Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
10/2002
10/01/2002US6458948 Process for producing carboxylic acid derivative and condensing agent comprising quaternary ammonium salt
10/01/2002US6458785 Aids therapy
10/01/2002US6458769 Amorphous lisinopril having the formula (s)-1-(n.sup.2 -(1-carboxy-3-phenylpropyl))-l-lysyl)-l-proline, wherein amorphous lisinopril has a glass transition point (tg) when dry, measured by thermal mehanical analysis
10/01/2002US6458767 Use of peptides inhibitory for thrombospondin dependent TGF-β activation in the treatment of kidney disease
10/01/2002US6458760 Comprising administering to said patient a therapeutically effective amount of a compound which is a specific inhibitor of either cathepsin b or cathepsin l, but which is not as effective inhibitor of calpain
10/01/2002US6458349 For treatment of leukemia, tumors, chronic infections, autoimmune disease, fibrotic disorders, psoriasis; for wound healing
10/01/2002CA2210258C Substituted oxazolidine calpain and/or cathepsin b inhibitors
10/01/2002CA2168113C Therapeutic peptide derivatives
10/01/2002CA2124087C Combinatorial strategies for polymer synthesis
10/01/2002CA2069256C Method of preparing .alpha.-l-aspartyl-l-phenylalanine methyl ester
09/2002
09/26/2002WO2002074792A1 Fo-6979 substances and process for producing the same
09/26/2002WO2002074761A1 Substituted n-arylsulfonyl-proline derivatives as potent cell adhesion inhibitors
09/26/2002WO2002074293A2 Methods for restoring cognitive function following systemic stress
09/26/2002WO2002074050A2 Asymmetric synthesis of (s, s, r)-(-)-actinonin and its analogs and uses therefor
09/26/2002WO2002036173A3 Simultaneous dual isotope imaging of cardiac perfusion and cardiac inflammation
09/26/2002WO2002030922A3 Dioxolane analogs for improved inter-cellular delivery
09/26/2002WO1997019953A8 New lh-rh antagonists with improved effectiveness
09/26/2002US20020137942 HIV protease inhibitors; administering to treat AIDS (acquired immune deficiency syndrome)
09/26/2002US20020137730 Positively charged non-natural amino acids, methods of making and using thereof in peptides
09/26/2002US20020137687 Novel compounds that inhibit tryptase activity
09/26/2002US20020137686 Inhibitors of the ICE/ced-3 family of cysteine proteases
09/26/2002US20020137672 Radiolabeled annexins
09/26/2002US20020137177 One or more amino acid residues being replaced by cysteine residues where at least some of cysteine residues are modified by replacing thiol hydrogen in cysteine residue with thiol side chain to form modified enzyme
09/26/2002CA2442717A1 Methods for restoring cognitive function following systemic stress
09/26/2002CA2441822A1 Asymmetric synthesis of (s, s, r)-(-)-actinonin and its analogs and uses therefor
09/25/2002EP1243594A1 Process for crystallizing N2-((S)-1-ethoxycarbonyl-3-phenylpropyl)-N6-trifluoroacetyl-L-lysyl-L-proline
09/25/2002EP1242365A1 Acyl pseudodipeptides which carry a functionalised auxiliary arm
09/25/2002EP1242363A2 Cd45 inhibitors
09/25/2002EP1242070A2 Treatment of ischemic brain injuries with brain targetted antioxidant compounds
09/25/2002EP0871656B1 Dolastatin derivatives, their preparation and use
09/25/2002CN1371388A Hexapeptide with stabilized disulfide bond and derivatives thereof regulating metabolism, proliferation differentiation and apoptosis
09/25/2002CN1371286A Use of cyclooxygenase-2 inhibitor matrix metallappoteinase inhibitor antineoplastic agent and optionally radiation as combination treatment of neoplasia
09/25/2002CN1370778A Beta-tetrahydro carboline carboxylic acid, its RGD conjugate, their synthesis and medical application
09/24/2002US6455705 Distillation-free; chemical intermediates for the production of angiotensin-converting enzyme (ace) inhibitors
09/24/2002US6455671 Thrombin inhibitors, the preparation and use thereof
09/24/2002US6455581 Inhibitors of hiv protease.
09/24/2002US6455500 Radiation therapy methods
09/24/2002US6455244 Methods for the detection of antibodies associated with autoimmune disorders and infectious agents employing immunoretroid peptides derived from antigens associated with said disorders and agents
09/24/2002CA2096223C Treatment for tissue ulceration
09/19/2002WO2002073208A2 Anti-epileptogenic agents
09/19/2002WO2002072629A1 Immunopotentiators
09/19/2002WO2002072618A1 Novel peptide ligands of leukocyte integrins
09/19/2002WO2002072617A1 Thiopeptide compounds
09/19/2002WO2002072616A2 Transfection complexes
09/19/2002WO2002072609A2 Neuroactive peptides for prevention and/or treatment of hypoxia and neuropathic pain
09/19/2002WO2002072151A1 Enzyme-activated cytostatic conjugates with integrin ligands
09/19/2002WO2002018341A3 Quinoline- (c=o) - (di-, tri- and tetrapeptide) derivatives as caspase inhibitors
09/19/2002WO2001025264A9 Substituted phosphinate based peptide derivatives
09/19/2002US20020133037 Artificial sweetener
09/19/2002US20020133001 Therapeutic agents and methods of use thereof for treating an amyloidogenic disease
09/19/2002US20020132779 Analogs of L-Glu-L-Trp having pharmacological activity
09/19/2002US20020132776 Inhibitors of transglutaminase
09/19/2002US20020132765 Powerful activity when administered orally and by injection so that they can be used in a hospital environment via injection, followed by an oral ambulatory treatment
09/19/2002US20020132300 Specific inhibitors of NFAT activation by calcineurin and their use in treating immune-related diseases
09/19/2002US20020132032 Alkylating aspartame with a benzene or benzodioxole aldehyde to produce a aspartyl dipeptide ester derivative; food or drink sweeteners
09/19/2002CA2470152A1 Transfection complexes comprising a novel peptide as cell surface receptor binding component
09/19/2002CA2441210A1 Novel peptide ligands of leukocyte integrins
09/19/2002CA2440834A1 Anti-epileptogenic agents
09/19/2002CA2440353A1 Thiopeptide compounds
09/19/2002CA2439897A1 Enzyme-activated cytostatic conjugates with integrin ligands
09/19/2002CA2439236A1 Immuno-enhancing agent
09/18/2002EP1240193A2 Peptide fragments of colostrinin
09/18/2002EP1240169A1 Peptide beta-turn mimetic compounds and processes for making them
09/18/2002EP1240152A1 Ox(adi)azolyl-hydroxamic acids useful as procollagen c-proteinase inhibitors
09/18/2002EP1239877A2 MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN $g(a) V?$g(b) 3? RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
09/18/2002CN1370181A Effectors of dipeptidyl peptidase IV for topical use
09/18/2002CN1370078A Prion protein peptides and uses thereof
09/17/2002US6451972 Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors
09/17/2002US6451971 Polypeptide cell adhesion inhibitors; antimetastasis and anticarcinogenic agents
09/17/2002US6451968 Hoogsteen type base pairing in triplex motif; diagnosis; heat resistance; detection of point mutations, restriction enzyme sites, and transcription inhibition
09/17/2002US6451853 Small molecules that elicit a polarized Th1 response and for modulation of cellular immunity
09/17/2002US6451761 N′N′-dichlorinated omega-amino acids and uses thereof
09/17/2002US6451760 Treatment of inflammation using a 2F1 polypeptide or an antibody thereto
09/17/2002CA2129976C Peptidyl derivatives as inhibitors of interleukin-1.beta. converting enzyme
09/12/2002WO2002070545A2 Siderophore analogues as tetra- or hexadentate iron chelators on the basis of amino acids or peptides, method for producing them and the use thereof
09/12/2002WO2002070511A1 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
09/12/2002WO2002070493A1 Bisaryl derivatives having fsh receptor modulatory activity
09/12/2002WO2002070018A2 Tetradentate peptide-chelate conjugates for colorectal cancer diagnosis
09/12/2002WO2002069905A2 Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-amp associated disorders
09/12/2002WO2002069884A2 A sunburn treatment and sunburn prevention method
09/12/2002WO2002050100A3 Diaminodicarboxylic acid: peptide-based gemini surfactant compounds used for drug delivery
09/12/2002WO2001016372A9 Methods of immobilizing ligands on solid supports and apparatus and methods of use therefor
09/12/2002US20020128473 Derivatives of octahydro-6, 10-dioxo-6H-pyridazino(1,2-a)(1,2)diazepine-1-carboxylic acid, useful for preperation of therapeutically active compounds
09/12/2002US20020128306 Programmed cell death; expansion of hematopoietic cells, for prolonging viability of an organ for transplantation, and maintaining viability of cell lines used in bioproduction
09/12/2002US20020128206 Such as 6-Amino-2-(2-((1-benzenesulfonyl-piperidine-4-carbonyl)-amino)-3-(1H-indol-3-yl)-propionylamino)-hexanoic acid tert-butyl ester for promotes secretion of growth hormone; gene expression
09/12/2002US20020127629 Imaging of enzymatic activity
09/12/2002US20020127320 Subjecting a 2-hydroxychroman compound and aspartame to a reductive alkylation reaction to produce N-(N-(3-(2-hydroxy-substituted phenyl)propyl)-L- alpha -aspartyl)-L-phenylalanine 1-methyl ester compound
09/12/2002CA2439691A1 Co-administration of melanocortin receptor agonist and phosphodiesterase inhibitor for treatment of cyclic-amp associated disorders
09/12/2002CA2439579A1 Tetradentate peptide-chelate conjugates for colorectal cancer diagnosis
09/12/2002CA2437594A1 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
09/12/2002CA2434184A1 Bisaryl derivatives having fsh receptor modulatory activity
09/11/2002EP1239037A1 PROCESS FOR PRODUCING KiSS-1 PEPTIDE
09/11/2002EP1238678A1 Enzyme-activated cytostatic conjugates with integrin ligands
09/11/2002EP1237878A2 4-pyrimidinyl-n-acyl-l-phenylalanines
09/11/2002EP1054892B1 Azole peptidomimetics as thrombin receptor antagonists
09/11/2002EP0853484B1 Novel mu opioid receptor ligands: agonists and antagonists
09/11/2002EP0603399B1 Endothelin-antagonizing peptide
09/11/2002CN1369015A Recombinant anti-CD 40 antibody and uses thereof
09/11/2002CN1090637C Cross-link cinnamic acid derivative and its preparation method
09/11/2002CN1090508C Storage stable water solution for infusion containing thrombin inhibitor