Patents
Patents for C07D 495 - Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms (21,336)
04/2003
04/16/2003EP1301493A2 Heterocycle carboxamides as antiviral agents
04/16/2003EP1301488A1 Squaric acid derivatives containing a bicyclic heteroaromatic ring as integrin antagonists
04/16/2003CN1411461A Thienopyridine derivatives and their preparing process and use
04/16/2003CN1105723C Spirocyclic metalloprotease inhibitors
04/15/2003US6548524 Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
04/15/2003US6548515 Use as anticancer agents
04/15/2003US6548493 Substituted heterocycle fused gamma-carbolines
04/15/2003CA2070573C Derivatives of amide analogs of certain methano bridged quinolizines
04/11/2003CA2506646A1 Serotonin transport inhibitors
04/10/2003WO2003028733A1 Tetracyclic indole derivatives as 5-ht receptor ligands
04/10/2003WO2002102793A3 Quinazolinediones as antibacterial agents
04/10/2003WO2002071827A3 Retinoid x receptor modulators
04/10/2003US20030069287 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
04/10/2003US20030069275 Substituted acid derivatives useful as antidiabetic and antiobesity agents and method
04/10/2003US20030069267 Modulators of protein tyrosine phosphatases (PTPases)
04/10/2003CA2453343A1 Tetracyclic indole derivatives as 5-ht receptor ligands
04/09/2003EP1299394A1 Method for preparing (+)-biotine
04/09/2003EP1299393A2 4-phenyl substituted tetrahydroisoquinolines and therapeutic use thereof
04/09/2003EP1299378A1 Tetrahydropyridino or piperidino heterocyclic derivatives
04/09/2003EP1299094A2 Selective androgen receptor modulators and methods for their identification, design and use
04/09/2003EP0892793B1 Substituted tetracyclic tetrahydrofuran derivatives
04/09/2003CN1105116C Thienopyrimidine with PDE V-inhibiting effect
04/09/2003CN1105113C Fungicidal pyrimidinones
04/08/2003USRE38073 Biosynthesis; using dehydration agent
04/08/2003US6545033 GABA receptor inhibitors
04/08/2003US6545014 Glaucoma; adjusting concentration of nitric oxide; hypotensive, antispasmodic, antiischemic, cardiotonic agents; bronchodilators; urogentital disorders; agonists, antagonists for endothelin receptors
04/08/2003US6544979 Fused imidazole derivatives for improving oral bioavailability of pharmaceutical agents
04/08/2003CA2112165C Bicyclic amine derivatives
04/08/2003CA2097824C Functionalized vinyl azoles and their use
04/03/2003WO2002092563A3 Protease inhibitors
04/03/2003US20030065182 Therapy for asthma, sexual disorders, hypotensive agents, analgesics
04/03/2003US20030065018 Substituted 4H-chromenes and analogs as activators of caspases and inducers of apoptosis and the use thereof
04/03/2003US20030065007 Analgesics; psychological disorders; antidepressants
04/03/2003US20030064997 Novel compounds
04/03/2003US20030064985 Prevent virus reproduction
04/03/2003US20030064982 Pyrazole compounds useful as protein kinase inhibitors
04/03/2003US20030064981 Anticancer agents; antidiabetic agents; Alzheimer's disease
04/03/2003US20030064979 Antiproliferative agent; antidiabetic agents
04/03/2003US20030064954 Gene therapy; vaccines; calcium channel blockers; cardiovascular disorders
04/03/2003DE20023184U1 New stable polymorphic forms of olanzapine, useful for treating psychotic conditions, mild anxiety and gastrointestinal conditions
04/02/2003EP1298133A1 Procedure for the alkylation of 3,4-dihydroxythiophene-2,5-dicarboxylic esters
04/02/2003EP1298132A1 Hydropyridine derivative acid addition salts
04/02/2003EP1296990A2 Dihydropyridine compounds for the inhibition of calcium-influx
04/02/2003EP1296972A1 Arylmethylamine derivatives for use as tryptase inhibitors
04/02/2003EP0770081B1 Heterocycle-condensed morphinoid derivatives
04/02/2003CN1407988A Method for producing thienopyrimidines
04/02/2003CN1407970A Urea compounds having muscarinic receptor antagonist activity
04/01/2003US6541669 Multibinding amine compounds which are beta 2 adrenergic receptor agonists useful in treatment and prevention of respiratory diseases such as asthma, bronchitis
04/01/2003US6541635 Silylprotected L-proline derivative or salt is deprotected in presence of a nonaqueous medium containing an organic solvent at a temperature of 5 degree C. to 40 degree C.
04/01/2003US6541630 Fungicides
04/01/2003US6541481 Substituted bicyclic derivatives useful as anticancer agents
04/01/2003US6541477 Inhibitors of p38-a kinase
04/01/2003US6541474 Administering a pharmaceutically effective dose of the heterocycle-containing carboxylic acid derivative or salt to a patient suffering form acute promyelocytic leukemia
04/01/2003US6541470 Have a potent antiviral activity against picornaviruses and rotaviruses.
03/2003
03/28/2003WO2002026745A1 Thienopyrimidine compounds and their salts and process for preparation of both
03/28/2003CA2423981A1 Thienopyrimidine compounds and salts thereof and process for the preparation of the same
03/27/2003WO2003024973A1 Spirocyclic-6,7-dihydro-5h-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
03/27/2003WO2003024971A1 6,7-dihydro-5h-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
03/27/2003WO2003024970A1 Compounds which inhibit the release of inflammatory cytokines
03/27/2003WO2003024962A1 Piperidine derivatives and their use as modulators of chemokine (especially ccr3) activity
03/27/2003WO2003024936A1 Substituted pyrazolo compounds for the treatment of inflammation
03/27/2003WO2003024448A2 Inhibitors of histone deacetylase
03/27/2003US20030060462 Therapeutic compounds
03/27/2003US20030059785 Detection of markers in nascent proteins
03/27/2003CA2465978A1 Inhibitors of histone deacetylase
03/27/2003CA2461073A1 6,7-dihydro-5h-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
03/27/2003CA2461072A1 Compounds which inhibit the release of inflammatory cytokines
03/27/2003CA2461071A1 Spirocyclic-6,7-dihydro-5h-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
03/26/2003EP1294729A1 2-aminoalkyl-thieno[2,3-d]pyrimidines
03/26/2003EP1294728A1 HMG-CoA REDUCTASE INHIBITORS AND METHOD
03/26/2003EP1294725A2 Multicyclic compounds and the use thereof as inhibitors of parp, vegfr2 and mlk3 enzymes
03/26/2003EP1294707A2 Thiophene derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
03/26/2003EP1294698A1 Fused azepine derivatives and their use as antidiuretic agents
03/26/2003CN1406239A Process for the production of thienopyrimidine derivatives
03/25/2003WO2003000254A1 Fused cyclic compounds and medicinal use thereof
03/25/2003US6538009 Pyrazole derivatives as anti-inflammatory/analgesic agents
03/25/2003US6538004 Potassium channel modulators relax smooth muscle cells and inhibit bladder contractions; treating nervous, eating, cardiovascular, gastrointestinal, and sexual disorders
03/25/2003US6538002 In particular, these compounds are useful as modulators of the chemokine receptors CCR-5 and/or CCR-3. as antiinflammatory agents
03/25/2003US6538000 9-(3-chloro-4-hydroxyphenyl)-5,6,7,9-tetrahydropyrazolo(5,1-b) quinazoline-8(4H)-one;for cardiovascular disorders
03/25/2003CA2423800A1 Fused cyclic compounds and medicinal use thereof
03/20/2003WO2003022856A1 Substituted 7-aza[2.2.1] bicycloheptanes for the treatment of diseases
03/20/2003WO2003022852A2 Furo-and thienopyrimidine derivatives as angiogenesis inhibitors
03/20/2003WO2003022848A2 Process for the preparation of diketopyrrolopyrroles
03/20/2003WO2003022847A2 Process for the direct preparation of pyrrolo[3,4-c]pyrroles
03/20/2003WO2003022214A2 Piperazine and homopiperazine compounds
03/20/2003WO2003022055A1 Pesticidal compositions
03/20/2003US20030055286 Il-8 receptor antagonists
03/20/2003US20030055269 Reacting a p-phenylacetic acid derivative in an acid halogenating reaction, reacting further with a malonic ester, magnesium alkoxide, sulfur and a nitriloacetic ester in the presence of a primary amine
03/20/2003US20030055130 New thiophenes and polymers derived therefrom
03/20/2003US20030055093 For therapy of cardiovascular diseases, stable or unstable angina pectoris, coronary heart disease, stable or unstable angina pectoris, coronary heart disease, Prinzmetal angina, acute coronary syndrome, heart failure, myocardial infarction
03/20/2003US20030055068 Pyrazole compounds useful as protein kinase inhibitors
03/20/2003US20030055044 Administering pyrazole derivative for inhibiting GSK-3 or Aurora activity in a patient
03/20/2003US20030055035 Useful in hyperpolarizing cell membranes, opening potassium channels, relaxing smooth muscle cells, and inhibiting bladder contractions
03/20/2003CA2460075A1 Substituted 7-aza[2.2.1] bicycloheptanes for the treatment of diseases
03/20/2003CA2457710A1 Process for the direct preparation of pyrrolo¬3,4-c|pyrroles
03/19/2003EP1293503A1 Triazole derivatives
03/19/2003EP1292573A2 Substituted thioacetamides
03/19/2003EP0799228B1 3-aryl-tetronic acid derivatives, the production thereof and the use thereof as anti-parasitic agents
03/19/2003CN1404470A 2-OXo-1-pyrrolidine derivatives, process for preparing them and their uses
03/19/2003CN1404469A 2-Oxo-1-pyrrolidine derivatives, processes for preparing them and their uses