| Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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| 08/14/2008 | CA2677015A1 Hcv inhibiting macrocyclic phenylcarbamates |
| 08/13/2008 | EP1956020A2 1-[2-(heterocyclyl-aminomethyl)-piperidin-1-YL]-1-(2-methyl-5-phenyl-heterocyclyl)-methanone derivatives and related compounds as orexin-1 antagonists for the treatment of obesity |
| 08/13/2008 | EP1954698A1 Spirocyclic compounds as hdac inhibitors |
| 08/13/2008 | EP1954132A2 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
| 08/13/2008 | EP1954128A2 Diphenylmethane derivatives as inhibitors of leukotriene biosynthesis |
| 08/13/2008 | EP1585749B1 Diazepinoindole derivatives as kinase inhibitors |
| 08/13/2008 | EP1572672B1 Benzoxazocines and their use as monoamine-reuptake inhibitors |
| 08/13/2008 | EP1495030B1 Non-steroidal progesterone receptor modulators |
| 08/13/2008 | EP1452528B1 Xanthine oxidase inhibitors |
| 08/13/2008 | CN101243093A New oxabispidine compounds for the treatment of cardiac arrhythmias |
| 08/13/2008 | CN101243068A Compounds for the treatment of multi-drug resistant bacterial infections |
| 08/13/2008 | CN101239953A Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans |
| 08/12/2008 | US7411063 Process for preparation of maytansinol |
| 08/12/2008 | US7410986 For therapy of inflammatory symptoms; tumors, ischemia and tumor |
| 08/12/2008 | US7410966 Use of and some novel imidazopyridines |
| 08/12/2008 | US7410933 Substituted thiene-3-ylsulphonylamino(thio)carbonyl-triazolin(thi)ones |
| 08/12/2008 | CA2398111C 4-pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy |
| 08/12/2008 | CA2359819C 2-oxy-benzoxazinone derivatives for the treatment of obesity |
| 08/07/2008 | WO2008093064A1 L-ALANINE DERIVATIVES AS α5 BETA 1 ANTAGONISTS |
| 08/07/2008 | WO2008092887A1 I-oxa-3-azaspiro (4.5) decan-2-one and 1-oxa-3, 8-diazaspiro (4.5) decan-2-one derivatives for the treatment of eating disorders |
| 08/07/2008 | US20080188511 Rapamycin; the 40-hydroxy position is derivatised as a carboxylic acid ester, as an ether, as a phosphate ester, as a phosphinate ester, as an acetal or as a gycosyl; transplantation rejection, graft vs. host disease, autoimmune disorders, inflammation, vascular, fibrotic diseases |
| 08/07/2008 | US20080188470 Oxazolidinone Derivatives as Antimicrobials |
| 08/07/2008 | US20080188371 use as pesticides and/or herbicides and/or microbicides; for the selective control of weeds; synergistic; low application rates and concentrations; in particular in cereals (especially wheat) |
| 08/06/2008 | EP1953154A1 Morpholine type cinnamide compound |
| 08/06/2008 | EP1951731A1 Azacyclohexane derivatives as inhibitors of stearoyl-coenzyme a delta-9 desaturase |
| 08/06/2008 | EP1951730A1 Heteroalkyl linked pyrimidine derivatives |
| 08/06/2008 | EP1951729A1 Oxygen linked pyrimidine derivatives |
| 08/06/2008 | EP1951228A2 Bicyclic spirohydantoin cgrp receptor antagonists |
| 08/06/2008 | CN101238136A Purification of tacrolimus on supports of vegetable origin |
| 08/06/2008 | CN101238135A Oxazolidinone-quinolone hybrids as antibacterial compounds |
| 08/06/2008 | CN101238134A Process for the preparation of sulfonic acid salts of oxabispidines |
| 08/06/2008 | CN101238131A Bridged piperazine and piperidine derivatives as CCR1 antagonists |
| 08/06/2008 | CN101235131A Method for preparing benzoxazine intermediate containing propargyl ether and resin thereof |
| 08/06/2008 | CN100408573C Pyrazole compounds useful as protein kinase inhibitors |
| 08/06/2008 | CN100408564C Pyrazole derivatives for treating HIV |
| 08/05/2008 | US7408063 1,8-annelated quinoline derivatives substituted with carbon-linked triazoles as farnesyl transferase inhibitors |
| 08/05/2008 | US7407972 e.g. 4,5-Dihydro-pyrazole-1,5-dicarboxylic acid 1-[(4-chloro-phenyl)-amide] 5-[(3-fluoro-2'-methanesulfonyl-biphenyl-4-yl)-amide]; anticoagulant, thrombolytic agent; thrombus formation within blood vessels; cardiovascular disease |
| 08/05/2008 | US7407968 Compounds |
| 08/05/2008 | US7407954 Thieno-(1,3)-oxazin-4-ones with lipase inhibiting activity |
| 08/05/2008 | US7407949 4-(2-Cyclopropyl-ethyl)-piperazine-1-carboxylic acid 2-methyl-4-(3-methyl-4,10-dihydro-3H-2,3,4,9-tetraaza-benzo[f]azulene-9-carbonyl)-benzylamide; inter alia, primary dysmenorrhoea, male erectile dysfunction |
| 08/05/2008 | CA2279319C Benzofurazan compounds which enhance ampa receptor activity |
| 08/05/2008 | CA2153984C Process for the manufacture of a tricyclic compound |
| 07/31/2008 | US20080182868 Novel chemical compounds |
| 07/31/2008 | US20080182867 Administering one or more rapamycin derivatives (including rapamycin and 40-O-(2-hydroxy)ethyl-rapamycin); lymphocytic leukemia, lymphoma, Epstein-Barr virus, inhibiting graft rejection and metastasis; drug screening |
| 07/31/2008 | US20080182842 L-alanine derivatives as a5beta1 antagonists |
| 07/30/2008 | EP1950206A1 Benzoxazocines and their use as monoamine-reuptake inhibitors |
| 07/30/2008 | EP1950199A1 Proline derivatives and use thereof as drugs |
| 07/30/2008 | EP1949100A1 Method of tacrolimus extraction and quantification using aqueous detergents |
| 07/30/2008 | EP1948666A1 Hiv integrase inhibitors |
| 07/30/2008 | EP1948660A1 Tetracyclic indole derivatives as antiviral agents |
| 07/30/2008 | EP1948626A1 Process for the preparation of delmopinol and derivatives thereof |
| 07/30/2008 | EP1948621A1 Hiv integrase inhibitors |
| 07/30/2008 | CN101233141A Ascomycin crystalline forms and preparation thereof |
| 07/30/2008 | CN101230066A Antidepressant piperidine derivatives of heterocycle-fused benzodioxans |
| 07/30/2008 | CN100406454C Pyrazole compounds useful as protein kinase inhibitors. |
| 07/29/2008 | US7405302 5-lipoxygenase-activating protein (FLAP) inhibitors |
| 07/29/2008 | US7405225 Substituted 3-amino-thieno[2,3-b]pyridine-2-carboxylic acid amide compounds and processes for preparing and their uses |
| 07/29/2008 | US7405212 Helix mimetics and composition and methods related thereto |
| 07/29/2008 | CA2432222C Pyrazole compounds useful as protein kinase inhibitors |
| 07/29/2008 | CA2432132C Pyrazole compounds useful as protein kinase inhibitors |
| 07/24/2008 | US20080176839 e.g. N-benzyl-2-(3,4-dichlorophenyl)-4-(6-fluoro-2-oxo-1,2-dihydro-1'H-spiro[3,1-benzoxazine-4,4'-piperidin]-1'-yl)-N-methylbutanamide; neurokinin 3 receptor antagonist; antidepressant, anxiolytic agent, analgesic; psychosis, Parkinson's disease, schizophrenia, attention deficit hyperactivity disorder |
| 07/24/2008 | US20080176829 e.g. 2,5-methylene-9-(phenylsulfonyl)-1,2,3,4,5,9-hexahydro[1,5]oxazocino[3,2-e]indole; serotonin receptors antagonist or partial agonist; metabolic diseases, e.g. obesity, insulin resisitance, type 2 diabetes, eating disorders; antidepressant, anxiolytic agent; cosmetics |
| 07/24/2008 | US20080175884 Polymer coatings as carriers for the drug delivery of a methosyaminocarbonyloxy derivative of rapamycin and another drug(s) such as an antiproliferative agent, anticoagulant, etc.; reduces restenosis in vasculature procedures to a level of 0-25%; coronary/periferal stents; grafts ; balloons |
| 07/23/2008 | EP1947102A1 Compositions comprising diazepinoindole derivatives as kinase inhibitors |
| 07/23/2008 | EP1945786A2 Fermentation processes for the preparation of tacrolimus |
| 07/23/2008 | EP1945647A2 Processes for preparation of maytansinol |
| 07/23/2008 | EP1945641A1 Hepatitis c virus inhibitors |
| 07/23/2008 | CN101228141A Tetrahydrobenzoxazines as stabilisers |
| 07/23/2008 | CN100403900C Mitotic kinesin inhibitors |
| 07/22/2008 | US7402593 (-)-5-methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridyl)methyl]sulfinyl]imidazo[4,5-b]pyridine; proton pump inhibitor (PPI) to treat gastro-oesophageal reflux, digestive bleeding and dyspepsia; enantiomer; long duration of action; longer half-life in plasma; oxidation of sulfide followed by salt formation |
| 07/22/2008 | US7402590 Spiroazacyclic compounds as monoamine receptor modulators |
| 07/22/2008 | US7402421 Recombinant methods and materials for producing epothilone and epothilone derivatives |
| 07/22/2008 | CA2436942C Method of manufacturing substance gm-95 |
| 07/17/2008 | WO2008086510A2 Process to make lestaurtinib |
| 07/17/2008 | WO2008086404A1 5-pyridinone substituted indazoles |
| 07/17/2008 | WO2008085480A1 A novel and economical process for preparing (s,s)-2, 8-diazabicyclo[4.3.0]nonane and its enantiomer |
| 07/17/2008 | WO2008062379A3 4- (2-oxo-oxazolidin-3yl)-phenoxymethyle derivativeas as antibacterials |
| 07/17/2008 | WO2008062379A2 4- (2-oxo-oxazolidin-3yl)-phenoxymethyle derivativeas as antibacterials |
| 07/17/2008 | US20080171868 CRYSTALLINE K-252b, SODIUM SALT, METHANOLATE PENTAHYDRATE |
| 07/17/2008 | US20080171867 (9S-(9 alpha ,10 beta ,12 alpha ))-2,3,9,10,11,12-hexahydro-10-hydroxy-10-(methoxycarbonyl)-9-methyl-9,12-epoxy-1H-diindolo[1,2,3-fg:3',2',1'-k1]pyrrolo[3,4-i][1,6]benzodiazocin-1-one bis(tetrahydrofuranate) |
| 07/17/2008 | US20080171866 CRYSTALLINE K-252a BIS(METHANOLATE) |
| 07/17/2008 | US20080171865 Method of targeting specific cell populations using cell-binding agent maytansinoid conjugates linked via a non-cleavable linker, said conjugates and methods of making said conjugates |
| 07/17/2008 | US20080171040 Antibody-drug conjugates and methods |
| 07/17/2008 | CA2673654A1 5-pyridinone substituted indazoles |
| 07/16/2008 | EP1943222A1 Antibacterial active 5-chinolin derivative |
| 07/16/2008 | EP1942899A2 Mitotic kinesin inhibitors |
| 07/16/2008 | EP1709044B1 Oxazolidinone-quinolone hybrid antibiotics |
| 07/16/2008 | EP1390372B1 1-oxa-3,9-diaza-spiro'5,5]undecan-2-ones derivatives and its use as antagonist of the neurikinin receptor |
| 07/16/2008 | CN101223179A Biologically active compounds obtainable from sorangium cellulosum |
| 07/16/2008 | CN101223175A Diazabenzo[de]anthracen-3-one compounds and methods for inhibiting PARP |
| 07/16/2008 | CN101223168A Heterocyclic JANUS kinase 3 inhibitors |
| 07/16/2008 | CN101220044A Telomerase inhibitor, preparation method and application thereof |
| 07/16/2008 | CN101220039A Chiral center aza ring carbene precursor salt with camphor framework, synthesizing method and uses thereof |
| 07/16/2008 | CN101220035A A kind of alkaloid, method for preparing the same and application in antineoplastic or antimicrobial aspects |
| 07/16/2008 | CN101220003A Propargylterminated compounds with benzoxazole ring and method for producing the same |
| 07/16/2008 | CN100402534C Tricycle compounds and its application in making medicine |
| 07/16/2008 | CN100402499C 2-iminopyrrolidine derivatives |
| 07/15/2008 | US7399866 2-(Imidazol-1-ylalkyl)-3H-quinazolin-4-one derivatives; mitotic kinesin KSP inhibitors; anticarcinogenic, antiinflammatory, and antiproliferative agents |
| 07/15/2008 | US7399765 Substituted diazabicycloalkane derivatives |
| 07/15/2008 | US7399480 Methods of administering tetrazole-containing rapamycin analogs with other therapeutic substances using medical devices |