Patents
Patents for C07D 495 - Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms (21,336)
12/2000
12/14/2000WO2000075145A1 Cell adhesion-inhibiting antiinflammatory compounds
12/14/2000CA2390948A1 Cell adhesion-inhibiting antiinflammatory compounds
12/13/2000EP1058549A1 THROMBIN OR FACTOR Xa INHIBITORS
12/13/2000EP0724583B1 Pyridazino quinoline compounds
12/13/2000CN1276723A Dithiolopyrrolones and their corresponding monoxides and dioxides as antineoplastic agent
12/13/2000CN1059443C Tetracylic 1,4-oxazine compound, its preparing method and medicinal composition contg. same
12/12/2000US6159981 3-substituted pyrido [3',4':4,5] Thieno [2,3-d] pyrimidine derivatives, and production and use of the same
12/12/2000US6159967 such as 1-(2-((2R)-(3,4-dichlorophenyl)-4-(3,4,5-trimethoxybenzoyl) morpholin-2-yl)ethyl)spiro(benzo(c)thiophene-1-(3H), 4'-piperidine)-(2S)-oxide; respiratory disease such as asthma
12/12/2000US6159963 Method for treating substance abuse
12/12/2000US6159962 3-substituted 3,4-dihydro-thieno[2,3-D]pyrimidine derivatives and production and use of the same
12/12/2000US6159904 Pyrazole derivatives
12/07/2000WO2000073313A1 New tricyclic amidine derivatives as inhibitors of nitric oxide synthase
12/07/2000WO2000073312A1 Compounds
12/07/2000WO2000073311A2 Tricyclic benzoylcyclohexanedione derivatives
12/07/2000WO2000072802A2 Water soluble multi-biotin-containing compounds
12/07/2000CA2372241A1 Tricyclic benzoylcyclohexanedione derivatives
12/06/2000EP1057814A1 Tetrahydrobenzindole derivatives
12/06/2000EP1056451A1 Bicyclic pyrrole derivatives as mcp-1 inhibitors
12/06/2000CN1275982A Novel heterocyclic compounds process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases
12/05/2000US6156781 Antiinflammatory agents for skin
12/05/2000US6156769 Antipruitus drugs for mammals
12/05/2000US6156747 Psychological, gastrointestinal, cardiovascular disorders
11/2000
11/30/2000WO2000071534A1 Heterocyclic substituted aminoazacycles useful as central nervous system agents
11/30/2000WO2000071524A1 2-nh-pyridones and pyrimidones as mrs inhibitors
11/30/2000CA2373793A1 Heterocyclic substituted aminoazacycles useful as central nervous system agents
11/29/2000EP1054887A1 Bicyclic pyridine and pyrimidine derivatives as neuropeptide y receptor antagonists
11/29/2000EP0632810B1 New biotinylation reagent
11/29/2000CN1058967C Novel pyridine compounds, processes for their preparation and pharmaceutical compositions thereof
11/29/2000CN1058841C Fungicidal oxazolidinones
11/28/2000US6153617 Used for reating cancer, restenosis, atherosclerosis, endometriosis, and psoriasis
11/28/2000US6153614 Piperazinyl pyrimidine dione compounds selective for adrenoceptors
11/23/2000WO2000069830A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
11/23/2000CA2373590A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
11/22/2000EP1053229A1 Condensed 4-thioxopyrimidine derivatives as microbicides
11/22/2000EP0736012B1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
11/22/2000CN1058718C Optically active benzothiepin derivative, its prepn. and use
11/21/2000US6150375 Inhibitors of both of the human 5ar isozymes; benign prostate hyperplasia, male pattern baldness, acne vulgaris, seborrhea, androgenic alopecia, hirsutism and prostate cancer; blocks the conversion of testosterone to 5-alpha-dihydrotestosterone
11/21/2000US6150370 1,3-dinitrocyclic compound treats numerous diseases caused by undesired metalloprotease activity, such as tumor metastasis, osteoarthritis, rheumatoid arthritis, skin inflammation, ulcerations, and periodontitis
11/21/2000US6150352 Antagonists of gonadotropin releasing hormone
11/21/2000US6150042 Material for organoelectro-luminescence device and use thereof
11/16/2000WO2000068233A1 Cyclohexenone dioxothiochromanoyl derivatives
11/16/2000CA2373165A1 Cyclohexenone dioxothiochromanoyl derivatives
11/15/2000EP1051415A1 Benzamide derivatives as vasopressin antagonists
11/15/2000EP1051176A1 SUBSTITUTED OXOAZAHETEROCYCLYL FACTOR Xa INHIBITORS
11/15/2000CN1058495C Polycyclic systems compound and derivatives thereof as neurotransmitter release enhancers useful in the treatment of cognitive disordes and medicine containing them and its use
11/14/2000US6147223 Lactacystin analogs
11/14/2000US6147110 Heterocyclic compounds
11/14/2000US6147089 Cholesteryl ester transfer protein inhibitors used to treat diseases which are exacerbated by low levels of hdl cholesterol and/or high levels of ldl-cholesterol and triglycerides, such as atherosclerosis and cardiovascular
11/14/2000US6147083 Novel substituted 1,2-ethanediamine derivatives which antagonize the pharmacological actions of the endogenous neuropeptide tachykinins known as neurokinins, useful for the treatment of asthma, etc.
11/09/2000CA2371632A1 Cyclocarbamate and cyclic amide derivatives
11/08/2000EP1050535A1 Fused pyrazine compounds
11/08/2000EP1049700A1 Chemokine receptor antagonists and methods of use therefor
11/08/2000EP1049694A1 Benzothiadiazoles and derivatives
11/08/2000EP1049675A1 Chemokine receptor antagonists and methods of use therefor
11/08/2000EP1049466A2 Carbonic anhydrase inhibitor for increasing oxygen tension in the optic nerve and retina
11/08/2000EP0842166B1 Process for synthesizing carbapenem side chain intermediates
11/07/2000CA2080223C Thiophene sulfonamides useful as carbonic anhydrase inhibitors
11/02/2000WO2000064904A1 5,7-bicyclic amidine derivatives useful as nitric oxide synthase inhibitors
11/02/2000EP1048658A1 Alicyclic acylated heterocyclic derivatives
11/02/2000EP1048651A1 Nitrogen-containing tetracyclic compounds
11/02/2000EP1048640A1 Apoptosis inhibitors
11/02/2000EP1047686A1 Substituted bicyclic lactones
11/02/2000EP1047675A1 Chemokine receptor antagonists and methods of use therefor
11/02/2000EP0713489B1 Photochromic heterocyclochromenes
10/2000
10/31/2000US6140507 Method for debenzylation of dibenzylbiotin
10/31/2000US6140325 Has endothelin antagonistic action; for treating liver hypofunction, acute renal insufficiency, cardiac infarction or liver insufficiency, vasoconstriction
10/26/2000WO2000063197A1 Hydroxamic acid derivative
10/26/2000WO2000034286A3 Process for the preparation of pyrimidinone derivatives
10/25/2000CN1271251A 2-methyl-thieno-benzodiazepine formulation
10/24/2000US6136985 CLA esters and uses thereof
10/24/2000US6136817 Opioid receptor antagonist compounds
10/24/2000US6136812 Methods of administering AMPA receptor antagonists to treat dyskinesias associated with dopamine agonist therapy
10/19/2000WO2000061587A1 Pyrido-thieno-diazepines, method for the production thereof and pharmaceutical compositions containing said pyrido-thieno-diazepines
10/19/2000WO2000061586A1 Bicyclic heteroaromatic compounds useful as lh agonists
10/19/2000WO2000061583A1 Xanthine derivatives and analogs as cell signaling inhibitors
10/19/2000WO2000061549A2 Pharmaceutical compounds
10/19/2000WO2000061541A2 Pharmaceutical compounds
10/19/2000WO2000061537A2 Pharmaceutical compounds
10/19/2000CA2370425A1 Pharmaceutical compounds
10/19/2000CA2370406A1 Pharmaceutical compounds
10/19/2000CA2369981A1 Therapeutic compounds for inhibiting interleukin-12 signaling and methods for using same
10/18/2000EP1044197A2 New piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides
10/18/2000EP1043991A1 Treatment for alzheimer's disease
10/18/2000EP1043977A1 Oral pharmaceutical pulsed release dosage form
10/18/2000EP1043976A1 Oral pharmaceutical extended release dosage form
10/18/2000CN1270593A Pyrimidin-4-one and pyrimidin-4-thione as fungicide
10/18/2000CN1270592A Spiroazabicyclic heterocyclic compounds
10/17/2000US6133459 Method and compositions providing enhanced chemiluminescence from 1,2-dioxetanes
10/17/2000US6133309 Treatment of T-helper cell type 2-mediated immune disease by retinoid antagonists
10/17/2000US6133296 Substituted pyridyl keto enols
10/17/2000US6133288 2,8-di(hydroxy)-5-((2-piperidin-1-yl)ethyoxy-1,4-phenylene)-)-5h -benzo-(e)naphtho(1,2-c)pyran; post-menopausal syndrome, osteoporosis, cardiovascular disorders; uterine fibrosis, endometriosis, and aortal smooth muscle cell proliferation
10/17/2000US6133283 Mono- or polyenic carboxylic acid derivatives
10/17/2000US6133275 3-phenylpyrrolidine alpha-1 adrenergic compounds
10/17/2000US6133257 Fused polycyclic 2-aminopyrimidine derivatives
10/12/2000WO2000059912A1 Thienopyrimidine compounds and salts thereof and process for the preparation of the same
10/12/2000WO2000059911A2 Tricyclic cyclohexanedione derivatives
10/12/2000WO2000059910A2 Tricyclic pyrazolone derivatives
10/12/2000WO2000059901A1 Substituted 1,4-dihydroindeno[1,2-c]pyrazoles as inhibitors of tyrosine kinase
10/12/2000WO2000059884A1 Pharmaceutically active compounds and methods of use thereof
10/12/2000WO2000059507A1 Obesity preventives