Patents
Patents for C07J 73 - Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms (1,160)
11/1992
11/10/1992US5162332 Selected 17 β-polyaroyl-4-aza-5 α-androst-1-en-3-ones as steroidal reductase inhibitors
10/1992
10/15/1992WO1992017489A1 Novel oxa- or azasteroid derivative
10/15/1992CA2107102A1 Novel oxa- or azasteroid derivatives
10/13/1992US5155107 17β-substituted-4-aza-5α-androstan-3-one derivatives and process for their preparation
09/1992
09/29/1992US5151430 Enzyme inhibitors, skin disorders and antiandrogens
09/29/1992US5151429 Enzyme inhibitors, skin disorders and antiandrogens
09/23/1992EP0504711A1 Compound UCA1064-B
08/1992
08/18/1992US5140022 3-acyclic or cyclicaminomethyl-17a-lower-alkyl-17a-aza-d-homo-5-alpha-androstanes
08/11/1992US5138063 17β-methoxycarbonyl-4-aza-androsten-1-en-3-ones
06/1992
06/24/1992CN1062145A Azasteroid compounds for treatment of prostatic hypertrophy, their preparation and use
06/09/1992US5120847 Chemical intermediate which can be dehydrohalogenation
06/09/1992US5120742 Androstanes as enzyme inhibitors
06/04/1992DE4038128A1 8-en-19, 11(beta)-ueberbrueckte steroide, deren herstellung und diese enthaltende pharmazeutische praeparate 8-ene-19, 11 (beta) -ueberbrueckte steroids, their production and pharmaceutical compositions containing them
05/1992
05/28/1992WO1992009618A1 8-ENE-19, 11β-BRIDGED STEROIDS, THEIR PREPARATION AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM
05/28/1992CA2097079A1 8-ene-19, 11.bet.beta.-bridged steroids, their preparation and pharma ceutical formulations containing them
05/26/1992US5116983 Dehydrogenation process intermediates
05/20/1992EP0485392A1 Androgen derivatives for use in the inhibition of sex steroid activity
05/06/1992EP0484094A2 Azasteroid compounds for the treatment of prostatic hypertrophy, their preparation and use
05/05/1992US5110939 Antiandrogens
04/1992
04/08/1992EP0478910A2 3-Substituted-aminomethyl-3-substituted-oxy-17A-methyl-17A-lower-alkyl-17A-aza-d-homo-5-alpha-androstanes
04/02/1992CA2046527A1 3-substituted-aminomethyl-3-substituted-oxy-17a-methyl-17a-lower-alkyl-17a-aza-d-homo-5-alpha androstanes
04/01/1992EP0478068A2 New process for making 17-beta alkanoyl 3-oxo-4-aza-5-alpha-androst-1-enes
04/01/1992EP0478066A2 New process for making 3-oxo-4-aza-androst-1-ene 17beta-ketones
04/01/1992EP0478065A2 New intermediate for making 3-oxo-4-aza-androst-1-ene 17beta-ketones
03/1992
03/25/1992CA2050824A1 Process for making 3-oxo-4-aza-androst-1-ene 17-.beta.-ketones
03/25/1992CA2050821A1 Process for making 17-.beta. alkanoyl 3-oxo-4-aza-5-alpha-androst- 1-enes
03/24/1992US5098908 Drugs for treatment of acne, seborrhea, female hirsurism and benign prostatic hypertropy
03/18/1992EP0474666A1 Oxidative preparation of a-nor-17 beta-carboxy-3,5-secoandrostan-5-one-3 oic acid.
03/04/1992EP0473226A2 Trialkysilyl trifluoromethanesulfonate mediated functionalization of 4-aza-5alpha-androstan-3-one steroids
03/04/1992EP0473225A2 Process for iodinating or brominating the alpha-methylenic carbon of a secondary amide
02/1992
02/25/1992US5091534 Electrophilic substitution
01/1992
01/28/1992US5084574 Dehydrogenation process
01/09/1992WO1992000010A1 Method of treating human prostatic adenocarcinoma
12/1991
12/27/1991EP0462668A2 New 17beta-aminobenzoyl-4-aza-5alpha-androst-1-en-3-ones as benign prostatic hypertrophy agents
12/27/1991EP0462665A2 Selected 17beta-polyaroyl-4-aza-5alpha-androst-1-en-3-ones as steroidal reductase inhibitors
12/27/1991EP0462664A2 Specific 17beta-thiobenzoyl-4-aza-5alpha-androst-1-en-3-ones as antiandrogenic agents
12/27/1991EP0462662A2 17beta-N-monosubstituted adamantyl/norbornanyl carbamoyl-4-aza-5alpha-androst-1-en-3-ones and androstan-3-ones
12/27/1991EP0462661A2 Novel 17beta-hydroxybenzoyl-4-aza-5alpha-androst-1-en-3-ones as testosterone reductase inhibitors
12/21/1991CA2058920A1 17.beta.-n-monosubstituted adamantyl/carbamoyl-4-aza-5.alpha.-androst-1-en-3-ones and androstan-3-ones as 5.alpha.-reductase
12/21/1991CA2044922A1 17.beta.-hydroxybenzoyl-4-aza-5.alpha.-androst-1-en-3-ones as testoste rone reductase inhibitors
12/21/1991CA2044921A1 Specific 17 .beta.-thiobenzoyl-4-aza-5 .alpha.-androst-1-en-3-ones as antiandrogenic agents
12/21/1991CA2044914A1 17.beta.-aminobenzoyl-4-5 .alpha.-androst-1-en-3-ones as benign prostatic hypertrophy agents
12/21/1991CA2044905A1 Selected 17 .beta.-polyaroyl-4-aza-5 .alpha.-androst-1-en-3-ones as steroidal reductase inhibitors
11/1991
11/28/1991WO1991012206A3 Aromatase-inhibiting steroids
10/1991
10/29/1991US5061803 Process for making 17-beta alkanoyl 3-oxo-4-aza-5-α-androst-1-enes
10/29/1991US5061802 17β-aminobenzoyl-4-aza-5α-androst-1-en-3-ones as benign prostatic hypertrophy agents
10/29/1991US5061801 Intermediate for making 3-oxo-4-aza-androst-1-ene 17β-ketones
09/1991
09/25/1991CN1054771A Process for preparation of 17beta-substituted-4-aza-5alpha-androstan-3-one derivatives
09/17/1991US5049562 Enzyme inhibitors, antiandrogens
09/02/1991WO1991013903A1 Heterocyclic steroid compounds
09/02/1991CA2077680A1 Heterocyclic steroid compounds
08/1991
08/22/1991WO1991012206A2 Aromatase-inhibiting steroids
08/10/1991WO1991012261A1 17β-SUBSTITUTED-4-AZA-5α-ANDROSTAN-3-ONE DERIVATIVES AND PROCESS FOR THEIR PREPARATION
08/10/1991CA2049318A1 17.beta.-substituted-4-aza-5.alpha.-androstan-3-one derivatives and process for their preparation
07/1991
07/16/1991US5032586 Enzyme inhibitors, steroid hormones
06/1991
06/04/1991US5021575 Treating with oxalyl chloride, brominating, dehydrobromination then deprotecting to yield isomers
06/04/1991CA1284636C 17.beta.-N-MONOSUBSTITUTED-CARBAMOYL-4-AZA-5.alpha.-ANDROSTAN-3-ONES
05/1991
05/22/1991EP0428366A2 Method for introducing a 1,2 double bond into azasteroids
04/1991
04/16/1991CA1282976C Increasing the yield of cereals by means of brassinolide derivatives
02/1991
02/27/1991EP0414529A2 7-Keto- and 7-Hydroxy-androsta-3,5-diene-3-carboxylic acid derivatives
02/27/1991EP0414491A2 17 Beta-acyl-4-aza-5 alpha-androst-1-ene-3-ones as 5 alpha-reductase inhibitors
02/27/1991EP0414490A2 17 Beta-acyl-4-aza-5 alpha-androst-1-ene-3-one as 5 alpha-reductase inhibitors
02/25/1991CA2023609A1 7-keto or hydroxy 3,5-diene steroids as inhibitors of steroid 5-–-reductase
02/22/1991CA2023158A1 17 beta-acyl-4-aza-5 alpha-androst-1-ene-3-ones as 5 alpha-reductase inhibitors
02/22/1991CA2023157A1 17 beta-acyl-4-aza-5 alpha-androst-1-ene-3-ones as 5 alpha-reductase inhibitors
02/21/1991WO1991001991A1 New topically active steroidal anti-inflammatory agents
01/1991
01/31/1991CA2000369A1 Topically active steroidal anti-inflammatory agents
01/24/1991WO1991000732A1 Androgen derivatives for use in the inhibition of sex steroid activity
01/24/1991CA2063378A1 Androgen derivatives for use in the inhibition of sex steroid activity
12/1990
12/01/1990WO1990015045A1 Oxidative preparation of a-nor-17 beta-carboxy-3,5-secoandrostan-5-one-3 oic acid
10/1990
10/09/1990US4961775 Brassinosteroid derivatives and plant growth regulators
09/1990
09/25/1990US4959097 23-Phenylsteroids
09/25/1990US4959093 Steroid, brassinolide derivative
07/1990
07/03/1990US4939247 Gamma-lactone derivatives and process of preparing same
05/1990
05/09/1990EP0367502A1 Methods of synthesizing benign prostatic hypertrophic agents
04/1990
04/03/1990US4914106 Controlling androgen-dependent diseases; preventing abortion; contraception
03/1990
03/27/1990US4912097 Novel 11 β-alkynylphenyl-10-nor-steroids
03/20/1990US4910192 Topically active steroidal anti-inflammatory agents
02/1990
02/14/1990CN1039594A Method for synthesizing epi-rape lactone and likes
12/1989
12/19/1989US4888336 Decrease dihydrotestosterone activity
12/12/1989US4886544 Plant growth regulators; alkenylation, oxidation, hydrolysis, acylation, lactonization
11/1989
11/29/1989EP0245170B1 19-nor or 19-nor d-homo steroids substituted at position 11 beta by a phenyl group substituted by an alkynyl group, process for their preparation, their use in medicaments and pharmaceutical compositions containing them
10/1989
10/17/1989US4874551 δ-lactone derivatives and process of preparing same
08/1989
08/29/1989US4861875 3α,5-cyclo-22,23-dihydroxy-5α-steroid compounds
08/22/1989US4859681 17 α-Acyl-4-aza-5a-androst-1-en-3-ones as 5 alpha-reductase inhibitors
07/1989
07/19/1989CN1033998A "22r, 23r,24s)-22,23-epoxy-2 alpha, 3 alpha-isopropylidenedioxy-beta-homo-7-oxa-5alpha stigmastan-6-one, process for preparation thereof and plant growth regulating composition contg. same
07/05/1989EP0322639A1 (22R,23R,24S)-22,23-Epoxy-2 alpha, 3 alpha-isopropylidenedioxy-B-homo-7-oxa-5 alpha-stigmastan-6-one, process for preparation thereof and plant growth regulating composition containing the same
07/04/1989US4845104 Oxidized analogs of 17β-N-monosubstituted-carbamoyl-4-aza-5-α-androstan-3-ones
06/1989
06/06/1989CA1255293A1 2-oxa- or -aza-pregnane compounds
05/1989
05/24/1989CN1033057A Brassinosteroid derivatives and plant growth regulators
05/17/1989EP0315921A1 Brassinosteroid derivatives and plant growth regulators
05/03/1989EP0314199A1 17 Beta-substituted-4-aza-5 alpha-androstenones and their use as 5 alpha-reductase inhibitors
04/1989
04/18/1989US4822803 Benzofuran 2-carboxylic acid hydrazides useful as inhibitors of leukotriene biosynthesis
01/1989
01/31/1989US4801607 Antiviral furanoditerpenoids
01/11/1989EP0298652A2 Dehydrogenation process and intermediates
11/1988
11/15/1988US4785103 Antiandrogens
10/1988
10/05/1988EP0285301A2 Antitumor and antiviral furanoditerpenoids
10/05/1988CN88101369A Preparation of 23-phenylsteroids and uses
09/1988
09/21/1988EP0282984A1 23-Phenylsteroids
08/1988
08/30/1988US4767442 Increasing the yield of cereals by means of brassinolide derivatives
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