Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
12/1985
12/03/1985US4556655 Antihypertensive compounds having both diuretic and angiotensin converting enzyme inhibitory activity
12/03/1985US4556652 Inhibitors of angiotensin, diuretics, treatment of congestive heart failure
11/1985
11/27/1985EP0162813A2 Pharmaceutical compositions containing a dipeptide
11/27/1985EP0162422A2 The novel physiologically active substance foroxymithine, a process and microorganisms for its production and its use as medicament
11/27/1985EP0162079A1 Use of arg-phe-amide derivatives
11/26/1985US4555511 Thieno [3,2,C]pyridines useful as antihypertensives
11/26/1985US4555508 Antihypertensive spiro-cyclic compounds
11/26/1985US4555503 N2 -(Substituted)carboxymethyl-N6 -(substituted)-lysyl-and αε-aminoalkyl)glycyl amino acid antihypertensive agents
11/26/1985US4555502 Aminoacyl-containing dipeptide derivatives useful as antihypertensives
11/26/1985US4555362 Method and intermediates for producing α-L-aspartyl-L-phenylalanine
11/26/1985CA1197165A1 Synthetic substrate and assay method of enzyme activity
11/21/1985WO1985005104A1 Fused 7-membered ring compounds and process for their preparation
11/21/1985EP0161801A2 Perhydrothiazepine derivatives, their preparation and their therapeutic use
11/21/1985EP0161588A2 Diamino acid derivatives
11/19/1985US4554351 Method for the total synthesis of cyclosporins, novel cyclosporins and novel intermediates and methods for their production
11/19/1985US4554289 Enzyme inhibitors, immunomodulators, antinflammatory agents
11/19/1985US4554272 Cholecystokinin inhibitors
11/19/1985US4554102 Cyanohydrination catalyst comprising non-crystalline or amorphous dipeptide
11/19/1985US4554100 Alkylamides of carboxyalkanoyl peptides and method for preparation thereof
11/19/1985CA1196911A1 Process for the preparation of compounds containing carboxylic acid amide groups, in particular of peptides
11/13/1985EP0161195A1 Method for the immunological determination of monoamines
11/13/1985EP0161017A1 Peptides
11/13/1985EP0161007A2 Retro - inverso C-Terminal hexapeptide analogues of substance P
11/12/1985US4552866 Use of diamino alcohols as analgesic agents
11/12/1985CA1196636A1 Benzazepin-2-ones
11/06/1985EP0048763B1 Sulfur-containing acylamino acids
11/05/1985US4551272 Derivatives of dipeptide and their use in determining the activity of carboxypeptidase A
10/1985
10/30/1985EP0159396A2 Carboxyalkyl peptide derivatives
10/29/1985US4549987 Aspartame synthesis
10/24/1985WO1985004657A1 Fused 7-membered ring compounds and process for their preparation
10/23/1985EP0159156A1 Hydroxy substituted ureido amino and imino acids
10/23/1985EP0159004A2 Antibiotics do-248-A and B and process for preparing the same
10/23/1985EP0158947A2 Amino thiol dipeptides
10/23/1985EP0158927A2 Process for the treatment of heart failure
10/23/1985EP0158843A1 A N-(6-substituted pyridine-2-carbonyl)-3-substituted histidine derivative, a method of preparing the same and its use as an anti-tumor agent
10/22/1985US4548932 3-Amino-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine derivatives
10/22/1985US4548926 Hypotensive peptides and their use
10/15/1985CA1195272A1 Process for preparation of aspartylphenylalanine alkyl esters
10/10/1985WO1985004408A1 Antibiotic tan-588, process for its preparation, and novel strainbelonging to genus empedobacter
10/10/1985WO1985004402A1 Fused 7-membered ring compounds and process for their preparation
10/09/1985EP0157753A1 New somatostatin compounds, process for their synthesis, preparation for veterinary use containing said compound and process for the treatment of animals
10/09/1985EP0157572A2 Acyltripeptide immunostimulants
10/09/1985EP0157409A2 Renin inhibitors containing 2-substituted statine
10/09/1985EP0157384A2 Substrates for hydrolases, process for their preparation and their use
10/02/1985EP0156455A2 Condensed seven-membered ring compounds, their production and use
10/02/1985EP0156322A2 Renin inhibitors containing peptide isosteres
10/02/1985EP0156321A2 Renin inhibitory peptides having improved solubility
10/02/1985EP0156320A2 Renin inhibitors containing homophe 8 and a C-terminal amide cycle
10/02/1985EP0156319A2 Renin inhibitors containing homophe 8
10/02/1985EP0156318A2 C-terminal amide cyclic renin inhibitors containing peptide isosteres
10/02/1985EP0156280A2 Process for the preparation of peptide intermediates poor in racemates, belonging to gonadorelin and gonadorelin analogues, their synthesis and intermediates obtained by this process
10/02/1985EP0156279A2 A novel process for the preparation of bestatin derivatives and intermediates thereof
10/02/1985EP0156063A2 Hypoglycaemic tetrapeptides
09/1985
09/25/1985EP0155809A2 Renin inhibitors containing statine or derivatives thereof
09/24/1985US4543350 Carcinostatic agent
09/18/1985EP0155165A2 Process for introducing phosphinoyl groups into amino groups
09/18/1985EP0154904A1 Acylamino oxo or hydroxy substituted alkylamino thiazines and thiazepines
09/18/1985EP0154886A2 Carboxyalkyl dipeptide derivatives, process for their preparation, agents containing them, and their use
09/12/1985WO1985003874A1 Method of treating depression in vertebrates
09/12/1985WO1985003873A1 Method of treating hypertension in vertebrates
09/12/1985WO1985003872A1 Method of lowering blood sugar level in vertebrates
09/12/1985WO1985003871A1 Method of prophylaxis or treatment of atherosclerosis
09/12/1985WO1985003870A1 A method of treating hypoglycemia in vertebrates
09/12/1985WO1985003869A1 Method of treating memory disorders of the elderly
09/11/1985EP0154472A2 Process for the production of L-aspartyl-L-phenylalanine ester
09/11/1985EP0154234A2 Substituted tyrosil alanine dipeptide amides
09/11/1985EP0153992A2 Water soluble derivatives of 3,5-diaceto amido-2,4,6-triiodobenzoic acid and process for their preparation and use
09/10/1985US4540682 Pharmaceutical peptides, preparation, use and intermediates
09/03/1985US4539312 Use of diamino ketones as analgesic agents
09/03/1985US4539155 New peptide, process for preparation thereof and use thereof
09/03/1985US4539147 3,5-dimethoxy-2,2-dimethylbenzyloxycarbonyl group to protect amine of aspartic acid
08/1985
08/27/1985US4537885 Substituted 1-carboxy-3-(carboxymethylamino)-2-one derivatives, angiotensin converting enzyme inhibitors
08/27/1985US4537714 Process for the preparation of lower alkyl esters of N-L-α-aspartyl-L-phenylalanine and of new intermediates for their preparation
08/27/1985US4537713 Process for the reduction of reducible groups and its use
08/21/1985EP0152255A2 New renin-inhibitory peptides and their use
08/21/1985EP0093128B1 Process for preparing of methyl ester of alpha-aspartyl phenyl alanine
08/20/1985US4536501 Angiotensin inhibitor diuretic, hypotensive agent
08/20/1985US4536476 From prokaryotic beta-lactam producing organism
08/20/1985US4536395 Amino acid derivatives and antihypertensive drugs containing them
08/20/1985CA1192078A1 Dipeptide sweetener sulfate and sulfonate salts
08/13/1985US4535176 Intermediates for substituted peptide compounds
08/13/1985US4534897 Drying on heated roll, controlled cooling below dew point
08/13/1985CA1191839A1 Branched amides of l-aspartyl-d-amino acid dipeptides
08/07/1985EP0150263A1 Derivatives of cis, endo-2-azabicyclo-[3.3.0]-octane-3-carboxylic acid, process for their preparation, medicaments containing them, and their use
08/07/1985EP0150227A1 Dipeptide derivatives and their use in determining the activity of carboxypeptidase A
08/06/1985US4533747 Leukotriene antagonists intermediates
08/06/1985US4533661 Certain 3-phosphinyl-amino-2-oxo-1H-azepine-1-acetic acid derivatives having anti-hypertensive activity
08/06/1985US4533657 Analgesic dipeptide amides and method of use and composition thereof
08/06/1985US4533656 Amide derivatives
08/06/1985US4533655 Analgesic dipeptide amides and method of use and compositions thereof
08/01/1985WO1985003301A1 Process for preparing aspartyl peptides and new aspartyc acid derivatives usable in the synthesis thereof
07/1985
07/31/1985EP0149615A1 New oligopeptide aldehydes useful as specific inhibitors of enterokinase
07/30/1985CA1191139A1 Aroyl amino acids
07/24/1985EP0149594A2 Enzymatic coupling of n-formyl amino acids and/or peptide residues
07/24/1985EP0149582A2 Process for the preparation of aspartyl peptides and derivatives of aspartic acid useful in their synthesis
07/24/1985EP0149263A2 Process for preparing alpha-L-aspartyl-L-phenylalanine methyl ester
07/23/1985US4530837 Containing tryptophan
07/23/1985US4530836 Containing tryptophan and methionine
07/16/1985US4529810 Preparation of optically-active alpha-substituted carboxylic esters and acids
07/10/1985EP0148133A2 Tripeptide compounds containing pyroglutamic acid and tryptophan, process for their production and therapeutic applications