Patents
Patents for C07J 73 - Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms (1,160)
02/2001
02/28/2001EP1077765A1 Photochemical and thermochemical solar syntheses using flat-bed solar collectors/solar reactors
02/14/2001EP0663924B1 17-beta-carboxanilides of 4-aza-5-alpha-androstan-3-ones as 5-alpha-reductase inhibitors
02/14/2001CN1061989C Compound of cholesteric lactone and analog, and its prepn method
01/2001
01/11/2001WO2001002422A1 PROCESS FOR OBTAINING 17β-(N-TERC-BUTYLCARBAMOYL)-3-ONE-4-AZA-STEROIDS
01/11/2001CA2342864A1 Process for obtaining 17.beta.-(n-terc-butylcarbamoyl)-3-one-4-aza-steroids
01/10/2001EP0649306B1 Ester derivatives of 4-aza-steroids
12/2000
12/27/2000EP0756481B1 17$g(b)-ARYL-4-AZA-STEROID DERIVATIVES
12/21/2000WO2000077025A1 NEW PROCESS FOR THE SYNTHESIS OF 17β-HYDROXY-17α-METHYL-2-OXA-5α-ANDROSTANE-3-ONE
11/2000
11/15/2000EP1051177A1 Steroid 3-o-sulphamate derivatives as inhibitors of oestrone sulphatase
11/15/2000CN1058499C 16-substituted-4-aza-androstane 5-alpha-reductase isoazyne 1 inhibitors
11/14/2000US6147213 Diastereomerically pure 3-oxo and 3-thioxo-4-aza-androstan derivatives and the use thereof as antiandrogens
11/14/2000CA2271974A1 2, 2-dibromo-azasteroids and their use in a method for introducing a 1, 2-double bond into azasteroids
11/08/2000EP0650495B1 Improved antiandrogens
11/07/2000US6143887 Process for the stereoselective synthesis of 16-substituted-4-aza-androstanones
11/01/2000CN1058018C Androsterone derivatives and its preparing process
10/2000
10/25/2000CN1271285A Remedial agent for baldness and other diseases
10/25/2000CN1057771C Androstenone derivative
10/17/2000US6133280 Androgen synthesis inhibitors
09/2000
09/28/2000WO2000056757A1 Immunomodulatory steroids, in particular the hemihydrate of 16.alpha.-bromoepiandrosterone
09/28/2000CA2365081A1 Immunomodulatory steroids, in particular the hemihydrate of 16.alpha.-bromoepiandrosterone
09/21/2000WO2000054779A1 OCULAR THERAPY IN KERATOCONJUCTIVITIS SICCA USING TOPICALLY APPLIED ANDROGENS OR TGF-$g(b)
09/21/2000CA2367643A1 Ocular therapy in keratoconjuctivitis sicca using topically applied androgens or tgf-.beta.
09/19/2000US6121449 Testosterone 5 alpha-reductase inhibitory activity; useful in therapy in the treatment of hyperandrogenic conditions
09/06/2000EP1032400A1 Prevention of precipitated acute urinary retention
09/05/2000US6114345 Phenylsubstituted 4-azasteroid fluoroderivatives
08/2000
08/29/2000US6110906 Androgen derivatives for use in the inhibition of sex steroid activity
08/23/2000EP1028734A1 $i(SPECIFIC) STEADY-STATE R-TYPE Ca?2+ CHANNEL BLOCKERS AND USE THEREOF
08/23/2000EP0759929B1 Oxidation of steroids having allylic groups
08/22/2000US6107289 Ocular therapy in keratoconjunctivitis sicca using topically applied androgens or TGF-β
08/16/2000EP0902790B1 Process for preparing steroids having a carboxamide side-chain
08/16/2000EP0641204B1 17-ethers and thioethers of 4-aza-steroids
08/02/2000EP0641208B1 4-azasteroid 5-alpha-reductase inhibitors
07/2000
07/19/2000EP1019060A1 Androgen synthesis inhibitors
07/11/2000US6087347 3-substituted-D-homo-1,3,5(10)-estratriene derivatives
06/2000
06/21/2000CN1053672C Azasteroid compounds for treating prostatic hypertrophy, their preparation and use
05/2000
05/10/2000EP0998930A1 Remedial agent for baldness and other diseases
04/2000
04/25/2000US6054598 Synthesis of 2-alkoxyestradiols
04/18/2000US6051726 Benzylation and bromination
04/05/2000EP0786011B1 Microbiological process for the preparation of 1-unsaturated 17-beta-carboxysubstituted 3-oxo-4-azaandrostan-3-ones
03/2000
03/22/2000CN1248263A Process for preparing carboxamido-4-azasteroids
03/15/2000EP0984979A1 Synthesis of 2-alkoxyestradiols
03/08/2000EP0983295A2 4-aza-steroids substituted in one or more of positions 7, 11 and 15 or with an unsaturated 14(15)-double bond as inhibitors of testosterone-5-alpha-reductase
02/2000
02/29/2000US6030981 Phenanthridine derivatives, methods of producing them and medicaments containing phenanthridine derivatives
02/09/2000EP0793671B1 Phenylsubstituted 4-azasteroid fluoroderivatives
01/2000
01/18/2000US6015806 Topical use in the treatment of androgen-dependent diseases associated with the skin.
01/12/2000EP0970105A1 Process for preparing carboxamido-4-azasteroids
01/05/2000EP0664812B1 17-beta-aryl ester carboxylates of 4-aza-5-alpha-androstane-3-ones
12/1999
12/14/1999US6001844 4-Azasteroids for treatment of hyperandrogenic conditions
12/07/1999US5998464 4-Oxa and 4-thia steroids
11/1999
11/30/1999US5994334 Androgen synthesis inhibitors
11/18/1999WO1999058551A1 Process for the stereoselective synthesis of 16-substituted-4-aza-androstanones
11/18/1999WO1999058550A1 7beta-methyl-16beta-((4-methylsulfonyl)-phenoxy)-4-aza-5alpha-androst-1-en-3-one as a 5-alpha-reductase isozyme 1 inhibitor
11/02/1999US5977126 Antiangrogens, enzyme inhbitors
10/1999
10/28/1999WO1999054032A1 Photochemical and thermochemical solar syntheses using flat-bed solar collectors/solar reactors
10/28/1999CA2328160A1 Photochemical and thermochemical solar syntheses using flat-bed solar collectors/solar reactors
10/12/1999US5965488 Plant growth regulating composition comprising epoxycyclohexane derivatives and brassinosteroids as well as method of regulating plant growth comprising the application thereof
10/05/1999US5962442 Administering a 3-oxo-4-azasteroid
09/1999
09/29/1999CN1230194A 3-substituted-d-homo-1,3,5 (10)-estratriene derivatives
09/08/1999EP0702027B1 Brassinosteroid derivatives and plant growth regulator containing the same
08/1999
08/24/1999US5942519 Administering androstene derivative 5-alpha reductase inhibitor
08/11/1999EP0934949A1 3-substituted-d-homo-1,3,5,(10)-estratriene derivatives
08/11/1999EP0649431B1 17-amino substituted 4-azasteroid 5-alpha-reductase inhibitors
08/03/1999US5932713 These novel genes are useful for the production of cotton fibers with improved characteristics.
07/1999
07/15/1999WO1999035161A1 Process for preparing carboxamido-4-azasteroids
07/15/1999CA2278487A1 Process for preparing carboxamido-4-azasteroids
07/13/1999US5922728 Phenylsubstituted 4-azasteroid fluoroderivatives
06/1999
06/16/1999EP0922770A2 A microbiological process for the transformation of 17beta-carboxy substituted 3-oxo-4-azasteroids and the use of such products as inhibitors of the enzyme 5alpha-reductase
06/10/1999WO1999027935A1 Steroid 3-o-sulphamate derivatives as inhibitors of oestrone sulphatase
06/08/1999US5910497 Treating acne vulgaris
05/1999
05/26/1999CN1217338A Process for synthesizing long-acting rapin lactones
05/26/1999CN1217337A Simple synthesizing process for rapin lactones and the like
05/06/1999WO1999021563A1 Prevention of precipitated acute urinary retention
05/06/1999CA2308070A1 Prevention of precipitated acute urinary retention
04/1999
04/21/1999EP0663402B1 7-substituted oxasteroid compound
04/14/1999EP0748221B1 7-substituted-4-aza-steroid derivatives as 5-alpha- reductase inhibitors
04/08/1999WO1999016449A1 SPECIFIC STEADY-STATE R-TYPE Ca2+ CHANNEL BLOCKERS AND USE THEREOF
03/1999
03/24/1999EP0902790A1 Process for preparing steroids having a carboxamide side-chain
03/23/1999US5886184 Finasteride processes
03/23/1999US5886005 4-Aza-19-norandrostane derivatives
03/17/1999CN1211256A 17-beta-cyclopropyl (amino/oxy 4-aza steroids as active inhibitors of testosterone 5-alpha-reductase and C17-20-lyase
03/10/1999CN1042431C Brassinosteroid derivatives and plant growth regulator containing the same
03/09/1999US5880110 Production of cotton fibers with improved fiber characteristics by treatment with brassinosteroids
03/03/1999CN1209319A Preparation method for medicinal composition containing aza-steroid compound for treating prostatic hyperplasia
02/1999
02/11/1999WO1999006050A1 Remedial agent for baldness and other diseases
02/11/1999CA2298851A1 Remedial agent for baldness and other diseases
02/04/1999WO1998050419A3 4-aza-steroids as inhibitors of testosterone-5-alpha-reductase
02/03/1999CN1041939C Androstenones
01/1999
01/07/1999EP0724592B1 16-substituted-4-aza-androstane 5-alpha-reductase isozyme 1 inhibitors
12/1998
12/09/1998CN1041096C Fluorinated 17 beta-substituted 4-aza-5 alpha-androstane-3-one derivatives
12/08/1998US5846976 Androstenone derivative
12/08/1998CA2164217C Brassinosteroid derivative and plant growth regulator using the same
12/02/1998EP0880540A1 17-beta-cyclopropyl(amino/oxy) 4-aza steroids as active inhibitors of testosterone 5-alpha-reductase and c17-20-lyase
12/01/1998US5843953 7-substituted 4-aza cholanic acid derivatives and their use
11/1998
11/18/1998EP0877554A1 Triterpene derivatives with immunosuppressant activity
11/12/1998WO1998050419A2 4-aza-steroids as inhibitors of testosterone-5-alpha-reductase
11/12/1998CA2287924A1 4-aza-steroids as inhibitors of testosterone-5-alpha-reductase
10/1998
10/28/1998EP0873315A1 Phenanthridine derivatives, methods of producing them and medicaments containing phenanthridine derivatives
10/28/1998EP0674651B1 Substituted 6-azaandrostenones
10/06/1998US5817802 Process for the stereoselective reduction of steroid enelactams
09/1998
09/30/1998EP0759929A4 Oxidation of steroids having allylic groups
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