic acids
11/10/1994CA2159834A1 Thrombin inhibitors
11/10/1994CA2139129A1 Peptidyl derivatives and their use as metalloproteinase inhibitors
11/10/1994CA2139128A1 Peptidyl derivatives as metalloproteinase inhibitors
11/09/1994EP0623592A1 Peptide analogs as irreversible interleukin-1beta protease inhibitors
11/09/1994CN1094712A Process for the preparation of intermediates useful in the preparation of pyranyl cyanoguanidine derivatives