| Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120) |
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| 08/12/2010 | US20100204288 Heteroaryl-Ureas and Their Use as Glucokinase Activators |
| 08/12/2010 | US20100204268 Processes for preparing different forms of (s)-(+)-clopidogrel bisulfate |
| 08/12/2010 | US20100203007 Novel benzodiazepine derivatives |
| 08/12/2010 | CA2750935A1 Heteroaryls and their use as pi3k inhibitors |
| 08/11/2010 | CN101801982A Macrocyclic indole derivatives for the treatment of hepatitis C infections |
| 08/11/2010 | CN101801981A Sirtuin modulating thiazolopyridine compounds |
| 08/11/2010 | CN101798317A N-substituted aminothiazole morphinan compound and preparation method and applications thereof |
| 08/11/2010 | CN101798316A Triazolothiadiazole compounds and preparation method and application thereof |
| 08/10/2010 | US7772261 Pyrazolo[4,3-d]thiazole derivatives, and preparation and therapeutic application thereof |
| 08/10/2010 | US7772260 Neuroprotectants; reduce side effect of neurotoxic agent; treatment of neuropathies resulting from chemotherapeutic agents used in the treatment of HIV and proliferative disease such as cancer and treatment of inflammatory diseases, neurodegenerative diseases |
| 08/10/2010 | US7772229 Oxabispidine compounds useful in the treatment of cardiac arrhythmias |
| 08/10/2010 | US7772198 cycstic fibrosis transmembrane conductance regulators (CFTR); for treatment of cystic fibrosis, asthma or diarrhea |
| 08/10/2010 | CA2451605C Diamine derivatives |
| 08/05/2010 | WO2010086481A1 New family of antichagasics derived from imidazo[4,5-c][1,2,6]thiadiazine 2,2-dioxide |
| 08/05/2010 | US20100197910 Process for preparation of prulifloxacin using novel intermediates |
| 08/04/2010 | CN101796056A heterocyclic inhibitors of c-met and uses thereof |
| 08/03/2010 | US7767824 5,5-dibenzylimidazo[2,1-b]thiazol-6(5H)-one, useful as cognition activators in connection with treatments on memory disturbance, memory acquirement and retention disturbance, for example in Alzheimer's disease |
| 08/03/2010 | US7767706 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication |
| 08/03/2010 | US7767670 Substituted 3-carboxamido isoxazoles as kinase modulators |
| 08/03/2010 | US7767659 Synthesis of naturally occurring ecteinascidins and related compounds |
| 07/29/2010 | WO2010085570A1 Poly (ADP-Ribose) Polymerase (PARP) Inhibitors |
| 07/29/2010 | WO2010084508A2 Process for the preparation of type i, type ii and type iii crystalline prulifloxacin |
| 07/29/2010 | WO2010014930A3 Piperidine derivatives as jak3 inhibitors |
| 07/29/2010 | WO2010004457A3 Process for the preparation of 3, 4-dihydro-2h-thien [3, 2-e] -1, 2-thiazin-4-ol 1, 1 -dioxide derivatives and intermediates |
| 07/29/2010 | US20100190774 Inhibitors of c-met and uses thereof |
| 07/29/2010 | CA2750777A1 Bicyclic heterocyclic spiro compounds |
| 07/29/2010 | CA2750106A1 Poly (adp-ribose) polymerase (parp) inhibitors |
| 07/28/2010 | CN101790527A benzothiophene inhibitors of rho kinase |
| 07/28/2010 | CN101790515A trans-3-aza-bicyclo[3.1.0]hexane derivatives |
| 07/27/2010 | US7763729 Bicyclic heteroaromatic derivatives |
| 07/27/2010 | US7763641 such as [(1S,2R)-2-hydroxy-3-[N-[4-(2-methylaminothiazol-4-yl)phenylsulfonyl]-N-(2-methylpropyl)amino]-1-(phenylmethyl)propyl]carbamic acid, [(3R,3aS,6aR)-hexahydrofuro[2,3-b]furan-3-yl]ester, used for treating human immunodeficiency virus infections |
| 07/27/2010 | US7763615 derivatives of ecteinascidins, particularly ecteinascidin 736, used for the treatment of lung, colon, kidney, prostate, cervical, ovarian, breast or pancreatic cancer, leukaemia or melanoma in mammals; reduced systemic toxicity and improved pharmacokinetics |
| 07/22/2010 | WO2010083141A1 Bicyclic compounds for the reduction of beta-amyloid production |
| 07/22/2010 | WO2010082612A1 Imidazothiazole derivative having proline ring structure |
| 07/22/2010 | WO2010082531A1 Active blood coagulation factor inhibitor |
| 07/22/2010 | WO2010082050A1 Macrocyclic and 7-aminoalkyl-substituted benzoxazocines for treatment of hepatitis c infections |
| 07/22/2010 | WO2010062038A3 Tyrosine kinase inhibitor compound, isomer thereof or pharmaceutically allowable salt thereof, and pharmaceutical composition containing the same |
| 07/22/2010 | US20100184808 3-aza-bicyclo[3.3.0]octane compounds |
| 07/22/2010 | US20100184794 Fused heterocyclic compound |
| 07/22/2010 | US20100184772 Sulfonamide substituted pyrazoline compounds, their preparation and use as cb1 modulators |
| 07/22/2010 | US20100184751 Heterocyclic compounds for the treatment of tuberculosis |
| 07/22/2010 | US20100183600 RAF Inhibitors and Their Uses |
| 07/22/2010 | CA2750009A1 Imidazothiazole derivatives having proline ring structure |
| 07/21/2010 | EP2207781A1 Thiazolopyrimidine p13k inhibitor compounds and methods of use |
| 07/21/2010 | EP2207774A1 Triazole derivatives as scd inhibitors |
| 07/21/2010 | EP1973920B1 Process for the preparation of 5-amino-3h-thiazolo [4,5-d] pyrimidin-2-one |
| 07/21/2010 | EP1399445B9 Substituted pyrroloquinolines and pyridoquinolines as serotonin agonists and antagonists |
| 07/21/2010 | CN101781321A Method for synthesizing Largazole and analog thereof |
| 07/20/2010 | US7759372 benzimidazole derivatives having antiviral activities, used optionally in combination with a polymerase inhibitor and/or a protease inhibitor |
| 07/20/2010 | US7759340 Antibacterial agents |
| 07/15/2010 | WO2010079238A1 Heterotricyclic compounds as positive allosteric modulators of metabotropic glutamate receptors |
| 07/15/2010 | US20100179190 Bicyclic pyrazolo protein kinase modulators |
| 07/15/2010 | US20100179141 Novel jnk inhibitors |
| 07/15/2010 | US20100179135 3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives |
| 07/15/2010 | CA2748843A1 Heterotricyclic compounds as positive allosteric modulators of metabotropic glutamate receptors |
| 07/14/2010 | EP2206715A1 Fused heterotetracyclic compounds and use thereof as hcv polymerase inhibitor |
| 07/14/2010 | EP1863812B1 Dipeptidyl peptidase-iv inhibiting compounds, methods of preparing the same, and pharmaceutical compositions containing the same as an active agent |
| 07/14/2010 | CN101778846A 1,2-diamido-ethylene derivatives as orexin antagonists |
| 07/13/2010 | US7754743 Heteroarylcarbamoylbenzene derivatives |
| 07/13/2010 | US7754719 Substituted piperidine derivatives as somatostatin SST1 receptor antagonists |
| 07/13/2010 | CA2567776C Vasopressin v1a antagonists |
| 07/13/2010 | CA2444611C Novel insecticidal azoles |
| 07/13/2010 | CA2409697C Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| 07/08/2010 | WO2010078408A1 Heteroaryl compounds useful as raf kinase inhibitors |
| 07/08/2010 | WO2010077852A2 Method of inducing cleavage of amyloid precursor protein to form a novel fragment |
| 07/08/2010 | WO2010077663A2 Substituted tetracyclic 1h-indeno (1,2-b) pyridine-2 (5h)-one analogs thereof and uses thereof |
| 07/08/2010 | WO2010076525A1 Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof |
| 07/08/2010 | US20100173917 Urea derivatives as abl modulators |
| 07/08/2010 | US20100173778 3-Biphenyl-substituted-3-substituted-4-ketolactam and ketolactone and their utilization as pesticide |
| 07/08/2010 | US20100172960 Pro-drugs of nsaias with very high skin and membranes penetration rates and their new medicinal uses |
| 07/08/2010 | CA2748413A1 Derivatives of 2-pyridin-2-yl-pyrazol-3(2h)-one, preparation and therapeutic use thereof |
| 07/08/2010 | CA2748274A1 Heteroaryl compounds useful as raf kinase inhibitors |
| 07/07/2010 | EP2203448A1 Phenothiazine derivative having a double bond, method for the production thereof, and use thereof as a pharmaceutical |
| 07/07/2010 | EP2203424A1 Indole compounds bearing aryl or heteroaryl groups having sphingosine-1-phosphate (s1p) receptor biological activity |
| 07/07/2010 | CN101772506A macrocycles and their uses |
| 07/07/2010 | CN101768172A Optical active compound of anti-infective prulifloxacin and preparation method thereof |
| 07/06/2010 | US7750160 inhibit p38, MAP kinase interacting serine/threonine kinase 2 (MKNK2 kinase) and serine-threonine kinases (STKs); treating proliferative diseases including cancer, leukemias; e.g. N-(isoxazolyl)urea compounds and thiourea compounds |
| 07/06/2010 | US7750034 Aminocyclohexanes as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes |
| 07/06/2010 | US7750021 3-{[2-(2-Trifluoromethyl-biphenyl-4-yl)-benzo[b]thiophen-5-ylmethyl]-amino}-propionic acid, useful in the treatment or prevention diseases associated with endothelial differentiation, G-protein-coupled (EDG) receptor mediated signal transduction, such as acute or chronic transplant rejection |
| 07/06/2010 | US7750020 3-Cyclopentyl-2-(4-cyclopropylsulfamoyl-phenyl)-N-(5-methoxy-thiazolo[5,4-b]pyridin-2-yl)-propionamide; antidiabetic agent; insulin resistance, impaired glucose tolerance, obesity; with other hypolipidemic agent, anti-obesity and hypotensive agent |
| 07/01/2010 | WO2010075204A2 Gamma secretase modulators |
| 07/01/2010 | WO2010054024A3 1, 2 -thiazol yl derivatives as cannabinoid receptor ligands |
| 07/01/2010 | US20100168418 Novel nitrogenated heterocyclic compound and salt thereof |
| 07/01/2010 | US20100168101 Oxindole hydrazide modulators of protein tyrosine phosphatases (ptps) |
| 07/01/2010 | US20100163813 Long wavelength shifted benzotriazole uv-absorbers and their use |
| 07/01/2010 | CA2747750A1 Gamma secretase modulators |
| 06/30/2010 | EP2202222A2 Indene derivatives, their preparation and use as medicaments |
| 06/30/2010 | EP2201019A1 Process for the preparation of 6-substituted-imidazo ý2,1-b¨thiazole-5-sulfonyl halide |
| 06/30/2010 | EP2201018A2 Solid forms comprising n-(5-tert-butyl-isoxazol-3-yl)-n'-{4-ý7-(2-morpholin-4-yl-ethoxy)imidazoý2,1-b¨ý1,3¨benzothiazol-2-yl¨phenyl}urea, compositions thereof, and uses therewith |
| 06/30/2010 | EP2200440A1 Antibacterial amide and sulfonamide substituted heterocyclic urea compounds |
| 06/30/2010 | CN101765594A 1, 3-thiazol-2 (3H) -ylidene compounds as cannabinoid receptor ligands |
| 06/30/2010 | CN101765593A 2-iminoisothiazole derivatives as cannabinoid receptor ligands |
| 06/29/2010 | US7745449 Thieno-[2,3-d]pyrimidine and thieno-pyridazine compounds and methods of use |
| 06/24/2010 | WO2010071853A1 Thiazolopyridine sirtuin modulating compounds |
| 06/24/2010 | WO2010071822A1 Piperidine and piperazine derivatives and methods of use thereof |
| 06/24/2010 | WO2010071819A1 Bicyclic heterocyclic derivatives and methods of use thereof |
| 06/24/2010 | WO2010071783A1 Thiazoles as cannabinoid receptor ligands |
| 06/24/2010 | WO2010071164A1 Activated blood coagulation factor x (fxa) inhibitor |
| 06/24/2010 | WO2010071121A1 Method for producing diamine derivative |
| 06/24/2010 | WO2010070452A1 Fused imidazole carboxamides as trpv3 modulators |