Patents
Patents for C07D 495 - Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms (21,336)
08/2002
08/21/2002CN1365363A thineopyranecarboxyamide derivatives
08/20/2002US6437132 Inhibitor of gonadotropin releasing hormone
08/20/2002US6436967 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
08/20/2002CA2257222C Amide derivatives
08/20/2002CA2240138C Quinazolin-4-one ampa antagonists
08/20/2002CA2077695C Hydropyridine derivatives having antithrombotic activity
08/15/2002WO2002062803A1 Thienopyrimidine derivative
08/15/2002WO2002062789A1 Pyrazole compounds useful as protein kinase inhibitors
08/15/2002WO2002062764A1 Fused heterocyclic compounds
08/15/2002WO2002062343A2 PHARMACEUTICAL FORMULATION COMPRISING PYRAZOLO[4,3-d]PYRIMIDINES AND ENDOTHELIN RECEPTOR ANTAGONISTS OR THIENOPYRIMIDINES AND ENDOTHELIN RECEPTOR ANTAGONISTS
08/15/2002WO2002042244A3 Synthesis of chiral intermediates useful in preparing pharmacologically active compounds
08/15/2002WO2002030860A3 Ketone compounds and compositions for cholesterol management and related uses
08/15/2002CA2437492A1 Fused heterocyclic compounds
08/15/2002CA2437085A1 Pharmaceutical formulation comprising pyrazolo[4,3-d]pyrimidines and endothelin receptor antagonists or thienopyrimidines and endothelin receptor antagonists
08/14/2002EP1230244A2 Pyrazolecarboxylic acid tricyclic derivatives, preparation and pharmaceutical compositions containing same
08/14/2002EP1230225A2 Pharmaceutically active 4-substituted pyrimidine derivatives
08/14/2002EP1229912A1 Protease inhibitors
08/14/2002EP1229911A1 Protease inhibitors
08/14/2002EP1087976B1 Polymorphic clopidogrel hydrogenesulphate form
08/14/2002EP0722439B1 Hiv protease inhibitors
08/14/2002DE10106457A1 DELTA·1·-Pyrroline DELTA · 1 · -Pyrrolines
08/13/2002US6433167 Triazolo-1,4-diazepine compounds and medicinal composition containing the same
08/13/2002US6433165 Chemokine receptor antagonists and methods of use therefor
08/13/2002US6432964 Fungicides
08/13/2002US6432955 Heterocyclic derivatives and their use as antithrombotic agents
08/13/2002US6432943 Method for treating sexual dysfunction
08/08/2002WO2002060906A2 Crystal modification of olanzapine
08/08/2002WO2002060894A2 Sulfonamide lactam inhibitors of factor xa
08/08/2002WO2002060872A1 Synthesis for the preparation of compounds for screening as potential tubulin binding agents
08/08/2002WO2002060858A1 Novel compound having maillard reaction inhibitory activity
08/08/2002WO2002060449A2 Pharmaceutical formulation containing pyrazolo[4,3-d]pyrimidine and nitrates or thienopyrimidines and nitrates
08/08/2002WO2002034716A3 Pyrrolidine modulators of ccr5 chemokine receptor activity
08/08/2002WO2002024650A3 Pyridinone and pyridinethione derivatives having hiv inhibiting properties
08/08/2002WO2002014269A3 2,4-substituted pyridine derivatives
08/08/2002WO2001093840A3 Ligands of integrin receptors
08/08/2002WO2001064685A3 Thienopyridine derivatives and their use as anti-inflammatory agents
08/08/2002US20020107411 Such as 25-hydroxy-3-aminopropoxyvitamin D3 biotinamide; kits
08/08/2002US20020107402 Aminoaryl oxazolidinone N-oxides
08/08/2002US20020107263 Squaric acid derivatives
08/08/2002CA2436774A1 Sulfonamide lactam inhibitors of factor xa
08/08/2002CA2436209A1 Pharmaceutical formulation containing pyrazolo[4,3-d]pyrimidine and nitrates or thienopyrimidines and nitrates
08/08/2002CA2435545A1 Synthesis for the preparation of compounds for screening as potential tubulin binding agents
08/07/2002EP1228063A2 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
08/07/2002EP1228060A1 Arylalkane, arylalkene and aryl azaalkane, medicaments containing said compounds and method for the production thereof
08/07/2002CN1362397A Dialkoyl-halogen phenyl substituted keto-enol
08/07/2002CN1088709C Amine compound and its acid addition salt
08/07/2002CN1088702C Disubstituted bicyclic heterocycles, their production and use as medicaments
08/06/2002US6429210 Orthorombic polymorph of clopidogrel hydrogen sulfate with improved stability and lower solubility; antithrombotic agent; specific crystal structure and thermodynamic properties
08/06/2002CA2231812C Cyclic nitrones and pharmaceutical compositions containing them
08/01/2002WO2002059128A2 Process for preparing clopidogrel
08/01/2002WO2002059112A2 Pyrazole compounds useful as protein kinase inhibitors
08/01/2002WO2002059111A2 Pyrazole compounds useful as protein kinase inhibitors
08/01/2002WO2002029409A3 Method of assaying pyrrole-containing biological compounds
08/01/2002WO2002012227A3 Indole, azaindole and indazole derivatives having vegf inhibiting activity
08/01/2002US20020103376 Dithiepino[6,5-b]pyridines, and related compositions and methods
08/01/2002US20020103234 Heterocycl-containing carboxylic acid derivative and drug containing the same
08/01/2002US20020103230 Heterocyclic compounds
08/01/2002US20020103213 Pyrimidone compounds which are inhibitors of the enzyme Lp-PLA2; use in treating atheroscelerosis
08/01/2002US20020102608 Library of indolinone compounds for use in the treatment of cancer
07/2002
07/31/2002EP1226193A2 Process for the preparation of ethylene polymers
07/31/2002EP1226146A2 Quinoline and naphthyridine carboxylic acid antibacterials
07/31/2002EP1226138A1 Fab i inhibitors
07/31/2002EP1226122A1 Bicyclic vasopressin agonists
07/31/2002EP1226119A2 Tyrosine kinase inhibitors
07/31/2002EP0527801B1 Thiophene sulfonamides useful as carbonic anhydrase inhibitors
07/31/2002CN1361779A New compounds
07/31/2002CN1361774A Heterocyclic substituted aminoazacycles useful as central nervous system agents
07/31/2002CN1361687A Phosphate transport inhibitors
07/31/2002CN1360891A Dithiolane amylene hepyrroleketone and its relative monoxide and dioxide using as antitumour agent
07/30/2002US6426350 Alpha-2 adrenoceptor antagonists; use treating nervous system disorders
07/30/2002US6426023 Benzopyrans annelated in C7-C8 with an aromatic heterocycle and compositions and (CO)polymer matrices containing them
07/30/2002CA2237357C Stable biotinylated biomolecule composition and methods
07/25/2002WO2002057271A2 Thienopyrimidine-based inhibitors of the src family
07/25/2002WO2002057259A2 Pyrazole compounds useful as protein kinase inhibitors
07/25/2002WO2002057242A2 Urea derivatives as integrin alpha 4 antagonists
07/25/2002WO2002020529A8 METHOD FOR OBTAINING 4-(N-ALKYLAMINE)-5, 6-DIHYDRO-4H-THIENO-(2,3-b)-THIOPYRAN-2-SULFAMIDE-7, 7-DIOXIDES AND INTERMEDIATE PRODUCTS
07/25/2002WO2002000653A3 Fused cyclic compounds as modulators of nuclear hormone receptor function
07/25/2002US20020099212 Sulfonamide compounds and pharmaceutical use thereof
07/25/2002US20020099073 5-(Benzoylaminomethyl)-2-(oxalyl-amino)-4,5,6,7-tetrahydro -thieno(2,3-c)pyridine-3-carboxylic acid for example; useful treating diabetes, type 2 diabetes, impaired glucose tolerance, insulin resistance, obesity
07/25/2002US20020099065 Novel 3, 5, and/or 6 substituted analogues of swainsonine, processes for their preparation and their use as therapeutic agents
07/25/2002US20020099055 Novel compounds
07/25/2002US20020098556 Generating preferential compound in culture; obtain genetically engineered bacteria, culturing, recover preferential compound
07/25/2002DE10101397A1 New reagent for biotinylation of substrates, useful e.g. in medical research, comprises biotin linked to a solid particle through N-alkyl-N-acylsulfonamide
07/25/2002CA2434939A1 Urea derivatives as integrin alpha 4 antagonists
07/25/2002CA2426775A1 Thienopyrimidine-based inhibitors of the src family
07/24/2002EP1224187A2 Certain alkylene diamine-substituted heterocycles
07/24/2002EP1224183A2 Heterocyclic sodium/proton exchange inhibitors and method
07/24/2002EP0820454B1 Anellated beta-carbolines
07/24/2002CN1360582A Quinazoline derivs.
07/23/2002US6423840 Forming n-acylamino compound
07/23/2002US6423711 Useful in diagnosis and therapy of anxiety, down syndrome, sleep, cognitive and seizure disorders, and overdose with benzodiazepine drugs and for enhancement of alertness
07/18/2002WO2002055524A1 THIENO(3,2-d)PYRIMIDINES AND FURANO(3,2-d)PYRIMIDINES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS
07/18/2002WO2002040455A8 Substituted amidoalkyl uracils and their use as inhibitors of the poly(adp-ribose) synthetase (pars)
07/18/2002WO2002012249A3 Substituted pyrrole compounds and their use as spla2 inhibitors
07/18/2002WO2002000623A3 Aryl fused substituted 4-oxy-pyridines
07/18/2002WO2001083480A3 Dihydropyridine compounds and methods of use
07/18/2002US20020094999 Highly selective butyrylcholinesterase inhibitors for the treatment and diagnosis of Alzheimer's disease and dementias
07/18/2002US20020094977 Benzo(3,4)pyrido(3,2-a)cycloctenes and benzo(3,4)pyrido-(3,2-a)oxocins, -thiocins or azocines; anticholesterol, antilipemic agents; lowering LDL cholesterol; increasing HDl cholesterol; hypertriglyceridemia and atherosclerosis
07/18/2002CA2434005A1 Thieno(3,2-d)pyrimidines and furano(3,2-d)pyrimidines and their use as purinergic receptor antagonists
07/17/2002EP1222193A2 Imidazole derivatives as phosphodiesterase vii inhibitors