Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960) |
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08/12/2014 | US8802712 Pyrazoloquinolines |
08/12/2014 | US8802695 Apoptosis signal-regulating kinase 1 inhibitors |
08/12/2014 | US8802674 Aminopyrimidine derivatives as LRRK2 modulators |
08/12/2014 | US8802667 Benzodiazepine derivatives |
08/07/2014 | US20140221379 N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS |
08/07/2014 | US20140221377 Quinuclidine Compounds as Alpha-7 Nicotinic Acetylcholine Receptor Ligands |
08/07/2014 | US20140221365 Alkylated piperazine compounds |
08/07/2014 | US20140221356 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
08/07/2014 | US20140221355 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
08/07/2014 | US20140221352 Compositions and methods for inhibition of the jak pathway |
08/07/2014 | US20140221350 Cyclohexyl-4H,6H-5-oxa-2,3,10b-triaza-benzo[e]azulenes as V1a antagonists |
08/07/2014 | US20140221348 Novel bicyclic antibiotics |
08/07/2014 | US20140221338 Novel macrocycles as factor xia inhibitors |
08/07/2014 | US20140221322 Heteroaryl substituted urea modulators of fatty acid amide hydrolase |
08/07/2014 | US20140221310 Flap modulators |
08/06/2014 | EP2762480A1 Oxazolidinone antibiotics containing fused ring |
08/06/2014 | EP2762140A1 Treatment of solid brain tumours with a rapamycin derivative |
08/06/2014 | EP2760872A1 Compounds for the treatment of hepatitis c |
08/06/2014 | EP2760871A1 Oxy-cyclohexyl-4h,6h-5-oxa-2,3,10b-triaza-benzo[e]azulenes as v1a antagonists |
08/06/2014 | EP2760870A1 Substituted bicyclic heteroaryl compounds |
08/06/2014 | EP2760867A1 Macrocyclic flt3 kinase inhibitors |
08/06/2014 | EP2760857A1 Pyrazol-4-yl-heterocyclyl-carboxamide compounds and methods of use |
08/06/2014 | EP2760453A1 Macrocyclic lrrk2 kinase inhibitors |
08/06/2014 | CN103974957A 具有整合酶抑制活性的多环吡啶酮衍生物 Having an integrase inhibitory activity of polycyclic pyridine derivatives |
08/06/2014 | CN103974948A 在治疗过度增殖性疾病中用作bub1激酶抑制剂的取代的苄基吲唑 Substituted bub1 kinase inhibitors used in the treatment of hyperproliferative diseases benzyl indazole |
08/06/2014 | CN103965213A 7,8-二氢-6H-[1,4]噁嗪[3,2-g]喹唑啉类衍生物及其制备方法和用途 7,8-dihydro -6H- [1,4] oxazine [3,2-g] quinazoline derivatives and their preparation and use |
08/06/2014 | CN103965212A 6,7,8,9-四氢-[1,4]氧氮杂卓[3,2-g]喹唑啉类衍生物及其制备方法和用途 6,7,8,9-tetrahydro - [1,4] oxazepine [3,2-g] quinazoline derivatives and their preparation and use |
08/06/2014 | CN103965211A 含喹唑啉结构的三环类衍生物及其制备方法和用途 Quinazoline structure containing tricyclic derivatives and their preparation and use |
08/06/2014 | CN102702225B 四酚芴基苯并噁嗪及其制备方法 Four benzene and phenol fluorene oxazine and its preparation method |
08/06/2014 | CN102498116B 取代的二氢苯并环烷氧基甲基噁唑并嘧啶酮、其制备及用途 Substituted dihydro-benzo cycloalkoxy methyloxazole and pyrimidone, their preparation and use |
08/06/2014 | CN101910152B 作为janus激酶抑制剂的4-吡唑基-n-芳基嘧啶-2-胺和4-吡唑基-n-杂芳基嘧啶-2-胺 As janus kinase inhibitors 4- pyrazolyl -n- aryl-pyrimidin-2-amine and 4-pyrazolyl -n- heteroaryl pyrimidin-2-amine |
08/05/2014 | US8796467 Compounds |
08/05/2014 | US8796454 Synthesis of [2.2.2]-diazabicyclic ring systems |
08/05/2014 | US8796299 NK1 antagonists |
08/05/2014 | US8796269 Crystalline 2-(3,5-Bis(trifluoromethyl)phenyl)-N-(4-(4-fluoro-2-methylphenyl)-6-((7S,9aS)-7-(hydroxymethyl)hexahydropyrazino[2,1-c][1,4]oxazin-8(1H)-yl)pyridin-3-yl)-N,2-dimethyl-propanamide of the formula (I), their use in therapy, and process for the preparation of the same |
08/05/2014 | US8796262 Fused heterocyclic derivatives as S1P modulators |
08/05/2014 | US8796261 Bromodomain inhibitors and uses thereof |
08/05/2014 | CA2565238C Amido compounds and their use as pharmaceuticals |
07/31/2014 | WO2014116611A1 Low temperature synthesis of rapamycin derivatives |
07/31/2014 | WO2014114929A1 Compounds and methods for treating bacterial infections |
07/31/2014 | US20140213571 Tetracyclic heterocycle compounds and methods of use thereof for the treatment of viral diseases |
07/31/2014 | US20140213553 Carbamoylpyridone derivatives |
07/30/2014 | EP2758406A1 Amino-oxazines and amino-dihydrothiazine compounds as beta-secretase modulators and methods of use |
07/30/2014 | CN103958525A 3,7-二取代八氢-2H-吡啶并[4,3-e][1,3]噁嗪-2-酮抗生素 3,7-substituted octahydro--2H- pyrido [4,3-e] [1,3] oxazin-2-one antibiotic |
07/30/2014 | CN103958524A 稠合的二环噁唑烷酮cetp抑制剂 Fused bicyclic oxazolidinone cetp inhibitors |
07/30/2014 | CN103958523A 作为双重活性H1反向激动剂/5-HT<sub>2A</sub>拮抗剂的(噻吩并[2,3-b][1,5]苯并氧氮杂*-4-基)哌嗪-1-基化合物 H1 dual activity as an inverse agonist / 5-HT <sub> 2A </ sub> antagonists (thieno [2,3-b] [1,5] benzoxazepine * 4-yl) piperazine 1-yl compound |
07/30/2014 | CN103958518A 杂环基吡啶基吡唑/杂环基嘧啶基吡唑 Heterocyclyl pyridyl pyrazole / heterocyclyl pyrimidinyl pyrazole |
07/30/2014 | CN103958506A 用作突变idh抑制剂的3-嘧啶-4-基-噁唑烷-2-酮化合物 Is used as an inhibitor of 3 mutations idh pyrimidin-4-yl - oxazolidin-2-one compounds |
07/30/2014 | CN103958495A 作为gpr-119的调节剂的新型化合物 Gpr-119 as a novel compound of modulators |
07/30/2014 | CN103951678A 三环三唑化合物 Tricyclic triazole compound |
07/30/2014 | CN103951677A 利福喷丁的制备方法 Rifapentine preparation |
07/30/2014 | CN102066384B 作为α-7烟碱乙酰胆碱受体配体的奎宁环化合物 As quinuclidine α-7 nicotinic acetylcholine receptor ligand compound |
07/29/2014 | US8791108 Inhibitors of human immunodeficiency virus replication |
07/29/2014 | US8791107 N-substituted oxazinopteridines and oxazinopteridinones |
07/29/2014 | US8790795 6,12-dinaphthylchrysene derivative and organic light-emitting device using the derivative |
07/29/2014 | US8790691 Modified drugs for use in liposomal nanoparticles |
07/24/2014 | WO2014110706A1 Thiophene-substituted tetracyclic compounds and methods of use thereof for treatment of viral diseases |
07/24/2014 | WO2014110705A1 Heterocycle-substitued tetracyclic compounds and methods of use thereof for treatment of viral diseases |
07/24/2014 | WO2014110688A1 Thiophene- sub stitued tetracyclic compounds and methods of use thereof for the treatment of viral diseases |
07/24/2014 | WO2014110687A1 Thiazolyl-substitued tetracyclic compounds and methods of use thereof for treatment of viral diseases |
07/24/2014 | US20140206872 Fluorescent dye |
07/24/2014 | US20140206683 Macrocyclic lrrk2 kinase inhibitors |
07/24/2014 | US20140206681 Btk inhibitors |
07/24/2014 | US20140206680 Substituted 6-aza-isoindolin-1-one derivatives |
07/24/2014 | US20140206679 Heterocyclic pyridone compound, and intermediate, preparation method and use thereof |
07/24/2014 | US20140206677 Compounds and methods for treating bacterial infections |
07/24/2014 | US20140206664 Heterocycle Amido Alkyloxy Substituted Quinazoline Derivative and Use Thereof |
07/24/2014 | US20140206663 Triazinone compounds |
07/24/2014 | US20140206618 Inhibitors of the Renal Outer Medullary Potassium Channel |
07/24/2014 | US20140205567 Macrocyclic Heterocyclic Compound for Inhibiting Hepatitis C Virus and Preparation and Use Thereof |
07/23/2014 | CN203725148U 临床动药用盐酸左氧氟沙星的合成搅拌加热装置 Clinical dynamic synthesis of medicinal Levofloxacin stirring heating device |
07/23/2014 | CN103936767A 一种制备化合物(1R,2S,6S,7S)-4,4-二甲基-9-苯甲基-3,5,8-三氧杂-9-氮杂三环[5.2.1.0<sup>2.6</sup>]葵烷的方法 A process for preparing the compound (1R, 2S, 6S, 7S) -4,4- dimethyl-9-benzyl -3,5,8- three-oxa-9-aza-tricyclo [5.2.1.0 <sup > 2.6 </ sup>] decane methods |
07/23/2014 | CN103936766A 一种5(4h)-吡啶酮并呋咱氧化物的合成方法 One kind of 5 (4h) - pyridone and furosemide oxide synthesis method we |
07/23/2014 | CN103936765A N-全芳香烃基双酚-双胺型四官能度芴基苯并噁嗪及其制备方法 N- wholly aromatic hydrocarbon bisphenol - double tetrafunctional fluorene amine benzene and oxazine and its preparation method |
07/23/2014 | CN103936764A N-半芳香烃基双酚-双胺型四官能度芴基苯并噁嗪及其制备方法 N- semi-aromatic hydrocarbon group bisphenol - double tetrafunctional fluorene amine benzene and oxazine and its preparation method |
07/23/2014 | CN103936763A 噁唑烷酮类化合物及其制备方法和用途 Oxazolidinone compounds and their preparation and use |
07/23/2014 | CN103936762A 吗啉并喹啉类化合物,其制备方法和用途 Morpholine and quinoline compounds, their preparation and use |
07/23/2014 | CN103936754A 一种苯并吡喃类化合物及其制备方法与应用 One kind of benzopyran compound and its preparation method and application |
07/23/2014 | CN102015726B 杂环衍生物 Heterocyclic derivatives |
07/23/2014 | CN101622240B 稠合取代氨基吡咯烷衍生物 Fused to an amino-substituted pyrrolidine derivatives |
07/22/2014 | US8785626 Benzoxazepin PI3K inhibitor compounds and methods of use |
07/22/2014 | US8785439 2,5,7-substituted oxazolopyrimidine derivatives |
07/22/2014 | US8784684 Polymerizable compound, polymerizable liquid crystalline composition, macromolecular compound and film |
07/17/2014 | WO2014110066A1 Macrocyclic benzofuran and azabenzofuran compounds for the treatment of hepatitis c |
07/17/2014 | WO2014110065A1 (THIENO[2,3-b][1,5]BENZOXAZEPIN-4-YL)PIPERAZIN-1-YL COMPOUNDS AS DUAL ACTIVITY H1 INVERSE AGONISTS/5-HT2A ANTAGONISTS |
07/17/2014 | US20140200654 Drug-delivery endovascular stent and method of forming the same |
07/17/2014 | US20140200344 Tricyclic heterocyclic compounds and jak inhibitors |
07/17/2014 | US20140200343 Process and intermediates for preparing macrolactams |
07/17/2014 | US20140200319 Fluorescent potassium ion sensors |
07/17/2014 | US20140200223 Inhibitors of beta-secretase |
07/17/2014 | US20140200216 Bicyclic aromatic carboxamide compounds useful as pim kinase inhibitors |
07/17/2014 | US20140200209 Polycyclic carbamoylpyridone derivative having hiv integrase inhibitory activity |
07/17/2014 | US20140199264 Tetracyclic xanthene derivatives and methods of use thereof for the treatment of viral diseases |
07/17/2014 | US20140199263 Heterocyclic-substituted benzofuran derivatives and methods of use thereof for the treatment of viral diseases |
07/16/2014 | CN103930427A 大环flt3 激酶抑制剂 Macrocyclic kinase inhibitors flt3 |
07/16/2014 | CN103923055A 一种制备(1s,2r,3s,4r)-2,3-o-亚异丙基-4-氨基环戊烷-1,2,3-三醇的方法 A method for the preparation of (1s, 2r, 3s, 4r) -2,3-o- isopropylidene-4-amino-cyclopentane-1,2,3-triol |
07/16/2014 | CN103922879A 一种脱除热敏性固体药物中残留溶剂的装置 An apparatus for heat-sensitive drugs in solid residual solvent removal |
07/16/2014 | CN103922878A 一种脱除热敏性固体药物中残留溶剂的方法 A process for removing residual solvent in the heat-sensitive solid pharmaceutical methods |
07/16/2014 | CN102015706B 作为11b-hsd1抑制剂的咪唑烷酮衍生物 Imidazolidinone derivatives as inhibitors of 11b-hsd1 |
07/16/2014 | CN101880280B 双环嘧啶酮以及其应用 Bicyclic pyrimidinone and their use |