Patents
Patents for C07C 237 - Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups (16,118)
07/1995
07/06/1995WO1995017903A1 Modular design and synthesis of oxazolone-derived molecules
07/06/1995WO1995017888A1 Phenylmethyl hexanamides, and the use thereof
07/06/1995CA2179810A1 Aminocarboxylic acid amides, process for preparing the same and their use as anti-arrhythmic agents
07/06/1995CA2155662A1 Anthranilic acid derivative
07/05/1995EP0661292A1 Orally active renin inhibitors
07/05/1995EP0661289A1 Vinyl carboxamide derivatives as insecticides and acaricides
07/05/1995EP0661267A1 Chelating agent for attaching metal ions to proteins
07/05/1995EP0661261A1 Phenyl or phenylalkyl substituted naphtalene derivatives having retinoid-like activity as well as anti-tumor activities
07/05/1995EP0661260A1 New bi-aromatic compounds derived from amides pharmaceutical compositions and cosmetic compositions containing them and their use
07/04/1995US5430162 7-(substituted)-8-(substituted)-9-substituted amino)-6-demethyl-6-deoxytetracyclines
07/04/1995US5430155 1,4-diamine-2,3-dihydroxy butanes
07/04/1995US5430151 Trifluoromethyl-containing pseudopeptides active against retroviruses
07/04/1995US5430044 Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties
07/04/1995US5430041 Amino acid derivatives having antiviral activity
07/04/1995US5430025 Elastase-inhibiting peptides bearing a C-terminal trifluoromethylketone moiety
07/04/1995CA2137997A1 Retinoid-like compounds
06/1995
06/30/1995CA2139044A1 Vinylcarboxylic acid derivatives
06/29/1995WO1995017418A2 NOVEL INTERMEDIATES FOR THE SYNTHESIS OF L-ASPARTYL-D-α-AMINOALKANOYL-(S)-N-α-ALKYLBENZYL AMIDES USEFUL AS ARTIFICIAL SWEETENERS
06/29/1995WO1995017093A1 New cryptophycins
06/29/1995CA2179490A1 New cryptophycins
06/29/1995CA2179376A1 Novel intermediates for the synthesis of l-aspartyl-d-.alpha.-aminoalkanoyl-(s)-n-.alpha.-alkylbenzyl amides useful as artificial sweeteners
06/28/1995EP0659174A1 Derivatives of valproic and 2-valproenoic acid amides and use as anticonvulsants
06/28/1995CN1104209A 2,4-diamino-3-hydroxycarboxylic acid derivatives
06/27/1995US5428073 Antimicrobial agents which are substituted 2-cyclohexan-1-yl-amine compounds.
06/27/1995US5428069 Treating cognition with, aminocyclopropanecarboxylic derivatives
06/27/1995US5427919 Hydrolytic enzyme inhibitors/inactivators and methods for using same
06/27/1995US5427774 A cationic sunscreen agents; water insolubility, receptivity, nonhydrolyzing, chemical resistance, stability
06/27/1995US5427773 Sunscreen agents
06/21/1995EP0658562A1 Pesticidal phosphoric and derivatives
06/21/1995EP0658538A1 Diagnosis, evaluation and treatment of coronary artery disease by exercise simulation using closed loop drug delivery of an exercise simulating agent beta agonist
06/21/1995CN1104018A Substituted (arylalkylaminobenzyl) aminopropionamide derivatives, their preparation and use anti-eptic, neuroprotective and antidepressant agents
06/21/1995CN1104017A Substituted (arylalkoxybenzyl) aminopropanamide derivatives, their preparation and use as anti-epileptic, neuroprotective and antidepressant agents
06/21/1995CN1028990C Hiv-inhibiting benzeneacetamide derivatives
06/20/1995US5426229 Ring-substituted 2-amino-1,2,3,4-tetra-hydronaphthalenes, 3-aminochromanes, and 3-aminothiochromanes
06/16/1995CA2137897A1 Biaromatic compounds derived from amides; pharmaceutical and cosmetic compositions containing the same and their uses
06/14/1995EP0657418A1 Acylamino-benzamides and fungicides containing them
06/14/1995EP0657029A1 Calcium receptor active molecules
06/14/1995EP0656884A1 Novel poly-iodated compounds, method of preparation and contrast product containing same
06/14/1995EP0656883A1 Cationic lipids
06/14/1995EP0496836B1 Synthesis and use of amino acid fluorides as peptide coupling reagents
06/14/1995EP0484328B1 Process for the preparation of 2,4,6-triiodo-5-amino-isophthalamide compounds
06/13/1995US5424292 5-aminosalicylic acid derivatives for the therapy of chronic inflammatory bowel diseases
06/08/1995WO1995015319A1 Paramagnetic chelates for nuclear magnetic resonance diagnosis
06/08/1995WO1995015311A1 Tachykinin antagonists
06/08/1995WO1995015306A1 Aryl halide substituted metallic complexes, pharmaceuticals containing these complexes, their use for diagnostic purposes, and methods for preparing the complexes and pharmaceuticals
06/08/1995CA2177994A1 Tachykinin antagonists
06/08/1995CA2177977A1 Aryl halide substituted metallic complexes, pharmaceuticals containing these complexes, their use for diagnostic purposes, and methods for preparing the complexes and pharmaceuticals
06/07/1995EP0656348A2 Aceric acid derivatives as medicaments
06/07/1995EP0656026A1 Polyarylates containing derivatives of the natural amino acid l-tyrosine
06/06/1995US5422004 Monocyclic or polycyclic aromatic amide moiety; increased enantioselectivity
06/01/1995WO1995014655A1 Diastereoselective synthesis of hydroxyethylene dipeptide isosteres
05/1995
05/31/1995EP0655069A1 Amphiphilic compounds derived from amino acids or peptides, their methods of synthesis and their application as drug delivery systems
05/31/1995EP0640067A4 Improved synthesis of ioversol.
05/30/1995US5420272 7-(substituted)-8-(substituted)-9-](substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
05/30/1995US5419894 Complexing agents, complexes and complex salts
05/30/1995US5419893 Aminopolycarboxylic acids and derivatives thereof for magnetic resonance imaging
05/26/1995WO1994027584A3 Arylating medicaments
05/24/1995EP0408654B1 Process for the preparation of 2,4,6-triiodo-5-amino-n-alkylisophthalamic acid
05/23/1995US5417882 Liquid-crystalline compounds
05/18/1995WO1995013059A1 Farnesyl derivatives and pharmaceutical compositions containing them
05/17/1995EP0652863A1 Non-peptidic surrogates of the ldv sequence and their use in the treatment of inflammation, autoimmune diseases and tumour progression
05/17/1995EP0513063B1 Process for production of ioversol
05/16/1995US5416223 Iodinated esters
05/16/1995US5416117 Cyclopropenone derivatives
05/16/1995US5416113 Bronchodilators
05/11/1995WO1995012603A1 Matrix metalloprotease inhibitors________________________________
05/11/1995WO1995012572A1 Cyclobutane derivatives as inhibitors of squalene synthetase and protein farnesyltransferase
05/11/1995CA2175667A1 Matrix metalloprotease inhibitors________________________________
05/11/1995CA2152822A1 Cyclobutane derivatives as inhibitors of squalene synthetase and protein farnesyltransferase
05/10/1995EP0652229A2 Oligopeptides with fungicidal activity
05/10/1995EP0652228A1 Urethanes and ureas that induce cytokine production
05/10/1995EP0651740A1 Amino acid linked nitrogen mustard derivatives and their use as prodrugs in the treatment of tumours
05/09/1995US5414099 Acid catalyst; also making phenyl esters by reacting the amido acids either with phenol in presence of acid catalyst and boric acid or with phenol ester of lower molecular weight carboxylic acid in presence of basic catalyst
05/09/1995US5413999 HIV protease inhibitors useful for the treatment of AIDS
05/09/1995US5413997 Triphenylmethane derivatives
05/04/1995WO1995011690A1 Desferrioxamine oral delivery system
05/03/1995EP0650595A1 Universal standard reagents, method of preparing same and use thereof
05/02/1995US5412145 P2'-modified hydroxamic acid collagenase inhibitors
05/02/1995US5411989 Nitric acid esters of cyclohexanol derivatives
04/1995
04/27/1995WO1995011221A1 Calcium receptor-active arylalkyl amines
04/26/1995EP0649443A1 Oxazolone derived materials
04/26/1995EP0649420A1 New process for the preparation of 3,3-diaryl acrylic acid amides.
04/26/1995EP0649409A1 Vinyl arenas having retinoid-like activity
04/26/1995EP0515510B1 Hydroquinone amino-acid esters, method of preparation, and pharmaceutical or cosmetic compositions containing them
04/25/1995CA1335375C Glycosaminoglycan salts, processes for the preparation thereof and pharmaceutical composition containing them
04/20/1995WO1995010552A1 Acrylamido functional disubstituted acetyl aryl ketone photoinitiators
04/20/1995CA2173228A1 Acrylamido functional disubstituted acetyl aryl ketone photoinitiators
04/19/1995EP0649057A2 A photographic processing composition and a processing process therewith
04/19/1995EP0648745A1 Arylalkylamine having anticonvulsant and neuroprotective properties
04/19/1995EP0648612A1 Reversible heat-sensitive recording material
04/19/1995EP0648489A1 Arylalkylamides having neuroprotective properties
04/19/1995EP0648206A1 Peptidyl derivatives and their use as metalloproteinase inhibitors
04/19/1995EP0648205A1 Peptidyl derivatives as metalloproteinase inhibitors
04/19/1995EP0648203A1 Novel polyiodinated compounds, preparation thereof and use thereof as radiological contrast agents
04/19/1995EP0638060A4 T-butyl cascade polymers.
04/18/1995US5407961 α-substituted benzenemethanamine derivatives and pharmaceutical use
04/18/1995US5407956 Hypotensive agents, kidney disorders
04/13/1995WO1995009843A1 Hiv protease inhibitors
04/13/1995WO1995009839A1 Cycloalkanediols and their use in preparing chiral compounds
04/13/1995WO1995009838A1 INHIBITORS OF β-AMYLOID PROTEIN PRODUCTION