Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
12/2009
12/03/2009US20090299060 Compounds and methods for inhibiting mitotic progression
12/03/2009US20090298904 Novel peptides from actinomadura namibiensis
12/03/2009US20090298856 2,3 Substituted fused bicyclic pyrimidin-4(3H)-ones modulating the function of the vanilliod-1receptor (VR1)
12/03/2009US20090298854 Indole acetic acid derivatives and their use as pharmaceutical agents
12/02/2009EP1626050B1 Sulfur-containing naphthoylimide derivatives
12/02/2009CN101595111A Selective glycosidase inhibitors and uses thereof
12/02/2009CN100563650C Indol-6 sulfonamide derivatives, their preparation and their use as 5-ht-6 modulators
12/01/2009US7626033 Compounds for the modulation of PPARγ activity
12/01/2009US7625924 Nicotinic alpha-7 receptor ligands and preparation and uses thereof
12/01/2009US7625913 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
12/01/2009US7625892 Pharmaceutical compositions for the treatment of diseases related to neurotrophines
12/01/2009US7625841 invention also relates to the preparation of the compounds, to their use as herbicides and to herbicidal compositions comprising the novel compounds.
11/2009
11/26/2009US20090292120 Benzimidazole compounds having gastric acid secretion inhibitory action
11/26/2009US20090291955 Azacyclohexane Derivatives as Inhibitors of Stearoyl-Coenzyme a Delta-9 Desaturase
11/26/2009US20090291948 Sulfonamide peri-substituted bicyclics for occlusive artery disease
11/25/2009CN101585849A Linked disulfide group substituted deuteroporphyrin, metal complexes, preparation method and uses thereof
11/25/2009CN100562521C Substituted thienopyrrole carboxylic acid amides, pyrrolothiazole carboxylic acid amides, and related analogs as inhibitors of casein kinase i epsilon
11/24/2009US7622490 Broadspecturm 2-amino-benzoxazole sulfonamide HIV protease inhibitors
11/24/2009US7622481 Gramnegative and Grampositive bacterial infections; substituted Piperidine derivatives specially optionally substituted pyrido [3,2, -b][1,4] thiazin-yl; 6-({(3R,4S)-3-Fluoro-1-[(R)-2-hydroxy-2-(2-methoxy-quinolin-8-yl)-ethyl]-piperidin-4-ylamino }-methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one; nontoxic
11/24/2009US7622479 For example, 2-(1,3-benzodioxol-5-yl)-6-phenyl-1H-imidazo[4,5-b]pyridinetyrosine; kinase-inhibiting activity; use in treatment of breast cancer, prostate cancer, lung cancer or pancreatic carcinoma
11/24/2009CA2408144C Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
11/19/2009WO2009140624A2 Glucokinase activators
11/19/2009WO2009140127A2 SYNTHESIS OF DIHYDROTHIENO[3,2-d]PYRIMIDINE DIOLS AND SIMILAR PYRIMIDINE DIOLS
11/19/2009WO2009139076A1 Lipoprotein lipase-activating compositions comprising benzene derivates
11/19/2009WO2009138793A1 Substituted quinazolines as blood platelet lowering agents
11/19/2009CA2724116A1 Glucokinase activators
11/19/2009CA2723958A1 Substituted quinazolines
11/19/2009CA2723455A1 Lipoprotein lipase-activating compositions comprising benzene derivates
11/18/2009EP2119719A1 Thiazepine derivative
11/18/2009EP1545453B1 Rifalazil for treating infections of clostridium difficile
11/18/2009CN101583365A Triazine derivatives and their therapeutical applications
11/17/2009US7619094 Ketoamides with cyclic P4's as inhibitors of NS3 serine protease of hepatitis C virus
11/17/2009US7618961 A sulfonylamino-tetrahydro(1,3)thiazolo(5,4-c)pyridinyl or benzothiazole derivatives, for treating diabetes, syndrome X, obesity, glaucoma, hyperlipidemia, hyperglycemia, hyperinsulinemia, osteoporosis, tuberculosis, dementia
11/17/2009US7618959 6-({2-[4-(6-Methoxy-[1,5]naphthyridin-4-yl)phenyl]ethylamino}methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one;bacterial infections; antibiotic resistance; Staphylococcus aureus, Streptococcus pneumoniae and pyogenes, Enterococcus; Haemophilus influenzae, Moraxella catarrhalis, E-coli
11/17/2009CA2535511C Compounds having thrombopoietin receptor agonism
11/17/2009CA2432181C Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists
11/12/2009WO2009136663A1 Fused heterocyclic derivatives and use thereof
11/12/2009WO2009136350A1 Novel class of spiro piperidines for the treatment of neurodegenerative diseases
11/12/2009WO2009135927A1 Substituted n-phenyl-2,3-dihydroimidazo[2,1-b]thiazole-5-sulfonamide derivatives as 5-ht6 ligands
11/12/2009WO2009135925A1 Substituted n-imidazo[2,1-b]thiazole-5-sulfonamide derivatives as 5-ht6 ligands
11/12/2009US20090281279 Rigidized trimethine cyanine dyes
11/12/2009US20090281123 Novel thiazolo (4,5-d) pyrimidine compounds novel compounds
11/12/2009US20090281082 Polo-like kinases (Plk1); 1-[1-(2-Chlorophenyl)ethyl]-7-imidazo[1,2-a]pyridin-3-yl-1,2,3,4-tetrahydrothieno[3,2-e][1,4]diazepin-5-one; 3-iodoimidazo[1,2-a]pyridine eractant; ANTITUMOR, ANTIPROLIFERATIVE
11/12/2009US20090281074 Drug compositions and methods for preventing and treating thrombosis or embolism
11/12/2009CA2721786A1 Novel class of spiro piperidines for the treatment of neurodegenerative diseases
11/12/2009CA2712586A1 Antibacterial fluoroquinolone analogs
11/11/2009EP2116547A1 Substituted N-imidazo(2, 1-b) thiazole-5-sulfonamide derivatives as 5-TH6 ligands
11/11/2009EP2116546A1 Substituted N-phenyl-2,3-dihydroimidazo[2,1-b]thiazole-5-sulfonamide derivatives as 5-HT6 ligands
11/11/2009EP2114937A1 Phenothiazin derivates, method for the production thereof and use thereof as pharmaceuticals
11/11/2009EP1477186B1 Antipruritics
11/11/2009CN100558355C Indol-5 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
11/05/2009WO2009134726A1 Substituted pyrimidine derivatives as histamine h4 receptor ligands
11/05/2009WO2009134203A1 New peptidomimetic compounds
11/05/2009WO2009133687A1 Cyclopentylacrylic acid amide derivative
11/05/2009US20090275623 Alpha-amino acid derivatives and medicaments containing the same as an active ingredient
11/05/2009CA2722938A1 New peptidomimetic compounds
11/05/2009CA2722733A1 Cyclopentylacrylamide derivative
11/04/2009EP1481077B1 Mitotic kinesin inhibitors
11/04/2009CN101573365A Compounds useful as protein kinase inhibitors
11/03/2009US7612205 Crystals of quinolinecarboxylic acid derivative solvate
11/03/2009US7612063 antibiotics, fungicides, viricides; treating microbial infections; fused rings based on 4-oxo-4H-pyrido[3,2,1-kl]benzo[g]-phenoxazine for example; Tumor suppression agents with reduced side effects; anticancer
11/03/2009US7612055 Macrocyclic lactams and pharmaceutical use thereof
11/03/2009CA2360767C Tricyclic benzodiazepines as vasopressin receptor antagonists
11/03/2009CA2316356C Benzoxazine compounds for enhancing synaptic response
10/2009
10/29/2009WO2009130560A1 Fused pyrimidineone compounds as trpv3 modulators
10/29/2009US20090270467 5-[(1S,3S,4R)-3-Amino-4-(2,4,5-trifluorophenyl)cyclohexyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-amine, used for treating insulin resistance, hyperglycemia and non-insulin dependent diabetes in mammals
10/29/2009US20090270446 Diamine derivatives
10/29/2009US20090270402 Novel triazolopyridazines
10/29/2009CA2720357A1 Fused pyrimidineone compounds as trpv3 modulators
10/28/2009EP1828207B1 Thiazolopyridinone derivates as mch receptor antagonists
10/28/2009CN101568536A 2-aza-bicyclo[3.1.0]hexane derivatives
10/28/2009CN101568533A 3-heteroaryl (amino or amido)-1- (biphenyl or phenylthiazolyl) carbonylpiperdine derivatives as orexin receptor inhibitors
10/28/2009CN101568527A 2-aminothiazole-4-carboxylic amides as protein kinase inhibitors
10/28/2009CN101565428A Preparation method of prulifloxacin
10/27/2009US7608717 3-[2-(dimethylamino)ethyl]-1-[(3-fluorophenyl)sulfonyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one; anxiety disorder or a cognitive disorder; central nervous system disorders; psychological disorders; neurodegenerative disorder; attention deficit disorder; obsessive compulsive disorder; Alzheimer's
10/27/2009CA2415966C Tetrahydro-heterocycloazepinyl pyrimidine derivatives
10/27/2009CA2415050C Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepines
10/22/2009WO2009129211A1 Inhibitors of phosphatidylinositol 3-kinase
10/22/2009WO2009128383A1 3-PHENYLPYRAZOLO[5,1-b]THIAZOLE COMPOUND
10/22/2009WO2009077956A3 HETEROCYCLIC INHIBITORS OF AN Hh-SIGNAL CASCADE, MEDICINAL COMPOSITIONS BASED THEREON AND METHODS FOR TREATING DISEASES CAUSED BY THE ABERRANT ACTIVITY OF AN Hh-SIGNAL SYSTEM
10/22/2009WO2008071961A8 2-quinolinone and 2-quinoxalinone- derivatives and their use as antibacterial agents
10/22/2009US20090264421 Methods and Compositions for Treating Cancer
10/22/2009US20090264411 Fused thiophene derivatives as mek inhibitors
10/22/2009CA2721670A1 3-phenylpyrazolo[5,1-b]thiazole compound
10/22/2009CA2721434A1 Inhibitors of phosphatidylinositol 3-kinase
10/21/2009EP1781673B1 Selected fused heterocyclics and uses thereof
10/21/2009EP1346993B1 Lactam compounds and medical use thereof
10/21/2009CN101563353A Antibacterial compounds and processes for its production
10/21/2009CN101563352A Antiviral indoles
10/21/2009CN101563349A Haloalkyl-substituted pyrimidinone derivatives
10/21/2009CN101563347A Vasopressin V1a antagonists
10/20/2009US7605169 Antibacterial agents
10/20/2009CA2408142C Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
10/15/2009WO2009126806A2 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene a4 hydrolase
10/15/2009WO2009126675A1 2-sulfonylamino-4-heteroaryl butyramide antagonists of ccr10
10/15/2009US20090259049 3-PHENYLPYRAZOLO[5,1-b]THIAZOLE COMPOUNDS
10/15/2009US20090258884 Substituted amides
10/15/2009US20090258857 Chemical compounds
10/15/2009US20090258854 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene A4 hydrolase
10/15/2009CA2721099A1 Thiazolopyridin-2-yloxy-phenyl and thiazolopyrazin-2-yloxy-phenyl amines as modulators of leukotriene a4 hydrolase
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