Patents
Patents for C07D 495 - Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms (21,336)
11/1999
11/16/1999US5986076 A conjugate is formed by bonding a bioreactive agent to the therapeutic agent with a bond that is selectively cleavable with electromagnetic radiation; useful for controlled release of drugs to treat the disorder
11/16/1999US5985884 Treatment and/or prophylaxis of diseases or conditions in which insulin resistance is the underlying pathophysiological mechanism such as type ii diabetes, impaired glucose tolerance, dyslipidaemia, hypertension, coronary heart disease
11/16/1999US5985799 Tricyclic n-heterocycles, their n-oxides, agriculturally-suitable salts and compositions, and methods of their use for controlling undesirable vegetation
11/16/1999CA2048896C Fluoroethylcamptothecin derivatives
11/11/1999WO1999057564A1 Method for immobilising and/or crystallising biological macromolecules on carbon nanotubes and uses
11/11/1999WO1999057122A1 3-phenylpyrrole alpha-1 adrenergic compounds
11/11/1999WO1999043682A9 2-(het-)aryl-4-(cyclic amino substituted) heteroaryl fused pyridine derivatives, their preparation and their use as (ant-)agonists for gaba (a) brain receptors
11/10/1999EP0955299A1 Benzothiophene, benzofurane and indole derivatives, process for their preparation and pharmaceutical compositions containing them
11/10/1999EP0954526A2 Serine protease inhibitors
11/10/1999EP0954522A1 Novel substituted naphthopyrans
11/10/1999EP0954305A2 Use of carbonic anhydrase inhibitors for treating macular edema
11/10/1999EP0553314B1 Process for the manufacture of spiroketals
11/10/1999CN1234802A Intermediates and process for preparing olanzapine
11/10/1999CN1234738A 奥氮平二水合物d Olanzapine dihydrate d
11/10/1999CN1046282C Photockromic heterocyclobenzopyrane and preparing method and use thereof
11/10/1999CN1046271C Substituted pyrimidines and fungicidal and pesticidal and anti-septic composition containing same
11/10/1999CN1046269C HIV protease inhibitors
11/09/1999US5981779 Enzyme linked immunoassays (elisas) (with biotin containing compounds) and fluorimetric and chemiluminometric assays (with fluorescein or chemiluminiscence containing compounds)
11/09/1999US5981576 (Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitors
11/09/1999US5981567 Substituted spiroheterocyclic 1h-3-aryl-pyrrolidine-2,4-dione derivatives and their use as pesticides
11/09/1999US5981540 Selective delta opioid agonists and antagonists; useful as analgesics and in treating general neurologic disorders
11/09/1999US5981539 Piperidine compounds as calcium channel blockers
11/04/1999WO1999055708A1 Condensed thienopyrimidines with phosphodiesterase-v inhibiting action
11/04/1999WO1999055673A1 Arylphenyl-substituted cyclic keto enols
11/04/1999WO1999055335A1 Substituted tricyclic pyrazole derivatives with protein kinase activity
11/04/1999DE19819023A1 Thienopyrimidine Thienopyrimidines
11/02/1999US5977132 Prolactin production inhibitory agent
11/02/1999US5977125 Mono-or polyenic carboxylic acid derivatives
11/02/1999US5977111 Thiopyran derivatives
11/02/1999US5977108 Leukemia
10/1999
10/28/1999WO1999054319A1 12,13-modified epothilone derivatives
10/28/1999WO1999054318A1 12,13-cyclopropane epothilone derivatives
10/28/1999WO1999054303A1 Optically active tetrahydrobenzindole derivatives
10/28/1999DE19818732A1 New aryl substituted cyclic ketoenol compounds useful for control of insects and as herbicides
10/28/1999CA2329319A1 Optically active tetrahydrobenzindole derivatives
10/28/1999CA2323609A1 12,13-cyclopropane epothilone derivatives
10/27/1999CN1045957C Tricyclic benzazepine, their application and preparation
10/26/1999US5973085 Monomers and composition which can be crosslinked and crosslinked polymers
10/26/1999US5972951 Tetracyclic spiro compounds, process for their preparation and their use as 5HT1D receptor antagonists
10/26/1999US5972932 Olanzapine or a salt or solvate thereof, and an opoid in a specific weight ratio; administering to provide mild pre-surgical anesthesia to provide amnesia while maintaining cooperation in mammals such as humans
10/26/1999CA2177576C Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
10/21/1999WO1999052910A1 Bicyclic hydroxamic acid derivatives
10/21/1999WO1999052876A1 Azacycloalkane derivatives, preparation and therapeutic application
10/21/1999WO1999032428A8 Synthesis of diamines
10/20/1999EP0950661A1 Substituted tricyclics useful in sPLA2 induced diseases
10/20/1999EP0949920A1 Highly selective butyrylcholinesterase inhibitors for the treatment and diagnosis of alzheimer's disease and dementias
10/20/1999CN1232450A 2- and 2,5-substd. phenylketoenols
10/19/1999US5969149 Reacting hexahydrofuro/3,4-d/imidazole-2,4-diones with hydrogen sulfide in presence of basic compound and sulfur
10/19/1999US5968937 For treatment and/or prevention of hypertension, cardiac insufficiency, coronary vasospasm, cardiac ischemia, renal vasospasm, liver cirrhosis, congestive heart failure, nephrotic syndrome, brain edema, cerebral ischemia
10/19/1999US5968930 Tricyclic diazepine vasopressin antagonists and oxytocin antagonists
10/19/1999CA2197298C Novel pyrimidine derivatives and processes for the preparation thereof
10/17/1999CA2269256A1 Substituted tricyclics
10/14/1999WO1999051587A1 Fused thiophene derivatives and drugs containing the same as the active ingredient
10/14/1999WO1999051580A1 Pyrazole inhibitors of cytokine production
10/14/1999WO1999051572A1 Sulfonamide derivatives
10/14/1999CA2327290A1 Sulfonamide derivatives
10/14/1999CA2327185A1 Pyrazole inhibitors of cytokine production
10/13/1999EP0948499A1 Heteroarylsulfonamide derivatives and pharmaceutical compositions containing them
10/12/1999US5965730 Selective phosphodiestearase iv inhibitor having bronchodialation and anti-inflammatory activity; prophylaxis and treatment of asthma
10/12/1999US5965692 Anticoagulants for treatment of thromobosis and hypercoagulability in blood and tissues
10/12/1999US5965565 Piperidines, pyrrolidines, and hexahydro-1h-azepines of given formula; can be used to promote growth of livestock and in humans treat physiological or medical conditions characterized by grwoth hormone defiency
10/07/1999WO1999037292A3 Carbonic anhydrase inhibitor for increasing oxygen tension in the optic nerve and retina
10/06/1999EP0946558A1 Ethylidene derivatives of tricyclic carbapenems
10/06/1999EP0946540A1 Substituted benzothiopyranes salts and their use as herbicides
10/06/1999EP0946523A1 Fused polycyclic 2-aminopyrimidine derivatives, their preparation and their use as protein tyrosine kinase inhibitors
10/06/1999EP0946179A1 Method for treating autism
10/06/1999EP0635508B1 Tetrahydropyridine derivative having substituents on three rings
10/06/1999CN1230962A 3-substituted pyrido [4',3' : 4, 5] thieno [2,3-D] pyrimidine derivatives, their preparation and their use
10/05/1999US5962469 Cyclic nitrones
10/05/1999US5962462 Spiro-substituted azacycles as modulators of chemokine receptor activity
10/05/1999US5962457 2,3 Disubstituted- (5,6)-heteroarylfused-pyrimidine-4-ones
10/05/1999US5962450 Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines and their use as medicaments
10/05/1999US5962448 Pyrroloazepine derivatives
09/1999
09/29/1999EP0944633A1 Substituted phenylketoenols and their use as pesticides and herbicides
09/29/1999EP0944386A1 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
09/29/1999CN1230196A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn.
09/28/1999US5958981 γ-diketone compounds with inhibitory activity against platelet aggregation
09/28/1999US5958936 For inducing antiandrogenic activity in warm-blooded animals, including humans
09/28/1999US5958924 Hypotensive agents, cardiovascular disorders, antiischemic agents, restenosis, anticoalugants, respiratory system disorders
09/22/1999EP0942911A1 Benzopyranopyrrole and benzopyranopyridine alpha-1 adrenergic compounds
09/22/1999CN1229412A Inhibitors of interleukin-1'beta' converting emzyme
09/22/1999CN1229082A Amine compound and its acid addition salt
09/22/1999CN1045206C Method for preparing cyclic amide derivative
09/21/1999US5955605 Biotinidase resistant biotin-DOTA conjugates
09/16/1999WO1999046268A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases)
09/16/1999WO1999046267A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999046266A1 Benzoxadiazocinyl arthropodicides
09/16/1999WO1999046244A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999WO1999046237A1 Modulators of protein tyrosine phosphatases
09/16/1999WO1999046236A1 Modulators of protein tyrosine phosphatases (ptpases)
09/16/1999CA2323493A1 Modulators of protein tyrosine phosphatases (ptpases)
09/15/1999EP0941994A1 Pyrazolopyrimidines and pyrazolotriazines with 5-HT6 receptor affinity
09/15/1999CN1228779A Spirocyclic metalloprotease inhibitors
09/15/1999CN1228777A Pyridyl alkene- and pyridyl alkine-acid amides as cytostatics and immunosuppressives
09/15/1999CN1228771A 1,3-diheterocyclic metalloprotease inhibitors
09/15/1999CN1228701A Heterocyclic compounds with thrombolytic activity and their use for treating thrombosis
09/15/1999CN1045084C Novel compound with platelet aggregation inhibitor activity and its use, and drug composition containing the same
09/14/1999US5952512 Production of optically active benzothiepin salts
09/14/1999US5952343 HIV protease inhibitors
09/14/1999US5952335 Antitumor agents