Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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07/15/2014 | US8779163 Synthesis of UDP-Glucose: N-acylsphingosine glucosyl transferase inhibitors |
07/15/2014 | US8778964 Hydroxy-substituted imidazo[1,2-a]-pyridinecarboxamides and their use |
07/15/2014 | US8778962 Treatment of solid tumors with rapamycin derivatives |
07/15/2014 | US8778961 O-methylated rapamycin derivatives for alleviation and inhibition of lymphoproliferative disorders |
07/15/2014 | US8778932 Dihydro-oxazolobenzodiazepinone compounds, a process for there preparation and pharmaceutical compositions containing them |
07/15/2014 | US8778920 3-cyano-quinoline derivatives with antiproliferative activity |
07/15/2014 | CA2674460C 3-substituted-h.2.31-benzotriazinone compound for enhancing glutamatergic synaptic responses |
07/15/2014 | CA2592119C Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-4-yl-amines as janus kinase inhibitors |
07/15/2014 | CA2563959C (1,10b-dihydro-2-(aminocarbonyl-phenyl)-5h-pyrazolo[1,5-c][1,3]benzoxazin-5-yl)phenyl methanone derivatives as hiv viral replication inhibitors |
07/10/2014 | US20140194415 Fatty acid synthase inhibitors |
07/10/2014 | US20140194408 Heteroaryl pyridone and aza-pyridone compounds |
07/10/2014 | US20140194349 HIV Protease Inhibiting Compounds |
07/09/2014 | EP2752417A1 Spiro-oxindole compounds and their uses as therapeutic agents |
07/09/2014 | EP2751115A1 (THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS |
07/09/2014 | CN101903377B 6H-二苯并[b,e]氧杂环庚烷衍生的非类固醇矿皮质激素受体拮抗剂 6H- dibenz [b, e] dioxepan-derived non-steroidal glucocorticoid receptor antagonists mines |
07/09/2014 | CN101541811B 吡唑并嘧啶衍生物 Pyrazolo pyrimidine derivatives |
07/08/2014 | US8772316 Substituted 6,7-dialkoxy-3-isoquinolinol derivatives as inhibitors of phosphodiesterase 10 (PDE10A) |
07/08/2014 | US8772307 Substituted spiro compounds and their use for producing pain-relief medicaments |
07/08/2014 | US8772301 Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof |
07/08/2014 | US8772283 Imidazo-oxazine compound or salt thereof |
07/08/2014 | US8772272 Pyrido-and pyrimidopyrimidine derivatives as anti-proliferative agents |
07/08/2014 | CA2735478C Malonyl-coa decarboxylase inhibitors useful as metabolic modulators |
07/08/2014 | CA2638095C New compounds |
07/08/2014 | CA2617107C Olanzapine analogs and methods of use thereof |
07/08/2014 | CA2568213C Composition and method for the treatment of tauopathies |
07/03/2014 | WO2014104407A1 Fused oxazole compounds and use thereof for pest control |
07/03/2014 | WO2014102817A1 Substituted phthalazin-1 (2h)-one derivatives as selective inhibitors of poly (adp-ribose) polymerase-1 |
07/03/2014 | WO2014102630A1 Solid form of dihydro-pyrido-oxazine derivative |
07/03/2014 | WO2014102589A1 Quinazolin-4(3h)-one-type piperidine compounds and uses thereof |
07/03/2014 | WO2014101765A1 Benzoxazine oxazolidinone compound, preparation method and application thereof |
07/03/2014 | US20140187772 Pyrazole compounds useful as protein kinase inhibitors |
07/03/2014 | US20140187769 Oxadiazoanthracene Compounds for the Treatment of Diabetes |
07/03/2014 | US20140187574 Use of rapamycin derivatives in vasculopathies and xenotransplantation |
07/03/2014 | US20140187542 Amino group-containing pyrrolidinone derivative |
07/02/2014 | EP2748170A1 1,4-diazabicyclo[3.2.2]nonanes as neuronal nicotinic acetylcholine receptor ligands |
07/02/2014 | EP2748158A1 Radiolabeled compounds and their use as radiotracers for quantitative imaging of phosphodiesterase (pde10a) in mammals |
07/02/2014 | CN103896963A 苯并噁嗪噁唑烷酮类化合物及其制备方法和用途 Benzoxazine oxazolidinone compound and its preparation and use |
07/02/2014 | CN103896816A 一种手性烯丙基硫醇羧酸酯及其合成方法 Chiral allyl mercaptan acid esters and synthetic method |
07/02/2014 | CN102234288B 唑他莫司的制备方法 Azole preparation tamoxifen Division |
07/02/2014 | CN102015686B 杂环化合物及其用途 Heterocyclic compounds and their use |
07/02/2014 | CN101784516B 作为凝血因子抑制剂的二肽类似物 As a coagulation factor inhibitor dipeptide analogs |
07/01/2014 | US8765799 Streptospirole derivatives |
06/26/2014 | WO2014100646A1 1,4-pyridone compounds |
06/26/2014 | WO2014100351A2 8'-hydroxy-dihydroergotamine compounds and compositions |
06/26/2014 | WO2014100323A1 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
06/26/2014 | WO2014099586A1 4-pyridinonetriazine derivatives as hiv integrase inhibitors |
06/26/2014 | WO2014098188A1 METHOD FOR PRODUCING cis-5-HYDROXY-2-PIPERIDINECARBOXYLIC ACID DERIVATIVE, AND METHOD FOR PURIFYING cis-5-HYDROXY-2-PIPERIDINECARBOXYLIC ACID |
06/26/2014 | WO2014097711A1 Organic electroluminescent element and electronic device |
06/26/2014 | WO2014097188A1 Compounds of 2,3-dihydro-4h-1,3-benzoxazine-4-one, method for preparing them and pharmaceutical form comprising them |
06/26/2014 | WO2014097147A1 Tricyclic compounds as cftr inhibitors |
06/26/2014 | WO2014096369A1 Spiroisoxazoline compounds having an activity potentiating the activity of an antibiotic |
06/26/2014 | WO2014094354A1 Preparation of maytansinoid esters |
06/26/2014 | WO2014094353A1 Maytansinoid derivatives |
06/26/2014 | US20140179917 Preparation of maytansinoid esters |
06/26/2014 | US20140179916 Forms of rifaximin and uses thereof |
06/26/2014 | US20140179705 8'-hydroxy-dihydroergotamine compounds and compositions |
06/26/2014 | US20140179704 8'-hydroxy-dihydroergotamine compounds and compositions |
06/26/2014 | US20140179695 Chromane compounds |
06/26/2014 | US20140179682 Metabotrophic glutamate receptor 5 modulators and methods of use thereof |
06/26/2014 | US20140179680 Substituted Imidazopyridines as HDM2 Inhibitors |
06/26/2014 | US20140179677 Therapeutic agent for ectopic pregnancy |
06/26/2014 | US20140179675 Quinolone compound |
06/26/2014 | US20140179674 Imidazopyridazinecarbonitriles useful as kinase inhibitors |
06/26/2014 | US20140179671 Fused ring azadecalin glucocorticoid receptor modulators |
06/26/2014 | US20140178415 Maytansinoid derivatives |
06/26/2014 | US20140178412 Compounds and methods for the treatment of egfr positive diseases |
06/25/2014 | EP2746285A1 Process for the preparation of aurora kinase inhibitors |
06/25/2014 | EP2744788A1 Benzopiperazine derivatives as cetp inhibitors |
06/25/2014 | CN103889974A 放射性标记的化合物和它们在哺乳动物中作为磷酸二酯酶(pde10a)的定量成像的放射示踪剂的用途 Radiolabeled compounds and their use as phosphodiesterase (pde10a) quantitative imaging radiotracer in a mammal The use |
06/25/2014 | CN103889951A 唑类衍生物 Azole derivative |
06/25/2014 | CN103881061A 一种双极性共聚物蓝光主体材料及其制备方法与有机电致发光器件 A bipolar copolymer blue host material and preparation method and organic electroluminescent devices |
06/25/2014 | CN103880862A 丙型肝炎病毒复制的抑制剂 Inhibitors of hepatitis C virus replication |
06/25/2014 | CN103880861A 一种作用于FGF受体的4,6-二甲基-噁唑并[5,4-d]嘧啶-5,7(4H,6H)-二酮衍生物 One kind of effect on FGF receptors 4,6-dimethyl - oxazolo [5,4-d] pyrimidine -5,7 (4H, 6H) - dione derivatives |
06/25/2014 | CN103880576A 一种脱除热敏性固体药物中残留溶剂的装置 An apparatus for heat-sensitive drugs in solid residual solvent removal |
06/25/2014 | CN102482258B α-螺旋模拟物和与其相关的方法 α- helix mimetics, and methods related thereto |
06/25/2014 | CN102333777B 含氮的稠合杂环化合物及其作为β淀粉样蛋白生成抑制剂的用途 Nitrogen-containing fused heterocyclic compounds and their use as inhibitors of β-amyloid protein production purposes |
06/25/2014 | CN101948475B 异黄酮衍生物-色烯(满)并噁嗪类化合物及其制备方法和应用 Isoflavone Derivatives - chromene (full) and oxazine compound and preparation method and application |
06/25/2014 | CN101759645B p38抑制剂及它们的使用方法 p38 inhibitors and methods for their use |
06/24/2014 | US8759513 Polymorphic form of rifaximin and process for its preparation |
06/24/2014 | US8759512 Methods of preparation of macrocyclic compounds |
06/24/2014 | US8759370 O-methylated rapamycin derivatives for alleviation and inhibition of lymphoproliferative disorders |
06/24/2014 | US8759341 Bi- and tricyclic indazole-substituted 1,4-dihydropyridine derivatives and uses thereof |
06/24/2014 | US8759337 Gamma secretase modulators |
06/19/2014 | WO2014092544A1 A sensor for determining calcium ions |
06/19/2014 | WO2014091415A1 Indole carboxamide derivatives as p2x7 receptor antagonists |
06/19/2014 | WO2014089904A1 Triazinone compounds |
06/19/2014 | US20140171639 Trpm8 antagonists and their use in treatments |
06/19/2014 | US20140171427 Heterocyclic chromene-spirocyclic piperidine amides as modulators of ion channels |
06/19/2014 | US20140171425 Quinazoline-2,4-dione derivatives |
06/19/2014 | US20140171412 Tricyclic compounds |
06/19/2014 | US20140171411 (THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS |
06/19/2014 | US20140171410 Batrachotoxin Analogues, Compositions, Uses, and Preparation Thereof |
06/19/2014 | US20140170111 Fused tetracycle derivatives and methods of use thereof for the treatment of viral diseases |
06/18/2014 | EP2742936A1 Fused heterocyclic compound and use thereof |
06/18/2014 | EP2742051A1 Amorphous form of dolutegravir |
06/18/2014 | EP2742042A1 Quinazoline-2,4-dione derivatives |
06/18/2014 | CN103874702A Novel substituted indole derivatives as gamma secretase modulators |
06/18/2014 | CN103864818A Preparation methods of drug intermediates |
06/18/2014 | CN103864754A Five-membered azole heterocycle compound, preparation method, drug composition and use thereof |
06/18/2014 | CN103864712A Method for synthesizing compound 3-(3-amino furazan-4-yl)-4-hydroxy-1-oxygen-2, 4-diaza-spiran-2-alkene |