Patents
Patents for C07D 495 - Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms (21,336)
03/2003
03/19/2003CN1103217C Aqueous eye drops containing apafant as active ingredient
03/18/2003US6534520 Antiviral compounds
03/18/2003US6534491 Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
03/13/2003WO2003020730A1 4-thioxo-4,7-dihydro-thieno[2,3-b]pyridine-5-carbothioamides as antiviral agents
03/13/2003WO2003020729A1 4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOXAMIDES AS ANT IVIRAL AGENTS
03/13/2003WO2003020728A1 4-THIOXO-4,7-DIHYDRO-THIENO[2,3-b]PYRIDINE-5-CARBOTHIOAMIDES AS ANTIVIRAL AGENTS
03/13/2003WO2003020727A1 GLYCINE-SUBSTITUTED THIENO [2,3-d]PYRIMIDINES WITH COMBINED LH AND FSH AGONISTIC ACTIVITY
03/13/2003WO2003020726A1 Thieno[2,3-d]pyrimidines with combined lh and fsh agonistic activity
03/13/2003WO2003020700A2 SUBSTITUTED INDENO[1,2-c]ISOQUINOLINE DERIVATIVES AND METHODS OF USE THEREOF
03/13/2003WO2003020264A1 Remedial agent for cancer and cancer preventive
03/13/2003WO2002096359A3 Piperazine pentanamide hiv protease inhibitors
03/13/2003WO2002076950A3 Imidiazole derivatives and their use as agonists selective at alpha 2b or 2b/2c adrenergic receptors
03/13/2003WO2002066469A3 Novel heterocyclic amide derivatives and their use as dopamine d3 receptor ligands
03/13/2003US20030050320 A therapeutic agent for treating hepatitis C, based on polymerase inhibitory activity
03/13/2003US20030047719 For use as semiconductors or charge transport materials in optical, electrooptical or electronic devices including field effect transistors, electroluminescent, photovoltaics, sensors and electrophotographic recording devices
03/13/2003CA2457534A1 Substituted indeno[1,2-c]isoquinoline derivatives and methods of use thereof
03/13/2003CA2452438A1 4-thioxo-4,7-dihydro-thieno¬2,3-b|pyridine-5-carbothioamides as antiviral agents
03/13/2003CA2452431A1 4-thioxo-4,7-dihydro-thieno¬2,3-b|pyridine-5-carboxamides as antiviral agents
03/12/2003EP1291023A1 Sustained release compositions
03/12/2003EP1289985A2 Beta-carboline derivatives useful as inhibitors of phosphodiesterase
03/12/2003EP1289980A1 Bicyclyl or heterobicyclylmethanesulfonylamino-substituted n-hydroxyformamides
03/12/2003EP1289563A2 Biotin derivatives
03/12/2003EP1289525A2 Tricyclic pyrazole derivatives as protein kinase inhibitors
03/11/2003US6531604 Useful as medicines having an osteogenesis promoting effect and chondrogensis promoting effect.
03/06/2003WO2003018590A1 Process for producing thienopyridine derivative
03/06/2003WO2003018548A2 Halogenated calixpyrroles, calixpyridinopyrroles and calixpyridines, and uses thereof
03/06/2003WO2003018012A1 Preventive agent/remedial agent for constipation predominant ibs
03/06/2003WO2003018002A2 Cyclopropyl and cyclobutyl epothilone analogs
03/06/2003WO2002042427A3 Mass tags for quantitative analysis
03/06/2003US20030045540 Nicotinic acetylcholine receptors antagonists; central nervous system disorder treatments
03/06/2003US20030045516 Chemokine receptor antagonists and methods of use therefor
03/06/2003US20030045432 Phenyl-substituted cyclic ketoenols
03/06/2003US20030044399 Method of treatment
03/06/2003CA2456280A1 Cyclopropyl and cyclobutyl epothilone analogs
03/05/2003EP1288206A1 Substituted benzenesulfonamide derivatives as prodrugs of COX-2 inhibitors
03/05/2003EP1288203A1 Cyclic nitrones and pharmaceutical compositions containing them
03/05/2003EP1287001A1 Thiophene derivatives useful as anticancer agents
03/05/2003EP1286994A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
03/05/2003EP1286973A2 Novel carbamates and carbamides, production and use thereof as endothelin receptor antagonists
03/05/2003EP1286673A2 Ligands of integrin receptors
03/05/2003EP1185534B1 Benzopyrans annelated in c7-c8 with an aromatic heterocycle and compositions and (co)polymer matrices containing them
03/05/2003EP0892791B1 N-[[4-(5-METHYL-3-PHENYLISOXAZOL-4-YL]PHENYL]SULFONYLPROPYLAMIDE and its SODIUMSALT AS PRODRUGS OF COX-2 INHIBITORS
03/05/2003EP0792273B1 Bicyclic oxazine and thiazine oxazolidinone antibacterials
03/05/2003EP0690863B1 Tetracyclic compounds as dopamine agonists
03/05/2003CN1400969A Fused imidazolium derivatives
03/05/2003CN1102594C Agent for suppressing interferencein immuno assaying
03/04/2003US6528662 Process for the preparation of 3, 4-alkylenedioxythiophene-2,5-dicarboxylic acid derivatives
03/04/2003US6528653 Thienopyrrolidinones
03/04/2003US6528627 Bridged aromatic substituted amine ligands with donor atoms
02/2003
02/27/2003WO2003016316A1 Diazacycloalkanes as oxytocin agonists
02/27/2003WO2003016302A1 Diamine derivatives
02/27/2003WO2003016248A2 Bicyclic hydroxamates as inhibitors of matrix metalloproteinases and/or tnf-$g(a) converting enzyme (tace)
02/27/2003WO2002100862A3 Novel substituted tetracyclic imidazole derivatives, processes for their preparation, pharmaceutical compositions comprising them and their use as a medicine
02/27/2003WO2002100851A3 Thiophene derivatives as antiviral agents for flavivirus infection
02/27/2003US20030040631 As chemical intermediates used for the preparation of S-alpha-ethyl-2-oxo-1-pyrrolidine acetamide
02/27/2003US20030040521 For controlling and preventing pests
02/27/2003CA2456841A1 Cyclohexyl and piperidine diamine derivatives useful as activated blood coagulation factor x inhibitors
02/27/2003CA2453962A1 Diazacycloalkanes as oxytocin agonists
02/26/2003EP1284977A1 Thienodibenzoazulene compounds as tumor necrosis factor inhibitors
02/26/2003EP1011726B1 Fused imidazole derivatives for improving oral bioavailability of pharmaceutical agents
02/26/2003EP0920431B1 Thienopyrimidines
02/26/2003CN1102144C Noval pyrimidine derivatives and prepn. processes thereof
02/25/2003US6525215 HIV protease inhibitors
02/25/2003US6525193 Aminoaryl oxazolidinone N-oxides
02/25/2003US6525070 Bipiperidine derivatives as modulators of CCR3 activity and as H1 antagonists
02/25/2003US6525042 Sulfonyl derivatives
02/25/2003US6525025 Controlling apoptosis; cardiovascular disorders; central nervous system disorders
02/20/2003WO2003013655A2 Carbonic anhydrase inhibitors
02/20/2003WO2003013522A1 Preventives/remedies for cholinergic neuropathy
02/20/2003WO2002072585A3 Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics
02/20/2003WO2002068399B1 Aryl carbamate derivatives, preparation and use thereof
02/20/2003WO2002030860A9 Ketone compounds and compositions for cholesterol management and related uses
02/20/2003US20030036612 Containing a ligand such as (3-methyl-4-trimethylsilyl-1-cyclopentadienyl)-7-(2,5-dimethyl -cyclopenta(1,2-b:4,3-b')-dithiophene)dimethylsilane
02/20/2003US20030036603 E.g., spiro(7-oxa-5-norbornene-2,3'- succinic anhydride, -tetrahydrofuran-2'-one, and -(2',2'-dimethyl)tetrahydrofuran))
02/20/2003US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease.
02/20/2003CA2456939A1 Carbonic anhydrase inhibitors
02/20/2003CA2456594A1 Preventives/remedies for cholinergic neuropathy
02/19/2003EP1119571B1 Tricyclic delta3-piperidines as alpha2-antagonists
02/19/2003EP0971931B1 Method for debenzylation of dibenzyl biotin
02/19/2003EP0799218B1 Diaryl-2-(5h)-furanones as cox-2 inhibitors
02/19/2003CN1101820C Method for debenzylation of dibenzyl biotin
02/19/2003CN1101680C Use of thienotriazolodia zepine to increase apolipoprotein A-I levels
02/18/2003US6521622 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
02/18/2003US6521620 Suppressing tumors, especially breast cancers; antiproli-ferative agents; arthritis, vascular restenosis, psoriasis and angiogenesis; extremely low cytotoxicity
02/13/2003WO2003011872A1 Platelet adp receptor inhibitors
02/13/2003WO2003011869A1 Radioligands and their use for identifying potassium channel modulators
02/13/2003WO2003011868A1 Thienopyrimidinediones and their use in the modulation of autoimmune disease
02/13/2003WO2003011858A1 Substituted isoindoles and e use thereof
02/13/2003US20030032652 Hydroxamic and carboxylic acid derivatives
02/13/2003CA2468925A1 Platelet adp receptor inhibitors
02/13/2003CA2455772A1 Substituted isoindoles and their use
02/13/2003CA2453274A1 Thienopyrimidinediones and their use in the modulation of autoimmune disease
02/12/2003EP0937078B1 Tricyclic carbapenem compounds
02/12/2003EP0926146B1 Chromene compounds
02/11/2003US6518427 Compounds are exceedingly water soluble which is useful in preparing pharmaceutical formulations of these compounds. They are also rapidly converted back to the parent amines in vivo, making them useful as prodrugs of the parent amines.
02/11/2003US6518286 Compounds
02/11/2003US6518267 Protease inhibitors
02/11/2003US6518265 1H-imidazopyridine derivatives
02/11/2003CA2205274C Novel 2,3 disubstituted-(5,6)-heteroarylfused-pyrimidine-4-ones
02/06/2003WO2003009852A1 Tyrosine kinase inhibitors