Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
12/1996
12/19/1996WO1996040286A1 Process for producing ioversol
12/19/1996WO1996040184A1 New cryptophycins from synthesis
12/19/1996WO1996040104A1 Hydroxyl ions as unique therapeutic agents and compounds that modulate ions, compounds
12/19/1996WO1996040097A1 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders
12/19/1996DE19521945A1 Kaskadenpolymere mit Iodaromaten Cascade polymers with iodoaromatics
12/19/1996DE19521412A1 Neue kationische und polykationische Amphiphile, diese enthaltende Reagenzien und deren Verwendung New cationic and polycationic amphiphiles containing these reagents and their use
12/19/1996CA2223978A1 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders
12/19/1996CA2223948A1 Chalcone retinoids and methods of use of same
12/19/1996CA2223925A1 Lipophilic contrast agents for use in hepatocyte-selective oil-in-water emulsions
12/17/1996US5585492 LTA4 Hydrolase inhibitors
12/17/1996US5585359 Inhibitors of farnesyl-protein transferase
12/17/1996US5585358 Derivatives of valproic acid amides and 2-valproenoic acid amides, method of making and use thereof as anticonvulsant agents
12/12/1996DE19521940A1 Iodhaltige lineare Polyamine und Polyamide The iodine-containing linear polyamines and polyamides
12/11/1996EP0747348A1 Aminoalkylcyclopropane derivative
12/11/1996EP0747346A2 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics
12/11/1996EP0747344A1 Process for the purification and crystallisation of iopamidol
12/10/1996US5583248 Amino acid derivatives having antiviral activity
12/10/1996US5583233 Retroviral protease inhibiting compounds
12/10/1996US5583232 Treating human immunodeficiency virus infections
12/10/1996US5583198 Amino acids, peptides or derivatives thereof coupled to fats
12/08/1996CA2176854A1 N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics
12/05/1996WO1996038435A1 Dopamine agonists
12/05/1996WO1996038406A1 Phenylalkanamide derivatives and agrohorticultural bactericides
12/05/1996DE19519508A1 Radio-halogenated benzamide derivs., useful in diagnosis and treatment of tumours
12/04/1996EP0745065A1 9-(substituted amino)-alpha-6-deoxy-5-oxy tetracycline derivatives, their preparation and their use as antibiotics
12/04/1996CN1033451C Alpha-substituted benzenemethanamine derivatives
12/03/1996US5580984 Retroviral protease inhibiting compounds
12/03/1996US5580481 Aqueous fabric softener composition, novel quaternary ammonium salt, and process for the preparation of said salt
11/1996
11/28/1996WO1996037461A1 Iodination process
11/27/1996EP0743853A1 Compounds active at a novel site on receptor-operated calcium channels useful for treatment of neurological disorders and diseases
11/27/1996EP0711180A4 Functionalized tripodal ligands for imaging applications
11/27/1996EP0646021B1 Purification of crude ioversol using continuous deionization
11/27/1996EP0489839B1 Novel hydrolytic enzyme inhibitors and substrates and assays, methods and kits embodying same
11/27/1996CN1136805A Aryl halide substituted metallic complexes, pharmaceuticals containing these complexes, their use for diagnostic purpose and complexs
11/27/1996CN1136556A Aromatic group substituted W-amino alkyl amide and alkyl amide
11/26/1996US5578594 Anticoagulants
11/26/1996US5578323 Proteinoid carriers and methods for preparation and use thereof
11/21/1996WO1996036620A1 Diaryldiamine derivatives and their use as delta opioid (ant)-agonists
11/21/1996WO1996036591A1 2-hydroxyphenylalkylamine derivatives and maillard reaction inhibitors
11/21/1996DE19518421A1 Aspartic acid oligomers and derivs. with high chelating capacity
11/21/1996CA2221380A1 Diaryldiamine derivatives and their use as delta opioid (ant)-agonists
11/21/1996CA2219944A1 2-hydroxyphenylalkylamine derivatives and maillard reaction inhibitors
11/20/1996EP0430968B1 Compounds, compositions and method for binding bio-affecting substances to surface membranes of bio-particles
11/19/1996US5576435 Process and intermediates for the preparation of excitatory amino acid receptor antagonists
11/19/1996US5575986 Chelating agent, complex compound of said chelating agent and metallic atom, and diagnostic agent comprising same
11/19/1996US5575905 Iodination process
11/14/1996WO1996035953A1 Combinatorial synthesis and high-throughput screening of a rev-inhibiting arylidenediamide array
11/14/1996CA2220576A1 Combinatorial synthesis and high-throughput screening of a rev-inhibiting arylidenediamide array
11/13/1996EP0741755A1 Polyaspartic acid having more than 50 % beta form and less than 50 % alpha form
11/13/1996EP0741697A1 Amino acid derivatives and their use as phospholipase a2 inhibitors
11/13/1996EP0741691A1 Polyhydroxy diamines and their use in detergent compositions
11/13/1996CN1135749A Iodinated derivatives, preparation and use thereof as contrast agents in x-ray radiology
11/12/1996US5574016 Anticoagulants and cardiovascular disorders
11/12/1996US5574015 Isosteric antiherpes peptide derivatives
11/12/1996US5573752 Aromatic amide compounds and metal chelates thereof
11/12/1996US5573748 Kit for use in preparing the chelate; container with glycylglycyl ligand, water soluble stannous salt, intermediate exchange ligand, water soluble technetium-99m pertechnetate
11/07/1996WO1996034852A1 Novel tetracycline derivatives
11/07/1996WO1996034851A1 Benzene, pyridine, naphtalene or benzophenone derivatives as inhibitors of squalene synthetase and protein farnesyltransferase
11/07/1996WO1996034850A1 Cyclobutane derivatives and their use as inhibitors of protein farnesyltransferase
11/07/1996WO1996034849A1 Tetralines bearing a phenyl substituant on the aromatic ring and their use in the treatment of epilepsy, stroke and brain or spinal trauma
11/07/1996CA2219277A1 Novel tetracycline derivatives
11/06/1996EP0740655A1 Metalloproteinase inhibitors
11/06/1996EP0740652A1 Metalloproteinase inhibitors
11/06/1996EP0740648A1 Lewis acid catalyzed ammonolysis of nylon
11/06/1996EP0706375A4 Proteinoid carriers
11/05/1996US5571941 Dissolving crude solid in secondary butanol, crystallization
11/05/1996US5571845 Nitroaniline derivatives and their use as anti-tumour agents
10/1996
10/30/1996EP0739486A1 Synthetic receptors, libraries and uses thereof
10/30/1996EP0739351A1 Monomeric diols and phosphate linked oligomers formed therefrom
10/30/1996EP0571593B1 New non ionic iodized agents for x-ray contrasting, method for preparing them and galenical compositions containing them
10/30/1996EP0538301B1 Hiv-inhibiting benzeneacetamide derivatives
10/30/1996CN1033142C Process for preparing pharmaceutical composition showing properties in against human immunodeficiency virus
10/29/1996US5569665 Peptidyl derivatives and their use as metalloproteinases inhibitors
10/29/1996US5569446 Therapeutic and diagnostic uses
10/24/1996WO1996033166A1 Hydroxamic and carboxylic acids as metalloprotease inhibitors
10/24/1996WO1996033165A1 Derivatives of succinamide and their use as metalloproteinase inhibitor
10/24/1996WO1996033162A1 Compounds containing a substantially planar, fused ring system with at least 4 aromatic rings and their use as a chiral stationary phase in enantiomeric separation
10/24/1996WO1996033161A1 Derivatives of succinamide and their use as metalloproteinase inhibitors
10/24/1996CA2218380A1 Novel hydroxamic and carbocylic acids as metalloprotease inhibitors
10/23/1996EP0738283A1 New polyaminocarboxylate chelators
10/23/1996EP0738155A1 Modular design and synthesis of oxazolone-derived molecules
10/23/1996EP0738149A1 1-aminoindan derivatives and compositions thereof
10/23/1996EP0738144A1 Phenylmethyl hexanamides, and the use thereof
10/23/1996EP0738138A1 Quaternary salts of para-dialkylamino benzamide derivatives
10/23/1996CN1134153A Matrix metalloprotease inhibitors
10/23/1996CN1133834A Cinnamic acid derivative
10/23/1996CN1033087C 7-(subtd.)-8-(substd.-9-|(substd.glycyl) amido¨-6-demethyl-6-deoxytetracyclines
10/22/1996US5567692 9-[(substituted glycyl) amido)]-6-demethyl-6-deoxytetracyclines
10/22/1996US5567597 Hydrolytic enzyme inhibitors/inactivators and methods for using same
10/22/1996US5567410 Compound capable of reversibly forming micelles containing hydrophilic polymer linked to hydrophobic polymer having covelantly bonded radiopaque molecules
10/22/1996CA1338672C Process for the synthesis of the levodopa
10/17/1996WO1996032102A1 Use of a cationic amphipathic compound as a transfection agent, vaccine additive or drug
10/17/1996WO1996020725A3 Peptide, peptide analog and amino acid analog protease inhibitors
10/17/1996CA2192597A1 Use of a cationic amphipathic compound as a transfection agent, vaccine additive or drug
10/15/1996US5565476 Renin inhibitors for treatment of congestive heart failure and hypertension
10/15/1996US5565418 Retroviral protease inhibiting compounds
10/15/1996US5565184 Administering as contrast agent stable complex with good relaxivity and osmolar characteristics
10/10/1996WO1996031527A1 Protease inhibiting succinic acid derivatives
10/10/1996WO1996031462A1 Benzamides for neurodegenerative disorder treatment
10/10/1996WO1996031461A1 Phenoxyethylamine derivatives having high affinity for the 5-ht1a receptor, preparation thereof, use thereof as drugs, and pharmaceutical compositions containing said derivatives