Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
01/2010
01/28/2010US20100022500 Macrocyclic Lactams and Pharmaceutical Use Thereof
01/28/2010CA2731738A1 Imaging agents useful for identifying ad pathology
01/27/2010EP2147914A1 Aminodihydrothiazine derivatives substituted with cyclic groups
01/27/2010EP1940849B1 Isothiazolopyridin-3-ylenamines for combating animal pests
01/27/2010CN101633667A Lornoxicam compound and purifying method thereof
01/27/2010CN100584846C Dealkylated derivatives of pyrrolo[2,1-b]benzothiazepines with atypical antipsychotic activity
01/26/2010US7652020 novel hydantoin derivatives to inhibit matrix metalloproteinases (MMPs), a disintegrin and metalloproteases (ADAMs) and/or tumor necrosis factor alpha converting enzyme (TACE) and in so doing prevent the release of tumor necrosis factor alpha (TNF- alpha ); autoimmune diseases; side effect reduction
01/26/2010US7652010 Azabicyclic aryl derivatives and their medical use
01/26/2010US7652008 Tricyclic benzopyran compound as anti-arrhythmic agents
01/21/2010WO2010009166A1 Oxindolyl inhibitor compounds
01/21/2010WO2010008843A1 Apoptosis signal-regulating kinase 1 inhibitors
01/21/2010WO2010008558A1 Compounds and methods of inducing apoptosis via interaction with chaperonin cct
01/21/2010WO2009137130A3 Antibacterial fluoroquinolone analogs
01/21/2010WO2009112677A3 Bicyclic derivatives of azabicyclic carboxamides, preparation thereof and therapeutic use thereof
01/21/2010WO2009069147A4 Improved process for preparation of triazol-benzodiazepine derivatives
01/21/2010US20100016386 Selective glycosidase inhibitors and uses thereof
01/21/2010US20100016304 Glucokinase activator
01/21/2010US20100016287 Compounds having affinity for dopamine d3 receptor and uses thereof"
01/21/2010US20100016233 Heterocyclic Aromatic Compounds Useful As Growth Hormone Secretagogues
01/21/2010CA2728228A1 Oxindolyl inhibitor compounds
01/19/2010US7649097 Tetracyclic arylsulfonyl indoles having serotonin receptor affinity useful as therapeutic agents, process for their preparation and pharmaceutical compositions containing them
01/19/2010US7648985 Oxabispidine compounds and their use in the treatment of cardiac arrhythmias
01/19/2010US7648980 3-{2-[3-fluoro-6-(methyloxy)-1,5-naphthyridin-4-yl]ethyl}-8-oxa-3-azabicyclo[3.2.1]oct-6-yl)amino]methyl}-2H-pyrido[3,2-b][1,4]thiazin-3(4H)-one; antibiotic resistance; Staphylococcus aureus, Streptococcus pneumoniae and pyogenes, Enterococcus; Haemophilus influenzae, Moraxella catarrhalis, E-coli
01/19/2010US7648975 Macrocyclic quinazoline derivatives as antiproliferative agents
01/19/2010CA2402751C Decahydro-isoquinolines
01/19/2010CA2239904C Inhibitors of interleukin-1.beta. converting enzyme
01/14/2010WO2010004507A1 Thiazolidine compounds as orexin receptor antagonists
01/14/2010WO2010003658A1 Macrocyclic indole derivatives useful as hepatitis c virus inhibitors
01/14/2010WO2009121872A3 Tetrahydroisoquinolines, pharmaceutical compositions containing them, and their use in therapy
01/14/2010US20100009977 Process for the preparation of (R)-(+)-4-(Ethylamino)-3,4-dihydro-2-(3-methoxypropyl)-2H-thieno[3,2-e]-1,2-thiazine-6-sulfonamide-1,1-dioxide.
01/14/2010US20100009969 Fused Oxazoles & Thiazoles As Histamine H3- Receptor Ligands
01/14/2010US20100008866 Cis-cyclohexyl substituted pyrimidinone derivatives
01/14/2010CA2729985A1 Thiazolidine compounds as orexin receptor antagonists
01/14/2010CA2729307A1 Macrocyclic indole derivatives useful as hepatitis c virus inhibitors
01/13/2010EP1641805B1 Thiazolo-, oxazalo and imidazolo-quinazoline compounds capable of inhibiting protein kinases
01/13/2010CN101624396A Spiro-compound containing thiadiazoline and furanring, preparation method and germicide application thereof
01/12/2010US7645881 Methods for treating hepatitis C
01/12/2010US7645766 Method for treatment of depression and depressive mood disorders
01/12/2010CA2407838C Pyrano, piperidino, and thiopyrano compounds and methods of use
01/07/2010WO2010003048A1 Benzimidazoles and related analogs as sirtuin modulators
01/07/2010WO2010000030A1 Thiazopyrimidinones and uses thereof
01/07/2010WO2009118712A3 Novel dihydroxypyrrolidine derivatives as anti-cancer agents
01/07/2010US20100004299 Imidazo[2,1-b]thiazoles and their use as pharmaceuticals
01/07/2010US20100004230 Azatricyclic compounds and their use
01/07/2010US20100004222 Amide Derivatives as Ion-Channel Ligands and Pharmaceutical Compositions and Methods of Using the Same
01/07/2010US20100004221 Thiazepine derivative
01/07/2010US20100004159 Substituted imidazolone derivatives, preparations and uses
01/07/2010CA2729649A1 Thiazopyrimidinones and uses thereof
01/07/2010CA2729128A1 Benzimidazoles and related analogs as sirtuin modulators
01/06/2010CN101619070A Preparation method of tenoxicam
01/06/2010CN100577651C Lactam compound and medicinal use thereof
01/05/2010US7642359 Pyrazolyl-substituted heterocycles and their use as phytosanitary products
12/2009
12/31/2009US20090326221 New oxabispidine compunds useful in the treatment of cardiac arrhythmias
12/31/2009US20090324744 Effective Antitumor Treatments
12/31/2009US20090324625 Heterocyclic Aromatic Compounds Useful As Growth Hormone Secretagogues
12/30/2009CN101613362A 3-carbonyl-6-ethoxycarbonyl-thiazole pyrimidine compound and synthesis method and application thereof
12/29/2009US7638529 Heterocyclic compounds, their preparation and their use as medicaments, in particular as anti-bacterial agents
12/29/2009US7638513 inhibitors of matrix metalloproteinases, aggrecanases, tumor necrosis factor-alpha converting enzyme, and tumor necrosis factors
12/29/2009CA2338543C Method of direct identification of compound efficacy at a g protein-coupled orphan receptor
12/24/2009US20090318704 Processes for the Preparation of N-(2-Acetyl-4,6-Dimethylphenyl)-3--2-Thiophenecarboxamide
12/24/2009US20090318513 Compounds exhibiting thrombopoietin receptor agonism
12/24/2009US20090318442 Thiazolyl-and oxazolyl-isoquinolinones and methods for using them
12/24/2009US20090318425 Apoptosis signal-regulating kinase 1 inhibitors
12/23/2009WO2009155402A1 Thiazolyl- and oxazolyl-isoquinolinones and methods for using them
12/23/2009EP1296972B1 Arylmethylamine derivatives for use as tryptase inhibitors
12/23/2009CN101611038A 2-quinolinone and 2-quinoxalinone- derivatives and their use as antibacterial agents
12/23/2009CN101611025A 5,6-ring annulated indole derivatives and methods of use thereof
12/23/2009CA2728454A1 Thiazolyl- and oxazolyl-isoquinolinones and methods for using them
12/23/2009CA2728408A1 Substituted pyridazine carboxamide compounds as kinase inhibitor compounds
12/23/2009CA2728046A1 S1p1 receptor agonists and use thereof
12/23/2009CA2727928A1 Inhibitors of janus kinases
12/22/2009US7635695 4-Amino-2-(4-methyl-thiophen-2-yl)thieno[3,2-c]pyridine-7-carboxylic acid amide; 4-amino-2-cyclopent-1-enyl-thieno[3,2-c]pyridine-7-carboxylic acid amide; for therapy and prophylaxis of disease or condition associated with inflammation, a metabolic disorder, infection, cancer or an immune disease
12/22/2009US7635394 Composition for the dyeing of keratin fibers comprising at least one 3-amino-pyrazolopyridine derivatives
12/22/2009CA2290744C Cyclic diamine compounds and medicine containing the same
12/17/2009WO2009151069A1 Imidazothiazole derivative having 4,7-diazaspiro[2.5]octane ring structure
12/17/2009WO2009150240A1 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
12/17/2009WO2009121036A3 Substituted aryl pyrimidinone derivatives
12/17/2009US20090312543 Pyrazole compounds useful as protein kinase inhibitors
12/17/2009US20090312374 Derivatives of 4,6-disubstituted 1,2,4-triazolo- 1,3,4-thiadiazole, a process and uses thereof
12/17/2009US20090312344 Arylpiperazine derivatives as adrenergic receptor antagonists
12/17/2009US20090312310 Imidazothiazole derivatives
12/17/2009CA2727062A1 Imidazopyridine derivatives as inhibitors of receptor tyrosine kinases
12/17/2009CA2727032A1 Novel tricyclic compounds
12/17/2009CA2726158A1 Compounds and compositions useful for the treatment of malaria
12/16/2009CN101605798A Imidazothiazole derivatives
12/15/2009US7632830 Lactam compounds and pharmaceutical use thereof
12/15/2009CA2529611C Pyrimidine derivatives for the treatment of abnormal cell growth
12/10/2009WO2009147616A1 [4-(1-amino-ethyl) -cyclohexyl] -methyl-amine and [6-(1-amino-ethyl) -tetrahydro- pyran-3-yl] -methyl-amine derivatives as antibacterials
12/10/2009WO2009147431A1 Thiazolo [5, 4-b] pyridine and oxazolo [5, 4-b] pyridine derivatives as antibacterial agents
12/10/2009US20090306057 [1,2,4]thiadiazine 1,1-dioxide compounds
12/10/2009CA2725689A1 Thiazolo [5,4-b] pyridine and oxazolo [5,4-b] pyridine derivatives as antibacterial agents
12/10/2009CA2725616A1 [4-(1-amino-ethyl) -cyclohexyl] -methyl-amine and [6-(1-amino-ethyl) -tetrahydro- pyran-3-yl] -methyl-amine derivatives as antibacterials
12/09/2009EP2130826A1 Annulins A, B, C or analogs as indoleamine 2,3-dioxygenase (IDO) inhibitors for treatment of cancer
12/09/2009EP2130820A1 Antipruritics
12/09/2009EP2129677A1 Heterocyclic cyclopamine analogs and methods of use thereof
12/09/2009EP1692140B1 Compositions useful as inhibitors of protein kinases
12/08/2009CA2422354C Pyrazole compounds useful as protein kinase inhibitors
12/08/2009CA2422342C Novel amide derivatives and medicinal use thereof
12/03/2009WO2009144159A1 Substituted pyridin-4-yl-methyl sulfonamidesas fungicides
12/03/2009WO2009069147A3 Improved process for preparation of triazol-benzodiazepine derivatives
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