Patents
Patents for C07J 73 - Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms (1,160)
11/1994
11/24/1994WO1994026767A1 Improved antiandrogens
11/24/1994CA2136303A1 Improved antiandrogens
11/23/1994CN1095383A Substituted 6-azaandrostenones
10/1994
10/25/1994US5359071 15-substituted 4-azasteroids
10/13/1994WO1994022900A1 AZA-ANDROSTANE-17β-CARBOXAMIDES
09/1994
09/29/1994WO1994014833A3 Substituted 6-azaandrostenones
09/29/1994WO1994011387A3 A process for the production of finasteride
09/15/1994WO1994020104A1 15-substituted 4-azasteroids
09/15/1994CA2157363A1 15-substituted 4-azasteroids
09/14/1994EP0474666B1 Oxidative preparation of a-nor-17 beta-carboxy-3,5-secoandrostan-5-one-3 oic acid
08/1994
08/30/1994US5342948 Antiandrogens; ozonation, amination, reduction of androstane derivative with acyl(urea or thiourea)
08/23/1994CA1331601C Dehydrogenation process
08/18/1994WO1994018225A1 15-oxasterols as hypocholesterolemics
08/17/1994EP0610472A1 Steroids with a fluorinated acylureidic type side chain
08/10/1994CN1090583A New finasteride processes
07/1994
07/27/1994EP0607400A1 Fluorinated 17-beta substituted-4-aza-5-alpha- andostran-3one derivatives.
07/26/1994CA1330987C (22r,23r,24s)-22,23-epoxy-2.-3.-isopropylidene-dioxy- .beta.-homo-7-oxa-5. -stigmastan-6-one, process for preparation thereof and plant growth regulating composition containing the same
07/07/1994WO1994014833A2 Substituted 6-azaandrostenones
07/07/1994WO1994014452A1 METHOD OF TREATMENT OF CHRONIC PROSTATITIS WITH 17β-N-MONOSUBSTITUTED-CARBAMOYL-4-AZA-5α-ANDROST-1-EN-3-ONES
07/07/1994CA2152053A1 Substituted 6-azaandrostenones
07/07/1994CA2151239A1 Method of treatment of chronic prostatitis with 17b-n- monosubstituted-carbamoyl-4-aza-5a-androst-1-en-3-ones
06/1994
06/28/1994US5324734 Antiandrogens
06/23/1994WO1994013691A1 Thio- and oxo-azasteroids, processes for the preparation thereof, use thereof as antiandrogens and pharmaceutical compositions containing them
06/01/1994EP0599376A2 A process for the production of finasteride
05/1994
05/26/1994WO1994011387A2 A process for the production of finasteride
05/26/1994WO1994011385A1 17-alpha-acyl steroids which inhibit 5-alpha-reductase
05/25/1994CN1087092A New 7 beta-substituted-4-aza-5 alpha-androstan-3-ones as 5 alpha-reductase inhibitors
04/1994
04/20/1994CN1085562A 7beta-substituted-4-aza-5alpha-cholestan-ones as 5-alpha-reductase inhibitors
04/19/1994US5304562 17β-substituted Aza-androstane derivatives
04/14/1994WO1994007909A1 NOVEL 17β-SUBSTITUTED 4-AZAANDROSTANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME
04/14/1994WO1994007908A1 Novel 7-substituted oxa- or azasteroid compound
04/14/1994WO1994007861A1 17β-CARBOXANILIDES OF 4-AZA-5α-ANDROSTAN-3-ONES AS 5α-REDUCTASE INHIBITORS
04/14/1994WO1994007860A1 17 β-ARYL ESTER CARBOXYLATES OF 4-AZA-5α-ANDROSTANE-3-ONES
04/14/1994CA2146164A1 Novel 17.beta.-substituted 4-azaandrostane derivatives, pharmaceutical compositions containing them and process for preparing same
04/14/1994CA2145643A1 Novel 7-substituted oxa-or azasteroid compound
04/13/1994EP0591165A1 Heterocyclic steroid compounds
04/13/1994CN1085224A Fluorinated 17beta-substituted 4-aza-5alpha-androstane-3-one derivatives
04/13/1994CN1085223A 17beta-substituted 4-aza-5alpha-androstan-3-one derivatives
04/12/1994US5302621 Azasteroid compounds for the treatment of prostatic hypertrophy, their preparation and use
04/05/1994US5300294 Administering a steroid 5-a-reductase inhibiting compound
03/1994
03/31/1994WO1994006425A1 OXIDIZATION METABOLITES OF 5α-23-METHYL-4-AZA-21-NOR-CHOL-1-ENE-3,20-DIONE
03/30/1994CN1084519A New process for producing 7 beta-substituted-aza-5 alpha-androstan-3-ones
02/1994
02/17/1994WO1994003476A1 17β-SUBSTITUTED 4-AZA-5α-ANDROSTAN-3-ONE DERIVATIVES
02/17/1994WO1994003475A1 FLUORINATED 17β-SUBSTITUTED 4-AZA-5α-ANDROSTAN-3-ONE DERIVATIVES
02/17/1994WO1994003474A1 Steroids with a fluorinated acylureidic type side chain
02/17/1994CA2120343A1 Fluorinated 17.beta.-substituted 4-aza-5.alpha.-androstan-3-one derivatives
02/17/1994CA2120339A1 17.beta.-substituted 4-aza-5.alpha.-androstan-3-one derivatives
02/16/1994EP0582713A1 Novel oxa- or azasteroid derivative
01/1994
01/11/1994US5278159 Aryl ester derivatives of 3-oxo-4-aza-androstane 17-β-carboxylates as 5-α-reductase inhibitors
01/11/1994CA1326013C Methods for synthesizing benign prostatic hypertropic agents and their intermediates
01/06/1994WO1994000121A1 17-acyl-4-aza-steroid-3-one as 5-alpha-reductase inhibitors
12/1993
12/07/1993CA1325006C Steroid 5-alpha-reductase inhibitors
12/01/1993EP0572166A1 New 7beta-substituted-4-aza-5a-androstan-3-ones as 5a-reductase inhibitors
12/01/1993EP0572165A1 New 7B-substituted-4-aza-5a-cholestan-ones as 5a-reductase inhibitors
11/1993
11/25/1993WO1993023420A1 NEW 7β-SUBSTITUTED-4-AZA-5α-ANDROSTAN-3-ONES AS 5α-REDUCTASE INHIBITORS
11/25/1993WO1993023419A1 NEW 7β-SUBSTITUTED-4-AZA-5α-CHOLESTAN-ONES AS 5α-REDUCTASE INHIBITORS
11/25/1993WO1993023376A1 NEW PROCESS FOR PRODUCING 7β-SUBSTITUTED-4-AZA-5α-ANDROSTAN-3-ONES
11/25/1993WO1993023053A1 INHIBITORS OF TESTOSTERONE 5α-REDUCTASE ACTIVITY
11/25/1993WO1993023051A1 New 17-ester, amide, and ketone derivatives of 3-oxo-4-azasteroids as 5a-reductase inhibitors
11/25/1993WO1993023050A1 NEW DELTA-17 AND DELTA-20 OLEFINIC AND SATURATED 17β-SUBSTITUTED-4-AZA-5α-ANDROSTAN-3-ONES AS 5α-REDUCTASE INHIBITORS
11/25/1993WO1993023048A1 4-azasteroid 5-alpha-reductase inhibitors
11/25/1993WO1993023042A1 17α AND 17β SUBSTITUTED ACYL 4 AZA STEROIDS
11/25/1993WO1993023041A1 Ester derivatives of 4-aza-steroids
11/25/1993WO1993023040A1 17-ethers and thioethers of 4-aza-steroids
11/25/1993WO1993023039A1 Substituted 4-aza-5a-androstan-ones as 5a-reductase inhibitors
11/25/1993WO1993023038A1 17-AMINO SUBSTITUTED 4-AZASTEROID 5α-REDUCTASE INHIBITORS
11/25/1993CA2136304A1 Inhibitors of testosterone 5.alpha.-reductase activity
11/25/1993CA2135174A1 17-ethers and thioethers of 4-aza-steroids
11/25/1993CA2135173A1 Ester derivatives of 4-aza-steroids
11/25/1993CA2135167A1 New 17-ester, amide, and ketone derivatives of 3-oxo-4- azasteroids as 5a-reductase inhibitors
11/25/1993CA2135057A1 17-amino substituted 4-azasteroid 5a-reductase inhibitors
11/25/1993CA2135056A1 New delta-17 and delta-20 olefinic and saturated 17b-substituted-4-aza-5a-andros-tan-3-ones as 5a-reductase inhibitors
11/25/1993CA2135055A1 4-azasteroid 5-alpha-reductase inhibitors
11/21/1993CA2096616A1 7beta-substituted-4-aza-5alpha-androstan-ones as 5alpha-reductase inhibitors
11/21/1993CA2096576A1 7beta-substituted-4-aza-5alpha-cholestan-ones as 5alpha-reductase inhibitors
08/1993
08/17/1993US5237065 Steroid 5-alpha-reductase inhibitors
08/17/1993US5237064 Process for producing 7β-substituted-aza-5αandrostan-3-ones
08/17/1993US5237061 17B-substituted 3-oxo-4-azasteroids, imidazolide intermediate
08/17/1993US5236929 Compound uca1064-b
07/1993
07/20/1993US5229511 From corresponding 17a-aza-D-homo-5-alpha-androstan-3-ol; muscle relaxants
07/13/1993US5227375 Androstanediones, estrogen-dependent diseases, anticancer
07/08/1993WO1993013124A1 Inhibitors of 5-alpha-testosterone reductase
07/08/1993CA2126203A1 Inhibitors of 5-alpha-testosterone reductase
06/1993
06/30/1993EP0548884A1 Biphosphonate derivative
06/30/1993EP0548774A1 Process for producing a lactone or an ester
06/27/1993CA2086026A1 Bisphosphonate derivative
06/23/1993EP0547691A1 The use of 17B-N-mono-substituted-carbamoyl-4-aza-5alpha-androst-1-en-3-ones for the preparation of a medicament for the prevention of prostatic carcinoma
06/23/1993EP0547690A1 Use of 17B-acyl-4-aza-5alpha-androst-1-en-3-ones for the preparation of a medicament for the prevention of prostatic carcinoma
06/23/1993EP0547687A1 17B-N-Substituted adamantyl/norbonanyl carbamoyl-4-aza-5a-and-rost-1-en-3-ones and androstan-3 ones
06/19/1993CA2085456A1 17beta-n-substituted adamantyl/norbornanyl carbamoyl-4-aza-5a -androst -1-en-3-ones and adrostan-3-ones as 5a-reductase inhibitors
06/18/1993CA2084798A1 Method of preventing prostatic carcinoma with 17beta -acyl-4-aza-5.- androst-1-ene-3-ones
06/15/1993US5219879 Heterocyclic steroid compounds
04/1993
04/21/1993EP0538192A1 New 17-beta-substituted aza-androstanderivatives
04/10/1993CA2080054A1 17beta-substituted aza-androstane derivatives
03/1993
03/16/1993CA1314541C 17.beta.-n-monosubstituted carbamoyl -4-aza-5.- androst-1-en-3-ones
02/1993
02/16/1993US5187278 Intermediates for antiandrogens
01/1993
01/20/1993WO1993002096A1 PROCESS FOR THE PREPARATION OF 17β-SUBSTITUTED-4-AZA-5α-ANDROSTAN-3-ONE DERIVATIVES
01/20/1993EP0523688A1 Process for the preparation of 17beta-substituted-4-aza-5alpha-androstan-3-one derivatives
01/20/1993CA2091983A1 Process for the preparation of 17.beta.-substituted-4-aza-5.alpha.-androstan-3-one derivatives
12/1992
12/15/1992CA1311469C --lactone derivatives and process of preparing same
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