Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
06/2009
06/03/2009EP2064209A1 Pyrrole derivatives with antibacterial activity
06/03/2009EP2064181A1 4, 5-ring annulated indole derivatives for treating or preventing of hcv and related viral infections
06/03/2009EP2064180A1 4,5-ring annulated indole derivatives for treating or preventing of hcv and related viral infections
06/03/2009EP1838715A4 Method for the preparation of maytansinoid esters
06/03/2009EP1694684A4 Process for making camptothecin derivatives
06/03/2009CN101448837A Novel epoxy compound and method for producing the same
06/03/2009CN100494202C Spirofuropyridine aryl derivatives
06/02/2009US7541378 tert-butyl 3-amino-1H-thieno[2,3-c]pyrazole-5-carboxylate; N-benzyl-3-[(4-fluorobenzoyl)amino]-1H-thieno[2,3-c]pyrazole-5-carboxamide; treats a disease caused associated with an altered (disregulated) protein kinase activity e.g cancer, cell proliferative disorders, Alzheimer's disease, viral infections
06/02/2009US7541367 3-benzoimidazolyl-pyrazolopyridines useful in treating kinase disorders
06/02/2009US7541365 heterocylic amines such as 2-(5-{3-[4-(4-Chloro-2-methyl-phenyl)-piperazin-1-yl]-propylidene}-5,11-dihydro-10-oxa-1-aza-dibenzo[a,d]cyclohepten-7-yl)-propan-2-ol, used for treating diseases associated with aberrant leukocyte recruitment and/or activation
06/02/2009US7541364 Compounds of the above formula are useful as analgesics for treating pain; as immunomodulators, to modulate the behavioral effects of drugs of abuse and to modulate the development of tolerance and dependence of mu agonists.
06/02/2009US7541346 Pancratistatin cyclic phosphate prodrugs and phenpanstatin cyclic phosphate prodrugs
06/02/2009US7541332 reporter system reflecting the transport process that transports GPI-anchored proteins to the cell wall was constructed and compounds inhibiting this process were discovered; antifungal agents; inhibiting expression of cell wall glycoproteins and preventing pathogens from showing pathogenicity
06/02/2009CA2474205C E2 displacement assay for identifying inhibitors of hpv
06/02/2009CA2258539C Ring-fused dihydropyranes, process for the preparation and use thereof
05/2009
05/29/2009CA2644817A1 Quartz glass micro-photoreactor and synthesis of 10-hydroxycamptothecin and 7-alkyl 10-hydroxycamptothecin
05/28/2009US20090137806 Dual nk1/nk3 receptor antagonists
05/28/2009US20090137604 corticotropin releasing factor receptor antagonists such as 8-(N-butyl-N-(2-butynyl)amino)-2-methyl-3-(2-chloro-4-methoxyphenyl)-6,7-dihydro-5H-cyclopenta[d]pyrazolo[1,5-a]pyrimidine, used for the treatment of nervous system, psychological, eating, sleep, and gastrointestinal disorders
05/28/2009US20090137586 Compounds for the treatment of inflammatory disorders
05/28/2009US20090137554 1,4,5,6-TETRAHYDRO -PYRROLO[2,3-d]AZEPINES AND -IMIDAZO[4,5-d]AZEPINES AS MODULATORS OF NUCLEAR RECEPTOR ACTIVITY
05/28/2009US20090136979 Class IIA Histone Deacetylase (HDAC) Substrate
05/28/2009US20090136596 P38 inhibitors and methods of use thereof
05/28/2009US20090136448 Antiviral 2-Carboxy-Thiophene Compounds
05/28/2009US20090134784 Carbazole-containing materials in phosphorescent light emitting diodes
05/28/2009CA2706391A1 Spiropiperidines for use as tryptase inhibitors
05/27/2009EP2062901A1 Fluoroboron compound having aromatic ring or salt thereof, and process for production of compound having cyclic ether-fused aromatic ring by using the same
05/27/2009EP2062898A2 Spirocyclic cyclohexane derivatives
05/27/2009EP2061770A1 Piperazine compounds with herbicidal action
05/27/2009EP1519915B1 Tricyclic steroid hormone nuclear receptor modulators
05/27/2009CN101443332A Anti-viral pyrimidine nucleoside derivatives
05/27/2009CN101440097A 1-(3',4',5'- trisubstituted phenyl)- isoquinoline compound and medical use thereof
05/27/2009CN101440096A 1-(3',4',5'- trisubstituted phenyl)- tetrahydroisoquinoline compound and its use
05/27/2009CN101440095A 3-oxa acridone, derivatives thereof and preparation
05/27/2009CN101440073A Aromatic chlorethazine piperazine quaternary ammonium salt derivatives, and preparation and use thereof
05/26/2009US7538220 silyl camptothecin derivatives for cancer and/or leukemia; cytotoxic; DNA-topoisomerase I inhibitors; antitumor agents; 7-trimethylsilyl-10-acetoxy camptothecin, 7-trimethylsilyl-11-fluoro camptothecin
05/26/2009US7538219 Soft anticholinergic zwitterions
05/26/2009US7538138 Histamine-3 receptor antagonists; 4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-4-yl)benzonitrile; acute myocardial infarction, asthma, psychological disorders, gastrointestinal disorders, inflammation, jet lag, cancer, septic shock, Tourette's syndrome, neurodegenerative disorders
05/26/2009US7538123 Indole derivative having piperidine ring
05/26/2009CA2533685C Nitrogen-containing fused heterocyclic carboxylic acid compounds
05/26/2009CA2387201C Tetrahydroquinoline derivatives
05/22/2009WO2009064835A1 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors
05/22/2009WO2009064792A1 Quinolone carboxylic acid-substituted rifamycin derivatives
05/22/2009WO2009064418A1 Substituted hydroxyethyl amine compounds as beta-secretase modulators and methods of use
05/22/2009WO2009063780A1 Organic transistor
05/22/2009WO2009062990A2 Equilibrative nucleoside transporter ent1 inhibitors
05/22/2009WO2009062605A1 Trisubstituted furopyrimidines and the use thereof as activators of the ip receptor
05/22/2009WO2009062289A1 Inhibitors of human immunodeficiency virus replication
05/22/2009WO2009062285A1 Inhibitors of human immunodeficiency virus replication
05/22/2009WO2009037542A3 Spirocyclic compounds as stearoyl coa desaturase inhibitors
05/22/2009WO2008136815A3 5, 6-ring annulated indole derivatives and use thereof
05/22/2009CA2707418A1 Inhibitors of human immunodeficiency virus replication
05/22/2009CA2705689A1 Trisubstituted furopyrimidines and the use thereof as activators of the ip receptor
05/22/2009CA2705318A1 Inhibitors of human immunodeficiency virus replication
05/22/2009CA2704599A1 4-pyrazolyl-n-arylpyrimidin-2-amines and 4-pyrazolyl-n-heteroarylpyrimidin-2-amines as janus kinase inhibitors
05/22/2009CA2704423A1 Equilibrative nucleoside transporter ent1 inhibitors
05/21/2009US20090131682 Supports for oligomer synthesis
05/21/2009US20090131672 3,4-cyclic phosphate prodrugs, including sodium-7-deoxynarcistatin, sodium-7-deoxy-transdihydronarcistatin, and sodium transdihydronarcistatin; anaticarcinogenic agent, antitumor agent; obtained via isolation from the medicinal plant species Narcissus (Amaryllidaceae), as precursors
05/21/2009US20090131502 Biologically active compounds
05/21/2009US20090131501 Alzheimer's disease; administering orally (+) phenserine; phenserine tartrate; racemic or enantiomerically pure; not toxic in a wide range of dosages
05/21/2009US20090131498 Enantioselective Synthesis of Merrilactone and Its Analogs
05/21/2009US20090131435 Heterocyclic inhibitors of mek and methods of use
05/21/2009US20090131419 Which modulates activity of amyloid precursor proteins; Alzheimer's disease
05/21/2009US20090131412 Novel 2-quinolone derivative
05/21/2009US20090130201 polymorphous forms of rifaximin, processes for their production and use thereof in the medicinal preparations
05/21/2009US20090126932 Reversible polymeric gelation for oilfield applications
05/20/2009EP2059519A2 Nitrogen-containing heterocyclic compounds and methods of use thereof
05/20/2009EP1270549B1 Polymer-immobilized alpha-iminoester
05/20/2009DE102007054786A1 Trisubstituierte Furopyrimidine und ihre Verwendung Trisubstituted Furopyrimidine and their use
05/20/2009CN101437827A Process for producing optically active chromene oxide compound
05/20/2009CN101437816A 2-aminopyridine analogs as glucokinase activators
05/19/2009US7534799 Pyridomorphinans, thienomorphinans and use thereof
05/19/2009US7534797 6,6-Bicyclic ring substituted heterobicyclic protein kinase inhibitors
05/19/2009US7534794 Certain arylaliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases
05/19/2009US7534793 (R)-2-{4-[(1H-Indol-2-ylmethyl)-amino]-piperidin-1-yl}-1-(6-methoxyquinolin-4-yl)-ethanol; effective against both gramnegative and grampositive bacteria
05/19/2009US7534790 Aminocyclohexyl ether compounds such as trans-[2-(4-morpholinyl)-1-(2-naphthenethoxy)]cyclohexane; arrhythmia, analgesia and local anesthesia
05/19/2009US7534767 4-amino-7-(2-C-methyl- beta -D-ribofuranosyl)-furo[3,2-d]pyrimidine; 7-amino-3-(2-C-methyl- beta -D-ribofuranosyl)-1H-pyrazolo[4,3-d]pyrimidine; -amino-7-(2-C-methyl- beta -D-ribofuranosyl)-5H-pyrrolo[3,2-d]pyrimidine; hepatitis C virus (HCV) infection
05/14/2009WO2009061597A1 Compounds for inhibiting ksp kinesin activity
05/14/2009WO2009060835A1 Novel ubiquilin-binding small molecule
05/14/2009WO2008118823A3 Compositions and methods for inhibition of the jak pathway
05/14/2009WO2007067711A3 Certain chemical entities, compositions, and methods for modulating trpv1
05/14/2009US20090124649 Aza spiro alkane derivatives as inhibitors of metalloproteases
05/14/2009US20090124648 Such as trans-N-[1-(2-fluorophenyl)-S-pyrazoly]-3-ox-ospiro[6-azaisobenzofuran-1(3H),1'-cyclohexane]-4'-carboxamide and novel salts, hydrates and polymorphs thereof; neuropeptide y5 (NPY5)
05/14/2009CA2702995A1 Compounds for inhibiting ksp kinesin activity
05/13/2009EP2058315A1 1H-Furo[3,2-C]Pyrazoles active as aurora kinase inhibitors
05/13/2009EP2058303A1 Method for producing piperidin-4-one-derivative
05/13/2009EP2057169A2 Compositions and methods of making a chlorin e6 derivative as a photoactive agent
05/13/2009EP2057162A2 Fused heterocyclic inhibitors of d-amino acid oxidase
05/13/2009EP2057124A2 Compounds and compositions as itpkb inhibitors
05/13/2009CN101432288A Process for production of camptothecin derivative
05/13/2009CN101429232A Hcv protease inhibitors
05/13/2009CN101429201A Lemon acid berbamine salt, preparation method and application thereof
05/13/2009CN101429200A Tricyclic benzopyran compound as anti-arrhythmic agents
05/13/2009CN100486973C Novel benzodioxoles
05/13/2009CN100486967C 5HT2C receptor modulators
05/12/2009US7531554 Useful as an anti-HIV agent that particularly shows an anti-HIV action based on an integrase inhibitory activity; for treatment or prophylaxis of AIDS; for example, 6-(2,3-dichlorobenzyl)-1-(2-hydroxyethyl)-4-oxo-1,4-dihydroquinoline-3-carboxylic acid
05/12/2009US7531550 Pseudobase benzo[c]phenanthridines with improved efficacy, stability, and safety
05/12/2009US7531536 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
05/12/2009CA2278553C Phenylsulfonylureas, processes for their preparation, and their use as herbicides and plant growth regulators
05/07/2009WO2009059272A1 Thienopyrimidines, thienopyridines, and pyrrolopyrimidines as b-raf inhibitors
05/07/2009WO2009058728A1 Thiazole derivatives as protein kinase inhibitors
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