Patents for C07B 53 - Asymmetric syntheses (6,231)
10/2006
10/19/2006WO2006109442A1 PROCESS FOR PRODUCTION OF OPTICALLY ACTIVE α-HYDROXYPHOSPHONIC ACIDS AND DERIVATIVES THEREOF, OPTICALLY ACTIVE ALUMINUM(SALALEN) COMPLEXES AND PROCESS FOR PRODUCTION OF THE COMPLEXES, AND PROCESS FOR PRODUCTION OF SALALEN LIGANDS
10/19/2006WO2006108903A1 Phosphinite thioglycosides, preparation method and use thereof as novel ligands in asymmetric catalysis
10/18/2006CN1847201A Amino group-containing chiral ionic liquid and its prepn process and application
10/18/2006CN1280258C Process for producing 4,5-diamino shikimic acid derivative
10/17/2006US7122680 3-Substituted oxindole β3 agonsists
10/17/2006US7122499 Osmium oxide carried by hydrophilic polymer
10/12/2006US20060229473 Ligands
10/12/2006US20060229457 Method for producing optically active compound
10/12/2006US20060229320 Enantiomers of 1-[(4-chlorophenyl) phenylmethyl]-4-[(4-methylphenyl) sulfonyl] piperazine
10/12/2006US20060229319 For treatment of allergies; antihistamines
10/12/2006DE10063410B4 Verfahren zur Herstellung von optisch aktiven Enonen von Cyclopentan und Zwischenprodukte dafür A process for the preparation of optically active enones of cyclopentane and intermediates therefor
10/11/2006EP1469851B1 Melanocortin receptor agonists
10/11/2006CN1845929A Process for producing penicillanic acid compound
10/11/2006CN1279040C Tryasolyl tropane derivatives for therapy
10/10/2006US7119197 Reacting racemic (+-)-10,11-dihydro-10-hydroxy-5H-dibenz/b,f/azepine-5-carboxamide with (2R,3R)-di-O,O'-substituted-tartaric acid anhydride; precipitation of less soluble diastereoisomeric 10-O-di-O,O'-substituted-tartrate half-ester; hydrolysis
10/05/2006WO2006104226A1 OPTICALLY ACTIVE QUATERNARY AMMONIUM SALT HAVING AXIAL ASYMMETRY AND PROCESS FOR PRODUCING α-AMINO ACID AND DERIVATIVE THEREOF WITH THE SAME
10/05/2006WO2006104120A1 Method for producing l-2-amino-4-(hydroxymethylphosphinyl)- butanoic acid
10/05/2006WO2006103986A1 Process for production of optically active fluoroproline derivative
10/05/2006WO2006103756A1 Process for production of optically active quinuclidinol
10/05/2006US20060224001 Hydrogenation catalysts
10/04/2006EP1707559A1 Method of enanthio-selective nucleophilic addition reaction for conversion of enamide to imine and method of synthesizing alpha amino-gamma-keto acid ester
10/04/2006EP1707556A1 Method of enantiometrically selective nucleophilic addition reaction to carbonyl of enamide and method of synthesizing optically active alpha-hydroxy-gamma-keto acid ester and hydroxydiketone
10/04/2006CN1842533A Phospinite-imidazolines and metal complexes thereof
10/04/2006CN1277807C Process for the preparation of aminoalcohol and (1S, 4Rú®or (1R, 4S)-1-amino-4-(methylol)-2-cyclopentene or its salts
10/03/2006US7115780 For therapy of ulcers, pancreatitis, obesity, urinary incontinence and pollakiuria
10/03/2006US7115769 Catalyzing the alkylation, forming a 2-alkylcysteine derivatives, a chemical intermediates for iron chelating agents
10/03/2006US7115590 Phosphoramidate, and mono-, di-, and tri-phosphate esters of (1R, cis)-4-(6-amino-9H-purin-9-yl)-2-cyclopentene-1-methanol as antiviral agents
09/2006
09/28/2006WO2006101092A1 Method of producing 3-hydroxybutyraldehyde derivative
09/28/2006WO2006099926A1 Process for preparing enantiopure e-(2s)-alkyl-5-halopent-4-enoic acids and esters
09/28/2006US20060217561 Synthesis of substituted thiazoline carboxylic acids
09/28/2006CA2602271A1 Method of producing 3-hydroxybutyraldehyde derivative
09/28/2006CA2599409A1 Process for preparing enantiopure e-(2s)-alkyl-5-halopent-4-enoic acids and esters
09/27/2006EP1200394B1 Process for preparing acids via alpha-chloroepoxy esters
09/21/2006US20060211862 Biotechnological resolution of racemic mixtures of 1-Amino-4-(hydroxymethyl)-2-cyclopentene using a hydrolase (lipase); optional formation of acyl derivatives
09/21/2006DE102005012408A1 Preparation of optically active 3-phenylpropionic acid derivative, useful to prepare halo-phenyl compound, comprises hydrogenating cis-isomer mixture of phenyl compound; crystallizing the enantiomer mixture and isolating the solid material
09/19/2006US7109350 Process for the preparation of optically active amines or salts thereof
09/19/2006US7109343 Metal catalysts and methods for making and using same
09/14/2006US20060205968 Process for producing optically active beta-amino acid derivatives
09/13/2006EP1325013B1 Catalyst for asymmetric (transfer) hydrogenation
09/13/2006CN1832953A Substituted ferrocenyldiphosphines as ligands for homogeneous hydrogenation catalysts
09/13/2006CN1832918A Process for producing optically active 1-alkyl-substituted 2,2,2-trifluoroethylamine
09/13/2006CN1274839C Process for preparation of enantiomerically enriched esters and alcohols
09/13/2006CN1274669C Fluorobenzamides suitable for the treatment of alzheimer's disease or senile dementia
09/12/2006US7105702 For use as catalysts in asymmetric reactions, such as, hydrogenation, hydride transfer, allylic alkylation, hydrosilylation, hydroboration, hydrovinylation, hydroformylation, olefin metathesis, hydrocarboxylation
09/12/2006US7105528 exhibit a surprising strong efficacy in lowering the intraocular pressure; excellent duration of action; excellent tolerability
09/08/2006WO2006093269A1 Optically active ammonium salt compound, production intermediate thereof and method for producing same
09/08/2006WO2006093142A1 Optically active ppar-activating compound intermediate and method for producing same
09/08/2006WO2006092884A1 Cyclic erythritol phosphoric acid derivative and asymmetric synthesis method using the same
09/08/2006WO2005117907A3 P-chiral phospholanes and phosphocyclic compounds and their use in asymmetric catalytic reactions
09/07/2006US20060199728 via iridium complex containing phosphoramidite ligand
09/07/2006DE102005010329A1 New diarylphenoxy-aluminum compound, obtained by a reaction of bis(diarylphenol) ligand with aluminum compound and/or aluminum compound, useful as a catalyst
09/06/2006EP0826652B1 Process for preparing asymmetric compound by using metal complex
09/06/2006CN1827214A Catalyst for asymmetric (transfer) hydrogenation
08/2006
08/31/2006DE102005007750A1 Preparation of optically active alkyl succinic acid monoalkyl esters comprising enantioselective hydrogenation of ester compound in presence of catalyst, which carries phospholane ligand
08/30/2006EP1180095B1 4-cyano-3-hydroxy butanoyl hydrazines, derivatives and process for the preparation thereof
08/30/2006CN1272310C Method for the production of optically active 2-amino-,2-chloro-,2-hydroxy or 2-alkoxy-1-alcohols
08/24/2006WO2006088142A1 Catalyst for asymmetric synthesis, ligand for use therein, and process for producing optically active compound through asymmetric synthesis reaction using them
08/24/2006WO2006087874A1 Process for producing optically active epoxy compound, complex for use in the process, and process for producing the same
08/24/2006DE102005007174A1 Verwendung von PIT-Emulsionen in biokatalytischen Reaktionen Use of PIT emulsions in biocatalytic reactions
08/24/2006CA2597883A1 Catalyst for asymmetric synthesis, ligand for use therein, and process for producing optically active compound through asymmetric synthesis reaction using them
08/23/2006EP1693364A1 Intermediates for the production of optically active cyclopropylamine derivatives and process for the production of the intermediates
08/23/2006EP1693362A1 Process for production of asymmetric alkyl compounds with alkali-treated solid carrier and alkali-treated solid carrier to be used in the process
08/23/2006EP1622920B1 Substituted ferrocenyldiphosphines as ligands for homogeneous hydrogenation catalysts
08/23/2006CN1823034A Process for producing optically active ss-hydroxy alpha aminocarboxylic acid derivative
08/22/2006US7094920 reacting oxy nitriles with solutions of inorganic acid in an alcohols, to form carbocyclic oxy esters and isomers, used as chemical intermediates for angiotensin converting enzyme inhibitors
08/22/2006US7094907 N,N-(optionally substituted)dialkylamino phosphines bound to an aromatic carbon are lithiated in ortho-position and the lithiated compounds are further converted to said bidentate ligands; oxidative dimerization; coupling
08/22/2006CA2179244C New bisphosphines as catalysts for asymmetric reactions
08/17/2006US20060183930 Chiral monophosphorus compounds
08/17/2006US20060183896 Optically active quaternary ammonium salt, process for producing the same, and process for producing optically active alpha-amino acid derivative with the same
08/17/2006DE102005005828A1 Makroporöses Kunststoffperlenmaterial Macroporous plastics bead material
08/16/2006EP1689760A1 Method for asymmetric synthesis
08/16/2006CN1269809C Process for ascorbic acids using alkaline earth silicate catalysts
08/16/2006CN1269808C Process for the preparation of vialoguestamin D analogs
08/16/2006CN1269793C Method for producing 3,3-diarylpropylamines
08/15/2006US7091195 Derived from plants; for preventing or inhibiting tumor growth
08/09/2006CN1814766A Preparing pravastatin
08/08/2006CA2188835C Novel compounds and methods for synthesis and therapy
08/03/2006WO2006080576A1 METHOD FOR ASYMMETRIC ALLYLATION OF α-IMINO ACID
08/03/2006WO2006080425A1 Process for production of optically active hydroxymethylated compounds and catalyst therefor
08/03/2006US20060173210 Process for producing optically active compound
08/02/2006EP1686114A1 Process for producing optically active 2-alkylcysteine, derivative thereof, and processes for production
08/02/2006EP1685092A2 Asymmetric reductive amination of keto acid derivatives for producing amino acid derivatives
08/02/2006CN1267441C Method for selective production of racemic metallocene complexes
08/02/2006CN1267438C antidepressant indoletetrahydropyridine derivatives of 2,3-dihydro-7h-[1,4] dioxino [2,3-3] indole
08/01/2006US7084278 stereoselective preparation of beta-hydroxy-beta-aryl-beta-heterocyclyl esters, e.g., tert-butyl 3-hydroxy-3-(4-chlorophenyl)-3-(pyridin-2-yl)propionate, by reacting a Reformatsky reagent with a aroylheterocycle (especially a benzoypyridine or a benzoylimidazole) in the presence of a cinchona alkaloid
08/01/2006US7084250 asymmetric hydrogenation of 2-[2-acetylamino-3-(4-cyanophenyl)acryloylamino]-2-cyclohexylacetic acid and conversion of the cyano group into the amidine, or a salt thereof, with a 3-(2-amino-2-carbamoylethyl)-1-methylpyridinium salt; claimed intermediates
08/01/2006CA2188400C Preparation of arthropodicidal oxadiazines
07/2006
07/27/2006US20060167267 Michael-type addition of a nucleophile to a dialkyl 2-methylidenylpropan-1,3-dioate and the conversion of a ester moiety into an amino moiety; S)-2-methylcysteine; desferrithiocin
07/27/2006US20060166337 Process for producing optically active erythro 3-cyclohexylserines
07/26/2006CN1266145C Synthesis of cannabinoids
07/26/2006CN1266136C Kinetic resolution of intermediate for preparing benazepril and its analogues
07/26/2006CN1266119C Preparation of acid by alpha-chlorination of epoxy resin
07/25/2006US7081544 Chiral ligands, transition metal complexes thereof, and the catalytic use of the same
07/25/2006US7081536 Complexes; used for catalyst
07/25/2006US7081533 Cycloaliphatic/aromatic diphosphines and use thereof in catalysis
07/20/2006WO2006075651A1 PROCESS FOR PRODUCING OPTICALLY ACTIVE β-HYDROXY-α-AMINOCARBOXYLIC ACID DERIVATIVE
07/20/2006WO2006075166A1 Metallocene-based phosphorus chiral phosphines
07/20/2006US20060161022 Chiral ligands for application in asymmetric syntheses
07/19/2006EP1451133A4 P-chiral phospholanes and phosphocyclic compounds and their use in asymmetric catalytic reactions
07/19/2006CN1264823C Process for preparing retroviral protease inhibitors and its intermediates
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