Patents
Patents for C07D 495 - Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms (21,336)
02/2000
02/16/2000CN1244529A Novel 8H-thiophene [2,3-b] pyrrolinezine-8-on compound, its preparing method and their medicinal compounds containing them
02/15/2000US6025371 Solid phase and combinatorial library syntheses of fused 2,4-pyrimidinediones
02/15/2000CA2119218C Enantioselective synthesis of 5,6-dihydro-(s)-4-(ethylamino)-(s)-6-methyl-4h-thieno 2,3-b thiopyran-2-sulfonamide 7,7-dioxide and related compounds
02/10/2000WO2000006529A1 Diketoacid-derivatives as inhibitors of polymerases
02/10/2000WO1999063944A3 Novel therapeutic agents that modulate estrogen receptors
02/10/2000CA2338490A1 Diketoacid-derivatives as inhibitors of polymerases
02/09/2000EP0977759A1 Crf antagonistic thiophenopyridines
02/09/2000EP0977754A1 Writable and erasable high-density optical storage media
02/09/2000EP0977752A1 Herbicidal pyrazoles
02/09/2000CN1244201A Heterocyclic metallocenes and polymerization catalysts
02/08/2000US6022307 Angiogenesis inhibitor
02/03/2000WO2000005234A1 NF-λB INHIBITORS CONTAINING INDAN DERIVATIVES AS THE ACTIVE INGREDIENT
02/03/2000WO2000004899A1 Ophthalmic compositions for treating ocular hypertension
02/03/2000WO2000004898A1 Ophthalmic compositions for treating ocular hypertension
02/03/2000WO2000004892A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/03/2000WO1999063936A3 Novel therapeutic agents that modulate endothelin receptors
02/03/2000WO1999063933A3 Multivalent agonists, partial agonists and antagonists of the gaba receptors
02/03/2000WO1999063929A3 Multibinding inhibitors of microsomal triglyceride transferase protein
02/03/2000CA2337399A1 Ophthalmic compositions for treating ocular hypertension
02/03/2000CA2337349A1 Ophthalmic compositions for treating ocular hypertension
02/03/2000CA2335062A1 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
02/02/2000EP0975639A1 Compounds
02/02/2000EP0975619A1 INTENSE COLOURING PHOTOCHROMIC 2$i(H)-NAPHTHO 1,2-$i(b)]PYRANS AND HETEROCYCLIC PYRANS
02/02/2000EP0975602A1 Imidazole and imidazoline derivatives and uses thereof
02/02/2000EP0975600A1 Heterocyclic derivatives and their use as antithrombotic agents
02/01/2000US6020487 Intermediates and process for preparing olanzapine
02/01/2000US6020343 (Methylsulfonyl)phenyl-2-(5H)-furanones as COX-2 inhibitors
02/01/2000US6020342 Fused imidazo[1,2-A]pyridines
01/2000
01/27/2000WO2000004027A1 Piperazynil pyrimidine dione compounds selective for adrenoceptors
01/27/2000WO2000004023A1 Anhydride modified cantharidin analogues useful in the treatment of cancer
01/27/2000WO1999063930A3 Novel angiotensin receptor modulators and their uses
01/27/2000CA2337771A1 Anhydride modified cantharidin analogues useful in the treatment of cancer
01/27/2000CA2336950A1 Piperazynil pyrimidine dione compounds selective for adrenoceptors
01/26/2000EP0973778A1 4,5,6,7-TETRAHYDRO-THIENO 3,2-c]PYRIDINE DERIVATIVES, THEIR PREPARATION AND USE
01/26/2000EP0973777A1 Furopyridine, thienopyridine, pyrrolopyridine and related pyrimidine, pyridazine and triazine compounds useful in controlling chemical synaptic transmission
01/26/2000EP0973772A1 Compounds
01/26/2000EP0778834B1 Diaryl bicyclic heterocycles as inhibitors of cyclooxygenase-2
01/26/2000CN1242773A Ticyclic carbapenem compound
01/25/2000US6018054 Intermediate compounds for preparing novel quinolone and naphthyridone derivatives which are substituted in the 7-position by a partially hydrogenated isoindolinyl ring, use as antibacterial agents and as feed additives
01/25/2000US6017768 For screening agonists or antagonists of alpha adrenergic receptors, dopamine receptors, sigma opiate receptors, potassium ion channels, carbonic anhydrase inhibitors; for treatment of glaucoma
01/20/2000WO2000002861A1 A3 adenosine receptor antagonists
01/20/2000WO2000002555A1 Methods and compositions for the treatment of chronic lymphocytic leukemia
01/20/2000WO1999059526A3 Protease inhibitors
01/20/2000CA2336932A1 Methods and compositions for the treatment of chronic lymphocytic leukemia
01/19/2000EP0971931A1 Method for debenzylation of dibenzyl biotin
01/19/2000EP0971914A2 NEUTRAL COLOURING PHOTOCHROMIC 2$i(H)-NAPHTHO 1,2-$i(b)]PYRANS AND HETEROCYCLIC PYRANS
01/19/2000EP0971748A2 Tetraaza- or n2s2- complexants, and their use in radiodiagnostics or radiotherapy
01/18/2000US6015912 Treating arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
01/18/2000US6015819 Administering adrenergic blocking agent; reduction of orthostatic fall in blood pressure side effect; fda orange book listed patent for silodosin
01/18/2000US6015817 Inhibitors of farnesyl-protein transferase
01/18/2000US6015810 Aqueous ophthalmic solution containing apafant as active ingredient
01/18/2000CA2000985C 1,4-diazepine derivative and its pharmaceutical use
01/13/2000WO2000002051A1 Trifunctional reagent for conjugation to a biomolecule
01/13/2000WO2000002050A1 Trifunctional reagent for conjugation to a biomolecule
01/13/2000WO2000001687A1 Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
01/13/2000CA2336739A1 Trifunctional reagent for conjugation to a biomolecule
01/13/2000CA2336315A1 Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
01/12/2000EP0970956A1 Pyrazole derivatives
01/12/2000EP0970086A1 Spiro compounds and the use thereof
01/12/2000EP0559891B1 Thienodiazepine compound and its use
01/11/2000US6013807 Amidation to produce compound having low toxicity and antitumor activity
01/11/2000US6013656 2-(arylalkenyl) azacycloalkane derivatives as ligands for sigma receptors
01/11/2000US6013655 Hypotensive agents; respiratory system diisorders
01/11/2000US6013652 Spiro-substituted azacycles as neurokinin antagonists
01/06/2000WO2000000493A1 Thienopyridine compounds, their production and use
01/06/2000CA2331399A1 Thienopyridine compounds, their production and use
01/05/2000CN1240450A Thienopyrimidine with phosphodiesterase V inhibiting effect
01/05/2000CN1240449A Substituted phenylketoenols and their use as pesticides and herbicides
01/05/2000CN1240440A Substituted benzothiopyranes salts and their use as herbicides
01/05/2000CN1240212A Process for reducing prochiral ketone to produce optically active alcohol of high optical purity
01/04/2000US6011029 Benzodiazepine compounds
12/1999
12/29/1999WO1999067228A1 Fluorophenyl resin compounds
12/29/1999WO1999067202A1 Process for preparation of pyrimidinone derivatives
12/29/1999WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors
12/29/1999WO1999066925A1 Protease inhibitors
12/29/1999EP0966470A1 Dioxino derivatives and their use as therapeutic agents
12/29/1999EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments
12/29/1999CA2335876A1 Protease inhibitors
12/29/1999CA2335760A1 Fluorophenyl resin compounds
12/29/1999CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors
12/28/1999US6008230 Treating bone diseases caused by abnormal bone metabolism in human being or animals as the inhibitors of bone resorption or the inhibitors of bone metastasis
12/23/1999WO1999065917A1 Use of diazepins for preparing medicines for treating pathological conditions or diseases involving one of the growth hormone release inhibiting factor receptors
12/23/1999WO1999065916A1 Thienodipyridine derivatives, production and use thereof
12/23/1999WO1999065915A1 Polymorphic clopidogrel hydrogenesulphate form
12/23/1999WO1999065910A1 Fused azepinone cyclin dependent kinase inhibitors
12/23/1999CA2335724A1 Use of diazepins for preparing medicines for treating pathological conditions or diseases involving one of the growth hormone release inhibiting factor receptors
12/23/1999CA2335106A1 Thienodipyridine derivatives, production and use thereof
12/22/1999EP0731795B1 Substituted pyrazolyl benzenesulfonamides for the treatment of inflammation
12/21/1999US6005083 Substituted metal chelating compounds for imaging and therapy
12/21/1999US6004971 Pentacyclic compounds, intermediates, processes, compositions, and methods
12/21/1999US6004964 Administering amide or sulfonamide derivative; analgesics
12/16/1999WO1999064425A1 Substituted thienocycloalkylpyrazoles: dopamine receptor subtype specific ligands
12/16/1999WO1999064420A1 β-CARBOLINE COMPOUNDS
12/16/1999WO1999064395A1 Heterocyclic amide compounds as cell adhesion inhibitors
12/16/1999WO1999064055A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht4 receptors
12/16/1999WO1999064054A1 Multibinding inhibitors of topoisomerase
12/16/1999WO1999064053A1 β3-ADRENERGIC RECEPTOR AGONISTS
12/16/1999WO1999064052A1 Novel leukotriene receptor antagonists and their uses
12/16/1999WO1999064051A1 Novel antibacterial compounds
12/16/1999WO1999064049A1 Novel antibacterial agents