Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
08/1981
08/04/1981CA1106388A1 Cyclic esters of 3,4-dihydroxy-thiophene-1,1-dioxide compounds and 3,4-dihydroxy-cyclopentadienone compounds
08/04/1981CA1106361A1 Peptide derivatives
07/1981
07/28/1981US4281180 Process for producing threo-3-amino-2-hydroxybutanoyl-aminoacetic acids, as well as novel intermediated therefor and process for producing them
07/28/1981CA1105926A1 L-pyroglutamyl-l-histidyl-glycine
07/28/1981CA1105924A1 Phenylalanine derivatives
07/21/1981US4279810 Easily split substrates for the quantification of proteases
07/14/1981US4278763 Indole or benzothiophene ester of amino acid or peptide
07/14/1981US4278762 Method for the quantitative determination of plasminogen activators
07/14/1981US4278595 Orally active MIF analogs with an effect on the central nervous system
07/14/1981CA1105006A1 Peptides
07/08/1981EP0031741A1 Substituted imino-acids, process for their preparation and their use as enzyme inhibitors
07/08/1981EP0031567A2 Tetrapeptidesemicarbazide derivatives and their production and use
07/07/1981US4277465 Enamine derivative
07/07/1981US4277395 Novel enzyme inhibitors
07/07/1981US4277394 Tetrapeptidehydrazide derivatives
07/01/1981EP0031104A1 Thiazolidine compounds, processes for their preparation and pharmaceutical compositions containing them
06/1981
06/30/1981US4276375 Contacting with chromogenic or fluorogenic substrate, spectrophotometry
06/30/1981US4276288 Dehydrooligopeptides, their production and their medicinal use
06/30/1981CA1104156A1 Analogues of bestatin
06/24/1981EP0030847A2 Pharmacologically active peptides, their preparation and pharmaceutical compositions containing them
06/24/1981EP0030845A2 Pharmacologically active peptides, their preparation and pharmaceutical compositions containing them
06/23/1981US4275153 Analytical fluorogenic substrates for proteolytic enzymes
06/23/1981US4275001 Process for the manufacture of LH-RH and LH-RH analogs using Glu-His(DnP)-OH
06/23/1981CA1103660A1 Carboxylic acid esters
06/16/1981US4273704 N-Adamantane-substituted tetrapeptide amides
06/16/1981CA1103239A1 Product and process for treating schizophrenia
06/10/1981EP0030076A1 Purification of L-aspartyl-L-phenylalanine alkyl esters
06/10/1981EP0029909A1 Process for the preparation of acid amides, use of the process and morpholino-ethyl isocyanide
06/03/1981EP0029488A1 Amino acid derivatives, process for their preparation and their use in treating hypertension
06/02/1981US4271068 Process for the manufacture of cystine-containing peptides
06/02/1981CA1102316A1 N su2 xx-arylsulfonyl-l-argininamides and the pharmaceutically acceptable salts thereof
05/1981
05/27/1981EP0029305A1 Process for the preparation of L-aspartic acid N-thiocarboxyanhydride
05/26/1981CA1101846A1 Derivatives of 4-hydroxy-phenylglycine
05/26/1981CA1101845A1 Addition compound of dipeptide derivative and amino acid derivative
05/26/1981CA1101844A1 Polypeptide
05/20/1981EP0028716A2 Motility increasing peptides and their use
05/20/1981EP0028627A1 Process for producing polypeptide alpha-thymosine and derivatives therefrom.
05/15/1981EP0034586A4 4-trifluoromethylcoumarin peptide derivatives and their use in proteinase assays.
05/12/1981US4267344 N-Substituted N-carboxyanhydrides of α-amino acids and their application in the preparation of peptides
05/12/1981CA1100948A2 Addition compound of dipeptide derivative and amino acid derivative
05/12/1981CA1100947A1 Psychopharmacologically active peptides and peptide derivatives, and the use thereof
05/12/1981CA1100944A1 Cephalosporins
05/05/1981US4265884 Therapeutically active polypeptides or acid addition salts thereof and a process for producing such compounds
05/05/1981US4265808 Pharmacologically active peptides
05/05/1981CA1100487A1 Process for the preparation of alpha-l-aspartyl-l- phenylalanine methyl ester
05/05/1981CA1100427A1 Process for recovering protease
04/1981
04/30/1981WO1981001145A1 Hydrolytic enzyme-activatible pro-drugs
04/28/1981US4264590 Antibacterial peptide
04/28/1981US4264491 Oligopeptide
04/22/1981EP0027319A2 Method for reductive elimination of protecting groups and preparative process using such method
04/22/1981EP0027260A2 Peptides, processes for their preparation and pharmaceutical compositions containing them
04/21/1981CA1099653A1 Process for recovering protease
04/15/1981EP0026867A1 Peptidylphosphonic acids, their preparation and use, and pharmaceutical preparations containing them
04/14/1981US4261979 Novel water-soluble compounds derived from extracts of streptomyces stimulosus, process for their production, their uses as immunological adjuvants and compositions containing them
04/14/1981US4261888 Organic compounds
04/14/1981US4261884 Desirable biological properties and stability to enzyme cleavage
04/14/1981US4261883 Novel N-aralkyl enkephalin amide analogs are provided having analgesic and opioid properties
04/08/1981EP0026464A2 Peptides, their production, their use, and pharmaceutical preparations
04/08/1981EP0026409A1 Combinations of active ingredients, pharmaceutical preparations, as well as their preparation
04/07/1981US4260682 High sensitivity assays for angiotensin converting enzyme
04/07/1981US4260601 Chemical compounds
04/07/1981CA1098850A1 Physiologically active peptides and a process for preparation thereof
04/01/1981EP0025842A2 Peptides, process for their preparation, their pharmaceutical compositions and their intermediates
03/1981
03/31/1981CA1098428A1 Specific chromogenic enzyme substrates
03/24/1981US4258193 For immobilization; immunoassay, crosslinking of proteins
03/24/1981US4258152 Pentapeptide modified resin
03/24/1981US4258151 Pentapeptide modified resin
03/24/1981US4257940 Valylleucyllysine derivatives, process for producing same and method for measuring activity of enzymes using same
03/24/1981US4257939 Substrates for determining enzyme activity
03/18/1981EP0025190A2 Chromogenic compounds and their use as enzymatic substrates
03/17/1981US4256897 Process for the preparation of L-aspartic acid N-thiocarboxyanhydride
03/17/1981US4256836 Reacting an n-substituted monoaminodicarboxylic acid with an amino carboxylic acid ester
03/17/1981US4256632 Novel derivatives of daunomycin
03/11/1981EP0024965A1 Fluorinated methyl beta-alanine derivatives, their preparation and pharmaceutical compositions containing them
03/11/1981EP0024739A2 Polyprenylpeptides and their production
03/11/1981EP0024664A1 Peptide amides and process for their preparation
03/03/1981US4254024 Tetrapeptides and derivatives having opiate activity
02/1981
02/24/1981US4252795 N-substituted dimeric cyclopeptide derivatives and preparation thereof
02/24/1981US4252715 Serine protease, oligopeptide for diagnostic determination of factor xa
02/17/1981US4251628 Hydrolysis of oligopeptides for radioisotope assay
02/17/1981US4251438 Piperazinone and piperazine polypeptides
02/10/1981US4250192 Novel substituted phenylacetic acid amide compounds
02/10/1981US4250183 Gastointestinal disorders; diseases of the pancreas, gall bladder, and liver
02/10/1981US4250086 Method and composition for preparation of H-SAR-LYS-SAR-GLN-NH2
02/10/1981US4250085 Phosphonate-containing oligopeptides, bactericides
02/03/1981US4248883 Antihypertension agents
02/03/1981CA1095040A1 N-substituted lactams
02/03/1981CA1095027A1 Dipeptide derivatives
01/1981
01/27/1981USRE30496 Tripeptide derivatives with central nervous system activity and preparation thereof
01/27/1981US4247454 Novel chromogenic thrombin substrates
01/27/1981US4247453 Folic acid derivatives for use in radioimmunoassay
01/20/1981CA1094052A1 Tetrapeptide amides and intermediates thereof
01/13/1981US4244947 Carba decapeptide derivatives of [TYR6 ]-somatostatin
01/13/1981US4244865 α hydroxy tripeptide substrates
01/07/1981EP0021766A2 Inhibitors of mammalian collagenase
01/07/1981EP0020481A1 Antibacterial peptide
01/06/1981USRE30473 Benzophenone glycinamide derivatives
01/06/1981US4243678 Gastrointestinal disorders, liver disorders
12/1980
12/30/1980US4242507 With n-hydroxybenzotriazoles and n-hydroxy oxo-substituted dihydrobenzotriazine, condensation agents
12/30/1980US4242329 Bradykinin-inhibiting tripeptide derivatives