Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
05/1984
05/15/1984US4448716 Dipeptide sweetener-metal complexes
05/15/1984US4448715 Tagged pyroglu-L-Phe-L-Arg derivatives, substrates and assays for kallikrein
05/09/1984EP0107907A2 Improvements in or relating to immunomodulating agents
05/09/1984EP0107860A1 Peptides, process for preparing the same and psychodepressant compositions containing the same
05/09/1984EP0028627B1 Process for producing polypeptide alpha-thymosine and derivatives therefrom
05/08/1984US4447419 Thiazole derivative, and pharmaceutical compositions containing it
05/08/1984CA1167044A1 Arylamine derivatives, production thereof and use thereof as microbicides
05/02/1984EP0107597A1 Chemical compounds and their use as sweetening agents
05/02/1984EP0107400A1 Hybrid plasmid and process for producing glutathione using said plasmid
05/02/1984EP0107095A1 1-N-alkylcarboxy-benzofused lactams useful as antihypertensive agents
04/1984
04/25/1984EP0106281A2 Analgesia-effecting 5-hydroxytryptophan derivatives
04/11/1984EP0105102A1 2-Aza-bicyclo(2,2,2)-octane-3-carboxylic-acid derivatives, process for their preparation, pharmaceutical preparations containing them and their application, and 2-aza-bicyclo(2,2,2)-octane-3-carboxylic acid as an intermediate and its preparation
04/10/1984US4442030 Process for preparing carboxyalkyl dipeptides
04/10/1984US4442029 Peptide synthesis using an isonitrile as activator
04/04/1984EP0104964A1 Peptide derivatives as inhibitors of acid proteases
04/04/1984EP0104546A2 Therapeutic dipeptides
04/04/1984EP0104461A2 Process for preparing antihypertensive 1-substituted cyclic lactam-2-carboxylic acids and their derivatives
04/03/1984US4440941 Aroyl-aminoacids, amides and esters thereof
04/03/1984US4440692 Adamantanyl-, blocking agent in peptide synthesis
04/03/1984US4440678 Tripeptide derivatives and their application in assaying enzymes
04/03/1984US4440677 Method and intermediates for producing α-L-aspartyl-L-phenylalanine
04/03/1984US4440676 Pentacoordinate phosphorane coupling agents
03/1984
03/28/1984EP0104041A1 Enzyme inhibitors
03/28/1984EP0103867A1 Phosphorus-containing peptide derivative
03/27/1984US4439460 Dipeptide sweetener sulfate and sulfonate salts
03/27/1984US4439425 Peptide derivatives
03/27/1984US4439364 Process for preparing antihypertensive 1-substituted cyclic lactam-2-carboxylic acids and their derivatives
03/27/1984US4439360 Retro-inverso analogues of C-terminal penta and hexapeptides of Substance P
03/21/1984EP0103077A2 Substituted dipeptides, methods for their production, pharmaceutical compositions containing them, method for making such pharmaceutical compositions
03/20/1984US4438270 α-Halomethyl derivatives of α-amino acids
03/20/1984US4438125 Arylamine derivatives and use as microbicides
03/20/1984US4438103 Organic compounds
03/20/1984US4438031 N-(Alkylsulfonyl)-L-proline amide and N-(alkylsulfonyl)-2-carboxylic acid amide-indoline derivatives
03/20/1984US4438029 Synthetic peptides
03/14/1984EP0102529A2 Process for preparation of aspartylphenylalanine alkyl esters
03/14/1984EP0102483A1 Process for preparing alpha-l-aspartyl-l-phenylalanine alkyl esters
03/13/1984US4436925 Addition compound of dipeptide derivative and amino acid derivative
03/13/1984US4436918 From a 2,5-dioxopyrrolidine compound
03/13/1984US4436726 N-Acylpeptide compound, processes for the preparation thereof and the pharmaceutical compositions
03/07/1984EP0102216A2 Biosynthesis of unnatural cephalosporins
02/1984
02/28/1984US4434151 Bifunctional chelating agents
02/28/1984US4434097 Process for the removal of the formyl group from N-formyl peptides and esters thereof
02/28/1984US4434096 Substrates for the quantitative determination of proteolytic enzymes
02/28/1984US4434095 Cyclic analogue of naturally-occurring phagocytosis-stimulant peptide - threonyl-cyclo-[-N.sup.ε -lysyl-prolyl-arginyl]
02/28/1984CA1162848A1 Method for enzyme immunoassay and peptide-enzyme conjugate and antibody therefor
02/21/1984US4432896 Detection of carboxypeptidase
02/14/1984US4431645 Antihypertensive agents
02/14/1984US4431644 Antihypertensive agents
02/14/1984US4431438 Herbicides
02/08/1984EP0099960A1 Process for the preparation of lower alkyl esters of N-L-alpha-aspartyl-L-phenyl alanine, and intermediates for their manufacture
02/07/1984CA1161839A1 Branched amides of l-aspartyl-d-amino acid dipeptides
02/07/1984CA1161838A1 Enkephalin derivatives
02/02/1984WO1984000365A1 Synthetic peptides and their preparation
02/01/1984EP0099855A1 Process for the preparation of a dipeptide ester from L-aspartic acid
02/01/1984EP0099709A2 Amide derivatives
02/01/1984EP0099585A1 Process for producing an addition compound of a dipeptide ester and an amino acid ester
01/1984
01/31/1984US4428940 Anti-hypertensive compounds and compositions
01/31/1984US4428938 Peptides affecting the immune regulation and a process for their preparation
01/31/1984US4428875 Compounds of dichlorodiethylaminophenylalanine with anti-tumor activity
01/31/1984US4428874 Tripeptide derivatives
01/31/1984CA1161451A1 .alpha.-ACETYLENIC AMINO ACIDS
01/31/1984CA1161450A1 Fluorinated methyl beta-alanine derivatives
01/31/1984CA1161432A1 Tripeptide derivatives and their application in assaying enzymes
01/31/1984CA1161431A1 Tripeptide derivatives
01/31/1984CA1161381A1 PROCESS FOR ESTERIFICATION OF .alpha.-L-ASPARTYL-L- PHENYLALANINE
01/25/1984EP0099286A1 Compound containing a tripeptide sequence of the threonyl-lysyl proline-type, or similar, useful as an anti-inflammatory, anti-allergic or antalgesic agent
01/25/1984EP0099057A2 N-acyl derivatives of peptides, their manufacture and use in combating diseases and means therefor
01/25/1984EP0099056A2 N-acyl derivatives of dipeptides, their manufacture and use in treating diseases, and means therefor
01/24/1984US4427660 Formyl-methionyl chemotatic peptide antibiotic conjugates useful in treating infections
01/24/1984US4427582 Antimicrobial disulfide prodrugs
01/24/1984US4427581 Peptide, process for preparation thereof and use thereof
01/24/1984CA1160973A1 Process for enzymatic production of peptides
01/19/1984WO1984000108A1 Compound containing a tripeptidic sequence of the threonyl-lysyl-proline type or the like, usable as an anti-inflammatory, anti-allergic or antalgic agent
01/18/1984EP0098520A1 L-alanyl-D-isoglutaminyl-adamantyl amide, process for its preparation and pharmaceutical compositions containing this compound
01/18/1984EP0098457A2 (1S,2R,3R)- and (1R,2S,3S)-nitrilo-1-carbonyl-3-methyl-2-oxy-heptanes and -hept-5-enes useful in the total synthesis of cyclosporins and processes for their production
01/18/1984EP0098456A2 Peptides comprising a (1S,2R,3R)- or (1R,2S,3S)-1-nitrilo-1-carbonyl-3-methyl-2-oxy-heptane or -hept-5-ene residue useful in the total synthesis of cyclosporins, and processes for their production
01/17/1984US4426532 α-(3-Cyano-propanoyl)-aminocarboxylic acid derivatives
01/17/1984US4426453 Derivatives of iodothyronine compounds and their use in an assay for the free iodothyronine compounds
01/17/1984US4426325 Process for the preparation of compounds containing carboxylic acid amide groups, in particular or peptides
01/17/1984US4426324 Immunopotentiating peptides
01/11/1984EP0097994A2 Method for the solid-phase synthesis of retro-inverso polypeptides
01/10/1984US4425333 Sulfur-containing acylamino acids
01/03/1984US4424354 Inhibitors of mammalian collagenase
01/03/1984US4424207 Enzyme inhibitors
12/1983
12/28/1983EP0097070A2 Process for preparing ellipticine derivatives, compounds so obtained and medicaments containing them
12/28/1983EP0096689A1 Method and reagent for detection of endotoxines or beta-1,3 glucanes from fungus or bacteria
12/27/1983US4423029 (S)-3-Amino-4-[(S,S)-1-(1-hydroxyethyl)alkyl amino]-4-oxo-butyric acid compounds suitable as non-nutritive sweetners
12/21/1983EP0096157A2 Substituted acyl derivatives of 1,2,3,4-tetrahydro-6,7-dimethoxy-3-isoquinolinecarboxylic acid
12/20/1983US4421765 Antiinflammatory agents
12/20/1983US4421745 Peptide
12/20/1983US4421744 Aminoacyl derivatives
12/13/1983US4420490 Substituted phenylacetic acid amide compounds
12/13/1983CA1158641A1 Anticoagulant agmatine derivatives and process for the preparation thereof
12/13/1983CA1158640A1 Therapeutically active polypeptides or acid addition salts and a process for producing such compounds
12/13/1983CA1158557A1 Hydrolytic enzyme-activatible pro-drugs
12/07/1983EP0095772A1 Dipetide sweetener sulfate and sulfonate salts
12/07/1983EP0095584A2 Substituted 4-phenoxy and 4-phenylthio prolines
12/07/1983EP0095557A1 Polypeptides with an antagonistic activity on substance P, process for their preparation, their use and process for the purification of polypeptides
12/06/1983CA1158237A1 Peptide amides and process for their manufacture
12/06/1983CA1158236A1 Process for the preparation of novel substituted phenylacetic acid amide compounds