Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
01/2003
01/30/2003WO2003007686A2 Use of copper chelators to inhibit the inactivation of protein c
01/30/2003WO2002048180A3 Peptides and/or proteins and use thereof for the production of a therapeutic and/or prophylactic medicament
01/30/2003WO2002045523A3 Protein hydrolysates enriched in peptides having a carboxy terminal proline residue
01/30/2003US20030023104 For prolonging or altering the activity of a compound which is a member of the chlorambucil family
01/30/2003CA2454418A1 Compositions and methods for use of bioactive agents derived from sulfated and sulfonated amino acids
01/30/2003CA2453987A1 Dolastatin 10 derivatives
01/30/2003CA2452322A1 Inhibitors of the ice/ced-3 family of cysteine proteases
01/29/2003EP1279665A2 A process for the preparation of perindopril, its analogous compounds and salts thereof using 2,5-dioxo-oxazolidine intermediate compounds
01/29/2003EP0910573B1 New amino acid derivatives and their use as thrombin inhibitors
01/29/2003CN1394199A Peptide derivatives and their pharmaceutically acceptable salts, processes for preparation of both, and use thereof
01/28/2003US6512111 A method for preparing compounds of formula (I) ) wherein cyclization is carried out in a basic medium and in the presence of a phosphonic acid derivative and the use of said method as an intermediate step for preparing a compound
01/28/2003US6512092 Solid phase peptide synthesis; in situ generation of amino acid chloride by deblocking; coupling sterically hindered amino acid residues
01/28/2003US6512001 D-proline derivatives
01/28/2003US6511663 Tri- and tetra-valent monospecific antigen-binding proteins
01/28/2003US6511648 Vitronectin receptor antagonist pharmaceuticals
01/28/2003CA2124375C Compounds containing a fused bicyclic ring and processes therefor
01/28/2003CA2110556C The elucidation and synthesis of antineoplastic tetrapeptide phenylamides of dolastatin 10
01/28/2003CA2110555C Tumor inhibiting tetrapeptide bearing modified phenethyl amides
01/23/2003WO2003006620A2 Linear and cyclic melanocortin receptor-specific peptides
01/23/2003WO2003006492A2 Biologically active peptides
01/23/2003WO2003006490A1 Bridged bicyclic serine protease inhibitors
01/23/2003WO2003006489A2 Prodrugs of excitatory amino acids
01/23/2003WO2003006444A2 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
01/23/2003WO2003006021A1 Alpha-hydroxyamide statine derivatives for the treatment of alzh eimer's disease
01/23/2003WO2002026775A3 Compositions and methods for regulating apoptosis
01/23/2003US20030018193 Beta-alanine derivatives and their use as receptor anatgonists
01/23/2003US20030018163 Acylation, amidation; using amine scavenger
01/23/2003US20030017996 Antilipemic agents, anticholesterol agents, cardiovascular disorders
01/23/2003US20030017995 Dialysis solutions and methods
01/23/2003US20030017993 Carbamyloxy compounds which inhibit leukocyte adhesion mediated by VLA-4
01/23/2003US20030017992 Crystalline forms
01/23/2003US20030017991 Substrates and assays for beta-secretase activity
01/23/2003US20030017990 Antiinflammatory agents, rheumatic diseases, antiarthritic agents, inflammatory bowel disorders
01/23/2003US20030017976 Anticancer agents; side effect reduction
01/23/2003US20030017964 Administration of agents via the PEPT-2 transporter
01/23/2003US20030017520 High-efficiency assay for protein mannosyl transferases
01/23/2003US20030017245 Novel aspartame powders
01/23/2003CA2707767A1 Biologically active peptides
01/23/2003CA2453515A1 Linear and cyclic melanocortin receptor-specific peptides
01/23/2003CA2453447A1 Alpha-hydroxyamide statine derivatives for the treatment of alzheimer's disease
01/23/2003CA2453169A1 Substituted amides, sulfonamides and ureas useful for inhibiting kinase activity
01/23/2003CA2452417A1 Compositions comprising the biologicially active peptide ysl
01/23/2003CA2449504A1 Bridged bicyclic serine protease inhibitors
01/22/2003EP1277761A2 Process for the preparation of peptides
01/22/2003EP1276758A2 A glycopeptide and preparation thereof
01/22/2003EP1276746A2 Process for preparing lipid ii and derivatives thereof
01/22/2003EP1276718A2 Small technetium-99m and rhenium labeled agents and methods for imaging tumors
01/22/2003EP1276491A1 Tamandarin and didemnin analogs and methods of making and using them
01/22/2003EP1107980B1 CRYSTALLINE FORMS OF EtO2C-CH2-(R)Cgl-Aze-Pab-OH
01/22/2003EP1030835B1 Urea derivatives and their use as integrin inhibitors
01/22/2003EP0865339B1 Metalloproteinase inhibitors
01/22/2003CN1392157A New anti-embolism medicine using small peptide arginine-glycine-aspartic acid (RGD) as leading compound
01/22/2003CN1392156A Synthesizing method for propyl-glutdipeptide
01/22/2003CN1099425C 新的肽衍生物 New peptide derivatives
01/21/2003US6509446 Recombinant genetic information (DNA or RNA), consisting a Chicken Anemia Virus (CAV)-specific nucleotide sequence, useful for diagonestics, vaccination or protein production
01/21/2003US6509330 Angiotensin converting enzyme (ACE); neutral endopeptidase (NEP); containing a dipeptide derived from an amino acid, or a conformationally restricted dipeptide mimic
01/21/2003US6509315 Didemnin analogs and fragments and methods of making and using them
01/21/2003US6509165 Detecting the ability of proinsulin peptide to preferentially stimulate the T-cells of diabetic subjects by measuring the ability of the T-cells to proliferate or ability of the T-cells to produce cytokines
01/21/2003US6509100 Fluorinated hydrogn bond stabilized surface modifying agents, articles made therefrom, methods for making and using the same
01/16/2003WO2003004517A2 Peyers's patch and/or m-celle targeting ligands
01/16/2003WO2003004516A1 Novel chromogenic substances and use thereof for the determination of carboxypeptidase activities
01/16/2003WO2002055185A3 Block copolymers for multifunctional self-assembled systems
01/16/2003WO2002031109A3 Intracellular delivery of biological effectors by novel transporter peptide sequences
01/16/2003WO2002012196A3 Lactam compounds and their use as inhibitors of serine proteases and method
01/16/2003US20030013881 Such as 4-((6-(3,5-difluoro-phenyl)-5-(S)-(3-dipropylcarb-amoyl-benzoyl-amino)-2-(R)-ethyl-4-(S)-hydroxy-hexanoylamino)-methyl)-cyclohexanecarboxylic acid for inhibiting secretase activity and cleavage of amyloid precursor protein
01/16/2003US20030013847 Pyruvate derivatives
01/16/2003US20030013846 Cytoprotective agents
01/16/2003US20030013725 Amino acid derivatives
01/16/2003US20030013700 Thrombin inhibitors
01/16/2003US20030013677 Anticancer agents
01/16/2003US20030013660 Dioxolane analogs for improved inter-cellular delivery
01/16/2003US20030013658 Small peptides and methods for treatment of asthma and inflammation
01/16/2003US20030013657 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
01/16/2003US20030013656 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
01/16/2003US20030012817 Modified amino acids and derivatives can form non-covalent mixtures with active biological agents and in an alternate embodiment can releasably carry active agents. Modified amino acids can also form drug containing microspheres.
01/16/2003CA2451741A1 Peyers's patch and/or m-celle targeting ligands
01/16/2003CA2450194A1 Novel chromogenic substances and use thereof for the determination of carboxypeptidase activities
01/15/2003EP1275657A1 Peptide derivatives and medicinal compositions
01/15/2003EP1274724A2 Macrocyclic ns3-serine protease inhibitors of hepatitis c virus comprising alkyl and aryl alanine p2 moieties
01/15/2003EP1274693A1 Method for producing 2,5-diketopiperazines, 2,5-diketopiperazines, dipeptides and the use thereof
01/15/2003EP1274682A2 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
01/15/2003EP1274323A1 Stability enhancement of sweeteners using salts containing divalent or trivalent cations
01/15/2003EP1015627A4 Method for detecting a target compound using a nucleic acid ligand
01/15/2003EP0907643B1 Compounds with growth hormone releasing properties
01/15/2003EP0880541B1 Derivatives of antibiotic ge2270 factors
01/15/2003CN1391580A Peptides
01/15/2003CN1391577A Pharmaceutical compositions comprising metal complexes
01/15/2003CN1391553A Novel intermediate for sweetener with high sweetness and process for producing the same
01/15/2003CN1098838C Substituted N-(indole-2-carbonyl)-beta-alanimamides and derivatives as antidiabetic agents
01/14/2003US6506906 Preparation and use of bifunctional molecules having DNA sequence binding specificity
01/14/2003US6506903 By reacting 4-methylthiazole with N-halosuccinimide in solvent in presence of 2,2-azobisisobutyronitrile; halogenation, catalysis
01/14/2003US6506786 HIV protease inhibitors based on amino acid derivatives
01/14/2003US6506761 Substituted hydrazinyl heteroaromatic inhibitors of thrombin
01/14/2003US6506760 Substituted hydrazinyl heteroaromatic inhibitors of thrombin
01/14/2003US6506759 Retroviral protease inhibitors
01/14/2003US6506754 Compounds as anticoagulants
01/14/2003US6506734 20(S) camptothecin glycoconjugates
01/14/2003US6506731 Elastin peptide analogs and methods of using same
01/14/2003US6506362 Peptides and peptide mimetics attached to labels and/or hydrophilic polymmers; treating hematological disorders, particularly thrombocytopenia resulting from chemotherapy, radiation therapy, or bone marrow transfusions
01/14/2003CA2250583C Process for the preparation of n-methyl-d-phenylalanyl-n-¬1-¬3-¬(aminoiminomethyl)amino|propyl|-3,3-difluoro-2-oxohexyl|-l-prolinamide