Patents for C07B 53 - Asymmetric syntheses (6,231)
05/2004
05/13/2004WO2004024684A3 Enantioselective amination and etherification
05/13/2004US20040092779 Comprising aromatic polyolefin having oxyalkyleneoxyaryl group; solvent and heat resistance; handling
05/13/2004US20040092388 Chemical and enantiomorph selectivity; high catalytic activity
05/12/2004EP1418170A2 Process for the preparation of optically active amino alcohols by optical resolution
05/12/2004EP1417199A1 Novel modifications of the trometamol salt of r-thioctic acid and method for producing the same
05/12/2004EP1341785A4 HYDROLYSIS OF R(R*,R*)]-2-(4-FLUOROPHENYL)-$g(b),$g(d) -DIHYDROXY-5-(1-METHYLETHYL)-3-PHENYL-4- (PHENYLAMINO)CARBONYL]-1H-PYRROLE-1-HEPTANOIC ACID ESTERS WITH CALCIUM HYDROXIDE
05/12/2004EP1131279B1 Industrial process for the production of l-carnitine
05/12/2004CN1496345A Chain oligolactic acid ester
05/12/2004CN1495189A Preparation method of phosphite ester and transition metal complex
05/12/2004CN1495164A Method for preparing chiral lactone
05/06/2004WO2004037838A1 Preparation of partially hydrogenated rac-ansa-metallocene complexes
05/06/2004WO2004037760A2 Process for producing optically active 2-alkoxy-1-(trifluoromethyl-substituted phenyl)ethanol derivatives
05/06/2004WO2003084942A3 Stereoselective alkylation of chiral 2-methyl-4-protected piperazines
05/06/2004US20040087437 Crown ether and perfluorinated sulfonyl lead derivative; high yield and optical selectivity under mild conditions; water tolerance; simple
05/06/2004EP1414569A2 Optically active catalysts comprising salen ligands and vanadium(iv), their preparation and use in the production of cyanhydrines
05/06/2004EP1414463A1 Asymmetric synthesis of kavalactones
05/06/2004EP1414384A2 Synthesis of epothilones and relates analogs
05/06/2004EP1335911B1 Synthesis of r(+)alpha-lipoic acid
05/06/2004EP1233828B1 Chiral catalysts for asymmetric acylation and related transformations
05/06/2004DE10250025A1 Production of new partially hydrogenated metallocene complexes, useful as catalysts for the polymerization of olefins, comprises reaction of transition metal complexes with cyclopentadienyl derivatives and hydrogenation
05/05/2004CN1494532A New asymmetric process for preparation of diarylmethylpiperazines derivatives and novel asymmetric diarylmetylamines as intermediates
05/05/2004CN1494524A Process for stereo selective synthesis of prostacyclin derivatives
05/05/2004CN1494456A Osmium oxide deposited on hydrophilic polymer support
05/05/2004CN1493576A Chiral diphosphorus compound and its transition metal compounding product
05/04/2004US6730629 Asymmetric phosphine ligand
05/04/2004CA2295993C Novel stereoselective processes for the preparation of gabapentin analogues
04/2004
04/29/2004WO2004035208A1 Mixtures of chiral monophosphorus compounds used as ligand systems for asymmetric transition metal catalysis
04/29/2004WO2003003972A3 Kinetic resolution of a intermediate useful in the production of benazepril and analogues thereof
04/29/2004US20040082820 Hydrogen transfer reduction; useful as intermediate for production of pharmaceuticals/agricultural chemicals
04/29/2004US20040082809 Reacting an anhydride with an alcohol; partial esterification
04/29/2004US20040082796 Reacting a substituted benzonitrile with a cysteine compound
04/29/2004US20040082647 Anticholesterol agents; controlling bile acid transfer into intestines
04/29/2004US20040082625 Osteoporosis, bone disorders
04/29/2004DE10247633A1 Mischungen von chiralen Monophosphor-Verbindungen als Ligandensysteme für die asymmetrische Übergangsmetallkatalyse Mixtures of chiral mono-phosphorus compounds as ligands for asymmetric systems transition metal catalysis
04/28/2004EP1413307A1 Therapeutically active levorotatory and dextrorotatory 1-(4-chlorophenyl)phenylmethyl piperazines
04/28/2004EP1412323A1 Protected 3,5-dihydroxy-2,2-dimethyl-valeronitriles for the synthesis of epothilones and derivatives and method for the production and use thereof
04/28/2004EP1200384B1 2-alkyl-5-halogen-pent-4-ene carboxylic acids and their production
04/28/2004EP1107936B1 Copper-catalysed enantioselective allylic substitution reactions
04/28/2004CN1147462C Improved process for preparation of non-hydroscopic salts of L(-)-Carnitine
04/27/2004US6727377 Asymmetric catalysis based on chiral phospholanes and hydroxyl phospholanes
04/27/2004US6727098 Circular dichroism
04/22/2004WO2003041728A9 Novel phenyl-propargylether derivatives
04/22/2004US20040077861 Asymmetric addition of organometallic compounds to chiral sulfinimine to give adducts in predominantly one diastereomer can subsequently be transferred into pure enantiomers of by cleavage of the chiral auxilliary
04/22/2004US20040077059 Process for the preparation of enantiomerically enriched esters and alcohols
04/21/2004EP1409691A2 Stereoselective preparation of cyclic l-amino acids
04/21/2004EP1409493A1 Method for producing non-chiral organic compounds containing optically active hydroxy groups
04/21/2004EP1409467A1 Synthesis of udp-glucose: n-acylsphingosine glucosyltransferase inhibitors
04/21/2004EP1409453A1 Novel diamines having a casr modulating activity
04/21/2004EP1409125A1 Microencapsulated catalyst, methods of preparation and methods of use thereof
04/21/2004EP1409122A2 Catalytic compositions and methods for asymmetric aldol reactions
04/21/2004EP1326846A4 Process for preparation of integrin receptor antagonist intermediates
04/21/2004EP1200387B1 Process for the cis-selective catalytic hydrogenation of cyclohexylidenamines
04/21/2004EP1154987B1 Phenylalaninol derivatives
04/20/2004US6723871 Asymmetric reduction of a beta-keto ester in the presence of a ruthenium-diamine complex
04/20/2004US6723868 Process for the preparation of aminoalcohol derivatives and their further conversion to (1R,4S)-4-((2-amino-6-chloro-5-formamido-4-pyrimidinyl)-amino)-2-cyclopentenyl-1-methanol
04/15/2004WO2004031198A1 Enantioselective reductive methods using chiral organostannanes
04/15/2004US20040072845 Enantiomers of 1-[ (4-chlorophenyl) phenylmethyl ] -4-[ (4-methylphenyl) sulfonyl] piperazine
04/15/2004US20040072680 Chiral phosphorus cyclic compounds for transition metal-catalyzed asymmetric reactions
04/15/2004DE10246740A1 Catalyst composition, useful for metal-catalyzed reactions e.g. asymmetric hydrogenation, comprises protein and interacting catalytic unit that includes a transition metal
04/14/2004EP1406860A1 Process for the preparation of 7-amino syn 3,5-dihydroxy heptanoic acid derivatives via 6-cyano syn 3,5-dihydroxy hexanoic acid derivatives
04/14/2004EP1305270B1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
04/14/2004EP1200419B1 Aminothiazole derivatives and their use as crf receptor ligands
04/14/2004CN1488760A Asymmetric synthesis method of antimer chiral silicon cyan aloohol
04/13/2004US6720454 Process for the cis-selective catalytic hydrogenation of cyclohexylidenamines
04/13/2004US6720439 Synthesis of ruthenium-hydride complexes and preparation procedures of chiral alcohols and ketones
04/13/2004US6720434 Process for preparing chiral compounds from recemic epoxides by using chiral salen catalysts
04/13/2004US6720357 Sulfonamide derivatives
04/13/2004US6720281 Chiral phosphorus ligands and the use thereof in the production of optically active products
04/08/2004WO2003097622A3 Synthesis of 2-alkylcysteines, 2-(hydroxylated phenyl)-4-alkylthiazoline-4-carboxylic acids and derivatives thereof
04/08/2004WO2003092578A3 Further syntheses of cyproterone acetate
04/08/2004US20040068140 Preparation of mandelic acid derivatives
04/08/2004US20040068126 Such as, hydrogenation, hydride transfer, allylic alkylation, hydrosilylation, hydroboration, hydrovinylation, hydroformylation, olefin metathesis, hydrocarboxylation, isomerization, cyclopropanation, Diels-Alder reaction, etc.
04/08/2004US20040068123 Introduction of t-butyldimethylsilyl(TBDMS) group as an alcohol protection group and construction of deprotection reaction condition not to produce by-products promise highly pure production of simvastatin
04/08/2004US20040068068 Optically active polymer with epoxide functions, method for preparing same, and use thereof
04/08/2004US20040067969 Syntheses of quinazolinones
04/08/2004US20040067928 Substituted propane-1,3-diamine derivatives and the pharmaceutical use thereof
04/07/2004EP1404700A2 Process for the production of 6,7-dihydroxy steroid compounds by allylic oxidation of steroid-5-ene compounds to steroid-5-ene-7-one compounds followed by hydroboration and oxidation and intermediates of this process
04/07/2004EP1404645A2 Method for producing optically active cyanohydrins and their corresponding acids
04/07/2004EP1404642A2 Synthesis and intermediates
04/07/2004EP1404639A1 Process for the preparation of intermediates useful in the synthesis of statin derivatives especially 7-amino 3,5-dihydroxy heptanoic acid derivatives, and intermediates thereof
04/07/2004EP1292602B1 New chiral salen catalyst and methods for the preparation of chiral compounds from racemic epoxides by using new catalyst
04/07/2004EP1131270B1 Process for converting an alcohol to the corresponding fluoride
04/07/2004CN1144878C Process for preparing optically pure (S)-3-hydroxy-gamma-butyrolactone
04/06/2004US6717011 Chiral diazaphospholidine ligands
04/06/2004US6716998 Such as (2r)-3,4-dihydro-2h-chromen-2-yl-methyl-4-methyl-benzenesulfonate; metathesis ring closing polymerization
04/01/2004WO2004026469A1 Active catalysts for stereoselective ring-opening reactions
04/01/2004WO2003095415A3 Aminated compounds bearing at least an allyl and a difluoromethyl and method used for synthesis thereof
04/01/2004US20040063999 Process for the production of optically active amino alcohols
04/01/2004CA2498893A1 Active catalysts for stereoselective ring-opening reactions
03/2004
03/31/2004EP1403262A1 Process for producing optically active alpha butyrolactone
03/31/2004EP1401803A2 Method for producing chiral amino acid derivatives
03/31/2004EP1401575A1 Hydroxylation of beta-dicarbonyls with zirconium catalysts
03/31/2004EP1299401B1 Chiral ligands for asymmetric catalysis
03/31/2004EP1289655A4 Novel chiral salen catalysts, and a process for preparing chiral compounds from racemic epoxides for using them
03/31/2004EP1282620B1 Azabicyclic carbamates and their use as alpha-7 nicotinic acetylcholine receptor agonists
03/31/2004EP1210324B1 Substituted cyclopentenes, their preparation and their use for chiral scaffolds
03/30/2004US6713652 Alkali metal or alkaline earth metal hydroxide in the presence of a polyol or amino alcohol
03/30/2004US6713435 Method for producing optically active lactone compounds by using salen cobalt complexes having a cis-β structure
03/25/2004WO2004024934A1 Process for producing optically active erythro 3-cyclohexylserines
03/25/2004WO2004024684A2 Enantioselective amination and etherification
1 ... 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 36 37 38 39 40 ... 63